Year |
Citation |
Score |
2020 |
Liu L, Kong C, Fumagalli M, Savková K, Xu Y, Huszár S, Sammartino JC, Fan D, Chiarelli LR, Mikušová K, Sun Z, Qiao C. Design, synthesis and evaluation of covalent inhibitors of DprE1 as antitubercular agents. European Journal of Medicinal Chemistry. 208: 112773. PMID 32898793 DOI: 10.1016/j.ejmech.2020.112773 |
0.333 |
|
2014 |
Xu Z, Yin W, Martinelli LK, Evans J, Chen J, Yu Y, Wilson DJ, Mizrahi V, Qiao C, Aldrich CC. Reaction intermediate analogues as bisubstrate inhibitors of pantothenate synthetase. Bioorganic & Medicinal Chemistry. 22: 1726-35. PMID 24507827 DOI: 10.1016/J.Bmc.2014.01.017 |
0.301 |
|
2007 |
Qiao C, Gupte A, Boshoff HI, Wilson DJ, Bennett EM, Somu RV, Barry CE, Aldrich CC. 5'-O-[(N-acyl)sulfamoyl]adenosines as antitubercular agents that inhibit MbtA: an adenylation enzyme required for siderophore biosynthesis of the mycobactins. Journal of Medicinal Chemistry. 50: 6080-94. PMID 17967002 DOI: 10.1021/Jm070905O |
0.371 |
|
2006 |
Qiao C, Ling KQ, Shepard EM, Dooley DM, Sayre LM. Mechanism-based cofactor derivatization of a copper amine oxidase by a branched primary amine recruits the oxidase activity of the enzyme to turn inactivator into substrate. Journal of the American Chemical Society. 128: 6206-19. PMID 16669691 DOI: 10.1021/Ja058838F |
0.581 |
|
2004 |
Lamplot Z, Sebela M, Malon M, Lenobel R, Lemr K, Havlis J, Pec P, Qiao C, Sayre LM. 1,5-diamino-2-pentyne is both a substrate and inactivator of plant copper amine oxidases. European Journal of Biochemistry / Febs. 271: 4696-708. PMID 15606757 DOI: 10.1111/J.1432-1033.2004.04434.X |
0.574 |
|
2004 |
Qiao C, Jeon HB, Sayre LM. Selective inhibition of bovine plasma amine oxidase by homopropargylamine, a new inactivator motif. Journal of the American Chemical Society. 126: 8038-45. PMID 15212554 DOI: 10.1021/Ja049568O |
0.601 |
|
2003 |
Jeon HB, Lee Y, Qiao C, Huang H, Sayre LM. Inhibition of bovine plasma amine oxidase by 1,4-diamino-2-butenes and -2-butynes. Bioorganic & Medicinal Chemistry. 11: 4631-41. PMID 14527560 DOI: 10.1016/S0968-0896(03)00521-2 |
0.596 |
|
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