Year |
Citation |
Score |
2021 |
Nuthakki VK, Mudududdla R, Bharate SB. Role of basic aminoalkyl chains in the lead optimization of Indoloquinoline alkaloids. European Journal of Medicinal Chemistry. 227: 113938. PMID 34710743 DOI: 10.1016/j.ejmech.2021.113938 |
0.702 |
|
2021 |
Abdullaha M, Ali M, Kour D, Mudududdla R, Khajuria P, Kumar A, Bharate SB. Tetramethoxystilbene Inhibits NLRP3 Inflammasome Assembly via Blocking the Oligomerization of Apoptosis-Associated Speck-like Protein Containing Caspase Recruitment Domain: and Evaluation. Acs Pharmacology & Translational Science. 4: 1437-1448. PMID 34423275 DOI: 10.1021/acsptsci.1c00126 |
0.461 |
|
2019 |
Nuthakki VK, Mudududdla R, Sharma A, Kumar A, Bharate SB. Synthesis and biological evaluation of indoloquinoline alkaloid cryptolepine and its bromo-derivative as dual cholinesterase inhibitors. Bioorganic Chemistry. 90: 103062. PMID 31220673 DOI: 10.1016/j.bioorg.2019.103062 |
0.71 |
|
2018 |
Derf A, Mudududdla R, Akintade D, Williams IS, Abdullaha M, Chaudhuri B, Bharate SB. Nonantioxidant Tetramethoxystilbene Abrogates α-Synuclein-Induced Yeast Cell Death but Not That Triggered by the Bax or βA4 Peptide. Acs Omega. 3: 9513-9532. PMID 31459084 DOI: 10.1021/acsomega.8b01154 |
0.441 |
|
2018 |
Derf A, Mudududdla R, Bharate SB, Chaudhuri B. Inhibitors of Aβ42-induced endoplasmic reticular unfolded protein response (UPR), in yeast, also rescue yeast cells from Aβ42-mediated apoptosis. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. PMID 30502452 DOI: 10.1016/j.ejps.2018.11.029 |
0.587 |
|
2018 |
Bharate SB, Mudududdla R, Mohanakrishnan D, Bharate SS, Vishwakarma RA, Sahal D. Orally Effective Aminoalkyl 10H-Indolo-[3,2-b]quinoline-11-carboxamide Kills the Malaria Parasite by Inhibiting Host Hemoglobin Uptake. Chemmedchem. PMID 30358112 DOI: 10.1002/Cmdc.201800579 |
0.609 |
|
2015 |
Mudududdla R, Guru SK, Wani A, Sharma S, Joshi P, Vishwakarma RA, Kumar A, Bhushan S, Bharate SB. 3-(Benzo[d][1,3]dioxol-5-ylamino)-N-(4-fluorophenyl)thiophene-2-carboxamide overcomes cancer chemoresistance via inhibition of angiogenesis and P-glycoprotein efflux pump activity. Organic & Biomolecular Chemistry. 13: 4296-309. PMID 25758415 DOI: 10.1039/C5Ob00233H |
0.694 |
|
2015 |
Sharma R, Abbat S, Mudududdla R, Vishwakarma RA, Bharatam PV, Bharate SB. ortho-Quinone methides: TFA-mediated generation in water and trapping with lactams and styrenes Tetrahedron Letters. 56: 4057-4059. DOI: 10.1016/J.Tetlet.2015.04.072 |
0.526 |
|
2015 |
Sharma R, Abbat S, Mudududdla R, Vishwakarma RA, Bharatam PV, Bharate SB. ChemInform Abstract: ortho-Quinone Methides: TFA-Mediated Generation in Water and Trapping with Lactams and Styrenes. Cheminform. 46: no-no. DOI: 10.1002/CHIN.201542194 |
0.417 |
|
2014 |
Mudududdla R, Sharma R, Abbat S, Bharatam PV, Vishwakarma RA, Bharate SB. Synthesis of 2-phenylnaphthalenes from styryl-2-methoxybenzenes. Chemical Communications (Cambridge, England). 50: 12076-9. PMID 25163506 DOI: 10.1039/C4Cc05151C |
0.675 |
|
2014 |
Mudududdla R, Sharma R, Guru SK, Kushwaha M, Gupta AP, Bharate SS, Aravinda S, Kant R, Bhushan S, Vishwakarma RA, Bharate SB. Trifluoroacetic acid catalyzed thiophenylmethylation and thioalkylmethylation of lactams and phenols via domino three-component reaction in water Rsc Advances. 4: 14081-14088. DOI: 10.1039/C3Ra47874B |
0.566 |
|
2013 |
Bharate SB, Bharate JB, Khan SI, Tekwani BL, Jacob MR, Mudududdla R, Yadav RR, Singh B, Sharma PR, Maity S, Singh B, Khan IA, Vishwakarma RA. Discovery of 3,3'-diindolylmethanes as potent antileishmanial agents. European Journal of Medicinal Chemistry. 63: 435-43. PMID 23517732 DOI: 10.1016/J.Ejmech.2013.02.024 |
0.737 |
|
2013 |
Bharate SB, Mudududdla R, Sharma R, Vishwakarma RA. The first method for C-devinylation of aromatic systems Tetrahedron Letters. 54: 2913-2915. DOI: 10.1016/J.Tetlet.2013.03.064 |
0.527 |
|
2013 |
Bharate SB, Mudududdla R, Sharma R, Vishwakarma RA. ChemInform Abstract: The First Method for C-Devinylation of Aromatic Systems. Cheminform. 44: no-no. DOI: 10.1002/CHIN.201337051 |
0.432 |
|
2012 |
Mudududdla R, Jain SK, Bharate JB, Gupta AP, Singh B, Vishwakarma RA, Bharate SB. ortho-Amidoalkylation of phenols via tandem one-pot approach involving oxazine intermediate. The Journal of Organic Chemistry. 77: 8821-7. PMID 22970791 DOI: 10.1021/Jo3017132 |
0.723 |
|
2012 |
Bharate SB, Mudududdla R, Bharate JB, Battini N, Battula S, Yadav RR, Singh B, Vishwakarma RA. Tandem one-pot synthesis of flavans by recyclable silica-HClO4 catalyzed Knoevenagel condensation and [4 + 2]-Diels-Alder cycloaddition. Organic & Biomolecular Chemistry. 10: 5143-50. PMID 22648274 DOI: 10.1039/C2Ob25376C |
0.728 |
|
2012 |
Bharate SB, Mupparapu N, Manda S, Bharate JB, Mudududdla R, Yadav RR, Vishwakarma RA. Efficient synthesis of 2,3-dihydroquinazolin-4(1H)-ones using heterogeneous solid acid catalysts: unexpected formation of 2,3-dihydro-2-(4-(tetrahydro-2H-pyran-2-yloxy)butyl)-quinazolin-4(1H)-one Arkivoc. 2012: 308-318. DOI: 10.3998/Ark.5550190.0013.826 |
0.72 |
|
2012 |
Yadav RR, Battini N, Mudududdla R, Bharate JB, Muparappu N, Bharate SB, Vishwakarma RA. Deformylation of indole and azaindole-3-carboxaldehydes using anthranilamide and solid acid heterogeneous catalyst via quinazolinone intermediate Tetrahedron Letters. 53: 2222-2225. DOI: 10.1016/J.Tetlet.2012.02.079 |
0.713 |
|
2012 |
Yadav RR, Battini N, Mudududdla R, Bharate JB, Muparappu N, Bharate SB, Vishwakarma RA. ChemInform Abstract: Deformylation of Indole and Azaindole-3-carboxaldehydes Using Anthranilamide and Solid Acid Heterogeneous Catalyst via Quinazolinone Intermediate. Cheminform. 43: no-no. DOI: 10.1002/CHIN.201232119 |
0.7 |
|
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