Year |
Citation |
Score |
2022 |
Basilaia M, Chen MH, Secka J, Gustafson JL. Atropisomerism in the Pharmaceutically Relevant Realm. Accounts of Chemical Research. PMID 36153960 DOI: 10.1021/acs.accounts.2c00500 |
0.343 |
|
2021 |
Cardenas MM, Saputra MA, Gordon DA, Sanchez AN, Yamamoto N, Gustafson JL. Catalytic atroposelective dynamic kinetic resolutions and kinetic resolutions towards 3-arylquinolines SAr. Chemical Communications (Cambridge, England). PMID 34515276 DOI: 10.1039/d1cc04335h |
0.318 |
|
2020 |
Dinh AN, Maddox SM, Vaidya SD, Saputra MA, Nalbandian CJ, Gustafson JL. Catalyst-Controlled Regioselective Chlorination of Phenols and Anilines through a Lewis Basic Selenoether Catalyst. The Journal of Organic Chemistry. PMID 33044067 DOI: 10.1021/acs.joc.0c01917 |
0.323 |
|
2020 |
Ortiz MA, Michaels H, Molina B, Toenjes S, Davis J, Diletta Marconi G, Hecht D, Gustafson JL, Javier Piedrafita F, Nefzi A. Discovery of cyclic guanidine-linked sulfonamides as inhibitors of LMTK3 kinase. Bioorganic & Medicinal Chemistry Letters. 127108. PMID 32192797 DOI: 10.1016/J.Bmcl.2020.127108 |
0.327 |
|
2020 |
Vaidya SD, Toenjes ST, Yamamoto N, Maddox SM, Gustafson JL. Catalytic Atroposelective Synthesis of N-Aryl Quinoid Compounds. Journal of the American Chemical Society. PMID 31944689 DOI: 10.1021/Jacs.9B12994 |
0.448 |
|
2020 |
Dinh A, Gustafson JL. A Catalytic Cycle of Discovery: Asymmetric Catalysis Gives Rise to New Chiral Catalyst Scaffolds Chem. 6: 810-812. DOI: 10.1016/J.Chempr.2020.03.020 |
0.439 |
|
2019 |
Toenjes ST, Garcia V, Maddox SM, Dawson GA, Ortiz MA, Piedrafita FJ, Gustafson JL. Leveraging atropisomerism to obtain a selective inhibitor of RET kinase with secondary activities towards EGFR mutants. Acs Chemical Biology. PMID 31424197 DOI: 10.1021/Acschembio.9B00407 |
0.409 |
|
2019 |
Dinh AN, Nguyen AD, Aceves EM, Albright ST, Cedano MR, Smith DK, Gustafson JL. Photocatalytic Oxidative C–H Thiolation: Synthesis of Benzothiazoles and Sulfenylated Indoles Synlett. 30: 1648-1655. DOI: 10.1055/S-0039-1690107 |
0.309 |
|
2018 |
Dinh AN, Noorbehesht RR, Toenjes ST, Jackson AC, Saputra MA, Maddox SM, Gustafson JL. Towards a Catalytic Atroposelective Synthesis of Diaryl Ethers via C()-H Alkylation Using Nitroalkanes. Synlett : Accounts and Rapid Communications in Synthetic Organic Chemistry. 29: 2155-2160. PMID 31178629 DOI: 10.1055/S-0037-1609581 |
0.363 |
|
2018 |
Maddox SM, Dawson GA, Rochester NC, Ayonon AB, Moore CE, Rheingold AL, Gustafson JL. Enantioselective Synthesis of Biaryl Atropisomers via the Addition of Thiophenols into Aryl-Naphthoquinones. Acs Catalysis. 8: 5443-5447. PMID 30455999 DOI: 10.1021/Acscatal.8B00906 |
0.411 |
|
2018 |
Nalbandian CJ, Brown ZE, Alvarez E, Gustafson JL. Lewis Base/Bronsted Acid Dual-Catalytic C-H Sulfenylation of Aromatics. Organic Letters. PMID 29762039 DOI: 10.1021/Acs.Orglett.8B01066 |
0.359 |
|
2018 |
Cardenas MM, Toenjes ST, Nalbandian CJ, Gustafson JL. Enantioselective Synthesis of Pyrrolopyrimidine Scaffolds through Cation-Directed Nucleophilic Aromatic Substitution. Organic Letters. PMID 29561161 DOI: 10.1021/Acs.Orglett.8B00579 |
0.466 |
|
2018 |
Toenjes ST, Gustafson JL. Atropisomerism in medicinal chemistry: challenges and opportunities. Future Medicinal Chemistry. PMID 29380622 DOI: 10.4155/Fmc-2017-0152 |
0.417 |
|
2017 |
Ottis P, Toure M, Cromm PM, Ko E, Gustafson JL, Crews CM. Assessing Different E3 Ligases for Small Molecule-induced Protein Ubiquitination and Degradation. Acs Chemical Biology. PMID 28767222 DOI: 10.1021/Acschembio.7B00485 |
0.358 |
|
2017 |
Nalbandian CJ, Miller EM, Toenjes ST, Gustafson JL. A conjugate Lewis base-Brønsted acid catalyst for the sulfenylation of nitrogen containing heterocycles under mild conditions. Chemical Communications (Cambridge, England). PMID 28084476 DOI: 10.1039/C6Cc09998J |
0.374 |
|
2017 |
Ayonon A, Nalbandian C, Guillemard L, Gustafson J. Benzylic bromination catalyzed by triphenylphosphine selenide via Lewis basic activation Tetrahedron Letters. 58: 2940-2943. DOI: 10.1016/J.Tetlet.2017.06.042 |
0.436 |
|
2016 |
Maddox SM, Dinh AN, Armenta F, Um J, Gustafson JL. The Catalyst-Controlled Regiodivergent Chlorination of Phenols. Organic Letters. PMID 27754679 DOI: 10.1021/Acs.Orglett.6B02650 |
0.414 |
|
2016 |
Maddox S, Hecht D, Gustafson JL. Enhancing the selectivity of kinase inhibitors in oncology: a chemical biology perspective. Future Medicinal Chemistry. PMID 26898835 DOI: 10.4155/Fmc.15.193 |
0.324 |
|
2016 |
Maligal-Ganesh RV, Xiao C, Goh TW, Wang LL, Gustafson J, Pei Y, Qi Z, Johnson DD, Zhang S, Tao F, Huang W. A Ship-in-a-Bottle Strategy to Synthesize Encapsulated Intermetallic Nanoparticle Catalysts: Exemplified for Furfural Hydrogenation Acs Catalysis. 6: 1754-1763. DOI: 10.1021/Acscatal.5B02281 |
0.338 |
|
2016 |
Kelly MJB, Fallot LB, Gustafson JL, Bergdahl BM. Water Mediated Wittig Reactions of Aldehydes in the Teaching Laboratory: Using Sodium Bicarbonate for the in Situ Formation of Stabilized Ylides Journal of Chemical Education. 93: 1631-1636. DOI: 10.1021/Acs.Jchemed.6B00206 |
0.321 |
|
2015 |
Smith DE, Marquez I, Lokensgard ME, Rheingold AL, Hecht DA, Gustafson JL. Exploiting Atropisomerism to Increase the Target Selectivity of Kinase Inhibitors. Angewandte Chemie (International Ed. in English). PMID 26276764 DOI: 10.1002/Anie.201506085 |
0.398 |
|
2015 |
Bondeson DP, Mares A, Smith IE, Ko E, Campos S, Miah AH, Mulholland KE, Routly N, Buckley DL, Gustafson JL, Zinn N, Grandi P, Shimamura S, Bergamini G, Faelth-Savitski M, et al. Catalytic in vivo protein knockdown by small-molecule PROTACs. Nature Chemical Biology. 11: 611-7. PMID 26075522 DOI: 10.1038/Nchembio.1858 |
0.401 |
|
2015 |
Buckley DL, Raina K, Darricarrere N, Hines J, Gustafson JL, Smith IE, Miah AH, Harling JD, Crews CM. HaloPROTACS: Use of Small Molecule PROTACs to Induce Degradation of HaloTag Fusion Proteins. Acs Chemical Biology. PMID 26070106 DOI: 10.1021/Acschembio.5B00442 |
0.399 |
|
2015 |
Maddox SM, Nalbandian CJ, Smith DE, Gustafson JL. A practical Lewis base catalyzed electrophilic chlorination of arenes and heterocycles. Organic Letters. 17: 1042-5. PMID 25671756 DOI: 10.1021/Acs.Orglett.5B00186 |
0.4 |
|
2015 |
Nalbandian CJ, Hecht DE, Gustafson JL. The Preorganization of Atropisomers to Increase Target Selectivity Synlett. DOI: 10.1055/S-0035-1561314 |
0.434 |
|
2015 |
Luca OR, Gustafson JL, Maddox SM, Fenwick AQ, Smith DC. Catalysis by electrons and holes: Formal potential scales and preparative organic electrochemistry Organic Chemistry Frontiers. 2: 823-848. DOI: 10.1039/C5Qo00075K |
0.318 |
|
2012 |
Buckley DL, Gustafson JL, Van Molle I, Roth AG, Tae HS, Gareiss PC, Jorgensen WL, Ciulli A, Crews CM. Small-molecule inhibitors of the interaction between the E3 ligase VHL and HIF1α. Angewandte Chemie (International Ed. in English). 51: 11463-7. PMID 23065727 DOI: 10.1002/Anie.201206231 |
0.374 |
|
2012 |
Tae HS, Sundberg TB, Neklesa TK, Noblin DJ, Gustafson JL, Roth AG, Raina K, Crews CM. Identification of hydrophobic tags for the degradation of stabilized proteins. Chembiochem : a European Journal of Chemical Biology. 13: 538-41. PMID 22271667 DOI: 10.1002/Cbic.201100793 |
0.323 |
|
2011 |
Gustafson JL, Lim D, Barrett KT, Miller SJ. Synthesis of atropisomerically defined, highly substituted biaryl scaffolds through catalytic enantioselective bromination and regioselective cross-coupling. Angewandte Chemie (International Ed. in English). 50: 5125-9. PMID 21520374 DOI: 10.1002/Anie.201101147 |
0.633 |
|
2010 |
Gustafson JL, Lim D, Miller SJ. Dynamic kinetic resolution of biaryl atropisomers via peptide-catalyzed asymmetric bromination. Science (New York, N.Y.). 328: 1251-5. PMID 20522769 DOI: 10.1126/Science.1188403 |
0.641 |
|
2010 |
Gustafson JL, Sigman MS, Miller SJ. Linear free-energy relationship analysis of a catalytic desymmetrization reaction of a diarylmethane-bis(phenol). Organic Letters. 12: 2794-7. PMID 20486656 DOI: 10.1021/Ol100927M |
0.463 |
|
2008 |
Lewis CA, Gustafson JL, Chiu A, Balsells J, Pollard D, Murry J, Reamer RA, Hansen KB, Miller SJ. A case of remote asymmetric induction in the peptide-catalyzed desymmetrization of a bis(phenol). Journal of the American Chemical Society. 130: 16358-65. PMID 19006301 DOI: 10.1021/Ja807120Z |
0.631 |
|
2007 |
Grotjahn DB, Larsen CR, Gustafson JL, Nair R, Sharma A. Extensive isomerization of alkenes using a bifunctional catalyst: an alkene zipper. Journal of the American Chemical Society. 129: 9592-3. PMID 17636924 DOI: 10.1021/Ja073457I |
0.397 |
|
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