Phillip R. Lazzara - Publications

Affiliations: 
2012- Loyola University Chicago, Chicago, IL, United States 

8 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2021 Zink KE, Ludvik DA, Lazzara PR, Moore TW, Mandel MJ, Sanchez LM. A Small Molecule Coordinates Symbiotic Behaviors in a Host Organ. Mbio. 12. PMID 33688014 DOI: 10.1128/mBio.03637-20  0.429
2020 Lazzara PR, Moore TW. Scaffold-hopping as a strategy to address metabolic liabilities of aromatic compounds. Rsc Medicinal Chemistry. 11: 18-29. PMID 33479602 DOI: 10.1039/c9md00396g  0.537
2020 Lazzara PR, Jain AD, Maldonado AC, Richardson B, Skowron KJ, David BP, Siddiqui Z, Ratia KM, Moore TW. Synthesis and Evaluation of Noncovalent Naphthalene-Based KEAP1-NRF2 Inhibitors. Acs Medicinal Chemistry Letters. 11: 521-527. PMID 32292559 DOI: 10.1021/Acsmedchemlett.9B00631  0.64
2020 Lazzara PR, Moore TW. Scaffold-hopping as a strategy to address metabolic liabilities of aromatic compounds Rsc Medicinal Chemistry. 11: 18-29. DOI: 10.1039/c9md00396g  0.523
2019 Lazzara PR, David BP, Ankireddy A, Richardson B, Dye K, Ratia KM, Reddy SP, Moore TW. Isoquinoline Kelch-like ECH-Associated Protein 1-Nuclear Factor (Erythroid-derived 2)-like 2 (KEAP1-NRF2) Inhibitors with High Metabolic Stability. Journal of Medicinal Chemistry. PMID 31682434 DOI: 10.1021/Acs.Jmedchem.9B01074  0.682
2019 Skowron KJ, Booker K, Cheng C, Creed S, David BP, Lazzara PR, Lian A, Siddiqui Z, Speltz TE, Moore TW. Steroid receptor/coactivator binding inhibitors: An update. Molecular and Cellular Endocrinology. 110471. PMID 31163202 DOI: 10.1016/J.Mce.2019.110471  0.627
2018 Richardson B, Jain AD, Potteti H, Lazzara PR, David BP, Tamatam C, Choma E, Skowron K, Dye K, Siddiqui Z, Wang YT, Krunic A, Reddy S, Moore TW. Replacement of a Naphthalene Scaffold in Kelch-like ECH-Associated Protein 1 (KEAP1)/Nuclear factor (erythroid-derived 2)-like 2 (NRF2)Inhibitors. Journal of Medicinal Chemistry. PMID 30122040 DOI: 10.1021/Acs.Jmedchem.8B01133  0.656
2016 Lazzara PR, Fitzpatrick KP, Eichman CC. Pd-Catalyzed Carboamination of Alkylidenecyclopropanes: Synthesis of Congested Pyrrolidines and Piperidines. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27661456 DOI: 10.1002/Chem.201604077  0.685
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