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Jerome Charles Bressi, Ph.D. - Publications

Affiliations: 
2000 University of Washington, Seattle, Seattle, WA 
Area:
medicinal enzymology
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9 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2010 Bressi JC, Jennings AJ, Skene R, Wu Y, Melkus R, De Jong R, O'Connell S, Grimshaw CE, Navre M, Gangloff AR. Exploration of the HDAC2 foot pocket: Synthesis and SAR of substituted N-(2-aminophenyl)benzamides. Bioorganic & Medicinal Chemistry Letters. 20: 3142-5. PMID 20392638 DOI: 10.1016/j.bmcl.2010.03.091  0.477
2002 Verlinde C, Bressi J, Choe J, Suresh S, Buckner F, Voorhis WV, Michels P, Gelb M, Hol W. Protein structure-based design of anti-protozoal drugs Journal of the Brazilian Chemical Society. 13: 843-844. DOI: 10.1590/S0103-50532002000600018  0.379
2002 Verlinde CLMJ, Bressi JC, Choe J, Suresh S, Buckner FS, Van Voorhis WC, Michels PAM, Gelb MH, Hol WGJ. Protein structure-based design of anti-protozoal drugs Journal of the Brazilian Chemical Society. 13: 843-848.  0.431
2001 Bressi JC, Verlinde CL, Aronov AM, Shaw ML, Shin SS, Nguyen LN, Suresh S, Buckner FS, Van Voorhis WC, Kuntz ID, Hol WG, Gelb MH. Adenosine analogues as selective inhibitors of glyceraldehyde-3-phosphate dehydrogenase of Trypanosomatidae via structure-based drug design. Journal of Medicinal Chemistry. 44: 2080-93. PMID 11405646 DOI: 10.1021/Jm000472O  0.585
2001 Suresh S, Bressi JC, Kennedy KJ, Verlinde CL, Gelb MH, Hol WG. Conformational changes in Leishmania mexicana glyceraldehyde-3-phosphate dehydrogenase induced by designed inhibitors. Journal of Molecular Biology. 309: 423-35. PMID 11371162 DOI: 10.1006/Jmbi.2001.4588  0.591
2001 Kennedy KJ, Bressi JC, Gelb MH. A disubstituted NAD+ analogue is a nanomolar inhibitor of trypanosomal glyceraldehyde-3-phosphate dehydrogenase. Bioorganic & Medicinal Chemistry Letters. 11: 95-8. PMID 11206479 DOI: 10.1016/S0960-894X(00)00608-9  0.569
2000 Bressi JC, Choe J, Hough MT, Buckner FS, Van Voorhis WC, Verlinde CL, Hol WG, Gelb MH. Adenosine analogues as inhibitors of Trypanosoma brucei phosphoglycerate kinase: elucidation of a novel binding mode for a 2-amino-N(6)-substituted adenosine. Journal of Medicinal Chemistry. 43: 4135-50. PMID 11063610 DOI: 10.1021/Jm000287A  0.587
2000 Golisade A, Bressi JC, Van Calenbergh S, Gelb MH, Link A. Polymer-assisted solution-phase synthesis of 2'-amido-2'-deoxyadenosine derivatives targeted at the NAD(+)-binding sites of parasite enzymes. Journal of Combinatorial Chemistry. 2: 537-44. PMID 11029179 DOI: 10.1021/Cc0000343  0.487
1998 Bernstein BE, Williams DM, Bressi JC, Kuhn P, Gelb MH, Blackburn GM, Hol WG. A bisubstrate analog induces unexpected conformational changes in phosphoglycerate kinase from Trypanosoma brucei. Journal of Molecular Biology. 279: 1137-48. PMID 9642090 DOI: 10.1006/Jmbi.1998.1835  0.561
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