Year |
Citation |
Score |
2024 |
Chetty LC, Kruger HG, Arvidsson PI, Maguire GEM, Govender T, Naicker T. The Oxidation of Electron-Rich Arenes Using a HO-Proline System. Acs Omega. 9: 37155-37162. PMID 39246484 DOI: 10.1021/acsomega.4c04383 |
0.453 |
|
2024 |
Chetty LC, Kruger HG, Arvidsson PI, Naicker T, Govender T. Investigating the efficacy of green solvents and solvent-free conditions in hydrogen-bonding mediated organocatalyzed model reactions. Rsc Advances. 14: 7992-7998. PMID 38454950 DOI: 10.1039/d4ra00679h |
0.456 |
|
2023 |
Shungube M, Hlophe AK, Girdhari L, Sabe VT, Peters BB, Reddy N, Omolabi KF, Chetty L, Arumugam T, Chuturgoon A, Kruger HG, Arvidsson PI, Qin HL, Naicker T, Govender T. Synthesis and biological evaluation of novel β-lactam-metallo β-lactamase inhibitors. Rsc Advances. 13: 18991-19001. PMID 37362332 DOI: 10.1039/d3ra02490c |
0.475 |
|
2023 |
Reddy N, Girdhari L, Shungube M, Gouws AC, Peters BK, Rajbongshi KK, Baijnath S, Mdanda S, Ntombela T, Arumugam T, Bester LA, Singh SD, Chuturgoon A, Arvidsson PI, Maguire GEM, et al. Neutralizing Carbapenem Resistance by Co-Administering Meropenem with Novel β-Lactam-Metallo-β-Lactamase Inhibitors. Antibiotics (Basel, Switzerland). 12. PMID 37106995 DOI: 10.3390/antibiotics12040633 |
0.445 |
|
2023 |
Peters BK, Reddy N, Shungube M, Girdhari L, Baijnath S, Mdanda S, Chetty L, Ntombela T, Arumugam T, Bester LA, Singh SD, Chuturgoon A, Arvidsson PI, Maguire GEM, Kruger HG, et al. In Vitro and In Vivo Development of a β-Lactam-Metallo-β-Lactamase Inhibitor: Targeting Carbapenem-Resistant . Acs Infectious Diseases. PMID 36786013 DOI: 10.1021/acsinfecdis.2c00485 |
0.444 |
|
2020 |
Lubanyana H, Arvidsson PI, Govender T, Kruger HG, Naicker T. Correction to "Improved Synthesis and Isolation of Bedaquiline". Acs Omega. 5: 24154. PMID 32984738 DOI: 10.1021/acsomega.0c03922 |
0.402 |
|
2020 |
Carlström KE, Chinthakindi PK, Espinosa B, Al Nimer F, Arnér ESJ, Arvidsson PI, Piehl F, Johansson K. Characterization of More Selective Central Nervous System Nrf2-Activating Novel Vinyl Sulfoximine Compounds Compared to Dimethyl Fumarate. Neurotherapeutics : the Journal of the American Society For Experimental Neurotherapeutics. PMID 32394330 DOI: 10.1007/S13311-020-00855-0 |
0.681 |
|
2020 |
Reddy N, Shungube M, Arvidsson PI, Baijnath S, Kruger HG, Govender T, Naicker T. A 2018-2019 patent review of metallo beta-lactamase inhibitors. Expert Opinion On Therapeutic Patents. PMID 32393078 DOI: 10.1080/13543776.2020.1767070 |
0.485 |
|
2020 |
Lubanyana H, Arvidsson PI, Govender T, Kruger HG, Naicker T. Improved Synthesis and Isolation of Bedaquiline. Acs Omega. 5: 3607-3611. PMID 32118176 DOI: 10.1021/acsomega.9b04037 |
0.498 |
|
2020 |
Rajbongshi KK, Ambala S, Govender T, Kruger HG, Arvidsson PI, Naicker T. Microwave-Accelerated N-Acylation of Sulfoximines with Aldehydes under Catalyst-Free Conditions Synthesis. 52: 1279-1286. DOI: 10.1055/S-0039-1691589 |
0.545 |
|
2020 |
Chinthakindi PK, Benediktsdottir A, Arvidsson PI, Chen Y, Sandström A. Solid Phase Synthesis of Sulfonimidamide Pseudopeptides and Library Generation European Journal of Organic Chemistry. 2020: 3796-3807. DOI: 10.1002/Ejoc.202000108 |
0.698 |
|
2019 |
Thota N, Makam P, Rajbongshi KK, Nagiah S, Abdul NS, Chuturgoon AA, Kaushik A, Lamichhane G, Somboro AM, Kruger HG, Govender T, Naicker T, Arvidsson PI. -Trifluoromethylthiolated Sulfonimidamides and Sulfoximines: Anti-microbial, Anti-mycobacterial, and Cytotoxic Activity. Acs Medicinal Chemistry Letters. 10: 1457-1461. PMID 31620233 DOI: 10.1021/Acsmedchemlett.9B00285 |
0.501 |
|
2019 |
Chinthakindi PK, Benediktsdottir A, Ibrahim A, Wared A, Aurell C, Pettersen A, Zamaratski E, Arvidsson PI, Chen Y, Sandström A. Synthesis of Sulfonimidamide-Based Amino Acid Building Blocks with Orthogonal Protecting Groups European Journal of Organic Chemistry. 2019: 1045-1057. DOI: 10.1002/Ejoc.201801541 |
0.711 |
|
2018 |
Khumalo MF, Akpan ED, Chinthakindi PK, Brasil EM, Rajbongshi KK, Makatini MM, Govender T, Kruger HG, Naicker T, Arvidsson PI. Synthesis of novel 1,2,4-thiadiazinane 1,1-dioxides three component SuFEx type reaction. Rsc Advances. 8: 37503-37507. PMID 35557800 DOI: 10.1039/c8ra07627h |
0.512 |
|
2018 |
Khumalo MF, Akpan ED, Chinthakindi PK, Brasil E, Rajbongshi KK, Makatini MM, Govender T, Kruger HG, Naicker T, Arvidsson PI. Synthesis of novel 1,2,4-thiadiazinane 1,1-dioxides via three component SuFEx type reaction Rsc Advances. 8: 37503-37507. DOI: 10.1039/C8Ra07627H |
0.766 |
|
2018 |
Peters BK, Razuwika R, Samipillai M, Arvidsson PI, Kruger HG, Govender T, Naicker T. An unexpected re-arrangement of the antibiotic carbapenem core to new 1,4-diazepin-5-one scaffolds Rsc Advances. 8: 190-193. DOI: 10.1039/C7Ra12688C |
0.52 |
|
2018 |
Chinthakindi PK, Arvidsson PI. Sulfonyl Fluorides (SFs): More Than Click Reagents? European Journal of Organic Chemistry. 2018: 3648-3666. DOI: 10.1002/Ejoc.201800464 |
0.7 |
|
2018 |
Nandi GC, Arvidsson PI. Sulfonimidamides: Synthesis and Applications in Preparative Organic Chemistry Advanced Synthesis & Catalysis. 360: 2976-3001. DOI: 10.1002/Adsc.201800273 |
0.314 |
|
2017 |
Ntshangase S, Shobo A, Kruger HG, Asperger A, Niemeyer D, Arvidsson PI, Govender T, Baijnath S. The downfall of TBA-354 - a possible explanation for its neurotoxicity via mass spectrometric imaging. Xenobiotica; the Fate of Foreign Compounds in Biological Systems. 1-23. PMID 28859520 DOI: 10.1080/00498254.2017.1375168 |
0.457 |
|
2017 |
Baijnath S, Moodley C, Ngcobo B, Singh SD, Kruger HG, Arvidsson PI, Naicker T, Pym A, Govender T. Clofazimine protects against mycobacterium tuberculosis dissemination in the CNS following an aerosol challenge in a murine model. International Journal of Antimicrobial Agents. PMID 28843822 DOI: 10.1016/J.Ijantimicag.2017.08.020 |
0.439 |
|
2017 |
Mdanda S, Baijnath S, Shobo A, Singh SD, Maguire GEM, Kruger HG, Arvidsson PI, Naicker T, Govender T. Lansoprazole-sulphide, pharmacokinetics of this promising anti-tuberculous agent. Biomedical Chromatography : Bmc. PMID 28623874 DOI: 10.1002/Bmc.4035 |
0.454 |
|
2017 |
Dutta J, Naicker T, Ebenhan T, Kruger HG, Arvidsson PI, Govender T. Synthetic approaches to radiochemical probes for imaging of bacterial infections. European Journal of Medicinal Chemistry. 133: 287-308. PMID 28395216 DOI: 10.1016/J.Ejmech.2017.03.060 |
0.477 |
|
2017 |
Chinthakindi PK, Govender KB, Kumar AS, Kruger HG, Govender T, Naicker T, Arvidsson PI. A Synthesis of "Dual Warhead" β-Aryl Ethenesulfonyl Fluorides and One-Pot Reaction to β-Sultams. Organic Letters. PMID 28075600 DOI: 10.1021/Acs.Orglett.6B03634 |
0.773 |
|
2017 |
Chinthakindi PK, Naicker T, Thota N, Govender T, Kruger HG, Arvidsson PI. Sulfonimidamide in medizinischer Chemie und Agrochemie Angewandte Chemie. 129: 4160-4170. DOI: 10.1002/Ange.201610456 |
0.755 |
|
2016 |
Chinthakindi PK, Naicker T, Thota N, Govender T, Kruger HG, Arvidsson PI. Gaining Momentum: Sulfonimidamides in Medicinal- and Agrochemistry. Angewandte Chemie (International Ed. in English). PMID 27958674 DOI: 10.1002/Anie.201610456 |
0.754 |
|
2016 |
Govender T, Arvidsson PI, Maguire GE, Kruger HG, Naicker T. Enantioselective Organocatalyzed Transformations of β-Ketoesters. Chemical Reviews. PMID 27463615 DOI: 10.1021/Acs.Chemrev.6B00156 |
0.551 |
|
2016 |
Chinthakindi PK, Kruger HG, Govender T, Naicker T, Arvidsson PI. On-water synthesis of biaryl sulfonyl fluorides. The Journal of Organic Chemistry. PMID 26900892 DOI: 10.1021/Acs.Joc.5B02770 |
0.749 |
|
2016 |
Makhathini SS, Das SK, Singh T, Arvidsson PI, Kruger HG, Gunosewoyo H, Govender T, Naicker T. Stereoselective synthesis towards unnatural proline-based amino acids Arkivoc. 2016: 134-144. DOI: 10.3998/Ark.5550190.P009.462 |
0.517 |
|
2016 |
CHIWUNZE TE, Azumah R, Ramtahal M, Somboro AM, Arvidsson PI, Kruger HG, Govender T, Naicker T. Organocatalyzed Mannich reactions on minocycline: Towards novel tetracycline antibiotics South African Journal of Chemistry. 69. DOI: 10.17159/0379-4350/2016/V69A9 |
0.547 |
|
2016 |
Naicker T, Albericio F, Dutta J, Chinthakindi P, Arvidsson P, de la Torre B, Kruger H, Govender T. A Facile Synthesis of NODASA-Functionalized Peptide Synlett. 27: 1685-1688. DOI: 10.1055/S-0035-1561970 |
0.766 |
|
2016 |
Chinthakindi PK, Nandi GC, Govender T, Kruger HG, Naicker T, Arvidsson PI. An Efficient Protecting-Group-Free Synthesis of Vinylic Sulfoximines via Horner–Wadsworth–Emmons Reaction Synlett. DOI: 10.1055/S-0035-1561573 |
0.774 |
|
2016 |
Chinthakindi PK, Nandi GC, Govender T, Kruger HG, Naicker T, Arvidsson PI. ChemInform Abstract: An Efficient Protecting-Group-Free Synthesis of Vinylic Sulfoximines via Horner-Wadsworth-Emmons Reaction. Cheminform. 47. DOI: 10.1002/CHIN.201642096 |
0.728 |
|
2015 |
Md Abdur Rauf S, Arvidsson PI, Albericio F, Govender T, Maguire GE, Kruger HG, Honarparvar B. The effect of N-methylation of amino acids (Ac-X-OMe) on solubility and conformation: a DFT study. Organic & Biomolecular Chemistry. 13: 9993-10006. PMID 26289381 DOI: 10.1039/C5Ob01565K |
0.529 |
|
2015 |
Borhade SR, Svensson R, Brandt P, Artursson P, Arvidsson PI, Sandström A. Preclinical characterization of acyl sulfonimidamides: potential carboxylic acid bioisosteres with tunable properties. Chemmedchem. 10: 455-60. PMID 25630705 DOI: 10.1002/Cmdc.201402497 |
0.328 |
|
2015 |
Somboro AM, Tiwari D, Bester LA, Parboosing R, Chonco L, Kruger HG, Arvidsson PI, Govender T, Naicker T, Essack SY. NOTA: a potent metallo-β-lactamase inhibitor. The Journal of Antimicrobial Chemotherapy. 70: 1594-6. PMID 25567963 DOI: 10.1093/Jac/Dku538 |
0.469 |
|
2015 |
Nandi GC, Kota SR, Wakchaure PB, Chinthakindi PK, Govender T, Kruger HG, Naicker T, Arvidsson PI. Pd-catalyzed C-N coupling of vinylbromides and sulfonimidamides: A facile synthesis of N′-vinylsulfonimidamides Rsc Advances. 5: 62084-62090. DOI: 10.1039/C5Ra10939F |
0.751 |
|
2015 |
Das SK, Bhatt N, Mujahid M, Arvidsson PI, Kruger HG, Naicker T, Govender T. Towards a stereoselective synthesis of α,α-disubstituted proline analogues Tetrahedron Letters. 56: 5172-5174. DOI: 10.1016/J.Tetlet.2015.07.065 |
0.547 |
|
2015 |
Nandi GC, Kota SR, Naicker T, Govender T, Kruger HG, Arvidsson PI. Cu(OAc)2-catalysed oxidative dual C-H/N-H activation of terminal alkynes and N-deprotected sulfonimidamides: An easy access to N-alkynylated sulfonimidamides European Journal of Organic Chemistry. 2015: 2861-2867. DOI: 10.1002/Ejoc.201500239 |
0.503 |
|
2015 |
Cele ZED, Arvidsson PI, Kruger HG, Govender T, Naicker T. Applied enantioselective aminocatalysis: α-heteroatom functionalization reactions on the carbapenem (β-lactam antibiotic) core European Journal of Organic Chemistry. 2015: 638-646. DOI: 10.1002/Ejoc.201403238 |
0.557 |
|
2015 |
Nandi GC, Kota SR, Wakchaure PB, Chinthakindi PK, Govender T, Kruger HG, Naicker T, Arvidsson PI. ChemInform Abstract: Pd-Catalyzed C-N Coupling of Vinylbromides and Sulfonimidamides: A Facile Synthesis of N′-Vinylsulfonimidamides. Cheminform. 46: no-no. DOI: 10.1002/CHIN.201548048 |
0.687 |
|
2014 |
Farahani MD, Honarparvar B, Albericio F, Maguire GE, Govender T, Arvidsson PI, Kruger HG. Proline N-oxides: modulators of the 3D conformation of linear peptides through "NO-turns". Organic & Biomolecular Chemistry. 12: 4479-90. PMID 24849849 DOI: 10.1039/C4Ob00433G |
0.526 |
|
2014 |
Khanyase S, Naicker T, Maguire GEM, Kruger HG, Arvidsson PI, Govender T. L-Proline organocatalyzed Michael synthesis of monobactam and carbapenem β-lactam cores Tetrahedron Asymmetry. 25: 969-973. DOI: 10.1016/J.Tetasy.2014.05.006 |
0.572 |
|
2014 |
Nandi GC, Kota SR, Govender T, Kruger HG, Arvidsson PI. Cu(OAc)2promoted Chan-Evans-Lam C-N cross coupling reactions on the N- and N′-nitrogen atoms of sulfonimidamides with aryl boronic acids Tetrahedron. 5428-5433. DOI: 10.1016/J.Tet.2014.06.122 |
0.534 |
|
2014 |
Wakchaure PB, Borhade SR, Sandström A, Arvidsson PI. Synthesis of Vinyl- and Aryl-Acyl Sulfonimidamides Through Pd-Catalyzed Carbonylation Using Mo(CO)6as ex situ CO Source European Journal of Organic Chemistry. 2015: 213-219. DOI: 10.1002/Ejoc.201403148 |
0.401 |
|
2014 |
Cele ZED, Pawar SA, Naicker T, Maguire GEM, Arvidsson PI, Kruger HG, Govender T. Organocatalytic mannich reactions on a carbapenem core - Synthesis of mannich bases and bicyclic diazanonanes European Journal of Organic Chemistry. 2014: 2253-2260. DOI: 10.1002/Ejoc.201301823 |
0.568 |
|
2013 |
Pawar SA, Alapour S, Khanyase S, Cele ZE, Chitti S, Kruger HG, Govender T, Arvidsson PI. Organocatalyzed stereospecific C-C bond formation of β-lactams. Organic & Biomolecular Chemistry. 11: 8294-7. PMID 24217690 DOI: 10.1039/C3Ob41858H |
0.511 |
|
2013 |
Borhade SR, Sandström A, Arvidsson PI. Synthesis of novel aryl and heteroaryl acyl sulfonimidamides via Pd-catalyzed carbonylation using a nongaseous precursor. Organic Letters. 15: 1056-9. PMID 23394148 DOI: 10.1021/Ol400049M |
0.336 |
|
2013 |
Makatini MM, Petzold K, Alves CN, Arvidsson PI, Honarparvar B, Govender P, Govender T, Kruger HG, Sayed Y, JerônimoLameira, Maguire GE, Soliman ME. Synthesis, 2D-NMR and molecular modelling studies of pentacycloundecane lactam-peptides and peptoids as potential HIV-1 wild type C-SA protease inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry. 28: 78-88. PMID 22339087 DOI: 10.3109/14756366.2011.633907 |
0.514 |
|
2013 |
Sawant RT, Stevenson J, Odell LR, Arvidsson PI. Organocatalytic asymmetric cross-aldol reaction of 2-chloroethoxy acetaldehyde: diversity-oriented synthesis of chiral substituted 1,4-dioxanes and morpholines Tetrahedron: Asymmetry. 24: 134-141. DOI: 10.1016/J.Tetasy.2012.12.004 |
0.393 |
|
2012 |
Yngve U, Söderman P, Svensson M, Rosqvist S, Arvidsson PI. Imidazopyridine-based inhibitors of glycogen synthase kinase 3: synthesis and evaluation of amide isostere replacements of the carboxamide scaffold. Chemistry & Biodiversity. 9: 2442-52. PMID 23161627 DOI: 10.1002/Cbdv.201200308 |
0.312 |
|
2012 |
Makatini MM, Petzold K, Arvidsson PI, Honarparvar B, Govender T, Maguire GE, Parboosing R, Sayed Y, Soliman ME, Kruger HG. Synthesis, screening and computational investigation of pentacycloundecane-peptoids as potent CSA-HIV PR inhibitors. European Journal of Medicinal Chemistry. 57: 459-67. PMID 22867528 DOI: 10.1016/J.Ejmech.2012.06.019 |
0.502 |
|
2012 |
Hemmaragala NM, Arvidsson PI, Maguire GE, Kruger HG, Govender T. Interaction of beta-amyloid interactions with peptide functionalized gold nanoparticles. Journal of Nanoscience and Nanotechnology. 12: 2179-84. PMID 22755035 DOI: 10.1166/Jnn.2012.5791 |
0.5 |
|
2012 |
Honarparvar B, Makatini MM, Pawar SA, Petzold K, Soliman ME, Arvidsson PI, Sayed Y, Govender T, Maguire GE, Kruger HG. Pentacycloundecane-diol-based HIV-1 protease inhibitors: biological screening, 2D NMR, and molecular simulation studies. Chemmedchem. 7: 1009-19. PMID 22544389 DOI: 10.1002/Cmdc.201100512 |
0.517 |
|
2012 |
Chakka SK, Cele ZED, Sosibo SC, Francis V, Arvidsson PI, Kruger HG, Maguire GEM, Govender T. Asymmetric conjugate addition of thioglycolate to a range of chalcones using tetrahydroisoquinoline (TIQ) N,N′-dioxide ligands Tetrahedron Asymmetry. 23: 616-622. DOI: 10.1016/J.Tetasy.2012.04.010 |
0.534 |
|
2012 |
Funes Maldonado M, Sehgelmeble F, Bjarnemark F, Svensson M, Åhman J, Arvidsson PI. Synthesis and arylation of unprotected sulfonimidamides Tetrahedron. 68: 7456-7462. DOI: 10.1016/J.Tet.2012.06.072 |
0.397 |
|
2012 |
Naicker T, Arvidsson PI, Kruger HG, Maguire GEM, Govender T. Microwave-assisted synthesis of guanidine organocatalysts bearing a tetrahydroisoquinoline framework and their evaluation in Michael addition reactions European Journal of Organic Chemistry. 3331-3337. DOI: 10.1002/Ejoc.201200303 |
0.585 |
|
2012 |
Honarparvar B, Makatini MM, Pawar SA, Petzold K, Soliman MES, Arvidsson PI, Sayed Y, Govender T, Maguire GEM, Kruger HG. Inside Cover: Pentacycloundecane-diol-Based HIV-1 Protease Inhibitors: Biological Screening, 2D NMR, and Molecular Simulation Studies (ChemMedChem 6/2012) Chemmedchem. 7: 938-938. DOI: 10.1002/Cmdc.201290025 |
0.464 |
|
2011 |
Makatini MM, Petzold K, Sriharsha SN, Ndlovu N, Soliman ME, Honarparvar B, Parboosing R, Naidoo A, Arvidsson PI, Sayed Y, Govender P, Maguire GE, Kruger HG, Govender T. Synthesis and structural studies of pentacycloundecane-based HIV-1 PR inhibitors: a hybrid 2D NMR and docking/QM/MM/MD approach. European Journal of Medicinal Chemistry. 46: 3976-85. PMID 21741133 DOI: 10.1016/J.Ejmech.2011.05.071 |
0.521 |
|
2011 |
Makatini MM, Petzold K, Sriharsha SN, Soliman ME, Honarparvar B, Arvidsson PI, Sayed Y, Govender P, Maguire GE, Kruger HG, Govender T. Pentacycloundecane-based inhibitors of wild-type C-South African HIV-protease. Bioorganic & Medicinal Chemistry Letters. 21: 2274-7. PMID 21429747 DOI: 10.1016/J.Bmcl.2011.02.105 |
0.524 |
|
2011 |
Naicker T, Arvidsson PI, Kruger HG, Maguire GEM, Govender T. Tetrahydroisoquinoline-based N-oxides as chiral organocatalysts for the asymmetric allylation of aldehydes European Journal of Organic Chemistry. 6923-6932. DOI: 10.1002/Ejoc.201100923 |
0.587 |
|
2010 |
Bose PP, Chatterjee U, Hubatsch I, Artursson P, Govender T, Kruger HG, Bergh M, Johansson J, Arvidsson PI. In vitro ADMET and physicochemical investigations of poly-N-methylated peptides designed to inhibit Abeta aggregation. Bioorganic & Medicinal Chemistry. 18: 5896-902. PMID 20659803 DOI: 10.1016/J.Bmc.2010.06.087 |
0.515 |
|
2010 |
Altaib MS, Arvidsson PI, Govender T, Maguire GE, Makatini M, Onajole OK, Kruger HG. Synthesis and NMR elucidation of novel pentacycloundecane-based peptides. Magnetic Resonance in Chemistry : Mrc. 48: 435-42. PMID 20474021 DOI: 10.1002/Mrc.2598 |
0.537 |
|
2010 |
Muthusamy K, Arvidsson PI, Govender P, Kruger HG, Maguire GE, Govender T. Design and study of peptide-based inhibitors of amylin cytotoxicity. Bioorganic & Medicinal Chemistry Letters. 20: 1360-2. PMID 20093026 DOI: 10.1016/J.Bmcl.2010.01.004 |
0.51 |
|
2010 |
Muthusamy K, Albericio F, Arvidsson PI, Govender P, Kruger HG, Maguire GE, Govender T. Microwave assisted SPPS of amylin and its toxicity of the pure product to RIN-5F cells. Biopolymers. 94: 323-30. PMID 20069542 DOI: 10.1002/Bip.21370 |
0.545 |
|
2010 |
Naicker T, Petzold K, Singh T, Arvidsson PI, Kruger HG, Maguire GEM, Govender T. Novel tetrahydroisoquinoline based organocatalysts for asymmetric Diels-Alder reactions: Insight into the catalytic mode using ROESY NMR and DFT studies Tetrahedron Asymmetry. 21: 2859-2867. DOI: 10.1016/J.Tetasy.2010.11.010 |
0.555 |
|
2009 |
Bose PP, Chatterjee U, Nerelius C, Govender T, Norström T, Gogoll A, Sandegren A, Göthelid E, Johansson J, Arvidsson PI. Poly-N-methylated amyloid β-peptide (Aβ) C-terminal fragments reduce Aβ toxicity in vitro and in Drosophila melanogaster Journal of Medicinal Chemistry. 52: 8002-8009. PMID 19908889 DOI: 10.1021/Jm901092H |
0.302 |
|
2009 |
Hartikka A, Hojabri L, Bose PP, Arvidsson PI. Synthesis and application of novel imidazole and 1H-tetrazolic acid containing catalysts in enantioselective organocatalyzed Diels–Alder reactions Tetrahedron: Asymmetry. 20: 1871-1876. DOI: 10.1016/J.Tetasy.2009.07.029 |
0.347 |
|
2008 |
Norgren AS, Arvidsson PI. Design and synthesis of glycosylated beta3-peptides capable of folding into the 3(14)-helical conformation in water. The Journal of Organic Chemistry. 73: 5272-8. PMID 18576687 DOI: 10.1021/Jo8003265 |
0.32 |
|
2008 |
Zhang S, Arvidsson PI. Facile Synthesis of N-protected Amino Acid Esters Assisted by Microwave Irradiation International Journal of Peptide Research and Therapeutics. 14: 219-222. DOI: 10.1007/S10989-008-9134-3 |
0.384 |
|
2007 |
Hubatsch I, Arvidsson PI, Seebach D, Luthman K, Artursson P. Beta- and gamma-di- and tripeptides as potential substrates for the oligopeptide transporter hPepT1. Journal of Medicinal Chemistry. 50: 5238-42. PMID 17887660 DOI: 10.1021/Jm070148U |
0.419 |
|
2007 |
Hartikka A, Arvidsson PI. Tetrazolic acid functionalized dihydroindol: rational design of a highly selective cyclopropanation organocatalyst. The Journal of Organic Chemistry. 72: 5874-7. PMID 17585815 DOI: 10.1021/Jo070519E |
0.326 |
|
2007 |
Hartikka A, Ślósarczyk AT, Arvidsson PI. Application of novel sulfonamides in enantioselective organocatalyzed cyclopropanation Tetrahedron: Asymmetry. 18: 1403-1409. DOI: 10.1016/J.Tetasy.2007.05.030 |
0.355 |
|
2007 |
Hojabri L, Hartikka A, Moghaddam FM, Arvidsson PI. A new imidazole-containing imidazolidinone catalyst for organocatalyzed asymmetric conjugate addition of nitroalkanes to aldehydes Advanced Synthesis and Catalysis. 349: 740-748. DOI: 10.1002/Adsc.200600316 |
0.373 |
|
2006 |
Norgren AS, Zhang S, Arvidsson PI. Synthesis and circular dichroism spectroscopic investigations of oligomeric beta-peptoids with alpha-chiral side chains. Organic Letters. 8: 4533-6. PMID 16986943 DOI: 10.1021/Ol061717F |
0.322 |
|
2006 |
Norgren AS, Büttner F, Prabpai S, Kongsaeree P, Arvidsson PI. Beta2-amino acids in the design of conformationally homogeneous cyclo-peptide scaffolds. The Journal of Organic Chemistry. 71: 6814-21. PMID 16930031 DOI: 10.1021/Jo060854N |
0.316 |
|
2006 |
Zhang S, Prabpai S, Kongsaeree P, Arvidsson PI. Poly-N-methylated alpha-peptides: synthesis and X-ray structure determination of beta-strand forming foldamers. Chemical Communications (Cambridge, England). 497-9. PMID 16432561 DOI: 10.1039/B513277K |
0.313 |
|
2006 |
Govender T, Arvidsson PI. Facile synthesis of Fmoc-N-methylated α- and β-amino acids Tetrahedron Letters. 47: 1691-1694. DOI: 10.1016/J.Tetlet.2006.01.085 |
0.378 |
|
2006 |
Govender T, Hojabri L, Moghaddam FM, Arvidsson PI. Organocatalytic synthesis of chiral benzopyrans Tetrahedron Asymmetry. 17: 1763-1767. DOI: 10.1016/J.Tetasy.2006.06.028 |
0.413 |
|
2005 |
Arvidsson PI, Ryder NS, Weiss HM, Hook DF, Escalante J, Seebach D. Exploring the antibacterial and hemolytic activity of shorter- and longer-chain beta-, alpha,beta-, and gamma-peptides, and of beta-peptides from beta2-3-aza- and beta3-2-methylidene-amino acids bearing proteinogenic side chains--a survey. Chemistry & Biodiversity. 2: 401-20. PMID 17191989 DOI: 10.1002/Cbdv.200590020 |
0.421 |
|
2005 |
Hedberg C, Källström K, Arvidsson PI, Brandt P, Andersson PG. Mechanistic insights into the phosphine-free RuCp*-diamine-catalyzed hydrogenation of aryl ketones: experimental and theoretical evidence for an alcohol-mediated dihydrogen activation. Journal of the American Chemical Society. 127: 15083-90. PMID 16248647 DOI: 10.1021/Ja051920Q |
0.337 |
|
2005 |
Zhang S, Govender T, Norström T, Arvidsson PI. An improved synthesis of Fmoc-N-methyl-alpha-amino acids. The Journal of Organic Chemistry. 70: 6918-20. PMID 16095315 DOI: 10.1021/Jo050916U |
0.308 |
|
2005 |
Norgren AS, Arvidsson PI. Functionalized foldamers: synthesis and characterization of a glycosylated beta-peptide 314-helix conveying the TN-antigen. Organic & Biomolecular Chemistry. 3: 1359-61. PMID 15827626 DOI: 10.1039/B503237G |
0.351 |
|
2005 |
Hartikka A, Arvidsson PI. 5-(Pyrrolidine-2-yl)tetrazole: Rationale for the Increased Reactivity of the Tetrazole Analogue of Proline in Organocatalyzed Aldol Reactions European Journal of Organic Chemistry. 2005: 4287-4295. DOI: 10.1002/Ejoc.200600266 |
0.36 |
|
2004 |
Hartikka A, Arvidsson PI. Rational design of asymmetric organocatalysts––increased reactivity and solvent scope with a tetrazolic acid Tetrahedron: Asymmetry. 15: 1831-1834. DOI: 10.1016/J.Tetasy.2004.04.029 |
0.333 |
|
2004 |
Büttner F, Erdélyi M, Arvidsson PI. cyclo(β‐Asp‐β3‐hVal‐β3‐hLys) – Solid‐Phase Synthesis and Solution Structure of a Water Soluble β‐Tripeptide. Preliminary Communication Helvetica Chimica Acta. 87: 2735-2741. DOI: 10.1002/Hlca.200490246 |
0.326 |
|
2003 |
Arvidsson PI, Ryder NS, Weiss HM, Gross G, Kretz O, Woessner R, Seebach D. Antibiotic and hemolytic activity of a beta2/beta3 peptide capable of folding into a 12/10-helical secondary structure. Chembiochem : a European Journal of Chemical Biology. 4: 1345-7. PMID 14661278 DOI: 10.1002/Cbic.200300698 |
0.424 |
|
2003 |
Hartikka A, Modin SA, Andersson PG, Arvidsson PI. Cinchona alkaloid derived ligands in catalytic asymmetric transfer hydrogenation. Organic & Biomolecular Chemistry. 1: 2522-6. PMID 12956071 DOI: 10.1039/B304060G |
0.308 |
|
2003 |
Arvidsson P, Frackenpohl J, Seebach D. Syntheses and CD-Spectroscopic Investigations of Longer-Chain -Peptides: Preparation by Solid-Phase Couplings of Single Amino Acids, Dipeptides, and Tripeptides Helvetica Chimica Acta. 86: 1522-1553. DOI: 10.1002/Hlca.200390133 |
0.494 |
|
2002 |
Wiegand H, Wirz B, Schweitzer A, Camenisch GP, Rodriguez Perez MI, Gross G, Woessner R, Voges R, Arvidsson PI, Frackenpohl J, Seebach D. The outstanding metabolic stability of a 14C-labeled beta-nonapeptide in rats--in vitro and in vivo pharmacokinetic studies. Biopharmaceutics & Drug Disposition. 23: 251-62. PMID 12214326 DOI: 10.1002/Bdd.334 |
0.391 |
|
2002 |
Hansson M, Arvidsson PI, Nilsson Lill SO, Ahlberg P. Stereoselective solvent induced 1,3-proton transfer of an allylic alkoxide to a homoallylic alkoxide catalysed by a chiral lithium amide Journal of the Chemical Society, Perkin Transactions 2. 763-767. DOI: 10.1039/B111676B |
0.319 |
|
2001 |
Arvidsson PI, Frackenpohl J, Ryder NS, Liechty B, Petersen F, Zimmermann H, Camenisch GP, Woessner R, Seebach D. On the antimicrobial and hemolytic activities of amphiphilic beta-peptides. Chembiochem : a European Journal of Chemical Biology. 2: 771-3. PMID 11948860 DOI: 10.1002/1439-7633(20011001)2:10<771::Aid-Cbic771>3.0.Co;2-# |
0.417 |
|
2001 |
Frackenpohl J, Arvidsson PI, Schreiber JV, Seebach D. The outstanding biological stability of beta- and gamma-peptides toward proteolytic enzymes: an in vitro investigation with fifteen peptidases. Chembiochem : a European Journal of Chemical Biology. 2: 445-55. PMID 11828476 DOI: 10.1002/1439-7633(20010601)2:6<445::Aid-Cbic445>3.0.Co;2-R |
0.435 |
|
2001 |
Gaul C, Arvidsson PI, Bauer W, Gawley RE, Seebach D. Computational, ReactIR-, and NMR-spectroscopic investigations on the chiral formyl anion equivalent N-(alpha-lithiomethylthiomethyl)-4-isopropyl-5,5-diphenyloxazolidin-2-one and related compounds. Chemistry (Weinheim An Der Bergstrasse, Germany). 7: 4117-25. PMID 11686589 DOI: 10.1002/1521-3765(20011001)7:19<4117::Aid-Chem4117>3.0.Co;2-I |
0.443 |
|
2001 |
Arvidsson PI, Rueping M, Seebach D. Design, machine synthesis, and NMR-solution structure of a β-heptapeptide forming a salt-bridge stabilised 314-helix in methanol and in water Chemical Communications. 649-650. DOI: 10.1039/B101085I |
0.587 |
|
2001 |
Seebach D, Rueping M, Arvidsson PI, Kimmerlin T, Micuch P, Noti C, Langenegger D, Hoyer D. Linear, peptidase-resistant β 2/β 3-Di- and α/β 3-tetrapeptide derivatives with nanomolar affinities to a human somatostatin receptor Helvetica Chimica Acta. 84: 3503-3510. DOI: 10.1002/1522-2675(20011114)84:11<3503::Aid-Hlca3503>3.0.Co;2-A |
0.549 |
|
2001 |
Seebach D, Schreiber J, Arvidsson P, Frackenpohl J. The Miraculous CD Spectra (and Secondary Structures?) ofβ-Peptides as They Grow Longer, Preliminary Communication Helvetica Chimica Acta. 84: 271-279. DOI: 10.1002/1522-2675(20010228)84:2<271::Aid-Hlca271>3.0.Co;2-O |
0.47 |
|
2001 |
Arvidsson PI, Rueping M, Seebach D. Design, machine synthesis, and NMR-solution structure of a β-heptapeptide forming a salt-bridge stabilised 314-helix in methanol and in water Chemical Communications. 649-650. |
0.436 |
|
1999 |
Arvidsson PI, Hilmersson G, Ahlberg P. Stereoselective diamine chelates of a chiral lithium amide dimer: New insights into the coordination chemistry of chiral lithium amides Journal of the American Chemical Society. 121: 1883-1887. DOI: 10.1021/Ja9827550 |
0.324 |
|
1999 |
Arvidsson PI, Davidsson O?, Hilmersson G. Enantioselective butylation of aliphatic aldehydes by mixed chiral lithium amide/n-BuLi dimers Tetrahedron Asymmetry. 10: 527-534. DOI: 10.1016/S0957-4166(99)00033-6 |
0.319 |
|
1999 |
Arvidsson PI, Hilmersson G, Davidsson O. Rational design of chiral lithium amides for asymmetric alkylation reactions - NMR spectroscopic studies of mixed lithium amide/alkyllithium complexes Chemistry - a European Journal. 5: 2348-2355. DOI: 10.1002/(Sici)1521-3765(19990802)5:8<2348::Aid-Chem2348>3.0.Co;2-A |
0.36 |
|
1999 |
Arvidsson PI, Ahlberg P, Hilmersson G. Intraaggregate fluxional lithium and carbanion exchanges in a chiral lithium amide/n-butyllithium mixed tetramer directly observed by multinuclear NMR Chemistry - a European Journal. 5: 1348-1354. DOI: 10.1002/(Sici)1521-3765(19990401)5:4<1348::Aid-Chem1348>3.0.Co;2-L |
0.303 |
|
1998 |
Zul-Qarnain Khan A, de Groot RW, Arvidsson PI, Davidsson Ö. A new chiral lithium amide based on (S)-2-[1-(3,3-dimethyl)pyrrolidinylmethyl]pyrrolidine—synthesis, NMR studies and use in the enantioselective deprotonation of cyclohexene oxide Tetrahedron: Asymmetry. 9: 1223-1229. DOI: 10.1016/S0957-4166(98)00085-8 |
0.324 |
|
1997 |
Hilmersson G, Arvidsson PI, Davidsson O, Håkansson M. Chiral lithium amide/solute complexes: X-ray crystallographic and NMR spectroscopic studies Organometallics. 16: 3352-3362. DOI: 10.1021/Om960989R |
0.303 |
|
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