Andrei K. Yudin, Ph.D. - Publications

Affiliations: 
Chemistry University of Toronto, Toronto, ON, Canada 
Area:
Organic synthesis
Website:
https://www.chem.utoronto.ca/ppl/faculty_profile.php?id=76

169 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2024 Diaz DB, Rowshanpour R, Saunders GJ, Dudding T, Yudin AK. The Role of Attractive Non-Covalent Interactions in Peptide Macrocyclization. The Journal of Organic Chemistry. PMID 38217516 DOI: 10.1021/acs.joc.3c02084  0.335
2023 Li Y, Fan WX, Luo S, Trofimova A, Liu Y, Xue JH, Yang L, Li Q, Wang H, Yudin AK. β-Boron Effect Enables Regioselective and Stereospecific Electrophilic Addition to Alkenes. Journal of the American Chemical Society. PMID 36947220 DOI: 10.1021/jacs.3c00860  0.301
2022 Tien CH, Lough AJ, Yudin AK. Iminologous epoxide ring-closure. Chemical Science. 13: 12175-12179. PMID 36349099 DOI: 10.1039/d2sc04496j  0.32
2022 Huh S, Saunders GJ, Yudin AK. Single Atom Ring Contraction of Peptide Macrocycles Using Cornforth Rearrangement. Angewandte Chemie (International Ed. in English). PMID 36346911 DOI: 10.1002/anie.202214729  0.353
2021 Kaldas SJ, Tien CH, Gomes GDP, Meyer S, Sirvinskas M, Foy H, Dudding T, Yudin AK. Oxidative Rearrangement of MIDA (-Methyliminodiacetic Acid) Boronates: Mechanistic Insights and Synthetic Applications. Organic Letters. PMID 33405935 DOI: 10.1021/acs.orglett.0c03823  0.324
2020 Yudin AK, Tien CH, Trofimova A, Holownia A, Kwak BS, Larson RT. Carboxyboronate as a Versatile in situ CO surrogate in Palladium-Catalyzed Carbonylative Transformations. Angewandte Chemie (International Ed. in English). PMID 33085182 DOI: 10.1002/anie.202010211  0.376
2020 Lebedev YN, Apte C, Cheng S, Lavigne C, Lough A, Seferos DS, Aspuru-Guzik A, Yudin AK. Boramidine: a Versatile Structural Motif for the Design of Fluorescent Heterocycles. Journal of the American Chemical Society. PMID 32602711 DOI: 10.1021/Jacs.0C05410  0.355
2020 Yudin AK. Synthetic half-reactions Chemical Science. DOI: 10.1039/D0Sc03876H  0.319
2019 Kaldas S, Kran E, Mück-Lichtenfeld C, Yudin A, Studer A. Reaction of Vinylaziridines with Arynes: Synthesis of Benzazepines and Branched Allyl Fluorides. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 31628755 DOI: 10.1002/Chem.201904727  0.448
2019 Yamaguchi A, Kaldas SJ, Appavoo SD, Diaz DB, Yudin AK. Conformationally stable peptide macrocycles assembled using the Petasis borono-Mannich reaction. Chemical Communications (Cambridge, England). PMID 31417998 DOI: 10.1039/C9Cc05934B  0.436
2019 Yudin AK, Holownia A, Tien CH, Diaz DB, Larson RT. Carboxyboronate: A Versatile C1-Building Block. Angewandte Chemie (International Ed. in English). PMID 31376232 DOI: 10.1002/Anie.201907486  0.463
2019 Tan J, Grouleff JG, Jitkova Y, Diaz DB, Griffith E, Shao W, Bogdanchikova AF, Poda G, Schimmer AD, Lee RE, Yudin AK. De novo design of boron-based peptidomimetics as potent inhibitors of human ClpP in the presence of human ClpX. Journal of Medicinal Chemistry. PMID 31187989 DOI: 10.1021/acs.jmedchem.9b00878  0.306
2019 Smolyar IV, Yudin AK, Nenajdenko VG. Heteroaryl Rings in Peptide Macrocycles. Chemical Reviews. PMID 31157971 DOI: 10.1021/Acs.Chemrev.8B00789  0.398
2018 Tan J, Yudin AK. Borylated reagents for multicomponent reactions. Drug Discovery Today. Technologies. 29: 51-60. PMID 30471674 DOI: 10.1016/J.Ddtec.2018.08.002  0.426
2018 Corless VB, Holownia A, Foy H, Mendoza-Sanchez R, Adachi S, Dudding T, Yudin AK. Synthesis of α-Borylated Ketones by Regioselective Wacker Oxidation of Alkenylboronates. Organic Letters. PMID 30129366 DOI: 10.1021/Acs.Orglett.8B02234  0.408
2018 Lee CF, Diaz DB, Holownia A, Kaldas SJ, Liew SK, Garrett GE, Dudding T, Yudin AK. Amine hemilability enables boron to mechanistically resemble either hydride or proton. Nature Chemistry. PMID 30061615 DOI: 10.1038/S41557-018-0097-5  0.385
2018 Belding L, Zaretsky S, Yudin AK, Dudding T. A Mechanistic Model for the Aziridine Aldehyde-driven Macrocyclization of Peptides. The Journal of Organic Chemistry. PMID 29966423 DOI: 10.1021/Acs.Joc.8B01198  0.44
2018 Appavoo S, Kaji T, Frost JR, Scully CC, Yudin AK. Development of Endocyclic Control Elements for Peptide Macrocycles. Journal of the American Chemical Society. PMID 29920073 DOI: 10.1021/Jacs.8B04412  0.379
2018 Soor HS, Appavoo SD, Yudin AK. Heterocycles: Versatile control elements in bioactive macrocycles. Bioorganic & Medicinal Chemistry. 26: 2774-2779. PMID 29735427 DOI: 10.1016/J.Bmc.2017.10.022  0.382
2018 Kaldas SJ, Rogova T, Nenajdenko VG, Yudin AK. Modular Synthesis of β-Amino Boronate Peptidomimetics. The Journal of Organic Chemistry. PMID 29631400 DOI: 10.1021/Acs.Joc.8B00325  0.443
2018 Kaldas SJ, Yudin AK. Achieving Skeletal Diversity in Peptide Macrocycles Through The Use of Heterocyclic Grafts. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 29363202 DOI: 10.1002/Chem.201705418  0.365
2018 Soor HS, Hansen J, Diaz DB, Appavoo S, Yudin AK. Solid-phase synthesis of peptide β-aminoboronic acids Peptide Science. 111: e24072. DOI: 10.1002/Pep2.24072  0.357
2018 Kaldas SJ, Yudin AK. Frontispiece: Achieving Skeletal Diversity in Peptide Macrocycles through The Use of Heterocyclic Grafts Chemistry - a European Journal. 24. DOI: 10.1002/Chem.201882861  0.324
2017 Zaretsky S, Yudin AK. Recent advances in the synthesis of cyclic pseudopeptides. Drug Discovery Today. Technologies. 26: 3-10. PMID 29249240 DOI: 10.1016/J.Ddtec.2017.11.004  0.424
2017 Tan J, Cognetta Iii AB, Diaz DB, Lum KM, Adachi S, Kundu S, Cravatt BF, Yudin AK. Multicomponent mapping of boron chemotypes furnishes selective enzyme inhibitors. Nature Communications. 8: 1760. PMID 29170371 DOI: 10.1038/S41467-017-01319-4  0.312
2017 Liew SK, Holownia A, Diaz DB, Cistrone PA, Dawson PE, Yudin AK. Borylated oximes: versatile building blocks for organic synthesis. Chemical Communications (Cambridge, England). PMID 28959806 DOI: 10.1039/C7Cc06579E  0.417
2017 Shao W, Kaldas SJ, Yudin AK. 3-Cyanoallyl boronates are versatile building blocks in the synthesis of polysubstituted thiophenes. Chemical Science. 8: 4431-4436. PMID 28936329 DOI: 10.1039/C7Sc00831G  0.402
2017 Mendoza-Sanchez R, Corless VB, Nguyen QNN, Bergeron-Brlek M, Frost J, Adachi S, Tantillo DJ, Yudin AK. Cyclols Revisited: Facile Synthesis of Medium-Sized Cyclic Peptides. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28771904 DOI: 10.1002/Chem.201703616  0.381
2017 Diaz DB, Yudin AK. The versatility of boron in biological target engagement. Nature Chemistry. 9: 731-742. PMID 28754930 DOI: 10.1038/Nchem.2814  0.305
2017 Chung BKW, White CJ, Yudin AK. Solid-phase synthesis, cyclization, and site-specific functionalization of aziridine-containing tetrapeptides. Nature Protocols. 12: 1277-1287. PMID 28538738 DOI: 10.1038/Nprot.2017.035  0.459
2017 Yudin AK, Kaldas SJ, O'Keefe KTV, Rodrigo MS. Amphoteric Borylketenimines: Versatile Intermediates in the Synthesis of Borylated Heterocycles. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28475819 DOI: 10.1002/Chem.201702008  0.454
2017 Belding L, Zaretsky S, Yudin AK, Dudding T. A mechanistic model for the aziridine aldehyde-driven macrocyclization of peptides. The Journal of Organic Chemistry. PMID 28273421 DOI: 10.1021/Acs.Joc.6B02899  0.441
2017 Lee CF, Holownia A, Bennett JM, Elkins JM, St Denis JD, Adachi S, Yudin AK. Oxalyl Boronates Enable Modular Synthesis of Bioactive Imidazoles. Angewandte Chemie (International Ed. in English). PMID 28267269 DOI: 10.1002/Anie.201611006  0.428
2017 Garrett GE, Diaz DB, Yudin AK, Taylor MS. Reversible covalent interactions of β-aminoboronic acids with carbohydrate derivatives. Chemical Communications (Cambridge, England). PMID 28106188 DOI: 10.1039/C6Cc09640A  0.302
2017 St. Denis JD, Liew SK, Scully CCG, Yudin AK. Activation of Alkynylzinc Reagents by a Hemiaminal-Driven Catalytic Microenvironment European Journal of Organic Chemistry. 2017: 419-423. DOI: 10.1002/Ejoc.201601554  0.464
2017 Kaldas SJ, O'Keefe KTV, Mendoza-Sanchez R, Yudin AK. Frontispiece: Amphoteric Borylketenimines: Versatile Intermediates in the Synthesis of Borylated Heterocycles Chemistry - a European Journal. 23. DOI: 10.1002/Chem.201784162  0.452
2016 Chung BKW, White CJ, Scully CCG, Yudin AK. The reactivity and conformational control of cyclic tetrapeptides derived from aziridine-containing amino acids. Chemical Science. 7: 6662-6668. PMID 28567256 DOI: 10.1039/C6Sc01687A  0.441
2016 Liew SK, Kaldas SJ, Yudin AK. A Linchpin Synthesis of 6-Hydroxyceramides from Aziridine Aldehydes. Organic Letters. 18: 6268-6271. PMID 27978678 DOI: 10.1021/Acs.Orglett.6B03067  0.414
2016 Frost JR, Scully CC, Yudin AK. Oxadiazole grafts in peptide macrocycles. Nature Chemistry. 8: 1105-1111. PMID 27874866 DOI: 10.1038/Nchem.2636  0.431
2016 Scully CC, White CJ, Yudin AK. The effect of backbone flexibility on site-selective modification of macrocycles. Organic & Biomolecular Chemistry. PMID 27735955 DOI: 10.1039/C6Ob01778A  0.427
2016 Diaz DB, Scully CC, Liew SK, Adachi S, Trinchera P, St Denis JD, Yudin AK. Synthesis of Aminoboronic Acid Derivatives from Amines and Amphoteric Boryl Carbonyl Compounds. Angewandte Chemie (International Ed. in English). PMID 27584917 DOI: 10.1002/Anie.201605754  0.497
2016 Liew SK, Holownia A, Tilley AJ, Carrera EI, Seferos DS, Yudin AK. A study of boratriazaroles - an underdeveloped class of heterocycles. The Journal of Organic Chemistry. PMID 27513290 DOI: 10.1021/Acs.Joc.6B01565  0.336
2016 Heine NB, Kaldas SJ, Belding L, Shmatova O, Dudding T, Nenajdenko VG, Studer A, Yudin AK. Synthesis of chiral piperazinones using amphoteric aziridine aldehyde dimers and functionalized isocyanides. The Journal of Organic Chemistry. PMID 27156711 DOI: 10.1021/Acs.Joc.6B00471  0.432
2016 Low KE, Ler S, Chen K, Campbell RL, Hickey JL, Tan J, Scully CC, Davies PL, Yudin AK, Zaretsky S. Rational design of calpain inhibitors based on calpastatin peptidomimetics. Journal of Medicinal Chemistry. PMID 27148623 DOI: 10.1021/Acs.Jmedchem.6B00267  0.314
2016 Hickey JL, Zaretsky S, St Denis MA, Kumar Chakka S, Morshed MM, Scully CC, Roughton AL, Yudin AK. Passive membrane permeability of macrocycles can be controlled by exocyclic amide bonds. Journal of Medicinal Chemistry. PMID 27120576 DOI: 10.1021/Acs.Jmedchem.6B00222  0.434
2015 Zaretsky S, Hickey JL, Tan J, Pichugin D, St Denis MA, Ler S, Chung BKW, Scully CCG, Yudin AK. Mechanistic investigation of aziridine aldehyde-driven peptide macrocyclization: the imidoanhydride pathway. Chemical Science. 6: 5446-5455. PMID 29861887 DOI: 10.1039/C5Sc01958C  0.42
2015 Yudin AK. Macrocycles: lessons from the distant past, recent developments, and future directions. Chemical Science. 6: 30-49. PMID 28553456 DOI: 10.1039/C4Sc03089C  0.356
2015 St Denis JD, Lee CF, Yudin AK. Access to Cyclic Amino Boronates via Rhodium-Catalyzed Functionalization of Alkyl MIDA Boronates. Organic Letters. PMID 26588176 DOI: 10.1021/Acs.Orglett.5B02861  0.422
2015 Adachi S, Liew SK, Lee CF, Lough A, He Z, Denis JD, Poda G, Yudin AK. Condensation-Driven Assembly of Boron-Containing Bis(Heteroaryl) Motifs Using a Linchpin Approach. Organic Letters. PMID 26551599 DOI: 10.1021/Acs.Orglett.5B02741  0.617
2015 Chung BK, Yudin AK. Disulfide-bridged peptide macrobicycles from nature. Organic & Biomolecular Chemistry. 13: 8768-79. PMID 26159878 DOI: 10.1039/C5Ob01115A  0.398
2015 Trinchera P, Corless VB, Yudin AK. Synthesis of Previously Inaccessible Borylated Heterocycle Motifs Using Novel Boron-Containing Amphoteric Molecules. Angewandte Chemie (International Ed. in English). PMID 26110917 DOI: 10.1002/Anie.201504271  0.423
2015 Zaretsky S, Rai V, Gish G, Forbes MW, Kofler M, Yu JC, Tan J, Hickey JL, Pawson T, Yudin AK. Twisted amide electrophiles enable cyclic peptide sequencing. Organic & Biomolecular Chemistry. PMID 26077966 DOI: 10.1039/C5Ob01050K  0.586
2015 Treder AP, Hickey JL, Tremblay MC, Zaretsky S, Scully CC, Mancuso J, Doucet A, Yudin AK, Marsault E. Solid-Phase Parallel Synthesis of Functionalised Medium-to-Large Cyclic Peptidomimetics through Three-Component Coupling Driven by Aziridine Aldehyde Dimers. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 9249-55. PMID 26014974 DOI: 10.1002/Chem.201500068  0.435
2015 Adachi S, Cognetta AB, Niphakis MJ, He Z, Zajdlik A, St Denis JD, Scully CC, Cravatt BF, Yudin AK. Facile synthesis of borofragments and their evaluation in activity-based protein profiling. Chemical Communications (Cambridge, England). 51: 3608-11. PMID 25633248 DOI: 10.1039/C4Cc09107H  0.559
2015 Zaretsky S, Tan J, Hickey JL, Yudin AK. Macrocyclic templates for library synthesis of peptido-conjugates. Methods in Molecular Biology (Clifton, N.J.). 1248: 67-80. PMID 25616326 DOI: 10.1007/978-1-4939-2020-4_5  0.406
2015 St. Denis JD, He Z, Yudin AK. Amphoteric α-Boryl Aldehyde Linchpins in the Synthesis of Heterocycles Acs Catalysis. 5: 5373-5379. DOI: 10.1021/Acscatal.5B00790  0.643
2015 Trinchera P, Corless VB, Yudin AK. Cover Picture: Synthesis of Previously Inaccessible Borylated Heterocycle Motifs Using Novel Boron-Containing Amphoteric Molecules (Angew. Chem. Int. Ed. 31/2015) Angewandte Chemie International Edition. 54: 8849-8849. DOI: 10.1002/Anie.201505831  0.392
2015 Trinchera P, Corless VB, Yudin AK. Titelbild: Synthesis of Previously Inaccessible Borylated Heterocycle Motifs Using Novel Boron-Containing Amphoteric Molecules (Angew. Chem. 31/2015) Angewandte Chemie. 127: 8975-8975. DOI: 10.1002/Ange.201505831  0.408
2014 St Denis JD, Zajdlik A, Tan J, Trinchera P, Lee CF, He Z, Adachi S, Yudin AK. Boron-containing enamine and enamide linchpins in the synthesis of nitrogen heterocycles. Journal of the American Chemical Society. 136: 17669-73. PMID 25422871 DOI: 10.1021/Ja510963K  0.604
2014 Belding L, Zaretsky S, Rotstein BH, Yudin AK, Dudding T. Shifting the energy landscape of multicomponent reactions using aziridine aldehyde dimers: a mechanistic study. The Journal of Organic Chemistry. 79: 9465-71. PMID 25264960 DOI: 10.1021/Jo501242R  0.722
2014 Zaretsky S, Adachi S, Rotstein BH, Hickey JL, Scully CC, St Denis JD, Courtemanche R, Yu JC, Chung BK, Yudin AK. Stereocontrolled disruption of the Ugi reaction toward the production of chiral piperazinones: substrate scope and process development. The Journal of Organic Chemistry. 79: 9948-57. PMID 25254948 DOI: 10.1021/Jo5018316  0.726
2014 Treder AP, Tremblay MC, Yudin AK, Marsault E. Solid-phase synthesis of piperazinones via disrupted Ugi condensation. Organic Letters. 16: 4674-7. PMID 25153611 DOI: 10.1021/Ol5023118  0.42
2014 Rotstein BH, Zaretsky S, Rai V, Yudin AK. Small heterocycles in multicomponent reactions. Chemical Reviews. 114: 8323-59. PMID 25032909 DOI: 10.1021/Cr400615V  0.755
2014 He Z, Zajdlik A, Yudin AK. α-Borylcarbonyl compounds: from transient intermediates to robust building blocks. Dalton Transactions (Cambridge, England : 2003). 43: 11434-51. PMID 24941221 DOI: 10.1039/C4Dt00817K  0.562
2014 White CJ, Hickey JL, Scully CC, Yudin AK. Site-specific integration of amino acid fragments into cyclic peptides. Journal of the American Chemical Society. 136: 3728-31. PMID 24533886 DOI: 10.1021/Ja412256F  0.375
2014 St Denis JD, Scully CC, Lee CF, Yudin AK. Development of the direct Suzuki-Miyaura cross-coupling of primary B-alkyl MIDA-boronates and aryl bromides. Organic Letters. 16: 1338-41. PMID 24527782 DOI: 10.1021/Ol500057A  0.392
2014 He Z, Zajdlik A, Yudin AK. Air- and moisture-stable amphoteric molecules: enabling reagents in synthesis. Accounts of Chemical Research. 47: 1029-40. PMID 24495255 DOI: 10.1021/Ar400210C  0.65
2014 Zajdlik A, He Z, St Denis JD, Yudin AK. Efficient preparation of α-aminoboronic acid derivatives via boroalkyl group migration Synthesis (Germany). 46: 445-454. DOI: 10.1055/S-0033-1340502  0.591
2014 Zaretsky S, Hickey JL, St. Denis MA, Scully CCG, Roughton AL, Tantillo DJ, Lodewyk MW, Yudin AK. Predicting cyclic peptide chemical shifts using quantum mechanical calculations Tetrahedron. 70: 7655-7663. DOI: 10.1016/J.Tet.2014.07.070  0.303
2014 Zaretsky S, Scully CCG, Lough AJ, Yudin AK. Corrigendum: Exocyclic Control of Turn Induction in Macrocyclic Peptide Scaffolds Chemistry - a European Journal. 20: 2983-2983. DOI: 10.1002/Chem.201400422  0.335
2013 Zaretsky S, Scully CC, Lough AJ, Yudin AK. Exocyclic control of turn induction in macrocyclic peptide scaffolds. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 17668-72. PMID 24259185 DOI: 10.1002/Chem.201303453  0.335
2013 Liew SK, He Z, St Denis JD, Yudin AK. Stereocontrolled synthesis of 1,2- and 1,3-diamine building blocks from aziridine aldehyde dimers. The Journal of Organic Chemistry. 78: 11637-45. PMID 23957736 DOI: 10.1021/Jo401489Q  0.647
2013 Zajdlik A, Wang Z, Hickey JL, Aman A, Schimmer AD, Yudin AK. α-Boryl isocyanides enable facile preparation of bioactive boropeptides. Angewandte Chemie (International Ed. in English). 52: 8411-5. PMID 23818141 DOI: 10.1002/Anie.201302818  0.304
2013 Dubovyk I, Watson ID, Yudin AK. Achieving control over the branched/linear selectivity in palladium-catalyzed allylic amination. The Journal of Organic Chemistry. 78: 1559-75. PMID 23327430 DOI: 10.1021/Jo3025253  0.81
2013 He Z, Dobrovolsky D, Trinchera P, Yudin AK. Synthesis of multisubstituted pyridines. Organic Letters. 15: 334-7. PMID 23273041 DOI: 10.1021/Ol303246B  0.65
2013 Chung BKW, Hickey JL, Scully CCG, Zaretsky S, Yudin AK. Bicycle synthesis through peptide macrocyclization using aziridine aldehydes followed by late stage disulfide bond installation Medchemcomm. 4: 1124-1128. DOI: 10.1039/C3Md00054K  0.462
2012 Scully CC, Rai V, Poda G, Zaretsky S, Burns DC, Houliston RS, Lou T, Yudin AK. Bending rigid molecular rods: formation of oligoproline macrocycles. Chemistry (Weinheim An Der Bergstrasse, Germany). 18: 15612-7. PMID 23124621 DOI: 10.1002/Chem.201203266  0.602
2012 He Z, Trinchera P, Adachi S, St Denis JD, Yudin AK. Oxidative geminal functionalization of organoboron compounds. Angewandte Chemie (International Ed. in English). 51: 11092-6. PMID 23038428 DOI: 10.1002/Anie.201206501  0.568
2012 St Denis JD, He Z, Yudin AK. Chemoselective palladium-catalyzed α-allylation of α-boryl aldehydes. Organic & Biomolecular Chemistry. 10: 7900-2. PMID 22911058 DOI: 10.1039/C2Ob26503F  0.581
2012 Assem N, Yudin AK. Convergent synthesis of aminomethylene peptidomimetics. Nature Protocols. 7: 1327-34. PMID 22722368 DOI: 10.1038/Nprot.2012.066  0.798
2012 Roxin Á, Chen J, Scully CC, Rotstein BH, Yudin AK, Zheng G. Conformational modulation of in vitro activity of cyclic RGD peptides via aziridine aldehyde-driven macrocyclization chemistry. Bioconjugate Chemistry. 23: 1387-95. PMID 22709546 DOI: 10.1021/Bc300239A  0.716
2012 He Z, Zajdlik A, St Denis JD, Assem N, Yudin AK. Boroalkyl group migration provides a versatile entry into α-aminoboronic acid derivatives. Journal of the American Chemical Society. 134: 9926-9. PMID 22662871 DOI: 10.1021/Ja304173D  0.797
2012 Assem N, Hili R, He Z, Kasahara T, Inman BL, Decker S, Yudin AK. Role of reversible dimerization in reactions of amphoteric aziridine aldehydes. The Journal of Organic Chemistry. 77: 5613-23. PMID 22662756 DOI: 10.1021/Jo3007418  0.791
2012 White CJ, Yudin AK. A versatile scaffold for site-specific modification of cyclic tetrapeptides. Organic Letters. 14: 2898-901. PMID 22612626 DOI: 10.1021/Ol301178R  0.368
2012 Rotstein BH, Winternheimer DJ, Yin LM, Deber CM, Yudin AK. Thioester-isocyanides: versatile reagents for the synthesis of cycle-tail peptides. Chemical Communications (Cambridge, England). 48: 3775-7. PMID 22430393 DOI: 10.1039/C2Cc16027G  0.71
2012 Jebrail MJ, Assem N, Mudrik JM, Dryden MDM, Lin K, Yudin AK, Wheeler AR. Combinatorial synthesis of peptidomimetics using digital microfluidics Proceedings of the 16th International Conference On Miniaturized Systems For Chemistry and Life Sciences, Microtas 2012. 1774-1776. DOI: 10.1556/Jfc-D-12-00012  0.794
2012 Rotstein BH, Yudin AK. Aziridine-2-carboxaldehyde dimers undergo homo-Ugi 4-component-5-center reactions Synthesis (Germany). 44: 2851-2858. DOI: 10.1055/S-0030-1260261  0.708
2012 Yudin AK. Synthesis of heterocycles using amphoteric molecules Chemistry of Heterocyclic Compounds. 48: 191-199. DOI: 10.1007/S10593-012-0982-6  0.426
2011 Cheung LL, He Z, Decker SM, Yudin AK. Skeletal fusion of small heterocycles with amphoteric molecules. Angewandte Chemie (International Ed. in English). 50: 11798-802. PMID 21990009 DOI: 10.1002/Anie.201106024  0.512
2011 Rotstein BH, Mourtada R, Kelley SO, Yudin AK. Solvatochromic reagents for multicomponent reactions and their utility in the development of cell-permeable macrocyclic peptide vectors. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 12257-61. PMID 21932287 DOI: 10.1002/Chem.201102096  0.711
2011 He Z, Yudin AK. Amphoteric α-boryl aldehydes. Journal of the American Chemical Society. 133: 13770-3. PMID 21809873 DOI: 10.1021/Ja205910D  0.635
2011 White CJ, Yudin AK. Contemporary strategies for peptide macrocyclization. Nature Chemistry. 3: 509-24. PMID 21697871 DOI: 10.1038/Nchem.1062  0.405
2011 Prakash GK, Wang F, Ni C, Shen J, Haiges R, Yudin AK, Mathew T, Olah GA. Conformational study of 9-dehydro-9-trifluoromethyl cinchona alkaloids via 19F NMR spectroscopy: emergence of trifluoromethyl moiety as a conformational stabilizer and a probe. Journal of the American Chemical Society. 133: 9992-5. PMID 21648459 DOI: 10.1021/Ja202373D  0.558
2011 Dubovyk I, Pichugin D, Yudin AK. Palladium-catalyzed ring-contraction and ring-expansion reactions of cyclic allyl amines. Angewandte Chemie (International Ed. in English). 50: 5924-6. PMID 21567674 DOI: 10.1002/Anie.201100612  0.798
2011 Siebert MR, Yudin AK, Tantillo DJ. The effect of strain on the RhI-catalyzed rearrangement of allylamines European Journal of Organic Chemistry. 553-561. DOI: 10.1002/Ejoc.201001132  0.397
2010 Rotstein BH, Rai V, Hili R, Yudin AK. Synthesis of peptide macrocycles using unprotected amino aldehydes. Nature Protocols. 5: 1813-22. PMID 21030956 DOI: 10.1038/Nprot.2010.127  0.778
2010 Jebrail MJ, Ng AH, Rai V, Hili R, Yudin AK, Wheeler AR. Synchronized synthesis of peptide-based macrocycles by digital microfluidics. Angewandte Chemie (International Ed. in English). 49: 8625-9. PMID 20715231 DOI: 10.1002/Anie.201001604  0.635
2010 Assem N, Natarajan A, Yudin AK. Chemoselective peptidomimetic ligation using thioacid peptides and aziridine templates. Journal of the American Chemical Society. 132: 10986-7. PMID 20666404 DOI: 10.1021/Ja104488D  0.795
2010 Cheung LL, Yudin AK. Synthesis of highly substituted cyclobutane fused-ring systems from N-vinyl beta-lactams through a one-pot domino process. Chemistry (Weinheim An Der Bergstrasse, Germany). 16: 4100-9. PMID 20186912 DOI: 10.1002/Chem.200902748  0.422
2010 Hili R, Rai V, Yudin AK. Macrocyclization of linear peptides enabled by amphoteric molecules. Journal of the American Chemical Society. 132: 2889-91. PMID 20155938 DOI: 10.1021/Ja910544P  0.634
2010 He Z, Yudin AK. A versatile synthetic platform based on strained propargyl amines. Angewandte Chemie (International Ed. in English). 49: 1607-10. PMID 20119999 DOI: 10.1002/Anie.200906066  0.514
2010 Baktharaman S, Afagh N, Vandersteen A, Yudin AK. Unprotected vinyl aziridines: facile synthesis and cascade transformations. Organic Letters. 12: 240-3. PMID 20017499 DOI: 10.1021/Ol902550Q  0.357
2010 Afagh NA, Yudin AK. Chemoselectivity and the curious reactivity preferences of functional groups. Angewandte Chemie (International Ed. in English). 49: 262-310. PMID 20014082 DOI: 10.1002/Anie.200901317  0.404
2010 YUDIN AK, SHARPLESS KB. ChemInform Abstract: Bis(trimethylsilyl) Peroxide Extends the Range of Oxorhenium Catalysts for Olefin Epoxidation. Cheminform. 29: no-no. DOI: 10.1002/chin.199810117  0.429
2010 PRAKASH GKS, YUDIN AK, DEFFIEUX D, OLAH GA. ChemInform Abstract: Synthetic Methods. Part 197. Facile Preparation of (Trifluoromethyl) tributyltin and Transtrifluoromethylation of Disilyl Sulfides to the Corresponding Trifluoromethylsilanes. Cheminform. 27: no-no. DOI: 10.1002/chin.199625163  0.392
2010 OLAH GA, RASUL G, YUDIN AK, BURRICHTER A, PRAKASH GKS, CHISTYAKOV AL, STANKEVICH IV, AKHREM IS, GAMBARYAN NP, VOL'PIN ME. ChemInform Abstract: Chemistry in Superacids. Part 21. Trihalomethyl Cations and Their Superelectrophilic Activation Cheminform. 27: no-no. DOI: 10.1002/chin.199624048  0.31
2010 PRAKASH GKS, DEFFIEUX D, YUDIN AK, OLAH GA. ChemInform Abstract: Considered Synthetic Methods and Reactions. Part 195. Convenient and Safe Electrochemical Synthesis of (Trifluoromethyl)trimethylsilane. Cheminform. 26: no-no. DOI: 10.1002/chin.199529038  0.344
2010 Jebrail MJ, Ng AHC, Rai V, Hili R, Yudin AK, Wheeler AR. Inside Cover: Synchronized Synthesis of Peptide-Based Macrocycles by Digital Microfluidics (Angew. Chem. Int. Ed. 46/2010) Angewandte Chemie International Edition. 49: 8536-8536. DOI: 10.1002/Anie.201004588  0.583
2010 Jebrail MJ, Ng AHC, Rai V, Hili R, Yudin AK, Wheeler AR. Innentitelbild: Synchronized Synthesis of Peptide-Based Macrocycles by Digital Microfluidics (Angew. Chem. 46/2010) Angewandte Chemie. 122: 8716-8716. DOI: 10.1002/Ange.201004588  0.586
2009 Hili R, Yudin AK. Amphoteric amino aldehydes reroute the aza-Michael reaction. Journal of the American Chemical Society. 131: 16404-6. PMID 19856916 DOI: 10.1021/Ja9072194  0.459
2009 Cheung LL, Yudin AK. Synthesis of aminocyclobutanes through ring expansion of N-vinyl-beta-lactams. Organic Letters. 11: 1281-4. PMID 19239262 DOI: 10.1021/Ol900118D  0.324
2009 De Iuliis MZ, Watson IDG, Yudin AK, Morris RH. A DFT investigation into the origin of regioselectivity in palladium-catalyzed allylic amination Canadian Journal of Chemistry. 87: 54-62. DOI: 10.1139/V08-078  0.349
2009 Jebrail MJ, Ng A, Rai V, Hili R, Yudin AK, Wheeler AR. Synchronized synthesis of cyclic peptides by digital microfluidics Proceedings of Conference, Microtas 2009 - the 13th International Conference On Miniaturized Systems For Chemistry and Life Sciences. 1297-1299.  0.537
2008 Rasmusson T, Martyn LJ, Chen G, Lough A, Oh M, Yudin AK. Aromatic fluorine as a versatile control element for the construction of molecules with helical chirality. Angewandte Chemie (International Ed. in English). 47: 7009-12. PMID 18671224 DOI: 10.1002/Anie.200801991  0.437
2008 Tsang DS, Yang S, Alphonse FA, Yudin AK. Stereoselective isomerisation of N-allyl aziridines into geometrically stable Z enamines by using rhodium hydride catalysis. Chemistry (Weinheim An Der Bergstrasse, Germany). 14: 886-94. PMID 17992683 DOI: 10.1002/Chem.200701322  0.391
2008 Hili R, Baktharaman S, Yudin AK. Synthesis of Chiral Amines Using α-Amino Aldehydes (Eur. J. Org. Chem. 31/2008) European Journal of Organic Chemistry. 2008: 5191-5191. DOI: 10.1002/Ejoc.200890084  0.384
2008 Hili R, Baktharaman S, Yudin AK. Synthesis of chiral amines using α-amino aldehydes European Journal of Organic Chemistry. 5201-5213. DOI: 10.1002/Ejoc.200800604  0.388
2007 Li X, Yudin AK. Epimerization- and protecting-group-free synthesis of peptidomimetic conjugates from amphoteric amino aldehydes. Journal of the American Chemical Society. 129: 14152-3. PMID 17963392 DOI: 10.1021/Ja076155P  0.434
2007 Dubovyk I, Watson ID, Yudin AK. Chasing the proton culprit from palladium-catalyzed allylic amination. Journal of the American Chemical Society. 129: 14172-3. PMID 17960935 DOI: 10.1021/Ja076659N  0.8
2007 Blyumin EV, Gallon HJ, Yudin AK. Construction of three contiguous tertiary stereocenters from aziridines in one step. Organic Letters. 9: 4677-80. PMID 17929932 DOI: 10.1021/Ol7015302  0.395
2007 Yudin AK, Hili R. Overcoming the demons of protecting groups with amphoteric molecules. Chemistry (Weinheim An Der Bergstrasse, Germany). 13: 6538-42. PMID 17623282 DOI: 10.1002/Chem.200700710  0.348
2007 Yu L, Kokai A, Yudin AK. Preparation and reactivity of versatile alpha-amino ketones. The Journal of Organic Chemistry. 72: 1737-41. PMID 17256911 DOI: 10.1021/Jo062401O  0.476
2007 Yang X, Yudin AK. Facile generation and synthetic utility of nitrogen-centered aziridinyl radicals Synlett. 2912-2918. DOI: 10.1055/S-2007-990960  0.376
2007 Yekta S, Cheung L, Yudin AK. Polyfluorinated phosphine ligands in the room temperature Suzuki cross-coupling reactions Tetrahedron Letters. 48: 8048-8051. DOI: 10.1016/J.Tetlet.2007.09.016  0.398
2006 He Z, Yudin AK. Palladium-catalyzed oxidative activation of arylcyclopropanes. Organic Letters. 8: 5829-32. PMID 17134283 DOI: 10.1021/Ol062476E  0.642
2006 Hili R, Yudin AK. Readily available unprotected amino aldehydes. Journal of the American Chemical Society. 128: 14772-3. PMID 17105264 DOI: 10.1021/Ja065898S  0.483
2006 Alphonse FA, Yudin AK. Rhodium-catalyzed stereoselective formation of Z-enamines from allylaziridines. Journal of the American Chemical Society. 128: 11754-5. PMID 16953604 DOI: 10.1021/Ja0632557  0.375
2006 Chen G, Sasaki M, Li X, Yudin AK. Strained enamines as versatile intermediates for stereocontrolled construction of nitrogen heterocycles. The Journal of Organic Chemistry. 71: 6067-73. PMID 16872190 DOI: 10.1021/Jo0607921  0.449
2006 Hili R, Yudin AK. Making carbon-nitrogen bonds in biological and chemical synthesis. Nature Chemical Biology. 2: 284-7. PMID 16710330 DOI: 10.1038/Nchembio0606-284  0.365
2006 Watson ID, Yu L, Yudin AK. Advances in nitrogen transfer reactions involving aziridines. Accounts of Chemical Research. 39: 194-206. PMID 16548508 DOI: 10.1021/Ar050038M  0.689
2006 Chen G, Sasaki M, Yudin AK. Facile preparation of allyl amines and pyrazoles by hydrazinolysis of 2-ketoaziridines Tetrahedron Letters. 47: 255-259. DOI: 10.1016/J.Tetlet.2005.11.039  0.412
2005 Watson ID, Yudin AK. New insights into the mechanism of palladium-catalyzed allylic amination. Journal of the American Chemical Society. 127: 17516-29. PMID 16332104 DOI: 10.1021/Ja055288C  0.7
2005 Dalili S, Yudin AK. Transition metal-catalyzed synthesis and reactivity of N-alkenyl aziridines. Organic Letters. 7: 1161-4. PMID 15760164 DOI: 10.1021/Ol050094N  0.455
2005 Siu T, Picard CJ, Yudin AK. Development of electrochemical processes for nitrene generation and transfer. The Journal of Organic Chemistry. 70: 932-7. PMID 15675851 DOI: 10.1021/Jo048591P  0.59
2005 Krasnova LB, Yudin AK. Novel nitrogen containing chelating ligands from aziridines -Preparation, coordination studies, and catalytic application in the cyclopropanation of styrene Canadian Journal of Chemistry. 83: 1025-1032. DOI: 10.1139/V05-113  0.387
2004 Watson ID, Styler SA, Yudin AK. Unusual selectivity of unprotected aziridines in palladium-catalyzed allylic amination enables facile preparation of branched aziridines. Journal of the American Chemical Society. 126: 5086-7. PMID 15099089 DOI: 10.1021/Ja049242F  0.681
2004 Krasnova LB, Yudin AK. p-Tolylsulfinyl amides: reagents for facile electrophilic functionalization of olefins. The Journal of Organic Chemistry. 69: 2584-7. PMID 15049664 DOI: 10.1021/Jo035518A  0.303
2004 Krasnova LB, Hili RM, Chernoloz OV, Yudin AK. Phenyliodine(III) diacetate as a mild oxidant for aziridination of olefins and imination of sulfoxides with N-aminophthalimide Arkivoc. 2005: 26-38. DOI: 10.3998/Ark.5550190.0006.404  0.398
2004 Caiazzo A, Dalili S, Picard C, Sasaki M, Siu T, Yudin AK. New methods for the synthesis of heterocyclic compounds Pure and Applied Chemistry. 76: 603-613. DOI: 10.1351/Pac200476030603  0.624
2004 Sasaki M, Yudin AK. One-pot reduction-aldol reaction of esters Synlett. 2443-2444. DOI: 10.1055/S-2004-834808  0.469
2004 Dalili S, Caiazzo A, Yudin AK. Aziridine-derived iminophosphine ligands in palladium-catalyzed allylic substitution Journal of Organometallic Chemistry. 689: 3604-3611. DOI: 10.1016/J.Jorganchem.2004.07.066  0.304
2004 Yekta S, Krasnova LB, Mariampillai B, Picard CJ, Chen G, Pandiaraju S, Yudin AK. Preparation and catalytic applications of partially fluorinated binaphthol ligands Journal of Fluorine Chemistry. 125: 517-525. DOI: 10.1016/J.Jfluchem.2003.11.024  0.392
2003 Sasaki M, Yudin AK. Oxidative cycloamination of olefins with aziridines as a versatile route to saturated nitrogen-containing heterocycles. Journal of the American Chemical Society. 125: 14242-3. PMID 14624549 DOI: 10.1021/Ja037726Q  0.415
2003 Watson ID, Yudin AK. Ring-opening reactions of nonactivated aziridines catalyzed by tris(pentafluorophenyl)borane. The Journal of Organic Chemistry. 68: 5160-7. PMID 12816471 DOI: 10.1021/Jo0343578  0.685
2003 Sasaki M, Dalili S, Yudin AK. N-arylation of aziridines. The Journal of Organic Chemistry. 68: 2045-7. PMID 12608835 DOI: 10.1021/Jo020696+  0.383
2003 Caiazzo A, Dalili S, Yudin AK. Lewis Acid-Catalyzed Dimerization of N-Unprotected Aziridines Synlett. 2198-2202. DOI: 10.1055/S-2003-42062  0.424
2003 Chen Y, Yudin AK. Synthesis of 3-aminoaspartic acid derivatives from glycine precursors Tetrahedron Letters. 44: 4865-4868. DOI: 10.1016/S0040-4039(03)01122-5  0.416
2002 Watson ID, Yudin AK. Selective functionalization of small organic molecules using electrophilic nitrogen sources. Current Opinion in Drug Discovery & Development. 5: 906-17. PMID 12478721  0.617
2002 Caiazzo A, Dalili S, Yudin AK. Design and development of cyclohexane-based P,N-ligands for transition metal catalysis. Organic Letters. 4: 2597-600. PMID 12123385 DOI: 10.1021/Ol026249Y  0.375
2002 Siu T, Yudin AK. Electrochemical imination of sulfoxides using N-aminophthalimide. Organic Letters. 4: 1839-42. PMID 12027627 DOI: 10.1021/Ol0257530  0.567
2002 Siu T, Yudin AK. Practical olefin aziridination with a broad substrate scope. Journal of the American Chemical Society. 124: 530-1. PMID 11804478 DOI: 10.1021/Ja0172215  0.59
2001 Siu T, Li W, Yudin AK. Parallel electrosynthesis of 1,2-diamines. Journal of Combinatorial Chemistry. 3: 554-8. PMID 11703151 DOI: 10.1021/Cc0100159  0.567
2001 Yudin AK, Siu T. Combinatorial electrochemistry. Current Opinion in Chemical Biology. 5: 269-72. PMID 11479118 DOI: 10.1016/S1367-5931(00)00202-7  0.516
2001 Yudin AK, Chiang JP, Adolfsson H, Copéret C. Olefin epoxidation with bis(trimethylsilyl) peroxide catalyzed by inorganic oxorhenium derivatives. Controlled release of hydrogen peroxide. The Journal of Organic Chemistry. 66: 4713-8. PMID 11421798 DOI: 10.1021/Jo010369M  0.772
2000 Adolfsson H, Copéret C, Chiang JP, Yudin AK. Efficient epoxidation of alkenes with aqueous hydrogen peroxide catalyzed by methyltrioxorhenium and 3-cyanopyridine. The Journal of Organic Chemistry. 65: 8651-8. PMID 11112586 DOI: 10.1021/Jo005623+  0.806
2000 Chen Y, Yekta S, Martyn LJ, Zheng J, Yudin AK. Regioselective substitution of fluorine in F(8)BINOL as a versatile route to new ligands with axial chirality Organic Letters. 2: 3433-6. PMID 11082001 DOI: 10.1021/Ol006428K  0.392
2000 Siu T, Li W, Yudin AK. Parallel electrosynthesis of alpha-alkoxycarbamates, alpha-alkoxyamides, and alpha-alkoxysulfonamides using the spatially addressable electrolysis platform (SAEP) Journal of Combinatorial Chemistry. 2: 545-9. PMID 11029180 DOI: 10.1021/Cc000035V  0.497
2000 Siu T, Yekta S, Yudin AK. New approach to rapid generation and screening of diverse catalytic materials on electrode surfaces Journal of the American Chemical Society. 122: 11787-11790. DOI: 10.1021/Ja002334U  0.548
2000 James L, Martyn P, Pandiaraju S, Yudin AK. Catalytic applications of F8BINOL: Asymmetric oxidation of sulfides to sulfoxides Journal of Organometallic Chemistry. 603: 98-104. DOI: 10.1016/S0022-328X(00)00172-8  0.371
2000 Siu T, Li W, Yudin AK. Parallel electrosynthesis of α-alkoxycarbamates, α-alkoxyamides, and α-alkoxysulfonamides using the Spatially Addressable Electrolysis Platform (SAEP) Journal of Combinatorial Chemistry. 2: 545-549.  0.444
1998 Copéret C, Adolfsson H, Khuong TAV, Yudin AK, Sharpless KB. A simple and efficient method for the preparation of pyridine N-oxides Journal of Organic Chemistry. 63: 1740-1741. DOI: 10.1021/Jo9723467  0.597
1998 Copéret C, Adolfsson H, Chiang JP, Yudin AK, Sharpless KB. A simple and efficient method for the preparation of pyridine-N-oxides II Tetrahedron Letters. 39: 761-764. DOI: 10.1016/S0040-4039(97)10619-0  0.778
1997 Prakash GK, Yudin AK. Perfluoroalkylation with Organosilicon Reagents. Chemical Reviews. 97: 757-786. PMID 11848888 DOI: 10.1021/Cr9408991  0.542
1997 Petasis NA, Yudin AK, Zavialov IA, Prakash GKS, Olah GA. Facile preparation of fluorine-containing alkenes, amides and alcohols via the electrophilic fluorination of alkenyl boronic acids and trifluoroborates Synlett. 606-608. DOI: 10.1055/S-1997-3228  0.331
1997 Petasis N, Yudin A, Zavialov I, Prakash G, Olah G. Facile Preparation of Fluorine-containing Alkenes, Amides and Alcohols via the Electrophilic Fluorination of Alkenyl Boronic Acids and Trifluoroborates Synlett. 1997: 606-608. DOI: 10.1055/s-1997-3228  0.407
1997 Yudin AK, Sharpless KB. Bis(trimethylsilyl) peroxide extends the range of oxorhenium catalysts for olefin epoxidation [2] Journal of the American Chemical Society. 119: 11536-11537. DOI: 10.1021/Ja973043X  0.491
1997 Yudin AK, Prakash GKS, Deffieux D, Bradley M, Bau R, Olah GA. Preparation of and fluoroalkylation with (chlorodifluoromethyl)trimethylsilane, difluorobis(trimethylsilyl)methane, and 1,1,2,2-tetrafluoro-1,2-bis(trimethylsilyl)ethane Journal of the American Chemical Society. 119: 1572-1581. DOI: 10.1021/Ja962990N  0.48
1996 Prakash GKS, Yudin AK, Deffieux D, Olah GA. Facile Preparation of (Trifluoromethyl)tributyltin and Transtrifluoromethylation of Disilyl Sulfides to the Corresponding Trifluoromethylsilanes1 Synlett. 1996: 151-153. DOI: 10.1055/S-1996-5355  0.476
1994 Surya Prakash GK, Deffieux D, Yudin AK, Olah GA. Convenient and Safe Electrochemical Synthesis of (Trifluoromethyl)trimethylsilane1a Synlett. 1994: 1057-1058. DOI: 10.1055/S-1994-34986  0.395
Show low-probability matches.