Year |
Citation |
Score |
2015 |
Parker EN, Song J, Kishore Kumar GD, Odutola SO, Chavarria GE, Charlton-Sevcik AK, Strecker TE, Barnes AL, Sudhan DR, Wittenborn TR, Siemann DW, Horsman MR, Chaplin DJ, Trawick ML, Pinney KG. Synthesis and biochemical evaluation of benzoylbenzophenone thiosemicarbazone analogues as potent and selective inhibitors of cathepsin L. Bioorganic & Medicinal Chemistry. PMID 26462052 DOI: 10.1016/J.Bmc.2015.09.036 |
0.833 |
|
2013 |
Song J, Jones LM, Chavarria GE, Charlton-Sevcik AK, Jantz A, Johansen A, Bayeh L, Soeung V, Snyder LK, Lade SD, Chaplin DJ, Trawick ML, Pinney KG. Small-molecule inhibitors of cathepsin L incorporating functionalized ring-fused molecular frameworks. Bioorganic & Medicinal Chemistry Letters. 23: 2801-7. PMID 23540644 DOI: 10.1016/J.Bmcl.2012.12.025 |
0.815 |
|
2012 |
Song J, Jones LM, Kumar GD, Conner ES, Bayeh L, Chavarria GE, Charlton-Sevcik AK, Chen SE, Chaplin DJ, Trawick ML, Pinney KG. Synthesis and biochemical evaluation of thiochromanone thiosemicarbazone analogues as inhibitors of cathepsin L. Acs Medicinal Chemistry Letters. 3: 450-3. PMID 24900494 DOI: 10.1021/Ml200299G |
0.732 |
|
2012 |
Chavarria GE, Horsman MR, Arispe WM, Kumar GD, Chen SE, Strecker TE, Parker EN, Chaplin DJ, Pinney KG, Trawick ML. Initial evaluation of the antitumour activity of KGP94, a functionalized benzophenone thiosemicarbazone inhibitor of cathepsin L. European Journal of Medicinal Chemistry. 58: 568-72. PMID 23168380 DOI: 10.1016/J.Ejmech.2012.10.039 |
0.713 |
|
2011 |
Trawick ML, Pinney KG, Chaplin DJ, Horsman MR, Chavarria GE, Arispe WM, Kumar GDK. Abstract 1416: Development and initial evaluation of the antitumor activity of a functionalized benzophenone thiosemicarbazone inhibitor of cathepsin L Cancer Research. 71: 1416-1416. DOI: 10.1158/1538-7445.Am2011-1416 |
0.784 |
|
2010 |
Kumar GD, Chavarria GE, Charlton-Sevcik AK, Yoo GK, Song J, Strecker TE, Siim BG, Chaplin DJ, Trawick ML, Pinney KG. Functionalized benzophenone, thiophene, pyridine, and fluorene thiosemicarbazone derivatives as inhibitors of cathepsin L. Bioorganic & Medicinal Chemistry Letters. 20: 6610-5. PMID 20933415 DOI: 10.1016/J.Bmcl.2010.09.026 |
0.831 |
|
2010 |
Kishore Kumar GD, Chavarria GE, Charlton-Sevcik AK, Arispe WM, Macdonough MT, Strecker TE, Chen SE, Siim BG, Chaplin DJ, Trawick ML, Pinney KG. Design, synthesis, and biological evaluation of potent thiosemicarbazone based cathepsin L inhibitors. Bioorganic & Medicinal Chemistry Letters. 20: 1415-9. PMID 20089402 DOI: 10.1016/J.Bmcl.2009.12.090 |
0.739 |
|
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