Year |
Citation |
Score |
2022 |
Bi C, Chadwick J, Davies ML, DelMonte AJ, Geng P, Glace AW, Green RA, Gurak JA, Haley MW, He BL, Inankur B, Jamison CR, Joe CL, Kolotuchin S, Lin D, ... ... Stevens JM, et al. Coupling-Condensation Strategy for the Convergent Synthesis of an Imidazole-Fused 2-Aminoquinoline NLRP3 Agonist. The Journal of Organic Chemistry. PMID 36516991 DOI: 10.1021/acs.joc.2c02395 |
0.617 |
|
2019 |
Fraunhoffer KJ, DelMonte AJ, Beutner GL, Bultman MS, Camacho K, Cohen B, Dixon DD, Fan Y, Fanfair D, Freitag AJ, Glace AW, Gonzalez-Bobes F, Gujjar M, Haley MW, Hickey MR, ... ... Stevens JM, et al. Rapid Development of a Commercial Process for Linrodostat, an Indoleamine 2,3-Dioxygenase (IDO) Inhibitor Organic Process Research & Development. 23: 2482-2498. DOI: 10.1021/Acs.Oprd.9B00359 |
0.599 |
|
2019 |
Mennen SM, Alhambra C, Allen CL, Barberis M, Berritt S, Brandt TA, Campbell AD, Castañón J, Cherney AH, Christensen M, Damon DB, Eugenio de Diego J, García-Cerrada S, García-Losada P, Haro R, ... ... Stevens JM, et al. The Evolution of High-Throughput Experimentation in Pharmaceutical Development and Perspectives on the Future Organic Process Research & Development. 23: 1213-1242. DOI: 10.1021/Acs.Oprd.9B00140 |
0.345 |
|
2019 |
Beutner GL, Cohen BM, DelMonte AJ, Dixon DD, Fraunhoffer KJ, Glace AW, Lo E, Stevens JM, Vanyo D, Wilbert C. Revisiting the Cleavage of Evans Oxazolidinones with LiOH/H2O2 Organic Process Research & Development. 23: 1378-1385. DOI: 10.1021/Acs.Oprd.9B00124 |
0.324 |
|
2019 |
Gonzalez FL, Wisniewski SR, Katipally K, Stevens JM, Rosso V, Mack B, Razler TM. Systematic Optimization of a Robust Telescoped Process for a BTK Inhibitor with Atropisomer Control by High-Throughput Experimentation, Design of Experiments, and Linear Regression Organic Process Research & Development. 23: 1143-1151. DOI: 10.1021/Acs.Oprd.8B00398 |
0.379 |
|
2018 |
Stevens JM, Parra-Rivera AC, Dixon DD, Beutner GL, DelMonte AJ, Frantz DE, Janey JM, Paulson J, Talley MR. Direct Lewis Acid-Catalyzed Conversion of Enantioenriched N-Acyl Oxazolidinones to Chiral Esters, Amides, and Acids. The Journal of Organic Chemistry. PMID 30412670 DOI: 10.1021/Acs.Joc.8B02451 |
0.359 |
|
2018 |
Wisniewski SR, Stevens JM, Yu M, Fraunhoffer KJ, Romero EO, Savage SA. Utilizing Native Directing Groups: Synthesis of a Selective IKur Inhibitor, BMS-919373, via a Regioselective C-H Arylation. The Journal of Organic Chemistry. PMID 30395712 DOI: 10.1021/Acs.Joc.8B02254 |
0.378 |
|
2018 |
Beutner GL, Young IS, Davies ML, Hickey MR, Park H, Stevens JM, Ye Q. TCFH-NMI: Direct Access to N-Acyl Imidazoliums for Challenging Amide Bond Formations. Organic Letters. PMID 29956545 DOI: 10.1021/Acs.Orglett.8B01591 |
0.311 |
|
2018 |
Beutner G, Carrasquillo R, Geng P, Hsiao Y, Huang EC, Janey J, Katipally K, Kolotuchin S, La Porte T, Lee A, Lobben P, Lora-Gonzalez F, Mack B, Mudryk B, Qiu Y, ... ... Stevens J, et al. Adventures in Atropisomerism: Total Synthesis of a Complex Active Pharmaceutical Ingredient with Two Chirality Axes. Organic Letters. PMID 29909639 DOI: 10.1021/Acs.Orglett.8B01218 |
0.388 |
|
2018 |
Coombs JR, Green RA, Roberts F, Simmons EM, Stevens JM, Wisniewski SR. Advances in Base-Metal Catalysis: Development of a Screening Platform for Nickel-Catalyzed Borylations of Aryl (Pseudo)halides with B2(OH)4 Organometallics. 38: 157-166. DOI: 10.1021/Acs.Organomet.8B00307 |
0.362 |
|
2017 |
deGruyter JN, Malins LR, Wimmer L, Clay KJ, Lopez-Ogalla J, Qin T, Cornella J, Liu Z, Che G, Bao D, Stevens JM, Qiao JX, Allen MP, Poss MA, Baran PS. CITU: A Peptide and Decarboxylative Coupling Reagent. Organic Letters. PMID 29115835 DOI: 10.1021/Acs.Orglett.7B03121 |
0.375 |
|
2013 |
Stevens JM, MacMillan DWC. Enantioselective α-alkenylation of aldehydes with boronic acids via the synergistic combination of copper(II) and amine catalysis Journal of the American Chemical Society. 135: 11756-11759. PMID 23889497 DOI: 10.1021/Ja406356C |
0.375 |
|
2009 |
Crimmins MT, Stevens JM, Schaaf GM. Total synthesis of irciniastatin A (Psymberin). Organic Letters. 11: 3990-3. PMID 19670853 DOI: 10.1021/Ol901655E |
0.611 |
|
2009 |
Voss ME, Ralph JM, Xie D, Manning DD, Chen X, Frank AJ, Leyhane AJ, Liu L, Stevens JM, Budde C, Surman MD, Friedrich T, Peace D, Scott IL, Wolf M, et al. Synthesis and SAR of vinca alkaloid analogues. Bioorganic & Medicinal Chemistry Letters. 19: 1245-9. PMID 19147348 DOI: 10.1016/J.Bmcl.2008.12.077 |
0.399 |
|
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