Year |
Citation |
Score |
2023 |
Sangadi DK, Sangadi A, Placeres-Uray F, Titus DJ, Johnstone T, Hogenkamp D, Gee KW, Atkins CM. Enhancing cognitive function in chronic TBI: The Role of α7 nicotinic acetylcholine receptor modulation. Experimental Neurology. 372: 114647. PMID 38070724 DOI: 10.1016/j.expneurol.2023.114647 |
0.72 |
|
2020 |
Belelli D, Hogenkamp D, Gee KW, Lambert JJ. Realising the therapeutic potential of neuroactive steroid modulators of the GABA receptor. Neurobiology of Stress. 12: 100207. PMID 32435660 DOI: 10.1016/J.Ynstr.2019.100207 |
0.436 |
|
2019 |
Titus DJ, Johnstone T, Johnson NH, London SH, Chapalamadugu M, Hogenkamp D, Gee KW, Atkins CM. Positive allosteric modulation of the α7 nicotinic acetylcholine receptor as a treatment for cognitive deficits after traumatic brain injury. Plos One. 14: e0223180. PMID 31581202 DOI: 10.1371/Journal.Pone.0223180 |
0.743 |
|
2019 |
Johnstone TBC, McCarren HS, Spampanato J, Dudek FE, McDonough JH, Hogenkamp D, Gee KW. Enaminone Modulators of Extrasynaptic αβδ γ-Aminobutyric Acid Receptors Reverse Electrographic Status Epilepticus in the Rat After Acute Organophosphorus Poisoning. Frontiers in Pharmacology. 10: 560. PMID 31178732 DOI: 10.3389/Fphar.2019.00560 |
0.379 |
|
2018 |
Johnstone TBC, Xie JY, Qu C, Wasiak DJ, Hogenkamp DJ, Porreca F, Gee KW. Positive Allosteric Modulators of Non-Benzodiazepine γ-Aminobutyric acida Receptor Subtypes for the Treatment of Chronic Pain. Pain. PMID 30204648 DOI: 10.1097/J.Pain.0000000000001392 |
0.401 |
|
2018 |
Reddy DS, Yoshimura RF, Ramanathan G, Carver C, Johnstone TB, Hogenkamp DJ, Gee KW. Role of β-specific GABA-A receptor isoforms in the development of hippocampus kindling epileptogenesis. Epilepsy & Behavior : E&B. 82: 57-63. PMID 29587186 DOI: 10.1016/J.Yebeh.2018.02.020 |
0.807 |
|
2017 |
Yoshimura RF, Tran MB, Hogenkamp DJ, Ayala NL, Johnstone T, Dunnigan AJ, Gee TK, Gee KW. Allosteric modulation of nicotinic and GABAA receptor subtypes differentially modify autism-like behaviors in the BTBR mouse model. Neuropharmacology. PMID 28842344 DOI: 10.1016/J.Neuropharm.2017.08.029 |
0.791 |
|
2017 |
Gee KW, Olincy A, Kanner R, Johnson L, Hogenkamp D, Harris J, Tran M, Edmonds SA, Sauer W, Yoshimura R, Johnstone T, Freedman R. First in human trial of a type I positive allosteric modulator of alpha7-nicotinic acetylcholine receptors: Pharmacokinetics, safety, and evidence for neurocognitive effect of AVL-3288. Journal of Psychopharmacology (Oxford, England). 269881117691590. PMID 28196430 DOI: 10.1177/0269881117691590 |
0.792 |
|
2015 |
Dasse O, Bilcer G, Putman D, Ng R, Gee K, Stevens KE, Tran M, Johnstone T, Yoshimura RF, Koelsch G, Kelly TA. APN0417: A potent and efficacious α7 nAChR positive allosteric modulator Biochemical Pharmacology. 97: 636. DOI: 10.1016/J.Bcp.2015.08.043 |
0.783 |
|
2015 |
Titus DJ, Concepcion F, Johnstone T, Hogenkamp D, Gee KW, Atkins CM. Positive allosteric modulation of the α7 nicotinic acetylcholine receptor reverses chronic cognitive deficits after TBI Biochemical Pharmacology. 97: 635. DOI: 10.1016/J.Bcp.2015.08.041 |
0.766 |
|
2014 |
Hogenkamp DJ, Tran MB, Yoshimura RF, Johnstone TB, Kanner R, Gee KW. Pharmacological profile of a 17β-heteroaryl-substituted neuroactive steroid. Psychopharmacology. 231: 3517-24. PMID 24682501 DOI: 10.1007/S00213-014-3494-5 |
0.75 |
|
2014 |
Yoshimura RF, Tran MB, Hogenkamp DJ, Johnstone TB, Xie JY, Porreca F, Gee KW. Limited central side effects of a β-subunit subtype-selective GABAA receptor allosteric modulator. Journal of Psychopharmacology (Oxford, England). 28: 472-8. PMID 24108410 DOI: 10.1177/0269881113507643 |
0.812 |
|
2014 |
Koelsch G, Meltzer LT, Yoshimura RF, Terry AV, Callahan PM, Bilcer G, Ng J, Ng R, Gee KW, Kelly TA. P4-373: APN1125: A NOVEL A7 NICOTINIC ACETYLCHOLINE RECEPTOR PARTIAL AGONIST Alzheimer's & Dementia. 10: P925-P925. DOI: 10.1016/J.Jalz.2014.07.142 |
0.736 |
|
2013 |
Hogenkamp DJ, Ford-Hutchinson TA, Li WY, Whittemore ER, Yoshimura RF, Tran MB, Johnstone TB, Bascom GD, Rollins H, Lu L, Gee KW. Design, synthesis, and activity of a series of arylpyrid-3-ylmethanones as type I positive allosteric modulators of α7 nicotinic acetylcholine receptors. Journal of Medicinal Chemistry. 56: 8352-65. PMID 24098954 DOI: 10.1021/Jm400704G |
0.806 |
|
2012 |
Chen S, Tusty M, Johnstone T, Hogenkamp D, Gee K, Brinton R. P2-395: Allopregnanolone analogues promote proliferation of neural progenitor cells Alzheimer's & Dementia. 8: P401-P401. DOI: 10.1016/J.Jalz.2012.05.1105 |
0.671 |
|
2011 |
Lotfipour S, Arnold MM, Hogenkamp DJ, Gee KW, Belluzzi JD, Leslie FM. The monoamine oxidase (MAO) inhibitor tranylcypromine enhances nicotine self-administration in rats through a mechanism independent of MAO inhibition. Neuropharmacology. 61: 95-104. PMID 21419142 DOI: 10.1016/J.Neuropharm.2011.03.007 |
0.366 |
|
2011 |
Johnstone TB, Gu Z, Yoshimura RF, Villegier AS, Hogenkamp DJ, Whittemore ER, Huang JC, Tran MB, Belluzzi JD, Yakel JL, Gee KW. Allosteric modulation of related ligand-gated ion channels synergistically induces long-term potentiation in the hippocampus and enhances cognition. The Journal of Pharmacology and Experimental Therapeutics. 336: 908-15. PMID 21159751 DOI: 10.1124/Jpet.110.176255 |
0.796 |
|
2010 |
Gee KW, Tran MB, Hogenkamp DJ, Johnstone TB, Bagnera RE, Yoshimura RF, Huang JC, Belluzzi JD, Whittemore ER. Limiting activity at beta1-subunit-containing GABAA receptor subtypes reduces ataxia. The Journal of Pharmacology and Experimental Therapeutics. 332: 1040-53. PMID 19940102 DOI: 10.1124/Jpet.109.161885 |
0.737 |
|
2010 |
HOGENKAMP DJ, TAHIR SH, HAWKINSON JE, UPASANI RB, ALAUDDIN M, KIMBROUGH CL, ACOSTA-BURRUEL M, WHITTEMORE ER, WOODWARD RM, LAN NC, GEE KW, BOLGER MB. ChemInform Abstract: Synthesis and in vitro Activity of 3β-Substituted-3α- hydroxypregnan-20-ones: Allosteric Modulators of the GABAA Receptor. Cheminform. 28: no-no. DOI: 10.1002/chin.199717196 |
0.323 |
|
2009 |
Gee K, Hogenkamp D, Johnstone T. Dual allosteric modulators of neuronal nicotinic-acetylcholine and GABAA receptors Biochemical Pharmacology. 78: 913-914. DOI: 10.1016/J.Bcp.2009.06.065 |
0.757 |
|
2007 |
Yoshimura RF, Hogenkamp DJ, Li WY, Tran MB, Belluzzi JD, Whittemore ER, Leslie FM, Gee KW. Negative allosteric modulation of nicotinic acetylcholine receptors blocks nicotine self-administration in rats. The Journal of Pharmacology and Experimental Therapeutics. 323: 907-15. PMID 17873105 DOI: 10.1124/Jpet.107.128751 |
0.777 |
|
2007 |
Hogenkamp DJ, Johnstone TB, Huang JC, Li WY, Tran M, Whittemore ER, Bagnera RE, Gee KW. Enaminone amides as novel orally active GABAA receptor modulators. Journal of Medicinal Chemistry. 50: 3369-79. PMID 17571865 DOI: 10.1021/Jm070083V |
0.771 |
|
2007 |
Ng HJ, Whittemore ER, Tran MB, Hogenkamp DJ, Broide RS, Johnstone TB, Zheng L, Stevens KE, Gee KW. Nootropic alpha7 nicotinic receptor allosteric modulator derived from GABAA receptor modulators. Proceedings of the National Academy of Sciences of the United States of America. 104: 8059-64. PMID 17470817 DOI: 10.1073/Pnas.0701321104 |
0.805 |
|
2006 |
Wang J, Hogenkamp DJ, Tran M, Li WY, Yoshimura RF, Johnstone TB, Shen WC, Gee KW. Reversible lipidization for the oral delivery of leu-enkephalin. Journal of Drug Targeting. 14: 127-36. PMID 16753826 DOI: 10.1080/10611860600648221 |
0.75 |
|
2004 |
Johnstone TB, Hogenkamp DJ, Coyne L, Su J, Halliwell RF, Tran MB, Yoshimura RF, Li WY, Wang J, Gee KW. Modifying quinolone antibiotics yields new anxiolytics. Nature Medicine. 10: 31-2. PMID 14647497 DOI: 10.1038/Nm967 |
0.787 |
|
2001 |
Vanover KE, Hogenkamp DJ, Lan NC, Gee KW, Carter RB. Behavioral characterization of Co 134444 (3alpha-hydroxy-21-(1'-imidazolyl)-3beta-methoxymethyl-5alpha- pregnan-20-one), a novel sedative-hypnotic neuroactive steroid. Psychopharmacology. 155: 285-91. PMID 11432691 DOI: 10.1007/S002130100695 |
0.328 |
|
1999 |
Vanover KE, Suruki M, Robledo S, Huber M, Wieland S, Lan NC, Gee KW, Wood PL, Carter RB. Positive allosteric modulators of the GABA(A) receptor: differential interaction of benzodiazepines and neuroactive steroids with ethanol. Psychopharmacology. 141: 77-82. PMID 9952068 DOI: 10.1007/S002130050809 |
0.384 |
|
1997 |
Wieland S, Belluzzi J, Hawkinson JE, Hogenkamp D, Upasani R, Stein L, Wood PL, Gee KW, Lan NC. Anxiolytic and anticonvulsant activity of a synthetic neuroactive steroid Co 3-0593. Psychopharmacology. 134: 46-54. PMID 9399366 DOI: 10.1007/S002130050424 |
0.383 |
|
1997 |
Carter RB, Wood PL, Wieland S, Hawkinson JE, Belelli D, Lambert JJ, White HS, Wolf HH, Mirsadeghi S, Tahir SH, Bolger MB, Lan NC, Gee KW. Characterization of the anticonvulsant properties of ganaxolone (CCD 1042; 3alpha-hydroxy-3beta-methyl-5alpha-pregnan-20-one), a selective, high-affinity, steroid modulator of the gamma-aminobutyric acid(A) receptor. The Journal of Pharmacology and Experimental Therapeutics. 280: 1284-95. PMID 9067315 |
0.334 |
|
1997 |
Hogenkamp DJ, Tahir SH, Hawkinson JE, Upasani RB, Alauddin M, Kimbrough CL, Acosta-Burruel M, Whittemore ER, Woodward RM, Lan NC, Gee KW, Bolger MB. Synthesis and in vitro activity of 3 beta-substituted-3 alpha-hydroxypregnan-20-ones: allosteric modulators of the GABAA receptor. Journal of Medicinal Chemistry. 40: 61-72. PMID 9016329 DOI: 10.1021/Jm960021X |
0.378 |
|
1996 |
Belelli D, Lambert JJ, Peters JA, Gee KW, Lan NC. Modulation of human recombinant GABAA receptors by pregnanediols. Neuropharmacology. 35: 1223-31. PMID 9014137 DOI: 10.1016/S0028-3908(96)00066-4 |
0.374 |
|
1996 |
Xue BG, Friend JM, Gee KW. Loreclezole modulates [35S]t-butylbicyclophosphorothionate and [3H]flunitrazepam binding via a distinct site on the GABAA receptor complex European Journal of Pharmacology. 300: 125-130. PMID 8741177 DOI: 10.1016/0014-2999(95)00856-X |
0.488 |
|
1995 |
Gee KW, McCauley LD, Lan NC. A putative receptor for neurosteroids on the GABA(A) receptor complex: The pharmacological properties and therapeutic potential of epalons Critical Reviews in Neurobiology. 9: 207-227. PMID 8581984 |
0.347 |
|
1995 |
McCauley LD, Gee KW. Influence of the estrus cycle on the discrimination of apparent neuroactive steroid site subtypes on the γ-aminobutyric acid(A) receptor complex in the rat Journal of Pharmacology and Experimental Therapeutics. 275: 1412-1417. PMID 8531110 |
0.315 |
|
1995 |
Lan NC, Chen JS, Johnson D, Gee KW. Differential effects of 4′-chlorodiazepam on expressed human GABAA receptors Journal of Neurochemistry. 64: 684-688. PMID 7830061 DOI: 10.1046/J.1471-4159.1995.64020684.X |
0.44 |
|
1995 |
McCauley LD, Park CH, Lan NC, Tomich JM, Shively JE, Gee KW. Benzodiazepines and peptides stimulate pregnenolone synthesis in brain mitochondria European Journal of Pharmacology. 276: 145-153. PMID 7781684 DOI: 10.1016/0014-2999(95)00036-K |
0.371 |
|
1995 |
Wang MD, Wahlström G, Gee KW, Bäckström T. Potency of lipid and protein formulation of 5 alpha-pregnanolone at induction of anaesthesia and the corresponding regional brain distribution. British Journal of Anaesthesia. 74: 553-7. PMID 7772431 DOI: 10.1093/Bja/74.5.553 |
0.321 |
|
1994 |
Hawkinson JE, Kimbrough CL, McCauley LD, Bolger MB, Lan NC, Gee KW. The neuroactive steroid 3 alpha-hydroxy-5 beta-pregnan-20-one is a two-component modulator of ligand binding to the GABAA receptor. European Journal of Pharmacology. 269: 157-63. PMID 7851492 DOI: 10.1016/0922-4106(94)90082-5 |
0.388 |
|
1994 |
Lan NC, Gee KW. Neuroactive steroid actions at the GABA(A) receptor Hormones and Behavior. 28: 537-544. PMID 7729823 DOI: 10.1006/Hbeh.1994.1052 |
0.507 |
|
1994 |
McCauley LD, Gee KW. Detection and Characterization of Epalon Receptors: Novel Recognition Sites for Neuroactive Steroids That Modulate the GABAA Receptor Complex Methods in Neurosciences. 22: 211-225. DOI: 10.1016/B978-0-12-185292-4.50019-X |
0.402 |
|
1993 |
Finn DA, Gee KW. A comparison of Ro 16-6028 with benzodiazepine receptor 'full agonists' on GABAA receptor function. European Journal of Pharmacology. 247: 233-7. PMID 7905829 DOI: 10.1016/0922-4106(93)90190-K |
0.458 |
|
1992 |
Cadoni C, Gee KW. Complex interactions between the steroid derivative RU 5135 and the GABAA-receptor complex European Journal of Pharmacology: Molecular Pharmacology. 227: 147-151. PMID 1330646 DOI: 10.1016/0922-4106(92)90122-C |
0.465 |
|
1992 |
McNeil RG, Gee KW, Bolger MB, Lan NC, Wieland S, Belelli D, Purdy RH, Paul SM. Neuroactive steroids that act at GABA(A) receptors Drug News and Perspectives. 5: 145-152. |
0.33 |
|
1991 |
Wieland S, Lan NC, Mirasedeghi S, Gee KW. Anxiolytic activity of the progesterone metabolite 5α-pregnan-3α-ol-20-one Brain Research. 565: 263-268. PMID 1688192 DOI: 10.1016/0006-8993(91)91658-N |
0.318 |
|
1991 |
Lan NC, Bolger MB, Gee KW. Identification and characterization of a pregnane steroid recognition site that is functionally coupled to an expressed GABAA receptor Neurochemical Research. 16: 347-356. PMID 1664061 DOI: 10.1007/Bf00966098 |
0.376 |
|
1991 |
Lan NC, Gee KW, Bolger MB, Chen JS. Differential responses of expressed recombinant human γ-aminobutyric acidA receptors to neurosteroids Journal of Neurochemistry. 57: 1818-1821. PMID 1655982 DOI: 10.1111/J.1471-4159.1991.Tb06388.X |
0.459 |
|
1990 |
Belelli D, Lan NC, Gee KW. Anticonvulsant steroids and the GABA/benzodiazepine receptor-chloride ionophore complex. Neuroscience and Biobehavioral Reviews. 14: 315-22. PMID 2172879 DOI: 10.1016/S0149-7634(05)80041-7 |
0.429 |
|
1990 |
Lan NC, Chen JS, Belelli D, Pritchett DB, Seeburg PH, Gee KW. A steroid recognition site is functionally coupled to an expressed GABA(A)-benzodiazepine receptor. European Journal of Pharmacology. 188: 403-6. PMID 2164942 DOI: 10.1016/0922-4106(90)90201-8 |
0.452 |
|
1990 |
Belelli D, McCauley L, Gee KW. Heterotropic cooperativity between putative recognition sites for progesterone metabolites and the atypical benzodiazepine Ro 5-4864. Journal of Neurochemistry. 55: 83-7. PMID 2113084 DOI: 10.1111/J.1471-4159.1990.Tb08824.X |
0.379 |
|
1990 |
McCauley L, Belelli D, Gee KW. Benzodiazepine receptor subtypes and receptor reserve capacity in rat brain European Journal of Pharmacology. 183: 2151. DOI: 10.1016/0014-2999(90)93675-G |
0.405 |
|
1990 |
Belelli D, McCauley L, Lan N, Bolger MB, Johnson D, Gee KW. Heterotropic cooperativity between recognition sites for steroids and 4'-chlorodiazepam (Ro5 4864) on the GABA/benzodiazepine receptor complex European Journal of Pharmacology. 183: 2024. DOI: 10.1016/0014-2999(90)92383-T |
0.413 |
|
1989 |
Belelli D, Bolger MB, Gee KW. Anticonvulsant profile of the progesterone metabolite 5 alpha-pregnan-3 alpha-ol-20-one. European Journal of Pharmacology. 166: 325-9. PMID 2792198 DOI: 10.1016/0014-2999(89)90077-0 |
0.409 |
|
1989 |
Ali SF, Newport GD, Scallet AC, Gee KW, Paule MG, Brown RM, Slikker W. Effects of chronic delta-9-tetrahydrocannabinol (THC) administration on neurotransmitter concentrations and receptor binding in the rat brain. Neurotoxicology. 10: 491-500. PMID 2576303 |
0.331 |
|
1989 |
Belelli D, Gee KW. 5 alpha-pregnan-3 alpha,20 alpha-diol behaves like a partial agonist in the modulation of GABA-stimulated chloride ion uptake by synaptoneurosomes. European Journal of Pharmacology. 167: 173-6. PMID 2550257 DOI: 10.1016/0014-2999(89)90760-7 |
0.348 |
|
1989 |
Gee KW, Joy DS, Belelli D. Complex interactions between pregnenolone sulfate and the t-butylbicyclophosphorothionate-labeled chloride ionophore in rat brain. Brain Research. 482: 169-73. PMID 2539882 DOI: 10.1016/0006-8993(89)90556-8 |
0.408 |
|
1988 |
Gee KW. Steroid modulation of the GABA/benzodiazepine receptor-linked chloride lonophore Molecular Neurobiology. 2: 291-317. PMID 2855977 DOI: 10.1007/Bf02935636 |
0.48 |
|
1988 |
Gee KW, Bolger MB, Brinton RE, Coirini H, McEwen BS. Steroid modulation of the chloride ionophore in rat brain: Structure-activity requirements, regional dependence and mechanism of action Journal of Pharmacology and Experimental Therapeutics. 246: 803-812. PMID 2841455 |
0.406 |
|
1988 |
Gee KW, Brinton RE, McEwen BS. Regional distribution of a Ro5 4864 binding site that is functionally coupled to the γ-aminobutyric acid/benzodiazepine receptor complex in rat brain Journal of Pharmacology and Experimental Therapeutics. 244: 379-383. PMID 2826772 |
0.343 |
|
1987 |
Gee KW, Chang WC, Brinton RE, McEwen BS. GABA-dependent modulation of the Cl- ionophore by steroids in rat brain European Journal of Pharmacology. 136: 419-423. PMID 3609126 DOI: 10.1016/0014-2999(87)90317-7 |
0.481 |
|
1986 |
Gee KW, Lawrence LJ, Yamamura HI. Modulation of the chloride ionophore by benzodiazepine receptor ligands: influence of gamma-aminobutyric acid and ligand efficacy. Molecular Pharmacology. 30: 218-25. PMID 3018479 |
0.332 |
|
1985 |
Lawrence LJ, Palmer CJ, Gee KW, Wang X, Yamamura HI, Casida JE. t-[3H]butylbicycloorthobenzoate: new radioligand probe for the gamma-aminobutyric acid-regulated chloride ionophore. Journal of Neurochemistry. 45: 798-804. PMID 2993514 DOI: 10.1111/J.1471-4159.1985.Tb04063.X |
0.322 |
|
1985 |
Gee KW, Lawrence LJ, Yamamura HI. Differential modulation of 35S-t-butylbicyclophosphorothionate (35S-TBPS) binding in rat brain by benzodiazepine (BZ) receptor ligands: Effect of GABA and ligand efficacy Federation Proceedings. 44. |
0.308 |
|
1984 |
Brinton RE, Gee KW, Wamsley JK, Davis TP, Yamamura HI. Regional distribution of putative vasopressin receptors in rat brain and pituitary by quantitative autoradiography. Proceedings of the National Academy of Sciences of the United States of America. 81: 7248-52. PMID 6095279 DOI: 10.1073/Pnas.81.22.7248 |
0.306 |
|
1984 |
Lawrence LJ, Gee KW, Yamamura HI. Benzodiazepine anticonvulsant action: gamma-aminobutyric acid-dependent modulation of the chloride ionophore. Biochemical and Biophysical Research Communications. 123: 1130-7. PMID 6091648 DOI: 10.1016/S0006-291X(84)80250-8 |
0.451 |
|
1984 |
Gee KW, Yamamura SH, Roeske WR, Yamamura HI. Benzodiazepine receptor heterogeneity: possible molecular basis and functional significance. Federation Proceedings. 43: 2767-72. PMID 6090222 |
0.317 |
|
1983 |
Gee KW, Killam EK, Hollinger MA. Effects of haloperidol-induced dopamine receptor supersensitivity on kindled seizure development. The Journal of Pharmacology and Experimental Therapeutics. 225: 70-6. PMID 6834278 |
0.645 |
|
1983 |
Wamsley JK, Gee KW, Yamamura HI. Comparison of the distribution of convulsant/barbiturate and benzodiazepine receptors using light microscopic autoradiography. Life Sciences. 33: 2321-9. PMID 6316061 DOI: 10.1016/0024-3205(83)90266-7 |
0.437 |
|
1983 |
Gee KW, Yamamura HI. Photoaffinity labeling of benzodiazepine receptors in rat brain with flunitrazepam alters the affinity of benzodiazepine receptor agonist but not antagonist binding. Journal of Neurochemistry. 41: 1407-13. PMID 6311986 DOI: 10.1111/J.1471-4159.1983.Tb00839.X |
0.364 |
|
1983 |
Ehlert FJ, Roeske WR, Gee KW, Yamamura HI. An allosteric model for benzodiazepine receptor function Biochemical Pharmacology. 32: 2375-2383. PMID 6311215 DOI: 10.1016/0006-2952(83)90679-2 |
0.458 |
|
1983 |
Mosberg HI, Hurst R, Hruby VJ, Gee K, Yamamura HI, Galligan JJ, Burks TF. Bis-penicillamine enkephalins possess highly improved specificity toward delta opioid receptors. Proceedings of the National Academy of Sciences of the United States of America. 80: 5871-4. PMID 6310598 DOI: 10.1073/Pnas.80.19.5871 |
0.342 |
|
1983 |
Mosberg HI, Hurst R, Hruby VJ, Galligan JJ, Burks TF, Gee K, Yamamura HI. Conformationally constrained cyclic enkephalin analogs with pronounced delta opioid receptor agonist selectivity. Life Sciences. 32: 2565-9. PMID 6304440 DOI: 10.1016/0024-3205(83)90239-4 |
0.381 |
|
1983 |
Gee KW, Brinton RE, Yamamura HI. PK 8165 and PK 9084, two quinoline derivatives with anxiolytic properties, antagonize the anticonvulsant effects of diazepam Brain Research. 264: 168-172. PMID 6303496 DOI: 10.1016/0006-8993(83)91138-1 |
0.447 |
|
1983 |
Yamamura HI, Gee KW, Brinton RE, Davis TP, Hadley M, Wamsley JK. Light microscopic autoradiographic visualization of [3H]-arginine vasopressin binding sites in rat brain. Life Sciences. 32: 1919-24. PMID 6300592 DOI: 10.1016/0024-3205(83)90072-3 |
0.308 |
|
1983 |
Gee KW, Ehlert FJ, Yamamura HI. Differential effect of γ-aminobutyric acid on benzodiazepine receptor subtypes labeled by [3H]propyl β-carboline-3-carboxylate in rat brain Journal of Pharmacology and Experimental Therapeutics. 225: 132-137. PMID 6300371 |
0.303 |
|
1983 |
Gee KW, Brinton RE, Yamamura HI. CL 218872 antagonism of diazepam induced loss of righting reflex: Evidence for partial agonistic activity at the benzodiazepine receptor Life Sciences. 32: 1037-1040. PMID 6298552 DOI: 10.1016/0024-3205(83)90936-0 |
0.452 |
|
1983 |
Gee KW, Yamamura HI. Selective anxiolytics: are the actions related to partial "agonist" activity or a preferential affinity for benzodiazepine receptor subtypes? Advances in Biochemical Psychopharmacology. 38: 1-9. PMID 6142598 |
0.357 |
|
1983 |
Brinton RE, Gee KW, Yamamura HI. CL 218872, PK 8165 and PK 9084: Selective anxiolytics that may act as partial agonist at the benzodiazepine receptor Federation Proceedings. 42. |
0.318 |
|
1982 |
Gee KW, Yamamura HI. Regional heterogeneity of benzodiazepine receptors at 37°C: An in vitro study in various regions of the rat brain Life Sciences. 31: 1939-1945. PMID 6294423 DOI: 10.1016/0024-3205(82)90032-7 |
0.423 |
|
1982 |
Gee KW, Yamamura HI. Differentiation of benzodiazepine receptor agonist and antagonist: Sparing of [3H]benzodiazepine antagonist binding following the photolabelling of benzodiazepine receptors European Journal of Pharmacology. 82: 239-241. PMID 6290239 DOI: 10.1016/0014-2999(82)90521-0 |
0.432 |
|
1982 |
Gee KW, Ehlert FJ, Yamamura HI. The influence of temperature and gamma-aminobutyric acid on benzodiazepine receptor subtypes in the hippocampus of the rat Biochemical and Biophysical Research Communications. 106: 1134-1140. PMID 6288041 DOI: 10.1016/0006-291X(82)91230-X |
0.405 |
|
1982 |
Morelli M, Gee KW, Yamamura HI. The effect of GABA on in vitro binding of two novel non-benzodiazepines, PK 8165 and CGS 8216, to benzodiazepine receptors in the rat brain Life Sciences. 31: 77-81. PMID 6287150 DOI: 10.1016/0024-3205(82)90403-9 |
0.454 |
|
1982 |
Gee KW, Yamamura HI. A novel pyrazoloquinoline that interacts with brain benzodiazepine receptors: Characterization of some in vitro and in vivo properties of CGS 9896 Life Sciences. 30: 2245-2252. PMID 6287145 DOI: 10.1016/0024-3205(82)90251-X |
0.439 |
|
1982 |
Mosberg HI, Hurst R, Hruby VJ, Galligan JJ, Burks TF, Gee K, Yamamura HI. [D-Pen2, L-Cys5]enkephalinamide and[D-Pen2, D-Cys5] enkephalinamide, conformationally constrained cyclic enkephalinamide analogs with delta receptor specificity. Biochemical and Biophysical Research Communications. 106: 506-12. PMID 6285922 DOI: 10.1016/0006-291X(82)91139-1 |
0.322 |
|
1982 |
Gee KW, Morelli M, Yamamura HI. The effect of temperature on CL 218872 and propyl beta-carboline-3-carboxylate inhibition of [3H]-flunitrazepam binding in rat brain Biochemical and Biophysical Research Communications. 105: 1532-1537. PMID 6125147 DOI: 10.1016/0006-291X(82)90962-7 |
0.397 |
|
1982 |
Gee KW, Horst WD, O'Brien R, Yamamura HI. High affinity inhibition of [3H]-Flunitrazepam binding to brain benzodiazepine receptors by CGS 9896, a novel pyrazoloquinoline Biochemical and Biophysical Research Communications. 105: 457-461. PMID 6124246 DOI: 10.1016/0006-291X(82)91456-5 |
0.338 |
|
1981 |
Gee KW, Hollinger MA, Killam EK. Effect of seizures kindled by subconvulsant doses of pentylenetetrazol on dopamine receptor binding and dopamine-sensitive adenylate cyclase in the rat. Experimental Neurology. 74: 265-75. PMID 6269870 DOI: 10.1016/0014-4886(81)90164-3 |
0.677 |
|
1981 |
Gee KW, Killam EK, Hollinger MA. The relationship of dopamine receptors to seizure development: Effects of haloperidol-induced supersensitivity Epilepsia. 22: 227. |
0.635 |
|
1980 |
Gee KW, Killam EK, Hollinger MA, Giri SN. Effect of anygdaloid kindling on dopamine-sensitive adenylate cyclase activity in rat brain. Experimental Neurology. 70: 192-9. PMID 7418769 DOI: 10.1016/0014-4886(80)90018-7 |
0.638 |
|
1980 |
Gee KW, Killam EK, Hollinger MA. The effects of chronic pentylenetetrazol on dopamine receptor binding in the rat brain Federation Proceedings. 39: 3895. |
0.657 |
|
1980 |
Gee KW, Killam EK, Hollinger MA, Giri SN. Alterations in dopamine-sensitive adenylate cyclase in the rat brain following amygdaloid kindling Pharmacologist. 22: No. 759. |
0.608 |
|
1979 |
Gee KW, Hollinger MA, Bowyer JF, Killam EK. Modification of dopaminergic receptor sensitivity in rat brain after amygdaloid kindling. Experimental Neurology. 66: 771-7. PMID 488251 DOI: 10.1016/0014-4886(79)90220-6 |
0.695 |
|
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