Year |
Citation |
Score |
2021 |
Zink KE, Ludvik DA, Lazzara PR, Moore TW, Mandel MJ, Sanchez LM. A Small Molecule Coordinates Symbiotic Behaviors in a Host Organ. Mbio. 12. PMID 33688014 DOI: 10.1128/mBio.03637-20 |
0.429 |
|
2020 |
Lazzara PR, Moore TW. Scaffold-hopping as a strategy to address metabolic liabilities of aromatic compounds. Rsc Medicinal Chemistry. 11: 18-29. PMID 33479602 DOI: 10.1039/c9md00396g |
0.537 |
|
2020 |
Lazzara PR, Jain AD, Maldonado AC, Richardson B, Skowron KJ, David BP, Siddiqui Z, Ratia KM, Moore TW. Synthesis and Evaluation of Noncovalent Naphthalene-Based KEAP1-NRF2 Inhibitors. Acs Medicinal Chemistry Letters. 11: 521-527. PMID 32292559 DOI: 10.1021/Acsmedchemlett.9B00631 |
0.64 |
|
2020 |
Lazzara PR, Moore TW. Scaffold-hopping as a strategy to address metabolic liabilities of aromatic compounds Rsc Medicinal Chemistry. 11: 18-29. DOI: 10.1039/c9md00396g |
0.523 |
|
2019 |
Lazzara PR, David BP, Ankireddy A, Richardson B, Dye K, Ratia KM, Reddy SP, Moore TW. Isoquinoline Kelch-like ECH-Associated Protein 1-Nuclear Factor (Erythroid-derived 2)-like 2 (KEAP1-NRF2) Inhibitors with High Metabolic Stability. Journal of Medicinal Chemistry. PMID 31682434 DOI: 10.1021/Acs.Jmedchem.9B01074 |
0.682 |
|
2019 |
Skowron KJ, Booker K, Cheng C, Creed S, David BP, Lazzara PR, Lian A, Siddiqui Z, Speltz TE, Moore TW. Steroid receptor/coactivator binding inhibitors: An update. Molecular and Cellular Endocrinology. 110471. PMID 31163202 DOI: 10.1016/J.Mce.2019.110471 |
0.627 |
|
2018 |
Richardson B, Jain AD, Potteti H, Lazzara PR, David BP, Tamatam C, Choma E, Skowron K, Dye K, Siddiqui Z, Wang YT, Krunic A, Reddy S, Moore TW. Replacement of a Naphthalene Scaffold in Kelch-like ECH-Associated Protein 1 (KEAP1)/Nuclear factor (erythroid-derived 2)-like 2 (NRF2)Inhibitors. Journal of Medicinal Chemistry. PMID 30122040 DOI: 10.1021/Acs.Jmedchem.8B01133 |
0.656 |
|
2016 |
Lazzara PR, Fitzpatrick KP, Eichman CC. Pd-Catalyzed Carboamination of Alkylidenecyclopropanes: Synthesis of Congested Pyrrolidines and Piperidines. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27661456 DOI: 10.1002/Chem.201604077 |
0.685 |
|
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