Micha Fridman - Publications

Affiliations: 
Tel Aviv University, Tel Aviv-Yafo, Tel Aviv District, Israel 

51 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2023 Haldar J, Garneau-Tsodikova S, Fridman M. Introduction to the themed collection on antimicrobial resistance. Rsc Medicinal Chemistry. 14: 1398-1399. PMID 37593571 DOI: 10.1039/d3md90016a  0.544
2022 Elias R, Basu P, Fridman M. Fluconazole-COX Inhibitor Hybrids: A Dual-Acting Class of Antifungal Azoles. Journal of Medicinal Chemistry. PMID 35084852 DOI: 10.1021/acs.jmedchem.1c01807  0.584
2020 Jaber QZ, Bibi M, Ksiezopolska E, Gabaldon T, Berman J, Fridman M. Elevated Vacuolar Uptake of Fluorescently Labeled Antifungal Drug Caspofungin Predicts Echinocandin Resistance in Pathogenic Yeast. Acs Central Science. 6: 1698-1712. PMID 33145409 DOI: 10.1021/Acscentsci.0C00813  0.337
2020 Jospe-Kaufman M, Siomin L, Fridman M. The relationship between the structure and toxicity of aminoglycoside antibiotics. Bioorganic & Medicinal Chemistry Letters. 127218. PMID 32360102 DOI: 10.1016/J.Bmcl.2020.127218  0.355
2020 Kovalerchik D, Singh RP, Schlesinger P, Mahajni A, Shefer S, Fridman M, Ilan M, Carmeli S. Bromopyrrole Alkaloids of the Sponge Collected Near the Israeli Mediterranean Coastline. Journal of Natural Products. PMID 32072810 DOI: 10.1021/Acs.Jnatprod.9B00863  0.343
2020 Zada SL, Baruch BB, Simhaev L, Engel H, Fridman M. Chemical Modifications Reduce Auditory Cell Damage Induced by Aminoglycoside Antibiotics. Journal of the American Chemical Society. PMID 31958945 DOI: 10.1021/Jacs.9B12420  0.345
2019 Elias R, Benhamou RI, Jaber QZ, Dorot O, Zada SL, Oved K, Pichinuk E, Fridman M. Antifungal activity, mode of action variability, and subcellular distribution of coumarin-based antifungal azoles. European Journal of Medicinal Chemistry. 179: 779-790. PMID 31288127 DOI: 10.1016/J.Ejmech.2019.07.003  0.372
2019 Fridman M, Louzoun Zada S, Jaber QZ. Guiding Drugs to Target- Harboring Organelles: Stretching Drug-Delivery to a Higher Level of Resolution. Angewandte Chemie (International Ed. in English). PMID 31237741 DOI: 10.1002/Anie.201906284  0.309
2018 Benhamou RI, Jaber QZ, Herzog IM, Roichman Y, Fridman M. Fluorescent Tracking of the Endoplasmic Reticulum in Live Pathogenic Fungal Cells. Acs Chemical Biology. PMID 30427174 DOI: 10.1021/Acschembio.8B00782  0.306
2018 Fridman M, Jaber QZ, Benhamou R, Herzog IM, Ben Baruch B. Cationic Amphiphiles Induce Macromolecule Denaturation and Organelle Decomposition in Pathogenic Yeast. Angewandte Chemie (International Ed. in English). PMID 30307679 DOI: 10.1002/Anie.201809410  0.336
2018 Louzoun Zada S, Green KD, Shrestha SK, Herzog IM, Garneau-Tsodikova S, Fridman M. Derivatives of Ribosome-Inhibiting Antibiotic Chloramphenicol Inhibit the Biosynthesis of Bacterial Cell Wall. Acs Infectious Diseases. PMID 29714997 DOI: 10.1021/Acsinfecdis.8B00078  0.609
2018 Kim D, Liu Y, Benhamou RI, Sanchez H, Simón-Soro Á, Li Y, Hwang G, Fridman M, Andes DR, Koo H. Bacterial-derived exopolysaccharides enhance antifungal drug tolerance in a cross-kingdom oral biofilm. The Isme Journal. PMID 29670217 DOI: 10.1038/S41396-018-0113-1  0.391
2018 Fridman M, Benhamou RI, Bibi M, Berman J. Localizing Antifungal Drugs to the Correct Organelle can Markedly Enhance their Efficacy. Angewandte Chemie (International Ed. in English). PMID 29575397 DOI: 10.1002/Anie.201802509  0.337
2018 Steinbuch KB, Benhamou RI, Levin L, Stein R, Fridman M. Increased Degree of Unsaturation in the Lipid of Antifungal Cationic Amphiphiles Facilitates Selective Fungal Cell Disruption. Acs Infectious Diseases. PMID 29419285 DOI: 10.1021/Acsinfecdis.7B00272  0.358
2017 Matzov D, Eyal Z, Benhamou RI, Shalev-Benami M, Halfon Y, Krupkin M, Zimmerman E, Rozenberg H, Bashan A, Fridman M, Yonath A. Structural insights of lincosamides targeting the ribosome of Staphylococcus aureus. Nucleic Acids Research. 45: 10284-10292. PMID 28973455 DOI: 10.1093/Nar/Gkx658  0.741
2017 Fridman M, Salta J, Benhamou RI, Herzog IM. Tuning the Effects of Bacterial Membrane Permeability through Photo-Isomerization of Antimicrobial Cationic Amphiphiles. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28727190 DOI: 10.1002/Chem.201703010  0.341
2017 Benhamou RI, Bibi M, Steinbuch KB, Engel H, Levin M, Roichman Y, Berman J, Fridman M. Real-Time Imaging of the Azole-Class of Antifungal Drugs in Live Candida Cells. Acs Chemical Biology. PMID 28472585 DOI: 10.1021/Acschembio.7B00339  0.318
2017 Neto CC, Penndorf KA, Feldman M, Meron-Sudai S, Zakay-Rones Z, Steinberg D, Fridman M, Kashman Y, Ginsburg I, Ofek I, Weiss EI. Characterization of non-dialyzable constituents from cranberry juice that inhibit adhesion, co-aggregation and biofilm formation by oral bacteria. Food & Function. PMID 28470309 DOI: 10.1039/C7Fo00109F  0.347
2017 Fridman M. Catalyst: The Role of Chemistry in Delivering the Next Antimicrobial Drugs Chem. 3: 8-10. DOI: 10.1016/J.Chempr.2017.06.004  0.326
2016 Herzog IM, Louzoun Zada S, Fridman M. Effects of 5-O-Ribosylation of Aminoglycosides on Antimicrobial Activity and Selective Perturbation of Bacterial Translation. Journal of Medicinal Chemistry. PMID 27509271 DOI: 10.1021/Acs.Jmedchem.6B00793  0.359
2016 Joseph R, Kaizerman D, Herzog IM, Hadar M, Feldman M, Fridman M, Cohen Y. Phosphonium pillar[5]arenes as a new class of efficient biofilm inhibitors: importance of charge cooperativity and the pillar platform. Chemical Communications (Cambridge, England). PMID 27503150 DOI: 10.1039/C6Cc05170G  0.354
2016 Fridman M, Benhamou RI, Steinbuch KB. Antifungal Imidazole-Decorated Cationic Amphiphiles with Markedly Low Hemolytic Activity. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27258738 DOI: 10.1002/Chem.201602198  0.365
2016 Shaul P, Benhamou RI, Herzog IM, Louzoun Zada S, Ebenstein Y, Fridman M. Synthesis and evaluation of membrane permeabilizing properties of cationic amphiphiles derived from the disaccharide trehalose. Organic & Biomolecular Chemistry. 14: 3012-5. PMID 26832956 DOI: 10.1039/C6Ob00031B  0.387
2016 Joseph R, Naugolny A, Feldman M, Herzog IM, Fridman M, Cohen Y. Cationic Pillararenes Potently Inhibit Biofilm Formation without Affecting Bacterial Growth and Viability. Journal of the American Chemical Society. PMID 26745311 DOI: 10.1021/Jacs.5B11834  0.382
2016 Steinbuch KB, Fridman M. Mechanisms of resistance to membrane-disrupting antibiotics in Gram-positive and Gram-negative bacteria Medchemcomm. 7: 86-102. DOI: 10.1039/C5Md00389J  0.422
2015 Benhamou RI, Shaul P, Herzog IM, Fridman M. Di-N-Methylation of Anti-Gram-Positive Aminoglycoside-Derived Membrane Disruptors Improves Antimicrobial Potency and Broadens Spectrum to Gram-Negative Bacteria. Angewandte Chemie (International Ed. in English). 54: 13617-21. PMID 26418734 DOI: 10.1002/Anie.201506814  0.396
2015 Shaul P, Steinbuch KB, Blacher E, Stein R, Fridman M. Exploring the Effects of Glycosylation and Etherification of the Side Chains of the Anticancer Drug Mitoxantrone. Chemmedchem. 10: 1528-38. PMID 26235383 DOI: 10.1002/Cmdc.201500274  0.304
2015 Berkov-Zrihen Y, Herzog IM, Benhamou RI, Feldman M, Steinbuch KB, Shaul P, Lerer S, Eldar A, Fridman M. Tobramycin and nebramine as pseudo-oligosaccharide scaffolds for the development of antimicrobial cationic amphiphiles. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 4340-9. PMID 25652188 DOI: 10.1002/Chem.201406404  0.424
2015 Gajadeera C, Willby MJ, Green KD, Shaul P, Fridman M, Garneau-Tsodikova S, Posey JE, Tsodikov OV. Antimycobacterial activity of DNA intercalator inhibitors of Mycobacterium tuberculosis primase DnaG. The Journal of Antibiotics. 68: 153-7. PMID 25248725 DOI: 10.1038/Ja.2014.131  0.605
2015 Blacher E, Ben Baruch B, Levy A, Geva N, Green KD, Garneau-Tsodikova S, Fridman M, Stein R. Inhibition of glioma progression by a newly discovered CD38 inhibitor. International Journal of Cancer. Journal International Du Cancer. 136: 1422-33. PMID 25053177 DOI: 10.1002/Ijc.29095  0.527
2015 Blacher E, Levy A, Baruch BB, Green KD, Garneau-Tsodikova S, Fridman M, Stein R. Targeting CD38 in the tumor microenvironment: A novel approach to treat glioma Cancer Cell & Microenvironment. 2. DOI: 10.14800/Ccm.486  0.522
2015 Baasov T, Fridman M, Werz DB. Carbohydrates: Special issue in honor of the 2014 wolf prize laureate in chemistry, professor Chi-Huey Wong Israel Journal of Chemistry. 55: 253. DOI: 10.1002/Ijch.201510003  0.511
2014 Baasov T, Fridman M. Foreword-The 17th European Carbohydrate Symposium-EuroCarb17. Carbohydrate Research. 389: 1. PMID 24726717 DOI: 10.1016/J.Carres.2014.03.013  0.495
2014 Herzog IM, Fridman M. Design and synthesis of membrane-targeting antibiotics: From peptides- to aminosugar-based antimicrobial cationic amphiphiles Medchemcomm. 5: 1014-1026. DOI: 10.1039/C4Md00012A  0.426
2013 Shaul P, Frenkel M, Goldstein EB, Mittelman L, Grunwald A, Ebenstein Y, Tsarfaty I, Fridman M. The structure of anthracycline derivatives determines their subcellular localization and cytotoxic activity. Acs Medicinal Chemistry Letters. 4: 323-8. PMID 24900668 DOI: 10.1021/Ml3002852  0.328
2013 Berkov-Zrihen Y, Green KD, Labby KJ, Feldman M, Garneau-Tsodikova S, Fridman M. Synthesis and evaluation of hetero- and homodimers of ribosome-targeting antibiotics: antimicrobial activity, in vitro inhibition of translation, and drug resistance. Journal of Medicinal Chemistry. 56: 5613-25. PMID 23786357 DOI: 10.1021/Jm400707F  0.644
2013 Berkov-Zrihen Y, Herzog IM, Feldman M, Sonn-Segev A, Roichman Y, Fridman M. Di-alkylated paromomycin derivatives: targeting the membranes of gram positive pathogens that cause skin infections. Bioorganic & Medicinal Chemistry. 21: 3624-31. PMID 23602621 DOI: 10.1016/J.Bmc.2013.03.046  0.382
2013 Herzog IM, Feldman M, Eldar-Boock A, Satchi-Fainaro R, Fridman M. Design of membrane targeting tobramycin-based cationic amphiphiles with reduced hemolytic activity Medchemcomm. 4: 120-124. DOI: 10.1039/C2Md20162C  0.391
2012 Herzog IM, Green KD, Berkov-Zrihen Y, Feldman M, Vidavski RR, Eldar-Boock A, Satchi-Fainaro R, Eldar A, Garneau-Tsodikova S, Fridman M. 6''-Thioether tobramycin analogues: towards selective targeting of bacterial membranes. Angewandte Chemie (International Ed. in English). 51: 5652-6. PMID 22499286 DOI: 10.1002/Anie.201200761  0.59
2012 Herzog IM, Green KD, Berkov‐Zrihen Y, Feldman M, Vidavski RR, Eldar‐Boock A, Satchi‐Fainaro R, Eldar A, Garneau‐Tsodikova S, Fridman M. Inside Cover: 6′′‐Thioether Tobramycin Analogues: Towards Selective Targeting of Bacterial Membranes (Angew. Chem. Int. Ed. 23/2012) Angewandte Chemie. 51: 5508-5508. DOI: 10.1002/Anie.201203240  0.339
2012 Herzog IM, Green KD, Berkov-Zrihen Y, Feldman M, Vidavski RR, Eldar-Boock A, Satchi-Fainaro R, Eldar A, Garneau-Tsodikova S, Fridman M. Innentitelbild: 6′′-Thioether Tobramycin Analogues: Towards Selective Targeting of Bacterial Membranes (Angew. Chem. 23/2012) Angewandte Chemie. 124: 5602-5602. DOI: 10.1002/Ange.201203240  0.569
2011 Breiner-Goldstein E, Evron Z, Frenkel M, Cohen K, Meiron KN, Peer D, Roichman Y, Flescher E, Fridman M. Targeting anthracycline-resistant tumor cells with synthetic aloe-emodin glycosides. Acs Medicinal Chemistry Letters. 2: 528-31. PMID 24900344 DOI: 10.1021/Ml2001104  0.349
2011 Shaul P, Green KD, Rutenberg R, Kramer M, Berkov-Zrihen Y, Breiner-Goldstein E, Garneau-Tsodikova S, Fridman M. Assessment of 6'- and 6'''-N-acylation of aminoglycosides as a strategy to overcome bacterial resistance. Organic & Biomolecular Chemistry. 9: 4057-63. PMID 21365081 DOI: 10.1039/C0Ob01133A  0.613
2010 Green KD, Chen W, Houghton JL, Fridman M, Garneau-Tsodikova S. Exploring the substrate promiscuity of drug-modifying enzymes for the chemoenzymatic generation of N-acylated aminoglycosides. Chembiochem : a European Journal of Chemical Biology. 11: 119-26. PMID 19899089 DOI: 10.1002/Cbic.200900584  0.593
2009 Green KD, Fridman M, Garneau-Tsodikova S. hChAT: a tool for the chemoenzymatic generation of potential acetyl/butyrylcholinesterase inhibitors. Chembiochem : a European Journal of Chemical Biology. 10: 2191-4. PMID 19637146 DOI: 10.1002/Cbic.200900309  0.522
2007 Fridman M, Balibar CJ, Lupoli T, Kahne D, Walsh CT, Garneau-Tsodikova S. Chemoenzymatic formation of novel aminocoumarin antibiotics by the enzymes CouN1 and CouN7. Biochemistry. 46: 8462-71. PMID 17580964 DOI: 10.1021/Bi700433V  0.592
2005 Hainrichson M, Pokrovskaya V, Shallom-Shezifi D, Fridman M, Belakhov V, Shachar D, Yaron S, Baasov T. Branched aminoglycosides: biochemical studies and antibacterial activity of neomycin B derivatives. Bioorganic & Medicinal Chemistry. 13: 5797-807. PMID 15993084 DOI: 10.1016/J.Bmc.2005.05.058  0.608
2005 Fridman M, Belakhov V, Lee LV, Liang FS, Wong CH, Baasov T. Dual effect of synthetic aminoglycosides: antibacterial activity against Bacillus anthracis and inhibition of anthrax lethal factor. Angewandte Chemie (International Ed. in English). 44: 447-52. PMID 15624157 DOI: 10.1002/Anie.200462003  0.596
2003 Fridman M, Belakhov V, Yaron S, Baasov T. A new class of branched aminoglycosides: pseudo-pentasaccharide derivatives of neomycin B. Organic Letters. 5: 3575-8. PMID 14507176 DOI: 10.1021/Ol035213I  0.609
2002 Fridman M, Solomon D, Yogev S, Baasov T. One-pot synthesis of glucosamine oligosaccharides. Organic Letters. 4: 281-3. PMID 11796070 DOI: 10.1021/Ol017054D  0.545
2001 Solomon D, Fridman M, Zhang J, Baasov T. A synthetic pentasaccharide with GTPase activity Organic Letters. 3: 4311-4314. PMID 11784205 DOI: 10.1021/Ol010257H  0.553
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