Year |
Citation |
Score |
2019 |
Agius MP, Ko KS, Johnson TK, Kwarcinski FE, Phadke S, Lachacz EJ, Soellner MB. Selective Proteolysis to Study the Global Conformation and Regulatory Mechanisms of c-Src Kinase. Acs Chemical Biology. PMID 31287657 DOI: 10.1021/Acschembio.9B00306 |
0.341 |
|
2016 |
Johnson TK, Soellner MB. Bivalent inhibitors of c-Src tyrosine kinase that bind a regulatory domain. Bioconjugate Chemistry. PMID 27266260 DOI: 10.1021/Acs.Bioconjchem.6B00243 |
0.352 |
|
2016 |
Gilani R, Phadke S, Bao LW, Lachacz E, Dziubinski M, Brandvold K, Steffey M, Kwarcinski F, Graveel CR, Kidwell KM, Merajver SD, Soellner MB. UM-164: a potent c-Src/p38 kinase inhibitor with in vivo activity against triple negative breast cancer. Clinical Cancer Research : An Official Journal of the American Association For Cancer Research. PMID 27154914 DOI: 10.1158/1078-0432.Ccr-15-2158 |
0.35 |
|
2016 |
Kwarcinski FE, Brandvold KR, Phadke S, Beleh OM, Johnson TK, Meagher JL, Seeliger MA, Stuckey JA, Soellner MB. Conformation-selective analogs of dasatinib reveal insight into kinase inhibitor binding and selectivity. Acs Chemical Biology. PMID 26895387 DOI: 10.1021/Acschembio.5B01018 |
0.358 |
|
2015 |
Larsen BJ, Sun Z, Lachacz E, Khomutnyk Y, Soellner MB, Nagorny P. Synthesis and Biological Evaluation of Lactimidomycin and Its Analogues. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 26577990 DOI: 10.1002/Chem.201503527 |
0.333 |
|
2015 |
Kwarcinski FE, Steffey ME, Fox CC, Soellner MB. Discovery of Bivalent Kinase Inhibitors via Enzyme-Templated Fragment Elaboration. Acs Medicinal Chemistry Letters. 6: 898-901. PMID 26286460 DOI: 10.1021/Acsmedchemlett.5B00167 |
0.416 |
|
2015 |
Brandvold KR, Santos SM, Breen ME, Lachacz EJ, Steffey ME, Soellner MB. Exquisitely Specific Bisubstrate Inhibitors of c-Src Kinase. Acs Chemical Biology. 10: 1387-91. PMID 25793938 DOI: 10.1021/Cb501048B |
0.632 |
|
2015 |
Breen ME, Soellner MB. Small molecule substrate phosphorylation site inhibitors of protein kinases: approaches and challenges. Acs Chemical Biology. 10: 175-89. PMID 25494294 DOI: 10.1021/Cb5008376 |
0.388 |
|
2015 |
Gilani RA, Brandvold KR, Bao LW, Phadke S, Steffey ME, Soellner MB, Merajver SD. Abstract 5536: KB-164, a novel and highly potent Src family kinase inhibitor, reduces cancer cell invasion and abrogates downstream oncogenic pathways in triple negative breast cancer Cancer Research. 75: 5536-5536. DOI: 10.1158/1538-7445.Am2015-5536 |
0.304 |
|
2014 |
Agius MP, Soellner MB. Modulating noncatalytic function with kinase inhibitors. Chemistry & Biology. 21: 569-71. PMID 24856138 DOI: 10.1016/J.Chembiol.2014.05.005 |
0.393 |
|
2014 |
Breen ME, Steffey ME, Lachacz EJ, Kwarcinski FE, Fox CC, Soellner MB. Substrate activity screening with kinases: discovery of small-molecule substrate-competitive c-Src inhibitors. Angewandte Chemie (International Ed. in English). 53: 7010-3. PMID 24797781 DOI: 10.1002/Anie.201311096 |
0.386 |
|
2014 |
Bremmer SC, McNeil AJ, Soellner MB. Enzyme-triggered gelation: targeting proteases with internal cleavage sites. Chemical Communications (Cambridge, England). 50: 1691-3. PMID 24394494 DOI: 10.1039/C3Cc48132H |
0.345 |
|
2013 |
Ko KS, Steffey ME, Brandvold KR, Soellner MB. Development of a chimeric c-Src kinase and HDAC inhibitor. Acs Medicinal Chemistry Letters. 4: 779-783. PMID 24015327 DOI: 10.1021/Ml400175D |
0.354 |
|
2013 |
Rabuck JN, Hyung SJ, Ko KS, Fox CC, Soellner MB, Ruotolo BT. Activation state-selective kinase inhibitor assay based on ion mobility-mass spectrometry. Analytical Chemistry. 85: 6995-7002. PMID 23845095 DOI: 10.1021/Ac4012655 |
0.412 |
|
2012 |
Kwarcinski FE, Fox CC, Steffey ME, Soellner MB. Irreversible inhibitors of c-Src kinase that target a nonconserved cysteine. Acs Chemical Biology. 7: 1910-7. PMID 22928736 DOI: 10.1021/Cb300337U |
0.376 |
|
2012 |
Brandvold KR, Steffey ME, Fox CC, Soellner MB. Development of a highly selective c-Src kinase inhibitor. Acs Chemical Biology. 7: 1393-8. PMID 22594480 DOI: 10.1021/Cb300172E |
0.372 |
|
2008 |
Tam A, Soellner MB, Raines RT. Electronic and steric effects on the rate of the traceless Staudinger ligation. Organic & Biomolecular Chemistry. 6: 1173-5. PMID 18362954 DOI: 10.1039/B802336K |
0.625 |
|
2007 |
Tam A, Arnold U, Soellner MB, Raines RT. Protein prosthesis: 1,5-disubstituted[1,2,3]triazoles as cis-peptide bond surrogates. Journal of the American Chemical Society. 129: 12670-1. PMID 17914828 DOI: 10.1021/Ja075865S |
0.722 |
|
2007 |
Tam A, Soellner MB, Raines RT. Water-soluble phosphinothiols for traceless staudinger ligation and integration with expressed protein ligation. Journal of the American Chemical Society. 129: 11421-30. PMID 17713909 DOI: 10.1021/Ja073204P |
0.666 |
|
2007 |
Soellner MB, Rawls KA, Grundner C, Alber T, Ellman JA. Fragment-based substrate activity screening method for the identification of potent inhibitors of the Mycobacterium tuberculosis phosphatase PtpB. Journal of the American Chemical Society. 129: 9613-5. PMID 17636914 DOI: 10.1021/Ja0727520 |
0.662 |
|
2006 |
Soellner MB, Tam A, Raines RT. Staudinger ligation of peptides at non-glycyl residues. The Journal of Organic Chemistry. 71: 9824-30. PMID 17168602 DOI: 10.1021/Jo0620056 |
0.686 |
|
2006 |
Soellner MB, Nilsson BL, Raines RT. Reaction mechanism and kinetics of the traceless Staudinger ligation. Journal of the American Chemical Society. 128: 8820-8. PMID 16819875 DOI: 10.1021/Ja060484K |
0.641 |
|
2005 |
Nilsson BL, Soellner MB, Raines RT. Chemical synthesis of proteins. Annual Review of Biophysics and Biomolecular Structure. 34: 91-118. PMID 15869385 DOI: 10.1146/Annurev.Biophys.34.040204.144700 |
0.688 |
|
2005 |
Smith BD, Soellner MB, Raines RT. Synthetic surfaces for ribonuclease adsorption. Langmuir : the Acs Journal of Surfaces and Colloids. 21: 187-90. PMID 15620301 DOI: 10.1021/La0480686 |
0.562 |
|
2003 |
Soellner MB, Dickson KA, Nilsson BL, Raines RT. Site-specific protein immobilization by Staudinger ligation. Journal of the American Chemical Society. 125: 11790-1. PMID 14505380 DOI: 10.1021/Ja036712H |
0.743 |
|
2003 |
Nilsson BL, Hondal RJ, Soellner MB, Raines RT. Protein assembly by orthogonal chemical ligation methods. Journal of the American Chemical Society. 125: 5268-9. PMID 12720426 DOI: 10.1021/Ja029752E |
0.75 |
|
2003 |
Smith BD, Soellner MB, Raines RT. Potent inhibition of ribonuclease A by oligo(vinylsulfonic acid). The Journal of Biological Chemistry. 278: 20934-8. PMID 12649287 DOI: 10.1074/Jbc.M301852200 |
0.616 |
|
2002 |
Soellner MB, Nilsson BL, Raines RT. Staudinger ligation of alpha-azido acids retains stereochemistry. The Journal of Organic Chemistry. 67: 4993-6. PMID 12098322 DOI: 10.1021/Jo025631L |
0.686 |
|
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