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Jetze J. Tepe - Publications

Affiliations: 
Chemistry Michigan State University, East Lansing, MI 
Area:
Organic Chemistry, Biochemistry, Molecular Biology
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63 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2022 Mehedi MSA, George DE, Tepe JJ. Sc(OTf)-Mediated One-Pot Synthesis of 3,4-Disubstituted 1-Pyrazoles and 3,5-Disubstituted Pyridines from Hydrazine or Ammonia with Epoxides. The Journal of Organic Chemistry. 87: 16820-16828. PMID 36475626 DOI: 10.1021/acs.joc.2c02544  0.818
2022 Savelson E, Tepe JJ. One-Pot Friedel-Crafts/Robinson-Gabriel Synthesis of the Indole-Oxazole Scaffold and Its Application to the Synthesis of Breitfussins C, G, and H. The Journal of Organic Chemistry. PMID 35235750 DOI: 10.1021/acs.joc.2c00033  0.303
2020 Keel KL, Tepe JJ. The preparation of (4H)-imidazol-4-ones and their application in the total synthesis of natural products Organic Chemistry Frontiers. 7: 3284-3311. PMID 33796321 DOI: 10.1039/D0Qo00764A  0.398
2020 Mehedi MSA, Tepe JJ. Sc(OTf)-Mediated One-Pot Synthesis of 2,3-Disubstituted Quinolines from Anilines and Epoxides. The Journal of Organic Chemistry. 85: 6741-6746. PMID 32319294 DOI: 10.1021/Acs.Joc.0C00803  0.813
2020 Mehedi SA, Tepe JJ. Recent Advances in the Synthesis of Imidazolines (2009–2020) Advanced Synthesis & Catalysis. DOI: 10.1002/Adsc.202000709  0.37
2019 Mehedi MSA, Tepe JJ. Diastereoselective One-Pot Synthesis of Oxazolines Using Sulfur Ylides and Acyl Imines. The Journal of Organic Chemistry. PMID 31117573 DOI: 10.1021/Acs.Joc.9B00883  0.802
2019 Giletto MB, Osmulski PA, Jones CL, Gaczynska ME, Tepe JJ. Pipecolic esters as minimized templates for proteasome inhibition. Organic & Biomolecular Chemistry. PMID 30778435 DOI: 10.1039/C9Ob00122K  0.362
2018 Gao S, Bethel TK, Kakeshpour T, Hubbell GE, Jackson JE, Tepe JJ. Substrate Controlled Regioselective Bromination of Acylated Pyrroles Using Tetrabutylammonium Tribromide (TBABr3). The Journal of Organic Chemistry. PMID 29969032 DOI: 10.1021/Acs.Joc.8B01251  0.322
2017 Osmulski PA, Cropper J, Giletto M, Jones C, Killer C, Jiang S, Tepe J, Chatterjee B, Huang T, Gaczynska ME. Anticancer applications of allosteric inhibitors of proteasome. Journal of Clinical Oncology. 35: e23066-e23066. DOI: 10.1200/Jco.2017.35.15_Suppl.E23066  0.305
2016 McDaniel TJ, Lansdell TA, Dissanayake AA, Azevedo LM, Claes J, Odom AL, Tepe JJ. Substituted quinolines as noncovalent proteasome inhibitors. Bioorganic & Medicinal Chemistry. PMID 27112450 DOI: 10.1016/J.Bmc.2016.04.005  0.4
2016 Osmulski PA, Karpowicz P, Jankowska E, Giletto M, Lansdell T, Tepe J, Huang TH, Gaczynska M. From Single Molecules to Single Cells: Biophysics of Interactions between Small Regulators and Proteasome Biophysical Journal. 110: 218a. DOI: 10.1016/J.Bpj.2015.11.1207  0.327
2015 Beck P, Lansdell TA, Hewlett NM, Tepe JJ, Groll M. Indolo-phakellins as β5-specific noncovalent proteasome inhibitors. Angewandte Chemie (International Ed. in English). 54: 2830-3. PMID 25581903 DOI: 10.1002/Anie.201410168  0.765
2015 Kuszpit MR, Giletto MB, Jones CL, Bethel TK, Tepe JJ. Hydroxyamination of olefins using Br-N-(CO2Me)2. The Journal of Organic Chemistry. 80: 1440-5. PMID 25574949 DOI: 10.1021/Jo502369D  0.77
2015 Beck P, Lansdell TA, Hewlett NM, Tepe JJ, Groll M. Indolo-Phakelline als β5-spezifische nichtkovalente Proteasom-Inhibitoren Angewandte Chemie. 127: 2872-2875. DOI: 10.1002/Ange.201410168  0.735
2013 Azevedo LM, Lansdell TA, Ludwig JR, Mosey RA, Woloch DK, Cogan DP, Patten GP, Kuszpit MR, Fisk JS, Tepe JJ. Inhibition of the human proteasome by imidazoline scaffolds. Journal of Medicinal Chemistry. 56: 5974-8. PMID 23789888 DOI: 10.1021/Jm400235R  0.73
2012 Lansdell TA, Hewlett NM, Skoumbourdis AP, Fodor MD, Seiple IB, Su S, Baran PS, Feldman KS, Tepe JJ. Palau'amine and related oroidin alkaloids dibromophakellin and dibromophakellstatin inhibit the human 20S proteasome. Journal of Natural Products. 75: 980-5. PMID 22591513 DOI: 10.1021/Np300231F  0.774
2012 Saleem RS, Lansdell TA, Tepe JJ. Synthesis and evaluation of debromohymenialdisine-derived Chk2 inhibitors. Bioorganic & Medicinal Chemistry. 20: 1475-81. PMID 22285028 DOI: 10.1016/J.Bmc.2011.12.054  0.791
2012 Nguyen TN, Saleem RS, Luderer MJ, Hovde S, Henry RW, Tepe JJ. Radioprotection by hymenialdisine-derived checkpoint kinase 2 inhibitors. Acs Chemical Biology. 7: 172-84. PMID 22004065 DOI: 10.1021/Cb200320C  0.769
2012 Nguyen TN, Tepe JJ. Current inhibitors of checkpoint kinase 2. Current Medicinal Chemistry. 18: 4368-74. PMID 21861812 DOI: 10.2174/092986711797200390  0.301
2012 Hovde S, Lansdell TA, Azevedo L, Tepe JJ, Henry RW. Abstract 2777: Suppression of multiple myeloma via non-canonical inhibition of NF-κB Cancer Research. 72: 2777-2777. DOI: 10.1158/1538-7445.Am2012-2777  0.332
2012 Hewlett NM, Tepe JJ. Erratum: Total synthesis of the natural product (±)-dibromophakellin and analogues (Organic Letters (2011) 13 (4552)) Organic Letters. 14. DOI: 10.1021/Ol300329H  0.769
2011 Qu K, Fisk JS, Tepe JJ. Azomethine ylide mediated inversion of configuration of quaternary imidazoline carbon: converting trans- to its cis- imidazolines. Tetrahedron Letters. 52: 4840-4842. PMID 21857756 DOI: 10.1016/J.Tetlet.2011.07.022  0.784
2011 Hewlett NM, Tepe JJ. Total synthesis of the natural product (±)-dibromophakellin and analogues. Organic Letters. 13: 4550-3. PMID 21797255 DOI: 10.1021/Ol201741R  0.786
2011 Kuszpit MR, Wulff WD, Tepe JJ. One-pot synthesis of 2-imidazolines via the ring expansion of imidoyl chlorides with aziridines. The Journal of Organic Chemistry. 76: 2913-9. PMID 21401025 DOI: 10.1021/Jo200101Q  0.804
2010 Saleem RS, Tepe JJ. Synthesis of 1,2,4-triazolines and triazoles utilizing oxazolones. The Journal of Organic Chemistry. 75: 4330-2. PMID 20481587 DOI: 10.1021/Jo100716M  0.804
2010 Tepe J, Saleem R. Heterocyclic Interconversion of Oxazolones into Triazolines and Triazoles Synfacts. 2010: 0997-0997. DOI: 10.1055/s-0030-1258006  0.807
2010 Hewlett NM, Hupp CD, Tepe JJ. ChemInform Abstract: Reactivity of Oxazol-5-(4H)-ones and Their Application Toward Natural Product Synthesis. Cheminform. 41. DOI: 10.1002/chin.201003123  0.786
2010 TEPE JJ, MADALENGOITIA JS, SLUNT KM, WERBOVETZ KW, SPOORS PG, MACDONALD TL. ChemInform Abstract: Inhibition of DNA Topoisomerase II by Azaelliptitoxins Functionalized in the Variable Substituent Domain. Cheminform. 27: no-no. DOI: 10.1002/chin.199637203  0.671
2009 Nguyen TN, Tepe JJ. Preparation of hymenialdisine, analogues and their evaluation as kinase inhibitors. Current Medicinal Chemistry. 16: 3122-43. PMID 19689287 DOI: 10.2174/092986709788803015  0.362
2009 Hupp CD, Tepe JJ. 1-Ethyl-3-(3-dimethylaminopropyl)carbodiimide hydrochloride-mediated oxazole rearrangement: gaining access to a unique marine alkaloid scaffold. The Journal of Organic Chemistry. 74: 3406-13. PMID 19331366 DOI: 10.1021/Jo900264P  0.798
2009 Kahlon DK, Lansdell TA, Fisk JS, Tepe JJ. Structural-activity relationship study of highly-functionalized imidazolines as potent inhibitors of nuclear transcription factor-kappaB mediated IL-6 production. Bioorganic & Medicinal Chemistry. 17: 3093-103. PMID 19328000 DOI: 10.1016/J.Bmc.2009.03.002  0.77
2009 Kahlon DK, Lansdell TA, Fisk JS, Hupp CD, Friebe TL, Hovde S, Jones AD, Dyer RD, Henry RW, Tepe JJ. Nuclear factor-κB mediated inhibition of cytokine production by imidazoline scaffolds Journal of Medicinal Chemistry. 52: 1302-1309. PMID 19220017 DOI: 10.1021/Jm8013162  0.75
2009 Hewlett NM, Hupp CD, Tepe JJ. Reactivity of oxazol-5-(4H)-ones and their application toward natural product synthesis Synthesis. 2825-2839. DOI: 10.1055/S-0029-1216924  0.809
2009 Mosey RA, Tepe JJ. New synthetic route to access (±) salinosporamide A via an oxazolone-mediated ene-type reaction Tetrahedron Letters. 50: 295-297. DOI: 10.1016/J.Tetlet.2008.10.154  0.817
2009 Mosey RA, Fisk JS, Tepe JJ. ChemInform Abstract: Stereoselective Syntheses of Quaternary Substituted α-Amino Acids Using Oxazol-5-(4H)-ones Cheminform. 40. DOI: 10.1002/chin.200922229  0.778
2009 Mosey RA, Tepe JJ. ChemInform Abstract: New Synthetic Route to Access (.+-.) Salinosporamide A via an Oxazolone-Mediated Ene-Type Reaction. Cheminform. 40. DOI: 10.1002/chin.200917204  0.804
2008 Hupp CD, Tepe JJ. Total synthesis of a marine alkaloid from the tunicate Dendrodoa grossularia. Organic Letters. 10: 3737-9. PMID 18680306 DOI: 10.1021/Ol801375K  0.791
2008 Mosey RA, Fisk JS, Friebe TL, Tepe JJ. Synthesis of tert-alkyl amino hydroxy carboxylic esters via an intermolecular ene-type reaction of oxazolones and enol ethers. Organic Letters. 10: 825-8. PMID 18232699 DOI: 10.1021/Ol702941F  0.812
2008 Mosey RA, Fisk JS, Tepe JJ. Stereoselective syntheses of quaternary substituted α-amino acids using oxazol-5-(4H)-ones Tetrahedron Asymmetry. 19: 2755-2762. DOI: 10.1016/J.Tetasy.2008.11.033  0.776
2007 Fisk JS, Mosey RA, Tepe JJ. The diverse chemistry of oxazol-5-(4H)-ones. Chemical Society Reviews. 36: 1432-40. PMID 17660876 DOI: 10.1039/B511113G  0.788
2007 Sharma V, Hupp CD, Tepe JJ. Enhancement of chemotherapeutic efficacy by small molecule inhibition of NF-kappaB and checkpoint kinases. Current Medicinal Chemistry. 14: 1061-74. PMID 17456020 DOI: 10.2174/092986707780362844  0.771
2007 Fisk JS, Tepe JJ. Intermolecular ene reactions utilizing oxazolones and enol ethers. Journal of the American Chemical Society. 129: 3058-9. PMID 17326632 DOI: 10.1021/Ja0627904  0.802
2006 Sharma V, Peddibhotla S, Tepe JJ. Sensitization of cancer cells to DNA damaging agents by imidazolines. Journal of the American Chemical Society. 128: 9137-43. PMID 16834387 DOI: 10.1021/Ja060273F  0.727
2005 Sharma V, Tepe JJ. Diastereochemical diversity of imidazoline scaffolds via substrate controlled TMSCl mediated cycloaddition of azlactones. Organic Letters. 7: 5091-4. PMID 16235965 DOI: 10.1021/Ol052118W  0.605
2005 Keni M, Tepe JJ. One-pot Friedel-Crafts/Robinson-Gabriel synthesis of oxazoles using oxazolone templates. The Journal of Organic Chemistry. 70: 4211-3. PMID 15876123 DOI: 10.1021/Jo0501590  0.468
2004 Sharma V, Lansdell TA, Peddibhotla S, Tepe JJ. Sensitization of tumor cells toward chemotherapy: enhancing the efficacy of camptothecin with imidazolines. Chemistry & Biology. 11: 1689-99. PMID 15610853 DOI: 10.1016/J.Chembiol.2004.10.006  0.727
2004 Peddibhotla S, Tepe JJ. Stereoselective synthesis of highly substituted Delta1-pyrrolines: exo-selective 1,3-dipolar cycloaddition reactions with azlactones. Journal of the American Chemical Society. 126: 12776-7. PMID 15469263 DOI: 10.1021/Ja046149I  0.761
2004 Sharma V, Tepe JJ. Potent inhibition of checkpoint kinase activity by a hymenialdisine-derived indoloazepine. Bioorganic & Medicinal Chemistry Letters. 14: 4319-21. PMID 15261294 DOI: 10.1016/J.Bmcl.2004.05.079  0.551
2004 Sharma V, Lansdell TA, Jin G, Tepe JJ. Inhibition of cytokine production by hymenialdisine derivatives. Journal of Medicinal Chemistry. 47: 3700-3. PMID 15214798 DOI: 10.1021/Jm040013D  0.544
2003 Peddibhotla S, Tepe JJ. Multicomponent Synthesis of Highly Substituted Imidazolines via a Silicon-Mediated 1,3-Dipolar Cycloaddition. Cheminform. 34. DOI: 10.1055/S-2003-40196  0.479
2003 Peddibhotla S, Cheng Z, DellaPenna D, Tepe JJ. Efficient two-step synthesis of methylphytylbenzoquinones: Precursor intermediates in the biosynthesis of vitamin E Tetrahedron Letters. 44: 237-239. DOI: 10.1016/S0040-4039(02)02564-9  0.703
2002 Peddibhotla S, Jayakumar S, Tepe JJ. Highly diastereoselective multicomponent synthesis of unsymmetrical imidazolines. Organic Letters. 4: 3533-5. PMID 12323062 DOI: 10.1021/Ol026703Y  0.739
2002 Beckerbauer L, Tepe JJ, Eastman RA, Mixter PF, Williams RM, Reeves R. Differential effects of FR900482 and FK317 on apoptosis, IL-2 gene expression, and induction of vascular leak syndrome. Chemistry & Biology. 9: 427-41. PMID 11983332 DOI: 10.1016/S1074-5521(02)00122-9  0.429
2002 Anderson KW, Tepe JJ. The first intermolecular Friedel-Crafts acylation with beta-lactams. Organic Letters. 4: 459-61. PMID 11820904 DOI: 10.1021/Ol010291W  0.332
2002 Anderson KW, Tepe JJ. Trifluoromethanesulfonic acid catalyzed Friedel-Crafts acylation of aromatics with β-lactams Tetrahedron. 58: 8475-8481. DOI: 10.1016/S0040-4020(02)01026-8  0.382
2002 Tepe JJ, Kosogof C, Williams RM. DNA interstrand cross-link formation by reductive activation of dehydropyrrolizidine progenitors Tetrahedron. 58: 3553-3559. DOI: 10.1016/S0040-4020(02)00311-3  0.472
2001 Beckerbauer L, Tepe JJ, Cullison J, Reeves R, Williams RM. FR900482 class of anti-tumor drugs cross-links oncoprotein HMG I/Y to DNA in vivo. Chemistry & Biology. 7: 805-12. PMID 11033083 DOI: 10.1016/S1074-5521(00)00028-4  0.447
2001 Kosogof C, Tepe JJ, Williams RM. DNA cross-linking by a phototriggered pyrrolic progenitor developed from monocrotaline Tetrahedron Letters. 42: 6641-6643. DOI: 10.1016/S0040-4039(01)01341-7  0.491
1999 Tepe JJ, Williams RM. Reductive Activation of a Hydroxylamine Hemiacetal Derivative of Dehydromonocrotaline: The First Reductively Activated Pyrrolizidine Alkaloid Capable of Cross-Linking DNA. Angewandte Chemie. 38: 3501-3503. PMID 10602221 DOI: 10.1002/(Sici)1521-3773(19991203)38:23<3501::Aid-Anie3501>3.0.Co;2-W  0.464
1999 Tepe JJ, Williams RM. DNA Cross-Linking by a Phototriggered Dehydromonocrotaline Progenitor Journal of the American Chemical Society. 121: 2951-2955. DOI: 10.1021/Ja983894K  0.475
1999 Tepe J, Williams R. Reduktive Aktivierung eines Hydroxylamin-Hemiacetal-Derivats von Dehydromonocrotalin: das erste reduktiv aktivierbare Pyrrolizidinalkaloid, das DNA-Stränge quervernetzen kann Angewandte Chemie. 111: 3711-3713. DOI: 10.1002/(Sici)1521-3757(19991203)111:23<3711::Aid-Ange3711>3.0.Co;2-A  0.416
1997 Madalengoitia JS, Tepe JJ, Werbovetz KA, Lehnert EK, Macdonald TL. Structure-activity relationship for DNA topoisomerase II-induced DNA cleavage by azatoxin analogues. Bioorganic & Medicinal Chemistry. 5: 1807-15. PMID 9354236 DOI: 10.1016/S0968-0896(97)00113-2  0.75
1996 Tepe JJ, Madalengoitia JS, Slunt KM, Werbovetz KW, Spoors PG, Macdonald TL. Inhibition of DNA topoisomerase II by azaelliptitoxins functionalized in the variable substituent domain. Journal of Medicinal Chemistry. 39: 2188-96. PMID 8667362 DOI: 10.1021/jm9508806  0.741
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