| Year |
Citation |
Score |
| 2016 |
Miyawaki S, Hirokami Y, Kinami K, Hoshino M, Minehira D, Miyamoto D, Nash RJ, Fleet GW, Adachi I, Toyooka N, Kato A. Strategy for designing selective α-l-rhamnosidase inhibitors: Synthesis and biological evaluation of l-DMDP cyclic isothioureas. Bioorganic & Medicinal Chemistry. PMID 27789075 DOI: 10.1016/J.Bmc.2016.10.015 |
0.402 |
|
| 2016 |
Glawar AF, Martínez RF, Ayers BJ, Hollas MA, Ngo N, Nakagawa S, Kato A, Butters TD, Fleet GW, Jenkinson SF. Structural essentials for β-N-acetylhexosaminidase inhibition by amides of prolines, pipecolic and azetidine carboxylic acids. Organic & Biomolecular Chemistry. PMID 27735004 DOI: 10.1039/C6Ob01549B |
0.352 |
|
| 2016 |
Liu Z, Yoshihara A, Jenkinson SF, Wormald MR, Estévez RJ, Fleet GW, Izumori K. Triacetonide of Glucoheptonic Acid in the Scalable Syntheses of d-Gulose, 6-Deoxy-d-gulose, l-Glucose, 6-Deoxy-l-glucose, and Related Sugars. Organic Letters. PMID 27487167 DOI: 10.1021/Acs.Orglett.6B02041 |
0.803 |
|
| 2016 |
Liu Z, Yoshihara A, Kelly C, Heap JT, Marqvorsen MH, Jenkinson SF, Wormald MR, Otero JM, Estévez A, Kato A, Fleet GW, Estévez RJ, Izumori K. 6-Deoxyhexoses from l-Rhamnose in the Search for Inducers of the Rhamnose Operon: Synergy of Chemistry and Biotechnology. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27439720 DOI: 10.1002/Chem.201602482 |
0.76 |
|
| 2016 |
Kelly CL, Liu Z, Yoshihara A, Jenkinson SF, Wormald MR, Otero JM, Estévez AM, Kato A, Marqvorsen MH, Fleet GW, Estevez RJ, Izumori K, Heap JT. Synthetic chemical inducers and genetic decoupling enable orthogonal control of the rhaBAD promoter. Acs Synthetic Biology. PMID 27247275 DOI: 10.1021/Acssynbio.6B00030 |
0.732 |
|
| 2016 |
Song YY, Kinami K, Kato A, Jia YM, Li YX, Fleet GW, Yu CY. First total synthesis of (+)-broussonetine W: glycosidase inhibition of natural product & analogs. Organic & Biomolecular Chemistry. PMID 27184090 DOI: 10.1039/C6Ob00720A |
0.375 |
|
| 2016 |
Wang HY, Kato A, Kinami K, Li YX, Fleet GW, Yu CY. Concise synthesis of calystegines B2 and B3via intramolecular Nozaki-Hiyama-Kishi reaction. Organic & Biomolecular Chemistry. PMID 27161660 DOI: 10.1039/C6Ob00697C |
0.345 |
|
| 2016 |
Qian BC, Kamori A, Kinami K, Kato A, Li YX, Fleet GW, Yu CY. Epimerization of C5 of an N-hydroxypyrrolidine in the synthesis of swainsonine related iminosugars. Organic & Biomolecular Chemistry. PMID 27093691 DOI: 10.1039/C6Ob00531D |
0.423 |
|
| 2016 |
Li YX, Kinami K, Hirokami Y, Kato A, Su JK, Jia YM, Fleet GW, Yu CY. Gem-difluoromethylated and trifluoromethylated derivatives of DMDP-related iminosugars: synthesis and glycosidase inhibition. Organic & Biomolecular Chemistry. PMID 26790356 DOI: 10.1039/C5Ob02474A |
0.381 |
|
| 2016 |
Kamori A, Kato A, Miyawaki S, Koyama J, Nash RJ, Fleet GW, Miura D, Ishikawa F, Adachi I. Dual action of acertannins as potential regulators of intracellular ceramide levels Tetrahedron: Asymmetry. 27: 1177-1185. DOI: 10.1016/J.Tetasy.2016.09.006 |
0.307 |
|
| 2016 |
Liu Z, Jenkinson SF, Kato A, Nakagawa S, Wormald MR, Yu C, Fleet GW. 3-Azidoazetidines as the first scaffolds for β-amino azetidine carboxylic acid peptidomimetics: azetidine iminosugars containing an acetamido group do not inhibit β- N -acetylhexosaminidases Tetrahedron: Asymmetry. 27: 872-881. DOI: 10.1016/J.Tetasy.2016.08.001 |
0.371 |
|
| 2015 |
Kato A, Nakagome I, Sato K, Yamamoto A, Adachi I, Nash RJ, Fleet GW, Natori Y, Watanabe Y, Imahori T, Yoshimura Y, Takahata H, Hirono S. Docking study and biological evaluation of pyrrolidine-based iminosugars as pharmacological chaperones for Gaucher disease. Organic & Biomolecular Chemistry. PMID 26633162 DOI: 10.1039/C5Ob02223A |
0.372 |
|
| 2015 |
Li YX, Shimada Y, Adachi I, Kato A, Jia YM, Fleet GW, Xiao M, Yu CY. Fluorinated and Conformationally Fixed Derivatives of L-HomoDMDP: Synthesis and Glycosidase Inhibition. The Journal of Organic Chemistry. 80: 5151-8. PMID 25909763 DOI: 10.1021/Acs.Joc.5B00571 |
0.446 |
|
| 2015 |
Liu Z, Jenkinson SF, Vermaas T, Adachi I, Wormald MR, Hata Y, Kurashima Y, Kaji A, Yu CY, Kato A, Fleet GW. 3-Fluoroazetidinecarboxylic Acids and trans,trans-3,4-Difluoroproline as Peptide Scaffolds: Inhibition of Pancreatic Cancer Cell Growth by a Fluoroazetidine Iminosugar. The Journal of Organic Chemistry. 80: 4244-58. PMID 25859886 DOI: 10.1021/Acs.Joc.5B00463 |
0.744 |
|
| 2015 |
Kato A, Zhang ZL, Wang HY, Jia YM, Yu CY, Kinami K, Hirokami Y, Tsuji Y, Adachi I, Nash RJ, Fleet GW, Koseki J, Nakagome I, Hirono S. Design and Synthesis of Labystegines, Hybrid Iminosugars from LAB and Calystegine, as Inhibitors of Intestinal α-Glucosidases: Binding Conformation and Interaction for ntSI. The Journal of Organic Chemistry. 80: 4501-15. PMID 25843107 DOI: 10.1021/Acs.Joc.5B00342 |
0.347 |
|
| 2015 |
Li YX, Shimada Y, Sato K, Kato A, Zhang W, Jia YM, Fleet GW, Xiao M, Yu CY. Synthesis and glycosidase inhibition of australine and its fluorinated derivatives. Organic Letters. 17: 716-9. PMID 25621897 DOI: 10.1021/Ol503728E |
0.416 |
|
| 2015 |
Kato A, Hirokami Y, Kinami K, Tsuji Y, Miyawaki S, Adachi I, Hollinshead J, Nash RJ, Kiappes JL, Zitzmann N, Cha JK, Molyneux RJ, Fleet GW, Asano N. Isolation and SAR studies of bicyclic iminosugars from Castanospermum australe as glycosidase inhibitors. Phytochemistry. 111: 124-31. PMID 25583438 DOI: 10.1016/J.Phytochem.2014.12.011 |
0.36 |
|
| 2014 |
Liu Z, Yoshihara A, Wormald MR, Jenkinson SF, Gibson V, Izumori K, Fleet GW. L-fucose from vitamin C with only acetonide protection. Organic Letters. 16: 5663-5. PMID 25310515 DOI: 10.1021/Ol502733X |
0.77 |
|
| 2014 |
Désiré J, Mondon M, Fontelle N, Nakagawa S, Hirokami Y, Adachi I, Iwaki R, Fleet GW, Alonzi DS, Twigg G, Butters TD, Bertrand J, Cendret V, Becq F, Norez C, et al. N- and C-alkylation of seven-membered iminosugars generates potent glucocerebrosidase inhibitors and F508del-CFTR correctors. Organic & Biomolecular Chemistry. 12: 8977-96. PMID 25277226 DOI: 10.1039/C4Ob00325J |
0.443 |
|
| 2014 |
Crabtree EV, MartÃnez RF, Nakagawa S, Adachi I, Butters TD, Kato A, Fleet GW, Glawar AF. Synthesis of the enantiomers of XYLNAc and LYXNAc: comparison of β-N-acetylhexosaminidase inhibition by the 8 stereoisomers of 2-N-acetylamino-1,2,4-trideoxy-1,4-iminopentitols. Organic & Biomolecular Chemistry. 12: 3932-43. PMID 24802185 DOI: 10.1039/C4Ob00097H |
0.358 |
|
| 2014 |
Ayers BJ, Glawar AF, MartÃnez RF, Ngo N, Liu Z, Fleet GW, Butters TD, Nash RJ, Yu CY, Wormald MR, Nakagawa S, Adachi I, Kato A, Jenkinson SF. Nine of 16 stereoisomeric polyhydroxylated proline amides are potent β-N-acetylhexosaminidase inhibitors. The Journal of Organic Chemistry. 79: 3398-409. PMID 24641544 DOI: 10.1021/Jo500157P |
0.757 |
|
| 2014 |
Ayers BJ, Hollinshead J, Saville AW, Nakagawa S, Adachi I, Kato A, Izumori K, Bartholomew B, Fleet GW, Nash RJ. Iteamine, the first alkaloid isolated from Itea virginica L. inflorescence. Phytochemistry. 100: 126-31. PMID 24534106 DOI: 10.1016/J.Phytochem.2014.01.012 |
0.389 |
|
| 2014 |
Martínez RF, Liu Z, Glawar AF, Yoshihara A, Izumori K, Fleet GW, Jenkinson SF. Short and sweet: (D)-glucose to (L)-glucose and (L)-glucuronic acid. Angewandte Chemie (International Ed. in English). 53: 1160-2. PMID 24310928 DOI: 10.1002/Anie.201309073 |
0.77 |
|
| 2013 |
Ayers BJ, Jenkinson SF, Fleet GW, Thompson AL. 2-N-Benzyl-2,6-dide-oxy-2,6-imino-3,4-O-iso-propyl-idene-d-allono-nitrile. Acta Crystallographica. Section E, Structure Reports Online. 69: o1772. PMID 24454220 DOI: 10.1107/S1600536813030584 |
0.351 |
|
| 2013 |
Zhu JS, Nakagawa S, Chen W, Adachi I, Jia YM, Hu XG, Fleet GW, Wilson FX, Nitoda T, Horne G, van Well R, Kato A, Yu CY. Synthesis of eight stereoisomers of pochonicine: nanomolar inhibition of β-N-acetylhexosaminidases. The Journal of Organic Chemistry. 78: 10298-309. PMID 24032658 DOI: 10.1021/Jo401694E |
0.46 |
|
| 2013 |
Glawar AF, Jenkinson SF, Newberry SJ, Thompson AL, Nakagawa S, Yoshihara A, Akimitsu K, Izumori K, Butters TD, Kato A, Fleet GW. An approach to 8 stereoisomers of homonojirimycin from (D)-glucose via kinetic & thermodynamic azido-γ-lactones. Organic & Biomolecular Chemistry. 11: 6886-99. PMID 23963282 DOI: 10.1039/C3Ob41334A |
0.416 |
|
| 2013 |
Risseeuw M, Overhand M, Fleet GW, Simone MI. A compendium of cyclic sugar amino acids and their carbocyclic and heterocyclic nitrogen analogues. Amino Acids. 45: 613-89. PMID 23955533 DOI: 10.1007/S00726-013-1521-1 |
0.354 |
|
| 2013 |
Jenkinson SF, Best D, Saville AW, Mui J, Martínez RF, Nakagawa S, Kunimatsu T, Alonzi DS, Butters TD, Norez C, Becq F, Blériot Y, Wilson FX, Weymouth-Wilson AC, Kato A, ... Fleet GW, et al. C-branched iminosugars: α-glucosidase inhibition by enantiomers of isoDMDP, isoDGDP, and isoDAB-L-isoDMDP compared to miglitol and miglustat. The Journal of Organic Chemistry. 78: 7380-97. PMID 23688199 DOI: 10.1021/Jo4005487 |
0.419 |
|
| 2013 |
Martínez RF, Araújo N, Jenkinson SF, Nakagawa S, Kato A, Fleet GW. (3R,4S,5R,6R,7S)-3,4,5,7-Tetrahydroxyconidine, an azetidine analogue of 6,7-diepicastanospermine and a conformationally constrained d-deoxyaltronojirimycin, from l-arabinose. Bioorganic & Medicinal Chemistry. 21: 4813-9. PMID 23545138 DOI: 10.1016/J.Bmc.2013.03.004 |
0.371 |
|
| 2013 |
Glawar AF, Jenkinson SF, Thompson AL, Nakagawa S, Kato A, Butters TD, Fleet GW. 3-Hydroxyazetidine carboxylic acids: non-proteinogenic amino acids for medicinal chemists. Chemmedchem. 8: 658-66. PMID 23468173 DOI: 10.1002/Cmdc.201200541 |
0.373 |
|
| 2013 |
Zhao WB, Nakagawa S, Kato A, Adachi I, Jia YM, Hu XG, Fleet GW, Wilson FX, Horne G, Yoshihara A, Izumori K, Yu CY. General synthesis of sugar-derived azepane nitrones: precursors of azepane iminosugars. The Journal of Organic Chemistry. 78: 3208-21. PMID 23458237 DOI: 10.1021/Jo400130P |
0.342 |
|
| 2012 |
Edgeley DS, Martínez RF, Jenkinson SF, Nash RJ, Fleet GW, Thompson AL. N-(2-Carb-oxy-eth-yl)-2,5-dide-oxy-2,5-imino-d-mannonic acid [(3R,4R,5R)-1-(2-carb-oxy-eth-yl)-3,4-dihy-droxy-5-hy-droxy-methyl-l-proline]. Acta Crystallographica. Section E, Structure Reports Online. 68: o2865-6. PMID 23125666 DOI: 10.1107/S1600536812037488 |
0.372 |
|
| 2012 |
Ayers BJ, Ngo N, Jenkinson SF, MartÃnez RF, Shimada Y, Adachi I, Weymouth-Wilson AC, Kato A, Fleet GW. Glycosidase inhibition by all 10 stereoisomeric 2,5-dideoxy-2,5-iminohexitols prepared from the enantiomers of glucuronolactone. The Journal of Organic Chemistry. 77: 7777-92. PMID 22928735 DOI: 10.1021/Jo301243S |
0.395 |
|
| 2012 |
Edgeley DS, Jenkinson SF, Lenagh-Snow G, Rutherford C, Fleet GW, Thompson AL. N-Benzyl-3,5-dide-oxy-3,5-imino-1,2-O-isopropyl-idene-β-l-lyxofuran-ose. Acta Crystallographica. Section E, Structure Reports Online. 68: o2410. PMID 22904864 DOI: 10.1107/S1600536812030656 |
0.412 |
|
| 2012 |
Araújo N, Jenkinson SF, MartÃnez RF, Glawar AF, Wormald MR, Butters TD, Nakagawa S, Adachi I, Kato A, Yoshihara A, Akimitsu K, Izumori K, Fleet GW. Synthesis from D-altrose of (5R,6R,7R,8S)-5,7-dihydroxy-8-hydroxymethylconidine and 2,4-dideoxy-2,4-imino-D-glucitol, azetidine analogues of swainsonine and 1,4-dideoxy-1,4-imino-D-mannitol. Organic Letters. 14: 4174-7. PMID 22839435 DOI: 10.1021/Ol301844N |
0.372 |
|
| 2012 |
Ayers BJ, Jenkinson SF, Fleet GW, Thompson AL. 2-N-Benzyl-2,6-dide-oxy-2,6-imino-3,4-O-isopropyl-idene-3-C-methyl-d-allono-nitrile. Acta Crystallographica. Section E, Structure Reports Online. 68: o1474. PMID 22590347 DOI: 10.1107/S1600536812016273 |
0.379 |
|
| 2012 |
Lenagh-Snow GM, Araújo N, Jenkinson SF, Martínez RF, Shimada Y, Yu CY, Kato A, Fleet GW. Azetidine iminosugars from the cyclization of 3,5-di-O-triflates of α-furanosides and of 2,4-di-O-triflates of β-pyranosides derived from glucose. Organic Letters. 14: 2142-5. PMID 22480242 DOI: 10.1021/Ol300669V |
0.308 |
|
| 2012 |
Lenagh-Snow GM, Jenkinson SF, Newberry SJ, Kato A, Nakagawa S, Adachi I, Wormald MR, Yoshihara A, Morimoto K, Akimitsu K, Izumori K, Fleet GW. Eight stereoisomers of homonojirimycin from D-mannose. Organic Letters. 14: 2050-3. PMID 22472134 DOI: 10.1021/Ol3005744 |
0.354 |
|
| 2011 |
Jenkinson SF, Parry LL, Wilson FX, Fleet GW, Watkin DJ. 6-De-oxy-3,4-O-isopropyl-idene-2-C-methyl-l-galactono-1,5-lactone. Acta Crystallographica. Section E, Structure Reports Online. 67: o2531-2. PMID 22059064 DOI: 10.1107/S1600536811034957 |
0.373 |
|
| 2011 |
Jenkinson SF, Lenagh-Snow GM, Fleet GW, Thompson AL. N-Benzyl-1,3-dide-oxy-1,3-imino-l-xylitol. Acta Crystallographica. Section E, Structure Reports Online. 67: o2452. PMID 22059020 DOI: 10.1107/S160053681103399X |
0.382 |
|
| 2011 |
Lenagh-Snow GM, Araujo N, Jenkinson SF, Rutherford C, Nakagawa S, Kato A, Yu CY, Weymouth-Wilson AC, Fleet GW. Inhibition of nonmammalian glycosidases by azetidine iminosugars derived from stable 3,5-di-O-triflates of pentoses. Organic Letters. 13: 5834-7. PMID 21985023 DOI: 10.1021/Ol2024482 |
0.406 |
|
| 2011 |
Zhang W, Sato K, Kato A, Jia YM, Hu XG, Wilson FX, van Well R, Horne G, Fleet GW, Nash RJ, Yu CY. Synthesis of fully substituted polyhydroxylated pyrrolizidines via Cope-House cyclization. Organic Letters. 13: 4414-7. PMID 21797200 DOI: 10.1021/Ol201749C |
0.375 |
|
| 2011 |
Jenkinson SF, Fleet GW, Nash RJ, Koike Y, Adachi I, Yoshihara A, Morimoto K, Izumori K, Kato A. Looking-glass synergistic pharmacological chaperones: DGJ and L-DGJ from the enantiomers of tagatose. Organic Letters. 13: 4064-7. PMID 21744786 DOI: 10.1021/Ol201552Q |
0.357 |
|
| 2011 |
Jenkinson SF, Fleet GW. Oxetanes from the ring contraction of alpha-triflates of gamma-lactones: oxetane nucleosides and oxetane amino acids. Chimia. 65: 71-5. PMID 21469449 DOI: 10.2533/Chimia.2011.71 |
0.379 |
|
| 2011 |
Li YX, Huang MH, Yamashita Y, Kato A, Jia YM, Wang WB, Fleet GW, Nash RJ, Yu CY. L-DMDP, L-homoDMDP and their C-3 fluorinated derivatives: synthesis and glycosidase-inhibition. Organic & Biomolecular Chemistry. 9: 3405-14. PMID 21423946 DOI: 10.1039/C0Ob01063D |
0.456 |
|
| 2011 |
Simone MI, Edwards AA, Tranter GE, Fleet GW. C-3 branched δ-3,5-cis- and trans-THF sugar amino acids: synthesis of the first generation of branched homooligomers. Amino Acids. 41: 643-61. PMID 21350854 DOI: 10.1007/S00726-011-0849-7 |
0.383 |
|
| 2011 |
da Cruz FP, Newberry S, Jenkinson SF, Wormald MR, Butters TD, Alonzi DS, Nakagawa S, Becq F, Norez C, Nash RJ, Kato A, Fleet GW. 4-C-Me-DAB and 4-C-Me-LAB - enantiomeric alkyl-branched pyrrolidine iminosugars - are specific and potent α-glucosidase inhibitors; acetone as the sole protecting group. Tetrahedron Letters. 52: 219-223. PMID 21157573 DOI: 10.1016/J.Tetlet.2010.10.173 |
0.372 |
|
| 2010 |
Simone MI, Edwards AA, Cowley AR, Fleet GW, Watkin DJ. (3R,4R,5R)-5-(Acetamido-meth-yl)-N-benzyl-3,4-dihy-droxy-tetra-hydro-furan-3-carboxamide. Acta Crystallographica. Section E, Structure Reports Online. 66: o2750-1. PMID 21588955 DOI: 10.1107/S1600536810039589 |
0.386 |
|
| 2010 |
Simone MI, Edwards AA, Parker SG, Tranter GE, Fleet GW, Watkin DJ. Penta-fluoro-phenyl (3R,4R,5S)-5-{[(3R,4R,5S)-5-azido-methyl-3,4-dimeth-oxy-2,3,4,5-tetra-hydro-furan-3-carboxamido]-meth-yl}-3,4-dimeth-oxy-2,3,4,5-tetra-hydro-furan-3-carboxyl-ate. Acta Crystallographica. Section E, Structure Reports Online. 66: o2699-700. PMID 21588915 DOI: 10.1107/S1600536810038559 |
0.352 |
|
| 2010 |
Jenkinson SF, Best D, Wilson FX, Fleet GW, Watkin DJ. (1R,2R,3S,6aS,7R,8R,9S,12aS)-1,2,3,7,8,9-Hexahydroxy-perhydro-dipyrido[1,2-a:1',2'-d]pyrazine-6,12-dione. Acta Crystallographica. Section E, Structure Reports Online. 66: o853. PMID 21580677 DOI: 10.1107/S1600536810009165 |
0.332 |
|
| 2010 |
Jenkinson SF, Lenagh-Snow GM, Izumori K, Fleet GW, Watkin DJ, Thompson AL. 2-Azido-3,4;6,7-di-O-isopropyl-idene-α-d-glycero-d-talo-heptopyran-ose. Acta Crystallographica. Section E, Structure Reports Online. 66: o525-6. PMID 21580298 DOI: 10.1107/S1600536810003995 |
0.379 |
|
| 2010 |
Dai N, Jenkinson SF, Fleet GW, Watkin DJ. 3,4-O-Isopropyl-idene-2-C-methyl-d-galactonolactone. Acta Crystallographica. Section E, Structure Reports Online. 66: o406-7. PMID 21579826 DOI: 10.1107/S1600536810001613 |
0.362 |
|
| 2010 |
Lenagh-Snow GM, Jenkinson SF, Stewart AJ, Fleet GW, Watkin DJ. 1-(1-Carboxy-methyl-1,4-anhydro-2,3-O-isopropyl-idene-α-d-erythrofuranos-yl)thymine. Acta Crystallographica. Section E, Structure Reports Online. 66: o404. PMID 21579824 DOI: 10.1107/S1600536810001704 |
0.383 |
|
| 2010 |
Jenkinson SF, Best D, Izumori K, Wilson FX, Weymouth-Wilson AC, Fleet GW, Thompson AL. 1-De-oxy-1-fluoro-l-galactitol. Acta Crystallographica. Section E, Structure Reports Online. 66: o1330. PMID 21579420 DOI: 10.1107/S1600536810016624 |
0.366 |
|
| 2010 |
Jenkinson SF, Best D, Izumori K, Wilson FX, Weymouth-Wilson AC, Fleet GW, Thompson AL. 6-De-oxy-6-fluoro-d-galactose. Acta Crystallographica. Section E, Structure Reports Online. 66: o1315. PMID 21579408 DOI: 10.1107/S1600536810016612 |
0.34 |
|
| 2010 |
Jenkinson SF, Dai N, Fleet GW, Watkin DJ. 2-Azido-2-de-oxy-3,4-O-isopropyl-idene-2-C-methyl-d-talono-1,5-lactone. Acta Crystallographica. Section E, Structure Reports Online. 66: o1221-2. PMID 21579248 DOI: 10.1107/S160053681001500X |
0.363 |
|
| 2010 |
Jenkinson SF, Crabtree EV, Glawar AF, Butters TD, Fleet GW, Watkin DJ. 2-Acetamido-N-benzyl-1,4-imino-1,2,4-tride-oxy-l-xylitol (N-benzyl-l-XYLNAc). Acta Crystallographica. Section E, Structure Reports Online. 66: o1147-8. PMID 21579195 DOI: 10.1107/S1600536810014145 |
0.367 |
|
| 2010 |
Jenkinson SF, Oña N, Romero A, Fleet GW, Thompson AL, Pino-González MS. 6-Azido-3-O-benzyl-6-de-oxy-N,N-diethyl-1,2-O-isopropyl-idene-d-glycero-α-d-gluco-heptofuran-uronamide. Acta Crystallographica. Section E, Structure Reports Online. 67: o38-9. PMID 21522748 DOI: 10.1107/S1600536810048944 |
0.369 |
|
| 2010 |
Hu XG, Bartholomew B, Nash RJ, Wilson FX, Fleet GW, Nakagawa S, Kato A, Jia YM, van Well R, Yu CY. Synthesis and glycosidase inhibition of the enantiomer of (-)-steviamine, the first example of a new class of indolizidine alkaloid. Organic Letters. 12: 2562-5. PMID 20438104 DOI: 10.1021/Ol1007718 |
0.4 |
|
| 2009 |
Jenkinson SF, Booth KV, Newberry S, Fleet GW, Izumori K, Morimoto K, Nash RJ, Jones L, Watkin DJ, Thompson AL. 2,6-Dide-oxy-2,6-imino-l-glycero-d-ido-heptitol. Acta Crystallographica. Section E, Structure Reports Online. 65: o1755-6. PMID 21583466 DOI: 10.1107/S1600536809025045 |
0.324 |
|
| 2009 |
Punzo F, Watkin DJ, Fleet GW. α-d-Tagatopyran-ose. Acta Crystallographica. Section E, Structure Reports Online. 65: o1393-4. PMID 21583239 DOI: 10.1107/S1600536809017656 |
0.326 |
|
| 2009 |
Jenkinson SF, Fenton JR, Booth KV, Fleet GW, Watkin DJ. (4S,5R,6R)-Methyl 4-hydr-oxy-4,5-iso-propyl-idenedioxy-4,5,6,7-tetra-hydro-1,2,3-triazolo[1,5-a]pyridine-3-carboxyl-ate. Acta Crystallographica. Section E, Structure Reports Online. 65: o610-1. PMID 21582263 DOI: 10.1107/S1600536809006357 |
0.364 |
|
| 2009 |
Booth KV, Jenkinson SF, Fleet GW, Watkin DJ. 2-De-oxy-2,3-O-isopropyl-idene-2,4-di-C-methyl-β-l-arabinose. Acta Crystallographica. Section E, Structure Reports Online. 65: o570. PMID 21582225 DOI: 10.1107/S1600536809005777 |
0.366 |
|
| 2009 |
Jenkinson SF, Best D, Weymouth-Wilson AC, Clarkson RA, Fleet GW, Watkin DJ. (1S)-1,2-O-Benzyl-idene-α-d-glucurono-6,3-lactone. Acta Crystallographica. Section E, Structure Reports Online. 65: o414-5. PMID 21582005 DOI: 10.1107/S1600536809002876 |
0.383 |
|
| 2009 |
Jenkinson SF, Wang C, Pino-González MS, Fleet GW, Watkin DJ. 7-Azido-N,N-diethyl-4,5-O-isopropyl-idene-4-C-methyl-3,6-anhydro-7-de-oxy-d-glycero-d-manno-heptonamide. Acta Crystallographica. Section E, Structure Reports Online. 65: o263. PMID 21581878 DOI: 10.1107/S1600536808044279 |
0.381 |
|
| 2009 |
Thompson AL, Michalik A, Nash RJ, Wilson FX, van Well R, Johnson P, Fleet GW, Yu CY, Hu XG, Cooper RI, Watkin DJ. Steviamine, a new class of indolizidine alkaloid [(1R,2S,3R,5R,8aR)-3-hydroxy-meth-yl-5-methyl-octa-hydro-indolizine-1,2-diol hydro-bromide]. Acta Crystallographica. Section E, Structure Reports Online. 65: o2904-5. PMID 21578486 DOI: 10.1107/S1600536809043827 |
0.324 |
|
| 2009 |
Best D, Jenkinson SF, Thompson AL, Watkin DJ, Wilson FX, Nash RJ, Fleet GW. (2S,3R,4R,5R)-3,4-Dihydr-oxy-5-(hydroxy-meth-yl)pyrrolidine-2-carboxylic acid [(2S,3R,4R,5R)-3,4-dihydr-oxy-5-(hydroxy-meth-yl)proline]. Acta Crystallographica. Section E, Structure Reports Online. 65: o2418-9. PMID 21577876 DOI: 10.1107/S1600536809035636 |
0.336 |
|
| 2009 |
Booth KV, Jenkinson SF, Fleet GW, Watkin DJ. 2,3-O-(S)-Benzyl-idene-2-C-methyl-d-ribono-1,4-lactone. Acta Crystallographica. Section E, Structure Reports Online. 65: o2199. PMID 21577602 DOI: 10.1107/S1600536809032796 |
0.39 |
|
| 2009 |
Rawlings AJ, Lomas H, Pilling AW, Lee MJ, Alonzi DS, Rountree JS, Jenkinson SF, Fleet GW, Dwek RA, Jones JH, Butters TD. Synthesis and biological characterisation of novel N-alkyl-deoxynojirimycin alpha-glucosidase inhibitors. Chembiochem : a European Journal of Chemical Biology. 10: 1101-5. PMID 19294724 DOI: 10.1002/Cbic.200900025 |
0.308 |
|
| 2009 |
Rountree JS, Butters TD, Wormald MR, Boomkamp SD, Dwek RA, Asano N, Ikeda K, Evinson EL, Nash RJ, Fleet GW. Design, synthesis, and biological evaluation of enantiomeric beta-N-acetylhexosaminidase inhibitors LABNAc and DABNAc as potential agents against Tay-Sachs and Sandhoff disease. Chemmedchem. 4: 378-92. PMID 19145603 DOI: 10.1002/Cmdc.200800350 |
0.367 |
|
| 2008 |
Jenkinson SF, Best D, Wilson FX, Fleet GW, Watkin DJ. (4R)-4-(2-Allyl-2H-1,2,3-triazol-4-yl)-1,2-O-isopropyl-idene-l-threose. Acta Crystallographica. Section E, Structure Reports Online. 64: o2361. PMID 21581334 DOI: 10.1107/S1600536808036416 |
0.383 |
|
| 2008 |
Booth KV, Jenkinson SF, Rao D, Simonisi T, Fleet GW, Izumori K, Watkin DJ. 6-Azido-6-de-oxy-α-l-galactose (6-azido-l-fucose) monohydrate. Acta Crystallographica. Section E, Structure Reports Online. 64: o1568-9. PMID 21203271 DOI: 10.1107/S1600536808022563 |
0.398 |
|
| 2008 |
Jenkinson SF, Booth KV, Yoshihara A, Morimoto K, Fleet GW, Izumori K, Watkin DJ. 1-De-oxy-d-galactitol (l-fucitol). Acta Crystallographica. Section E, Structure Reports Online. 64: o1429. PMID 21203146 DOI: 10.1107/S1600536808020345 |
0.342 |
|
| 2008 |
Booth KV, Jenkinson SF, Fleet GW, Gullapalli P, Yoshihara A, Izumori K, Watkin DJ. 6-De-oxy-α-l-talopyran-ose. Acta Crystallographica. Section E, Structure Reports Online. 64: o1385. PMID 21203105 DOI: 10.1107/S1600536808019582 |
0.363 |
|
| 2008 |
Jenkinson SF, Cruz FP, Booth KV, Fleet GW, Izumori K, Yu CY, Watkin DJ. 1-De-oxy-d-arabinitol. Acta Crystallographica. Section E, Structure Reports Online. 64: o1010-1. PMID 21202536 DOI: 10.1107/S1600536808012555 |
0.359 |
|
| 2008 |
Jenkinson SF, Booth KV, Gullapalli P, Morimoto K, Izumori K, Fleet GW, Watkin DJ. 1-De-oxy-l-mannitol (6-de-oxy-l-mannitol or l-rhamnitol). Acta Crystallographica. Section E, Structure Reports Online. 64: o1705-6. PMID 21201694 DOI: 10.1107/S1600536808024586 |
0.366 |
|
| 2008 |
Jenkinson SF, Booth KV, Best D, Fleet GW, Watkin DJ. tert-Butyl 2-de-oxy-4,5-O-isopropyl-idene-d-gluconate. Acta Crystallographica. Section E, Structure Reports Online. 64: o2011-2. PMID 21201208 DOI: 10.1107/S160053680803064X |
0.362 |
|
| 2008 |
da Cruz FP, Booth KV, Fleet GW, Watkin DJ. 3-O-Benzhydryl-2,5-dide-oxy-2,5-imino-2-C-methyl-l-lyxono-1,4-lactone. Acta Crystallographica. Section E, Structure Reports Online. 64: o1902-3. PMID 21201113 DOI: 10.1107/S1600536808027888 |
0.393 |
|
| 2008 |
Jenkinson SF, Rule SD, Booth KV, Fleet GW, Watkin DJ, Petursson S. 2-O-Benzhydryl-3,4-(S)-O-benzyl-idene-d-lyxono-1,4-lactone. Acta Crystallographica. Section E, Structure Reports Online. 64: o26. PMID 21200976 DOI: 10.1107/S1600536807059739 |
0.335 |
|
| 2008 |
Rao D, Gullapalli P, Yoshihara A, Jenkinson SF, Morimoto K, Takata G, Akimitsu K, Tajima S, Fleet GW, Izumori K. Direct production of L-tagatose from L-psicose by Enterobacter aerogenes 230S. Journal of Bioscience and Bioengineering. 106: 473-80. PMID 19111643 DOI: 10.1263/Jbb.106.473 |
0.375 |
|
| 2008 |
Minami Y, Kuriyama C, Ikeda K, Kato A, Takebayashi K, Adachi I, Fleet GW, Kettawan A, Okamoto T, Asano N. Effect of five-membered sugar mimics on mammalian glycogen-degrading enzymes and various glucosidases. Bioorganic & Medicinal Chemistry. 16: 2734-40. PMID 18258441 DOI: 10.1016/J.Bmc.2008.01.032 |
0.334 |
|
| 2008 |
Lopez-Ortega B, Jenkinson SF, Claridge TD, Fleet GW. Oxetane amino acids: synthesis of tetrameric and hexameric carbopeptoids derived from l-ribo 4-(aminomethyl)-oxetan-2-carboxylic acid Tetrahedron: Asymmetry. 19: 976-983. DOI: 10.1016/J.Tetasy.2008.03.030 |
0.437 |
|
| 2008 |
Claridge TD, Lopez-Ortega B, Jenkinson SF, Fleet GW. Secondary structural investigations into homo-oligomers of δ-2,4-cis oxetane amino acids Tetrahedron: Asymmetry. 19: 984-988. DOI: 10.1016/J.Tetasy.2008.03.029 |
0.316 |
|
| 2007 |
Jenkinson SF, Hotchkiss DJ, Cowley AR, Fleet GW, Watkin DJ. (S)-3-Dimethyl-amino-2-{(4S,5R)-5-[(R)-2,2-dimethyl-1,3-dioxolan-4-yl]-2,2-dimethyl-1,3-dioxolan-4-yl}-2-hydroxy-propanoic acid. Acta Crystallographica. Section E, Structure Reports Online. 64: o294-5. PMID 21200859 DOI: 10.1107/S1600536807066676 |
0.407 |
|
| 2007 |
Kato A, Kato N, Adachi I, Hollinshead J, Fleet GW, Kuriyama C, Ikeda K, Asano N, Nash RJ. Isolation of glycosidase-inhibiting hyacinthacines and related alkaloids from Scilla socialis. Journal of Natural Products. 70: 993-7. PMID 17536859 DOI: 10.1021/Np0700826 |
0.311 |
|
| 2007 |
Otero JM, Soengas RG, Estévez JC, Estévez RJ, Watkin DJ, Evinson EL, Nash RJ, Fleet GW. Preliminary studies on the transformation of nitrosugars into branched chain iminosugars: synthesis of 1,4-dideoxy-4-C-hydroxymethyl-1,4-imino-pentanols. Organic Letters. 9: 623-6. PMID 17286369 DOI: 10.1021/Ol062887V |
0.776 |
|
| 2007 |
Jones NA, Jenkinson SF, Soengas R, Izumori K, Fleet GW, Watkin DJ. The concomitant crystallization of two polymorphs of 1-deoxy-alpha-D-tagatose. Acta Crystallographica. Section C, Crystal Structure Communications. 63: o7-10. PMID 17206062 DOI: 10.1107/S0108270106048591 |
0.621 |
|
| 2007 |
Hotchkiss DJ, Soengas R, Booth KV, Weymouth-Wilson AC, Eastwick-Field V, Fleet GW. Green aldose isomerisation: 2-C-methyl-1,4-lactones from the reaction of Amadori ketoses with calcium hydroxide Tetrahedron Letters. 48: 517-520. DOI: 10.1016/J.Tetlet.2006.11.137 |
0.629 |
|
| 2007 |
Hotchkiss DJ, Kato A, Odell B, Claridge TD, Fleet GW. Homochiral carbon branched piperidines from carbon branched sugar lactones: 4-C-methyl-deoxyfuconojirimycin (DFJ) and its enantiomer—removal of glycosidase inhibition Tetrahedron: Asymmetry. 18: 500-512. DOI: 10.1016/J.Tetasy.2007.02.001 |
0.392 |
|
| 2006 |
Jockusch RA, Talbot FO, Rogers PS, Simone MI, Fleet GW, Simons JP. Carbohydrate amino acids: the intrinsic conformational preference for a beta-turn-type structure in a carbopeptoid building block. Journal of the American Chemical Society. 128: 16771-7. PMID 17177427 DOI: 10.1021/Ja0607133 |
0.312 |
|
| 2006 |
Fleet GW, Johnson SW, Jones JH. Cyclic oligomers of oxetane-based dipeptide isosteres derived from L-rhamnose. Journal of Peptide Science : An Official Publication of the European Peptide Society. 12: 559-61. PMID 16710869 DOI: 10.1002/Psc.759 |
0.45 |
|
| 2006 |
Clinch K, Evans GB, Fleet GW, Furneaux RH, Johnson SW, Lenz DH, Mee SP, Rands PR, Schramm VL, Taylor Ringia EA, Tyler PC. Syntheses and bio-activities of the L-enantiomers of two potent transition state analogue inhibitors of purine nucleoside phosphorylases. Organic & Biomolecular Chemistry. 4: 1131-9. PMID 16525558 DOI: 10.1039/B517883E |
0.418 |
|
| 2006 |
Håkansson AE, Horne G, Fleet GW, Watkin DJ. (6S)-Methyl-L-swainsonine [(1R,2S,6S,8S,8aS)-6-methyloctahydroindolizine-1,2,8-triol] Acta Crystallographica Section E Structure Reports Online. 63: o210-o212. DOI: 10.1107/S1600536806052111 |
0.396 |
|
| 2006 |
Parker S, Watkin D, Mayes B, Storer R, Jenkinson S, Fleet G. 2-Deoxy-2-fluoro-2-C-methyl-D-ribono-1,4-lactone (fluoromethylrib) Acta Crystallographica Section E Structure Reports Online. 62: o1208-o1210. DOI: 10.1107/S1600536806006337 |
0.364 |
|
| 2006 |
Hotchkiss DJ, Jenkinson SF, Storer R, Heinz T, Fleet GW. Amadori ketoses with calcium hydroxide and the Kiliani reaction on 1-deoxy ketoses: two approaches to the synthesis of saccharinic acids Tetrahedron Letters. 47: 315-318. DOI: 10.1016/J.Tetlet.2005.11.018 |
0.398 |
|
| 2005 |
Blériot Y, Gretzke D, Krülle TM, Butters TD, Dwek RA, Nash RJ, Asano N, Fleet GW. Looking glass inhibitors: efficient synthesis and biological evaluation of D-deoxyfuconojirimycin. Carbohydrate Research. 340: 2713-8. PMID 16274755 DOI: 10.1016/J.Carres.2005.10.002 |
0.396 |
|
| 2005 |
Watson KA, Chrysina ED, Tsitsanou KE, Zographos SE, Archontis G, Fleet GW, Oikonomakos NG. Kinetic and crystallographic studies of glucopyranose spirohydantoin and glucopyranosylamine analogs inhibitors of glycogen phosphorylase. Proteins. 61: 966-83. PMID 16222658 DOI: 10.1002/Prot.20653 |
0.309 |
|
| 2005 |
Johnson SW, Jenkinson SF, Angus D, Pérez-Victoria I, Claridge TD, Fleet GW, Jones JH. The synthesis of oligomers of oxetane-based dipeptide isosteres derived from L-rhamnose or D-xylose. Journal of Peptide Science : An Official Publication of the European Peptide Society. 11: 303-18. PMID 15968624 DOI: 10.1002/Psc.622 |
0.47 |
|
| 2005 |
Johnson SW, Jenkinson SF, Pérez-Victoria I, Edwards AA, Claridge TD, Tranter GE, Fleet GW, Jones JH. Conformational studies of oligomeric oxetane-based dipeptide isosteres derived from L-rhamnose or D-xylose. Journal of Peptide Science : An Official Publication of the European Peptide Society. 11: 517-24. PMID 15884104 DOI: 10.1002/Psc.658 |
0.403 |
|
| 2005 |
Claridge TD, Long DD, Baker CM, Odell B, Grant GH, Edwards AA, Tranter GE, Fleet GW, Smith MD. Helix-forming carbohydrate amino acids. The Journal of Organic Chemistry. 70: 2082-90. PMID 15760191 DOI: 10.1021/Jo0480040 |
0.544 |
|
| 2005 |
Soengas R, Izumori K, Simone MI, Watkin DJ, Skytte UP, Soetaert W, Fleet GW. Kiliani reactions on ketoses: branched carbohydrate building blocks from D-tagatose and D-psicose Tetrahedron Letters. 46: 5755-5759. DOI: 10.1016/J.Tetlet.2005.06.030 |
0.645 |
|
| 2005 |
Simone MI, Soengas R, Newton CR, Watkin DJ, Fleet GW. Branched tetrahydrofuran α,α-disubstituted-δ-sugar amino acid scaffolds from branched sugar lactones: a new family of foldamers? Tetrahedron Letters. 46: 5761-5765. DOI: 10.1016/J.Tetlet.2005.06.029 |
0.631 |
|
| 2005 |
Asano N, Ikeda K, Yu L, Kato A, Takebayashi K, Adachi I, Kato I, Ouchi H, Takahata H, Fleet GW. The l-enantiomers of d-sugar-mimicking iminosugars are noncompetitive inhibitors of d-glycohydrolase? Tetrahedron: Asymmetry. 16: 223-229. DOI: 10.1016/J.Tetasy.2004.11.067 |
0.414 |
|
| 2004 |
Yu CY, Asano N, Ikeda K, Wang MX, Butters TD, Wormald MR, Dwek RA, Winters AL, Nash RJ, Fleet GW. Looking glass inhibitors: L-DMDP, a more potent and specific inhibitor of alpha-glucosidases than the enantiomeric natural product DMDP. Chemical Communications (Cambridge, England). 1936-7. PMID 15340609 DOI: 10.1039/B406035K |
0.361 |
|
| 2004 |
Edwards AA, Ichihara O, Murfin S, Wilkes R, Whittaker M, Watkin DJ, Fleet GW. Tetrahydrofuran-based amino acids as library scaffolds. Journal of Combinatorial Chemistry. 6: 230-8. PMID 15002972 DOI: 10.1021/Cc034054R |
0.363 |
|
| 2004 |
Chung YK, Claridge TD, Fleet GW, Johnson SW, Jones JH, Lumbard KW, Stachulski AV. An unsaturated peptidomimetic assembly derived from a carbohydrate. Journal of Peptide Science : An Official Publication of the European Peptide Society. 10: 1-7. PMID 14959886 DOI: 10.1002/Psc.488 |
0.367 |
|
| 2004 |
Hotchkiss D, Soengas R, Simone MI, van Ameijde J, Hunter S, Cowley AR, Fleet GW. Kiliani on ketoses: branched carbohydrate building blocks from d-fructose and l-sorbose Tetrahedron Letters. 45: 9461-9464. DOI: 10.1016/J.Tetlet.2004.10.086 |
0.673 |
|
| 2004 |
Mayes BA, Simon L, Watkin DJ, Ansell CW, Fleet GW. Huge (14-, 21-, 28-, 35-, 56- and 70-membered ring) macrocyclic lactams––a novel family of carbopeptoid-cyclodextrins Tetrahedron Letters. 45: 157-162. DOI: 10.1016/J.Tetlet.2003.10.103 |
0.339 |
|
| 2004 |
Jenkinson (née Barker) SF, Harris T, Fleet GW. Oxetane cis- and trans β-amino-acid scaffolds from d-xylose by efficient SN2 reactions in oxetane rings: methyl and hydroxymethyl analogues of the antibiotic oxetin, an oxetane β-amino-acid Tetrahedron: Asymmetry. 15: 2667-2679. DOI: 10.1016/J.Tetasy.2004.07.031 |
0.391 |
|
| 2003 |
Mons S, Fleet GW. An approach to the generation of simple analogues of the antitumour agent spicamycin. Organic & Biomolecular Chemistry. 1: 3685-91. PMID 14649899 DOI: 10.1039/B307795K |
0.307 |
|
| 2003 |
Smith MD, Claridge TD, Sansom MS, Fleet GW. Bend ribbon-forming tetrahydrofuran amino acids. Organic & Biomolecular Chemistry. 1: 3647-55. PMID 14649895 DOI: 10.1039/B307707C |
0.546 |
|
| 2003 |
Wang MX, Liu Y, Gao HY, Zhang Y, Yu CY, Huang ZT, Fleet GW. Ring-chain tautomerism in organic synthesis: synthesis of heterocyclic enamines from a novel and practical formal ring transformation reaction of lactones. The Journal of Organic Chemistry. 68: 3281-6. PMID 12688802 DOI: 10.1021/Jo026560T |
0.334 |
|
| 2003 |
Sanjayan GJ, Stewart A, Hachisu S, Gonzalez R, Watterson MP, Fleet GW. Templated scaffolds of cis- and trans-tetrahydrofuran γ-amino acids: γ-azido-β-hydroxy-tetrahydrofuran-2-carboxylates from pentono-δ-lactones Tetrahedron Letters. 44: 5847-5851. DOI: 10.1016/S0040-4039(03)01415-1 |
0.357 |
|
| 2003 |
Hunter DF, Fleet GW. Towards hydroxylated nylon 6: oligomers from a protected 6-amino-6-deoxy-d-allonate Tetrahedron: Asymmetry. 14: 3831-3839. DOI: 10.1016/J.Tetasy.2003.10.008 |
0.401 |
|
| 2002 |
Yamashita T, Yasuda K, Kizu H, Kameda Y, Watson AA, Nash RJ, Fleet GW, Asano N. New polyhydroxylated pyrrolidine, piperidine, and pyrrolizidine alkaloids from Scilla sibirica. Journal of Natural Products. 65: 1875-81. PMID 12502331 DOI: 10.1021/Np020296H |
0.348 |
|
| 2002 |
Mellor HR, Nolan J, Pickering L, Wormald MR, Platt FM, Dwek RA, Fleet GW, Butters TD. Preparation, biochemical characterization and biological properties of radiolabelled N-alkylated deoxynojirimycins. The Biochemical Journal. 366: 225-33. PMID 11982484 DOI: 10.1042/Bj20020466 |
0.338 |
|
| 2002 |
Yasuda K, Kizu H, Yamashita T, Kameda Y, Kato A, Nash RJ, Fleet GW, Molyneux RJ, Asano N. New sugar-mimic alkaloids from the pods of Angylocalyx pynaertii. Journal of Natural Products. 65: 198-202. PMID 11858756 DOI: 10.1021/Np010360F |
0.387 |
|
| 2002 |
Stewart AJ, Evans RM, Weymouth-Wilson AC, Cowley AR, Watkin DJ, Fleet GW. 2-Deoxy-l-ribose from an l-arabinono-1,5-lactone Tetrahedron: Asymmetry. 13: 2667-2672. DOI: 10.1016/S0957-4166(02)00738-3 |
0.392 |
|
| 2001 |
Asano N, Yasuda K, Kizu H, Kato A, Fan JQ, Nash RJ, Fleet GW, Molyneux RJ. Novel alpha-L-fucosidase inhibitors from the bark of Angylocalyx pynaertii (Leguminosae). European Journal of Biochemistry / Febs. 268: 35-41. PMID 11121099 DOI: 10.1046/J.1432-1327.2001.01837.X |
0.412 |
|
| 2000 |
Ikeda K, Takahashi M, Nishida M, Miyauchi M, Kizu H, Kameda Y, Arisawa M, Watson AA, Nash RJ, Fleet GW, Asano N. Homonojirimycin analogues and their glucosides from Lobelia sessilifolia and Adenophora spp. (Campanulaceae). Carbohydrate Research. 323: 73-80. PMID 10782288 DOI: 10.1016/S0008-6215(99)00246-3 |
0.327 |
|
| 2000 |
Asano N, Nishida M, Miyauchi M, Ikeda K, Yamamoto M, Kizu H, Kameda Y, Watson AA, Nash RJ, Fleet GW. Polyhydroxylated pyrrolidine and piperidine alkaloids from Adenophora triphylla var. japonica (Campanulaceae). Phytochemistry. 53: 379-82. PMID 10703061 DOI: 10.1016/S0031-9422(99)00555-5 |
0.322 |
|
| 2000 |
Butters T, van den Broek L, Fleet G, Krulle T, Wormald M, Dwek R, Platt F. Molecular requirements of imino sugars for the selective control of N-linked glycosylation and glycosphingolipid biosynthesis Tetrahedron: Asymmetry. 11: 113-124. DOI: 10.1016/S0957-4166(99)00468-1 |
0.363 |
|
| 2000 |
Johnson SW, Angus D, Taillefumier C, Jones JH, Watkin DJ, Floyd E, Buchanan J, Fleet GW. Two epimerisations in the formation of oxetanes from l-rhamnose: towards oxetane-containing peptidomimetics Tetrahedron: Asymmetry. 11: 4113-4125. DOI: 10.1016/S0957-4166(00)00360-8 |
0.429 |
|
| 1999 |
Smith MD, Fleet GW. Designing secondary structures: 5-azidomethyl tetrahydrofuran-2-carboxylates as carbohydrate-derived dipeptide isosteres. Journal of Peptide Science : An Official Publication of the European Peptide Society. 5: 425-41. PMID 10580642 DOI: 10.1002/(Sici)1099-1387(199910)5:10<425::Aid-Psc222>3.0.Co;2-O |
0.387 |
|
| 1999 |
Kato A, Adachi I, Miyauchi M, Ikeda K, Komae T, Kizu H, Kameda Y, Watson AA, Nash RJ, Wormald MR, Fleet GW, Asano N. Polyhydroxylated pyrrolidine and pyrrolizidine alkaloids from Hyancinthoides non-scripta and Scilla campanulata. Carbohydrate Research. 316: 95-103. PMID 10515698 DOI: 10.1016/S0008-6215(99)00043-9 |
0.307 |
|
| 1999 |
Martı́n A, Butters TD, Fleet GW. Synthesis and biological evaluation of enantiomeric rhamnose analogues of the antitumour agent spicamycin—is the mode of action by modification of N-linked glycoproteins? Tetrahedron: Asymmetry. 10: 2343-2360. DOI: 10.1016/S0957-4166(99)00240-2 |
0.426 |
|
| 1999 |
Watterson MP, Pickering L, Smith MD, Hudson SJ, Marsh PR, Mordaunt JE, Watkin DJ, Newman CJ, Fleet GW. 3-Azidotetrahydrofuran-2-carboxylates: monomers for five-ring templated β-amino acid foldamers? Tetrahedron: Asymmetry. 10: 1855-1859. DOI: 10.1016/S0957-4166(99)00205-0 |
0.523 |
|
| 1999 |
Martin A, Watterson MP, Brown AR, Imtiaz F, Winchester BG, Watkin DJ, Fleet GW. 6R- and 6S-6C-Methylmannose from d-mannuronolactone. Inhibition of phosphoglucomutase and phosphomannomutase: agents for the study of the primary metabolism of mannose Tetrahedron: Asymmetry. 10: 355-366. DOI: 10.1016/S0957-4166(98)00492-3 |
0.447 |
|
| 1999 |
Lee RE, Smith MD, Pickering L, Fleet GW. An approach to combinatorial library generation of galactofuranose mimics as potential inhibitors of mycobacterial cell wall biosynthesis: Synthesis of a peptidomimetic of uridine 5′-diphosphogalactofuranose (UDP-Galf) Tetrahedron Letters. 40: 8689-8692. DOI: 10.1016/S0040-4039(99)01844-4 |
0.508 |
|
| 1999 |
Smelt KH, Harrison AJ, Biggadike K, Müller M, Prout K, Watkin DJ, Fleet GW. Components for a combinatorial library of rigid azabicyclic α-L-fucose mimics: First X-ray crystal structure of a stable monoalkylated triazene formed by hydrogenation of an azide Tetrahedron Letters. 40: 3259-3262. DOI: 10.1016/S0040-4039(99)00378-0 |
0.411 |
|
| 1999 |
Smelt KH, Blériot Y, Biggadike K, Lynn S, Lane AL, Watkin DJ, Fleet GW. Photobromination of a bicyclic mimic of α-L-fucose; components for a combinatorial library of rigid fucose analogues Tetrahedron Letters. 40: 3255-3258. DOI: 10.1016/S0040-4039(99)00377-9 |
0.415 |
|
| 1998 |
Asano N, Nishida M, Kato A, Kizu H, Matsui K, Shimada Y, Itoh T, Baba M, Watson AA, Nash RJ, Lilley PM, Watkin DJ, Fleet GW. Homonojirimycin isomers and N-alkylated homonojirimycins: structural and conformational basis of inhibition of glycosidases. Journal of Medicinal Chemistry. 41: 2565-71. PMID 9651160 DOI: 10.1021/Jm970836L |
0.31 |
|
| 1998 |
Asano N, Kato A, Miyauchi M, Kizu H, Kameda Y, Watson AA, Nash RJ, Fleet GW. Nitrogen-containing furanose and pyranose analogues from Hyacinthus orientalis. Journal of Natural Products. 61: 625-8. PMID 9599261 DOI: 10.1021/Np9705726 |
0.342 |
|
| 1998 |
Long DD, Smith MD, Marquess DG, Claridge TD, Fleet GW. A solid phase approach to oligomers of carbohydrate amino-acids: Secondary structure in a trimeric furanose carbopeptoid Tetrahedron Letters. 39: 9293-9296. DOI: 10.1016/S0040-4039(98)02089-9 |
0.519 |
|
| 1998 |
Estevez JC, Fairbanks AJ, Fleet GW. Synthesis of tetrahydropyrans from sugar lactones Tetrahedron. 54: 13591-13620. DOI: 10.1016/S0040-4020(98)00837-0 |
0.726 |
|
| 1998 |
Wang Y, Fleet GW, Zhao L. 1,1,3,3-Tetraisopropyldisiloxane-1,3-diyl (TIPS) migration facilitates one-pot formation of enantiomerically pure methyl 2,3-epoxy-D-xylonate Carbohydrate Research. 307: 159-162. DOI: 10.1016/S0008-6215(98)00019-6 |
0.343 |
|
| 1997 |
Bell A, Pickering L, Finn M, de la Fuente C, Krülle T, Davis B, Fleet G. Caesium Trifluoroacetate Displacement of Triflates in the Inversion of Alcohols Synlett. 1997: 1077-1078. DOI: 10.1055/S-1997-1541 |
0.416 |
|
| 1997 |
Watterson MP, Martin A, Krülle TM, Estevez JC, Fleet GW. Mannuronolactone acetonide: easy access to C-3 OH and C-5 OH of mannose Tetrahedron: Asymmetry. 8: 4111-4120. DOI: 10.1016/S0957-4166(97)00604-6 |
0.673 |
|
| 1997 |
Krülle TM, de la Fuente C, Pickering L, Aplin RT, Tsitsanou KE, Zographos SE, Oikonomakos NG, Nash RJ, Griffiths RC, Fleet GW. Triazole carboxylic acids as anionic sugar mimics? Inhibition of glycogen phosphorylase by a d-glucotriazole carboxylate Tetrahedron: Asymmetry. 8: 3807-3820. DOI: 10.1016/S0957-4166(97)00561-2 |
0.413 |
|
| 1996 |
Blériot Y, Veighey CR, Smelt KH, Cadefau J, Stalmans W, Biggadike K, Lane AL, Müller M, Watkin DJ, Fleet GW. The first example of a : Inhibition of glucokinase Tetrahedron: Asymmetry. 7: 2761-2772. DOI: 10.1016/0957-4166(96)00356-4 |
0.412 |
|
| 1996 |
Brandstetter TW, Wormald MR, Dwek RA, Butters TD, Platt FM, Tsitsanou KE, Zographos SE, Oikonomakos NG, Fleet GW. A galactopyranose analogue of hydantocidin Tetrahedron: Asymmetry. 7: 157-170. DOI: 10.1016/0957-4166(95)00432-7 |
0.337 |
|
| 1995 |
Watson KA, Mitchell EP, Johnson LN, Cruciani G, Son JC, Bichard CJ, Fleet GW, Oikonomakos NG, Kontou M, Zographos SE. Glucose analogue inhibitors of glycogen phosphorylase: from crystallographic analysis to drug prediction using GRID force-field and GOLPE variable selection. Acta Crystallographica. Section D, Biological Crystallography. 51: 458-72. PMID 15299833 DOI: 10.1107/S090744499401348X |
0.314 |
|
| 1995 |
Davis B, Brandstetter TW, Smith C, Hackett L, Winchester BG, Fleet GW. Tetrazoles of manno- and rhamno-furanoses Tetrahedron Letters. 36: 7507-7510. DOI: 10.1016/S0040-4020(99)00138-6 |
0.607 |
|
| 1995 |
Brandstetter TW, Davis B, Hyett D, Smith C, Hackett L, Winchester BG, Fleet GW. Tetrazoles of manno- and rhamno-pyranoses: inhibition of glycosidases by tetrazoles and other mannose mimics Tetrahedron Letters. 36: 7511-7514. DOI: 10.1016/0040-4039(95)01519-1 |
0.579 |
|
| 1995 |
Pilar Vázquez-Tato M, Seijas JA, Fleet GW, Mathews CJ, Hemmings PR, Brown D. Synthesis of (3S,5S)-quinuclidine-3,5-diol and of [3S-(3α,3aα,7aα)]-octahydro-2-furo[2,3-c]pyridinol from D-arabinose Tetrahedron. 51: 959-974. DOI: 10.1016/0040-4020(94)01009-O |
0.665 |
|
| 1994 |
Watson KA, Mitchell EP, Johnson LN, Son JC, Bichard CJ, Orchard MG, Fleet GW, Oikonomakos NG, Leonidas DD, Kontou M. Design of inhibitors of glycogen phosphorylase: a study of alpha- and beta-C-glucosides and 1-thio-beta-D-glucose compounds. Biochemistry. 33: 5745-58. PMID 8180201 DOI: 10.1021/Bi00185A011 |
0.334 |
|
| 1994 |
Oikonomakos NG, Kontou M, Zographos SE, Tsitoura HS, Johnson LN, Watson KA, Mitchell EP, Fleet GW, Son JC, Bichard CJ. The design of potential antidiabetic drugs: experimental investigation of a number of beta-D-glucose analogue inhibitors of glycogen phosphorylase. European Journal of Drug Metabolism and Pharmacokinetics. 19: 185-92. PMID 7867660 DOI: 10.1007/Bf03188920 |
0.322 |
|
| 1994 |
Bichard CJ, Wheatley JR, Fleet GW. Acetonides of heptonolactones: Kiliani ascension of 3-O-benzyl-D-glucose and 3-O-benzyl-D-allose Tetrahedron: Asymmetry. 5: 431-440. DOI: 10.1016/S0957-4166(00)86215-1 |
0.337 |
|
| 1994 |
Wheatley JR, Beacham AR, de Q. Lilley PM, Watkin DJ, Fleet GW. Ketals of L-rhamnoheptonolactones: Potential mimics of L-rhamnose Tetrahedron: Asymmetry. 5: 2523-2534. DOI: 10.1016/S0957-4166(00)80399-7 |
0.396 |
|
| 1994 |
Fairbanks AJ, Hui A, Skead BM, Lilley PMQ, Lamont R, Storer R, Saunders J, Watkin DJ, Fleet GW. Polyhydroxylated cyclohexane and cyclopentane α-amino acids from cyclisations of an azidolactone Tetrahedron Letters. 35: 8891-8894. DOI: 10.1016/S0040-4039(00)78527-3 |
0.585 |
|
| 1994 |
Estevez JC, Ardron H, Wormald MR, Brown D, Fleet GW. Spirocyclic peptides at the anomeric position of mannofuranose Tetrahedron Letters. 35: 8889-8890. DOI: 10.1016/S0040-4039(00)78526-1 |
0.616 |
|
| 1994 |
Estevez JC, Estevez RJ, Ardron H, Wormald MR, Brown D, Fleet GW. Tri- and tetra-peptides incorporating an α-amino acid at the anomeric position of mannofuranose Tetrahedron Letters. 35: 8885-8888. DOI: 10.1016/S0040-4039(00)78525-X |
0.711 |
|
| 1994 |
Hsia KY, Ward P, Brian Lamont R, de Q. Lilley PM, Watkin DJ, Fleet GW. Formation of highly substituted cyclopentanes from radical and anionic Michael cyclisations of α-iodo-γ- and -δ-lactones Tetrahedron Letters. 35: 4823-4826. DOI: 10.1016/S0040-4039(00)76978-4 |
0.355 |
|
| 1994 |
Estevez JC, Fairbanks AJ, Hsia KY, Ward P, Fleet GW. Tetrahydropyran derivatives from γ- and δ-hexonolactones Tetrahedron Letters. 35: 3361-3364. DOI: 10.1016/S0040-4039(00)76908-5 |
0.535 |
|
| 1993 |
Winchester B, al Daher S, Carpenter NC, Cenci di Bello I, Choi SS, Fairbanks AJ, Fleet GW. The structural basis of the inhibition of human alpha-mannosidases by azafuranose analogues of mannose. The Biochemical Journal. 290: 743-9. PMID 8457203 DOI: 10.1042/Bj2900743 |
0.577 |
|
| 1993 |
Molyneux RJ, Pan YT, Tropea JE, Elbein AD, Lawyer CH, Hughes DJ, Fleet GW. 2-Hydroxymethyl-3,4-dihydroxy-6-methyl-pyrrolidine (6-deoxy-DMDP), an alkaloid beta-mannosidase inhibitor from seeds of Angylocalyx pynaertii. Journal of Natural Products. 56: 1356-64. PMID 8229017 DOI: 10.1021/Np50098A020 |
0.337 |
|
| 1993 |
Ardron H, Butters TD, Platt FM, Wormald MR, Dwek RA, Fleet GW, Jacob GS. Synthesis of 1,5-dideoxy-3-O-(α-D-mannopyranosyl)-1,5-imino-D-mannitol and 1,5-dideoxy-3-O-(α-D-glucopyranosyl)-1,5-imino-D-mannitol: Powerful inhibitors of endomannosidase Tetrahedron: Asymmetry. 4: 2011-2024. DOI: 10.1016/S0957-4166(00)82250-8 |
0.379 |
|
| 1993 |
Bichard CJ, Bruce I, Hughes DJ, Girdhar A, Fleet GW, Watkin DJ. Benzylidene acetals of heptonolactones Tetrahedron: Asymmetry. 4: 1579-1589. DOI: 10.1016/S0957-4166(00)80363-8 |
0.357 |
|
| 1993 |
Fairbanks AJ, Ford PS, Watkin DJ, Fleet GW. Synthesis of 1-epihydantocidin from d-ribose Tetrahedron Letters. 34: 3327-3330. DOI: 10.1016/S0040-4039(00)73695-1 |
0.591 |
|
| 1993 |
Skead BM, Fleet GW, Saunders J, Brian Lamont R. Cyclic sulphates of δ-lactones in the synthesis of tetrahydrofurans tetrahydropyrans and cyclohexanes Tetrahedron Letters. 34: 6115-6118. DOI: 10.1016/S0040-4039(00)61744-6 |
0.344 |
|
| 1993 |
Fairbanks AJ, Elliott RP, Smith C, Hui A, Way G, Storer R, Taylor H, Watkin DJ, Winchester BG, Fleet GW. Synthesis of cyclopentane spirohydantoins by aldol cyclisations: An approach to highly substituted α-cyclopentane amino acids Tetrahedron Letters. 34: 7953-7956. DOI: 10.1016/S0040-4039(00)61521-6 |
0.609 |
|
| 1993 |
Mantell SJ, Ford PS, Watkin DJ, Fleet GW, Brown D. 3-Hydroxymuscarines from L-Rhamnose Tetrahedron. 49: 3343-3358. DOI: 10.1016/S0040-4020(01)90162-0 |
0.422 |
|
| 1992 |
Collyer CA, Goldberg JD, Viehmann H, Blow DM, Ramsden NG, Fleet GW, Montgomery FJ, Grice P. Anomeric specificity of D-xylose isomerase. Biochemistry. 31: 12211-8. PMID 1457418 DOI: 10.1021/Bi00163A034 |
0.344 |
|
| 1992 |
Bruce I, Fleet GW, di Bello IC, Winchester B. Iminoheptitols as glycosidase inhibitors: Synthesis of α-homomannojirimycin, 6-epi-α-homomannojirimycin and of a highly substituted pipecolic acid Tetrahedron. 48: 10191-10200. DOI: 10.1016/S0040-4020(01)89047-5 |
0.386 |
|
| 1992 |
Myerscough PM, Fairbanks AJ, Jones AH, Bruce I, Choi SS, Fleet GW, Al-Daher SS, di Bello IC, Winchester B. Inhibition of α-mannosidases by seven carbon sugars: Synthesis of some seven carbon analogues of mannofuranose Tetrahedron. 48: 10177-10190. DOI: 10.1016/S0040-4020(01)89046-3 |
0.564 |
|
| 1992 |
Fairbanks AJ, Carpenter NC, Fleet GW, Ramsden NG, Cenci de Bello I, Winchester BG, Al-Daher SS, Nagahashi G. Synthesis of, and lack of inhibition of a rhamnosidase by, both enantiomers of deoxyrhamnojirimycin and rhamnolactam: β-mannosidase inhibition by δ-lactams Tetrahedron. 48: 3365-3376. DOI: 10.1016/0040-4020(92)85012-4 |
0.435 |
|
| 1991 |
Martin JL, Veluraja K, Ross K, Johnson LN, Fleet GW, Ramsden NG, Bruce I, Orchard MG, Oikonomakos NG, Papageorgiou AC. Glucose analogue inhibitors of glycogen phosphorylase: the design of potential drugs for diabetes. Biochemistry. 30: 10101-16. PMID 1931942 DOI: 10.1107/S0108767378095409 |
0.326 |
|
| 1991 |
Fleet GW, Seijas JA, Vázquez-Tato M. Synthesis of the necine base platynecine from glucose Tetrahedron. 47: 525-530. DOI: 10.1016/S0040-4020(01)90508-3 |
0.651 |
|
| 1991 |
Ana AC, Kaplan MAC, Maia JGS, Gottlieb OR, Nash RJ, Fleet G, Pearce L, Watkin DJ, Scofield AM. Isolation of 7a-epialexaflorine from leaves of alexa grandiflora a unique pyrrolizidine amino acid with a carboxylic acid substituent at C-3 Tetrahedron. 47: 5637-5640. DOI: 10.1016/S0040-4020(01)80994-7 |
0.32 |
|
| 1991 |
Choi S, Witty D, Fleet G, Myer P, Storer R, Wailis C, Watkin D, Pearce L. Approach to oxetane and furan nucleosides with an anomeric carbon substituent: Nucleophilic substitution at highly hindered α-bromo-oxetane- and -tetrahydrofuran-carboxylates Tetrahedron Letters. 32: 3569-3572. DOI: 10.1016/0040-4039(91)80836-U |
0.333 |
|
| 1991 |
Elliott RP, Fleet GW, Pearce L, Smith C, Watkin DJ. A reductive aldol strategy for the synthesis of very highly substituted cyclopentanes from sugar lactones Tetrahedron Letters. 32: 6227-6230. DOI: 10.1016/0040-4039(91)80795-8 |
0.35 |
|
| 1991 |
Choi S, Bruce I, Fairbanks A, Fleet G, Jones A, Nash R, Fellows L. Alexines from heptonolactones Tetrahedron Letters. 32: 5517-5520. DOI: 10.1016/0040-4039(91)80072-E |
0.501 |
|
| 1991 |
Fairbanks AJ, Fleet GW, Jones AH, Bruce I, Al Daher S, di Bello IC, Winchester B. Synthesis from a heptonolactone and effect on glycosidases of (1S,2R,6R,7S)-1,2,6,7-tetrahydroxypyrrolizidine Tetrahedron. 47: 131-138. DOI: 10.1016/0040-4020(91)80015-T |
0.588 |
|
| 1990 |
Axamawaty MT, Fleet GW, Hannah KA, Namgoong SK, Sinnott ML. Inhibition of the alpha-L-arabinofuranosidase III of Monilinia fructigena by 1,4-dideoxy-1,4-imino-L-threitol and 1,4-dideoxy-1,4-imino-L-arabinitol. The Biochemical Journal. 266: 245-9. PMID 2310375 DOI: 10.1042/Bj2660245 |
0.379 |
|
| 1990 |
Fleet GW, Ramsden NG, Nash RJ, Fellows LE, Jacob GS, Molyneux RJ, di Bello IC, Winchester B. Synthesis of the enantiomers of 6-epicastanospermine and 1,6-diepicastanospermine from D- and L-gulonolactone. Carbohydrate Research. 205: 269-82. PMID 2276139 DOI: 10.1016/0008-6215(90)80146-T |
0.373 |
|
| 1990 |
Winchester B, Barker C, Baines S, Jacob GS, Namgoong SK, Fleet G. Inhibition of alpha-L-fucosidase by derivatives of deoxyfuconojirimycin and deoxymannojirimycin. The Biochemical Journal. 265: 277-82. PMID 2137330 DOI: 10.1042/Bj2650277 |
0.374 |
|
| 1990 |
Winchester BG, Cenci di Bello I, Richardson AC, Nash RJ, Fellows LE, Ramsden NG, Fleet G. The structural basis of the inhibition of human glycosidases by castanospermine analogues. The Biochemical Journal. 269: 227-31. PMID 2115770 DOI: 10.1042/Bj2690227 |
0.344 |
|
| 1990 |
Fleet GW, Witty DR. Synthesis of homochiral β-hydroxy-α-aminoacids [(2S,3R,4R)-3,4-dihydroxyproline and (2S,3R,4R)-3,4-dihydroxypipecolic aicd] and of 1,4-dideoxy-1,4-imino-D-arabinitol [DAB1] and fagomine [1,5-imino-1,2,5-trideoxy-D-arabino-hexitol] Tetrahedron: Asymmetry. 1: 119-136. DOI: 10.1016/S0957-4166(00)86337-5 |
0.341 |
|
| 1990 |
Wilson F, Fleet G, Witty D, Vogt K, Wang Y, Storer R, Myers P, Wallis C. Synthesis of the oxetane nucleosides α- an β-noroxetanocin Tetrahedron: Asymmetry. 1: 525-526. DOI: 10.1016/S0957-4166(00)80540-6 |
0.341 |
|
| 1990 |
Elliott RP, Fleet GW, Young SG, Ramsden NG, Smith C. High yield reduction of 2-O-trifluoromethanesulphonate esters of α-hydroxylactones to the corresponding 2-deoxylactones by lithium iodide trihydrate Tetrahedron Letters. 31: 3785-3788. DOI: 10.1016/S0040-4039(00)97471-9 |
0.338 |
|
| 1990 |
Wilson F, Fleet G, Vogt K, Wang Y, Witty D, Choi S, Storer R, Myers P, Wallis C. Synthesis of oxetanocin Tetrahedron Letters. 31: 6931-6934. DOI: 10.1016/S0040-4039(00)97210-1 |
0.393 |
|
| 1990 |
Fleet GW, Carpenter NM, Petursson S, Ramsdena NG. Synthesis of deoxynojirimycin and of nojirimycin δ-lactam Tetrahedron Letters. 31: 409-412. DOI: 10.1016/S0040-4039(00)94568-4 |
0.36 |
|
| 1990 |
Fleet GW, Ramsden NG, Carpenter NM, Peturssona S, Aplin RT. Some comments on an allegedly “facile synthesis of nojirimycin” Tetrahedron Letters. 31: 405-408. DOI: 10.1016/S0040-4039(00)94567-2 |
0.325 |
|
| 1990 |
Bruce I, Fleet GW, Girdhar A, Haraldsson M, Peach JM, Watkin DJ. Retention and apparent inversion during azide displacement of α-triflates of 15-lactones Tetrahedron. 46: 19-32. DOI: 10.1016/S0040-4020(01)97581-7 |
0.351 |
|
| 1989 |
Daher SA, Fleet G, Namgoong SK, Winchester B. Change in specificity of glycosidase inhibition by N-alkylation of amino sugars. Biochemical Journal. 258: 613-615. PMID 2706004 DOI: 10.1042/Bj2580613 |
0.4 |
|
| 1989 |
Bello ICd, Fleet G, Namgoong SK, Tadano KI, Winchester B. Structure-activity relationship of swainsonine. Inhibition of human α-mannosidases by swainsonine analogues Biochemical Journal. 259: 855-861. PMID 2499316 DOI: 10.1042/Bj2590855 |
0.33 |
|
| 1989 |
Carpenter NM, Fleet GW, Cenci di Bello I, Winchester B, Fellows LE, Nash RJ. Synthesis of the mannosidase inhibitors swainsonine and 1,4-dideoxy-1,4-imino-D-mannitol and of the ring contracted swainsonines, (1S, 2R, 7R, 7aR)-1,2,7-trihydroxypyrrolizidine and (1S, 2R, 7S, 7aR)-1,2,7-trihydroxypyrrolizidine Tetrahedron Letters. 30: 7261-7264. DOI: 10.1016/S0040-4039(01)93953-X |
0.326 |
|
| 1989 |
Fleet GW, Ramsden NG, Witty DR. A practical synthesis of deoxymannojirimycin and of (2s,3R,4R,5R)-3,4,5-trihydroxypipecolic acid from D-glucose Tetrahedron. 45: 327-336. DOI: 10.1016/0040-4020(89)80060-2 |
0.369 |
|
| 1989 |
Fleet GW, Ramsden NG, Witty DR. Practical synthesis of deoxymannojirimycin and mannonolactam from L-gulonolactone. Tetrahedron. 45: 319-326. DOI: 10.1016/0040-4020(89)80059-6 |
0.41 |
|
| 1988 |
Fleet GW, Haraldsson M, Nash RJ, Fellows LE. Synthesis from D-glucose of alexine [(1R,2R,3R,7S,8S)-3-hydroxymethyl-1,2,7-trihydroxypyrrolizidine], 3-epialexine and 7-epialexine Tetrahedron Letters. 29: 5441-5444. DOI: 10.1016/S0040-4039(00)82890-7 |
0.303 |
|
| 1988 |
Fleet GW, Seijas JA, Vazquez Tato M. Synthesis of - and -1-amino-3-hydroxymethyl-cyclobutane-1-carboxylic acids Tetrahedron. 44: 2077-2080. DOI: 10.1016/S0040-4020(01)90351-5 |
0.635 |
|
| 1988 |
Fleet GW, Ramsden NG, Molyneux RJ, Jacob GS. Synthesis of 6-epicastanospermine and 1,6-diepicastanospermine from L-gulonolactone and synthesis of L-6-epicastanospermine and L-1,6-diepicastanospermine from D-gulonolactone Tetrahedron Letters. 29: 3603-3606. DOI: 10.1016/0040-4039(88)85305-X |
0.35 |
|
| 1988 |
Fleet GW, Ramsden NG, Witty DR. Short syntheses of D-deoxymannojirimycin and D-mannonolactam from L-gulonolactone and of L-deoxymannojirimycin and L-mannonolactam from D-gulonolactone Tetrahedron Letters. 29: 2871-2874. DOI: 10.1016/0040-4039(88)85234-1 |
0.398 |
|
| 1987 |
Fleet GW, Seymour LC. Synthesis of intermediates for stereospecific synthesis of α- and β-C-nucleosides: Ring contraction of protected 2-0-trifluoromethanesulphonates of galacto- and altro-pyranosides Tetrahedron Letters. 28: 3015-3018. DOI: 10.1016/S0040-4039(00)96272-5 |
0.41 |
|
| 1987 |
Fleet GW, Fellows L, Smith PW. Synthesis of deoxymannojirimycin fagomine deoxynojirimycin 2-acetamido-1,5-imino-1,2,5-trideoxy-D-mannitol 2-acetamido-1,5-imino-1,2,5-trideoxy-D-glucitol 2S,3R,4R,5R-trihydroxypipecolic acid and 2S,3R,4R,5S-trihydroxypipecolic acid from methyl 3-O-benzyl-2,6-dideoxy-2,6-imino-α-D-mannofuranoside Tetrahedron. 43: 979-990. DOI: 10.1016/S0040-4020(01)90035-3 |
0.363 |
|
| 1987 |
Fleet GW, Smith PW. Methyl 2-azido-3-O-benzyl-2-deoxy-α-D-mamnofuranoside as a divergent intermediate for the synthesis of polyhydroxylated piperidines and pyrrolidines: synthesis of 2,5-dideoxy-2,5-imino-D-mannitol [2R,5R-dihydroxymethyl-3R,4R-dihydroxypyrrolidine] Tetrahedron. 43: 971-978. DOI: 10.1016/S0040-4020(01)90034-1 |
0.376 |
|
| 1987 |
Bashyal BP, Chow H, Fleet GW. Synthesis of 2s, 4s, 5s -dihydroxypipecolic acid and bulgecinine [2s,4s,5r-4-hydroxy-5- (hydroxymethyl)proline] from d-glucuronolactone, a strategy for the synthesis of 2s,4s-4-hydroxy-α-amino acids Tetrahedron. 43: 423-430. DOI: 10.1016/S0040-4020(01)89973-7 |
0.337 |
|
| 1987 |
Bashyal BP, Fleet GW, Gough MJ, Smith PW. Synthesis of the α-Mannosidase inhibitors swainsonine [(1S, 2R, 8R, 8aR)-1,2,8-trihydroxyoctahydroindolizine] and 1,4-dideoxy-1,4-imino-d-mannitol from mannose Tetrahedron. 43: 3083-3093. DOI: 10.1016/S0040-4020(01)86850-2 |
0.372 |
|
| 1986 |
Dho J, Fleet G, Peach J, Prout K, Smith P. Synthesis of 2R,3S,4R-dihydroxyproline from D-ribonolactone Tetrahedron Letters. 27: 3203-3204. DOI: 10.1016/S0040-4039(00)84754-1 |
0.332 |
|
| 1986 |
Fleet GW, James K, Lunn RJ, Mathews CJ. An enantiospecific synthesis of S-quinuclidinol from D-glucose Tetrahedron Letters. 27: 3057-3058. DOI: 10.1016/S0040-4039(00)84715-2 |
0.392 |
|
| 1986 |
Fleet GW, James K, Lunn RJ. Enantiospecific synthesis of S-quinuclidinol from D-glucose: A strategy for the synthesis of chiral quinuclidines. Tetrahedron Letters. 27: 3053-3056. DOI: 10.1016/S0040-4039(00)84714-0 |
0.403 |
|
| 1986 |
Fleet GW, Smith PW. The synthesis from d-xylose of the potent and specific enantiomeric glucosidase inhibitors, 1,4-dideoxy-1,4-imino-d-arabinitol and 1,4-dideoxy-1,4-imin Tetrahedron. 42: 5685-5692. DOI: 10.1016/S0040-4020(01)88174-6 |
0.447 |
|
| 1985 |
Fleet GW, Smith PW. Enantiospecific syntheses of deoxymannojirimycin, fagomine and 2r,5r-dihydroxymethyl-3r,4r-dihydroxypyrrolidine from D-glucose Tetrahedron Letters. 26: 1469-1472. DOI: 10.1016/S0040-4039(00)99073-7 |
0.345 |
|
| 1985 |
Evans SV, Hayman AR, Fellows LE, Shing TK, E.Derome A, Fleet GW. Lack of glycosidase inhibition by, and isolation from xanthocercis zambesiaca (leguminosae) of, 4-O-(β-D-glucopyranosyl)-fagomine [1,2,5-trideoxy-4-O-(β-D-glucopyranosyl)-1,5-imino-D- arabino-hexitol], a novel glucoside of a polyhydroxylated piperidine alkaloid Tetrahedron Letters. 26: 1465-1468. DOI: 10.1016/S0040-4039(00)99072-5 |
0.36 |
|
| 1985 |
Fleet G, Nicholas S, Smith P, Evans S, Fellows L, Nash R. Potent competitive inhibition of α-galactosidase and α-glucosidase activity by 1,4-dideoxy-1,4-iminopentitols: syntheses of 1,4-dideoxy-1,4-imino-d-lyxitol and of both enantiomers of 1,4-dideoxy-1,4-iminoarabinitol Tetrahedron Letters. 26: 3127-3130. DOI: 10.1016/S0040-4039(00)98636-2 |
0.404 |
|
| 1985 |
Evans S, Fellows L, Shing T, Fleet G. Glycosidase inhibition by plant alkaloids which are structural analogues of monosaccharides Phytochemistry. 24: 1953-1955. DOI: 10.1016/S0031-9422(00)83099-X |
0.353 |
|
| 1985 |
Evans SV, Shing TK, Aplin RT, Fellows LE, Fleet GW. Sulphate ester of trans-4-hydroxypipecolic acid in seeds of Peltophorum Phytochemistry. 24: 2593-2596. DOI: 10.1016/S0031-9422(00)80675-5 |
0.333 |
|
| 1984 |
Fleet G, Gough M, Smith P. Enantiospecific Synthesis of Swainsonine, (1S, 2R, 8R, 8aR)-1,2,8-trihydroxyoctahydroindolizine, from D-mannose Tetrahedron Letters. 25: 1853-1856. DOI: 10.1016/S0040-4039(01)90059-0 |
0.371 |
|
| 1984 |
Fleet G, Gough M, Shing T. Syntheses of 1,5-dideoxy-1,5-imino-D-mannitol from D-mannose and from D-glucose Tetrahedron Letters. 25: 4029-4032. DOI: 10.1016/0040-4039(84)80058-1 |
0.368 |
|
| 1983 |
Fleet G, Gough M, Shing T. Enantiospecific total synthesis of pseudomonic acids from arabinose Tetrahedron Letters. 24: 3661-3664. DOI: 10.1016/S0040-4039(00)88195-2 |
0.332 |
|
| 1983 |
Fleet G, Shing T. Enantiospecific synthesis of (3s-hydroxy-2s-methyl) butyltriphenylphosphonium iodide, a precursor for the chiral side chain of pseudomonic acid C Tetrahedron Letters. 24: 3657-3660. DOI: 10.1016/S0040-4039(00)88194-0 |
0.385 |
|
| 1982 |
Fleet G, Spensley C. Model studies on the synthesis of pseudomonic acids Tetrahedron Letters. 23: 109-112. DOI: 10.1016/S0040-4039(00)97547-6 |
0.399 |
|
| 1982 |
Fleet G, Gough M. Enantiospecific syntheses of intermediates in the total synthesis of pseudomonic acids Tetrahedron Letters. 23: 4509-4512. DOI: 10.1016/S0040-4039(00)85640-3 |
0.423 |
|
| 1981 |
Fleet G, Harding P. Selectivity in the acid catalysed reduction of carbonyl compounds to alcohols by bis(triphenylphosphine)copper(I) tetrahydroborate: Reduction of aldehydes in the presence of ketones Tetrahedron Letters. 22: 675-678. DOI: 10.1016/S0040-4039(01)92520-1 |
0.321 |
|
| 1979 |
Fleet G, Harding P. Convenient synthesis of bis(triphenylphosphine) copper(I) tetrahydroborate and reduction of acid chlorides to aldehydes Tetrahedron Letters. 20: 975-978. DOI: 10.1016/S0040-4039(01)86066-4 |
0.327 |
|
| 1973 |
Corey E, Fleet G. Chromium trioxide-3, 5-dimethylpyrazole complex as a reagent for oxidation of alcohols to carbonyl compounds Tetrahedron Letters. 14: 4499-4501. DOI: 10.1016/S0040-4039(01)87260-9 |
0.372 |
|
| 1973 |
Corey E, Fleet G, Kato M. A biogenetic approach to the synthesis of a prostanoid precursor. Tetrahedron Letters. 14: 3963-3966. DOI: 10.1016/S0040-4039(01)87084-2 |
0.428 |
|
| 1972 |
Fleet GW, Knowles JR, Porter RR. The antibody binding site. Labelling of a specific antibody against the photo-precursor of an aryl nitrene. The Biochemical Journal. 128: 499-508. PMID 4117794 DOI: 10.1042/Bj1280499 |
0.489 |
|
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