Ari M.P. Koskinen, Ph.D. - Publications

Chemistry Aalto University, Espoo, Finland 
organic synthesis, natural products, chemical biology

165 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2019 Konstantinova OV, Koskinen AMP. Synthesis of the C1-C12 Fragment of Calyculin C Synthesis. 51: 285-295. DOI: 10.1055/S-0037-1610387  0.64
2015 Van Adrichem AJ, Fagerholm A, Turunen L, Lehto A, Saarela J, Koskinen A, Repasky GA, Wennerberg K. Discovery of MINC1, a GTPase-activating protein small molecule inhibitor, targeting MgcRacGAP Combinatorial Chemistry and High Throughput Screening. 18: 3-17. DOI: 10.2174/1386207318666141205112730  1
2015 Rembiak A, Koskinen AMP. Versatile Synthesis of Symmetrical Carbazole Based Ligand Precursors via Regioselective Aromatic Bromination Synthesis. 47: 3347-3353. DOI: 10.1055/S-0034-1378825  0.64
2015 Sundqvist T, Oasmaa A, Koskinen A. Upgrading fast pyrolysis bio-oil quality by esterification and azeotropic water removal Energy and Fuels. 29: 2527-2534. DOI: 10.1021/Acs.Energyfuels.5B00238  1
2015 Lood CS, Nieger M, Koskinen AMP. Enantiospecific gram scale synthesis of (S)-eleagnine Tetrahedron. 71: 5019-5024. DOI: 10.1016/J.Tet.2015.05.063  1
2015 Lood CS, Laine AE, Högnäsbacka A, Nieger M, Koskinen AMP. Synthesis of chiral (indol-2-yl)methanamines and insight into the stereochemistry protecting effects of the 9-phenyl-9-fluorenyl protecting group European Journal of Organic Chemistry. 2015: 3793-3805. DOI: 10.1002/Ejoc.201500391  1
2015 Ihanainen NE, Kumpulainen ETT, Koskinen AMP. Palladium-catalyzed direct C-H arylation of dicyanobenzenes European Journal of Organic Chemistry. 2015: 3226-3229. DOI: 10.1002/Ejoc.201500288  0.04
2015 Koskinen AMP, Kataja AO. The Tishchenko Reaction Organic Reactions. 105-410. DOI: 10.1002/0471264180.Or086.02  1
2014 Huy PH, Westphal JC, Koskinen AM. Concise, stereodivergent and highly stereoselective synthesis of cis- and trans-2-substituted 3-hydroxypiperidines - development of a phosphite-driven cyclodehydration. Beilstein Journal of Organic Chemistry. 10: 369-83. PMID 24605158 DOI: 10.3762/Bjoc.10.35  1
2014 Laine AE, Lood C, Koskinen AM. Pharmacological importance of optically active tetrahydro-β-carbolines and synthetic approaches to create the C1 stereocenter. Molecules (Basel, Switzerland). 19: 1544-67. PMID 24473212 DOI: 10.3390/Molecules19021544  1
2014 Koskinen AM. Boron enolate chemistry toward the syntheses of polyketide stereotetrads. Chemical Record (New York, N.Y.). 14: 52-61. PMID 24420331 DOI: 10.1002/Tcr.201300033  0.01
2014 Karjalainen OK, Koskinen AMP. Scalable synthesis of (-)-trans-3-hydroxypipecolic acid via a useful chiral building block Tetrahedron. 70: 2444-2448. DOI: 10.1016/J.Tet.2014.02.020  1
2014 Lood CS, Koskinen AMP. Harmicine, a Tetracyclic Tetrahydro-β-Carboline: From the First Synthetic Precedent to Isolation from Natural Sources to Target-Oriented Synthesis (Review)* Chemistry of Heterocyclic Compounds. DOI: 10.1007/S10593-014-1602-4  1
2014 Lood CS, Koskinen AMP. Synthesis of (S)- and (R)-harmicine from proline: An approach toward tetrahydro-β-carbolines European Journal of Organic Chemistry. 2014: 2357-2364. DOI: 10.1002/Ejoc.201301903  1
2013 Passiniemi M, Koskinen AM. Garner's aldehyde as a versatile intermediate in the synthesis of enantiopure natural products. Beilstein Journal of Organic Chemistry. 9: 2641-59. PMID 24367429 DOI: 10.3762/Bjoc.9.300  1
2013 Huy PH, Koskinen AM. Efficient, stereodivergent access to 3-piperidinols by traceless P(OEt)3 cyclodehydration. Organic Letters. 15: 5178-81. PMID 24090120 DOI: 10.1021/Ol4026588  1
2013 Karjalainen OK, Nieger M, Koskinen AM. Diastereoselective intramolecular allyl transfer from allyl carbamate accompanied by 5-endo-trig ring closure. Angewandte Chemie (International Ed. in English). 52: 2551-4. PMID 23341176 DOI: 10.1002/Anie.201209443  1
2013 Pelss A, Koskinen AMP. Stereocontrolled construction of decahydro quinoline ring systems: The case of lepadin alkaloids (Review) Chemistry of Heterocyclic Compounds. 49: 226-240. DOI: 10.1007/S10593-013-1239-8  1
2012 Karjalainen OK, Koskinen AM. Diastereoselective synthesis of vicinal amino alcohols. Organic & Biomolecular Chemistry. 10: 4311-26. PMID 22535485 DOI: 10.1039/C2Ob25357G  1
2012 Koskinen AMP. Asymmetric Synthesis of Natural Products Asymmetric Synthesis of Natural Products. DOI: 10.1002/9781118347300  0.01
2011 Passiniemi M, Koskinen AM. Asymmetric synthesis of Pachastrissamine (Jaspine B) and its diastereomers via η3-allylpalladium intermediates. Organic & Biomolecular Chemistry. 9: 1774-83. PMID 21264408 DOI: 10.1039/C0Ob00643B  1
2011 Karjalainen OK, Koskinen AM. Rapid and practical synthesis of (-)-1-deoxyaltronojirimycin. Organic & Biomolecular Chemistry. 9: 1231-6. PMID 21186396 DOI: 10.1039/C0Ob00747A  1
2011 Passiniemi M, Myllymäki MJ, Vuokko J, Koskinen AMP. Demethylation of aromatic methyl ethers using ionic liquids under microwave irradiation Letters in Organic Chemistry. 8: 48-52. DOI: 10.2174/157017811794557741  1
2011 Koskinen AMP. Chirospecific synthesis: Catalysis and chiral pool hand in hand Pure and Applied Chemistry. 83: 435-443. DOI: 10.1351/Pac-Con-10-10-09  0.01
2011 Passiniemi M, Koskinen AMP. Enantioselective synthesis of Boc-protected norfuranomycins Tetrahedron Letters. 52: 6736-6738. DOI: 10.1016/J.Tetlet.2011.10.007  1
2010 Karppanen EJ, Koskinen AM. The 9-phenyl-9-fluorenyl group for nitrogen protection in enantiospecific synthesis. Molecules (Basel, Switzerland). 15: 6512-47. PMID 20877241 DOI: 10.3390/Molecules15096512  0.01
2010 Habrant D, Koskinen AM. Towards the total synthesis of calyculin C: preparation of the C(9)-C(25) spiroketal-dipropionate unit. Organic & Biomolecular Chemistry. 8: 4364-73. PMID 20683542 DOI: 10.1039/C0Ob00092B  1
2010 Habrant D, Rauhala V, Koskinen AM. Conversion of carbonyl compounds to alkynes: general overview and recent developments. Chemical Society Reviews. 39: 2007-17. PMID 20502799 DOI: 10.1039/B915418C  1
2010 Koivisto JJ, Kumpulainen ET, Koskinen AM. Conformational ensembles of flexible beta-turn mimetics in DMSO-d6. Organic & Biomolecular Chemistry. 8: 2103-16. PMID 20401387 DOI: 10.1039/B921794K  1
2010 Karjalainen OK, Passiniemi M, Koskinen AM. Short and straightforward synthesis of (-)-1-deoxygalactonojirimycin. Organic Letters. 12: 1145-7. PMID 20170191 DOI: 10.1021/Ol100037C  1
2010 Fagerholm AE, Habrant D, Koskinen AM. Calyculins and related marine natural products as serine-threonine protein phosphatase PP1 and PP2A inhibitors and total syntheses of calyculin A, B, and C. Marine Drugs. 8: 122-72. PMID 20161975 DOI: 10.3390/Md80100122  1
2010 Käsnänen H, Myllymäki MJ, Minkkilä A, Kataja AO, Saario SM, Nevalainen T, Koskinen AM, Poso A. 3-Heterocycle-phenyl N-alkylcarbamates as FAAH inhibitors: design, synthesis and 3D-QSAR studies. Chemmedchem. 5: 213-31. PMID 20024981 DOI: 10.1002/Cmdc.200900390  1
2010 Kataja AO, Koskinen AMP. Asymmetric organocatalytic Michael addition of Meldrum's acid to nitroalkenes: Probing the mechanism of bifunctional thiourea organocatalysts Arkivoc. 2010: 205-223. DOI: 10.3998/Ark.5550190.0011.216  1
2010 Sauerland SJK, Castillo-Meléndez JA, Nättinen K, Rissanen K, Koskinen AMP. Enantioselective synthesis of homosphingosine derivatives from L-aspartic acid Synthesis. 757-762. DOI: 10.1055/S-0029-1219081  1
2010 Passiniemi M, Koskinen AMP. A short and efficient synthesis of (2S,3S,4S)-tert-butyl 3,4-dihydroxy-2-(methoxymethyl)-5-oxopyrrolidine-1-carboxylate Synthesis. 2816-2822. DOI: 10.1055/S-0029-1218843  1
2009 Kumpulainen ET, Koskinen AM. Catalytic activity dependency on catalyst components in aerobic copper-TEMPO oxidation. Chemistry (Weinheim An Der Bergstrasse, Germany). 15: 10901-11. PMID 19746477 DOI: 10.1002/Chem.200901245  1
2009 Pelss A, Kumpulainen ET, Koskinen AM. Highly chemoselective copper-catalyzed conjugate reduction of stereochemically labile alpha,beta-unsaturated amino ketones. The Journal of Organic Chemistry. 74: 7598-601. PMID 19739611 DOI: 10.1021/Jo9017588  1
2009 Myllymäki MJ, Käsnänen H, Kataja AO, Lahtela-Kakkonen M, Saario SM, Poso A, Koskinen AM. Chiral 3-(4,5-dihydrooxazol-2-yl)phenyl alkylcarbamates as novel FAAH inhibitors: Insight into FAAH enantioselectivity by molecular docking and interaction fields. European Journal of Medicinal Chemistry. 44: 4179-91. PMID 19539407 DOI: 10.1016/J.Ejmech.2009.05.012  1
2009 Reux B, Nevalainen T, Raitio KH, Koskinen AM. Synthesis of quinolinyl and isoquinolinyl phenyl ketones as novel agonists for the cannabinoid CB2 receptor. Bioorganic & Medicinal Chemistry. 17: 4441-7. PMID 19477133 DOI: 10.1016/J.Bmc.2009.05.013  1
2009 Minkkilä A, Myllymäki MJ, Saario SM, Castillo-Melendez JA, Koskinen AM, Fowler CJ, Leppänen J, Nevalainen T. The synthesis and biological evaluation of para-substituted phenolic N-alkyl carbamates as endocannabinoid hydrolyzing enzyme inhibitors. European Journal of Medicinal Chemistry. 44: 2994-3008. PMID 19232787 DOI: 10.1016/J.Ejmech.2009.01.007  1
2009 Koskinen AMP, Kallatsa OA, Nissinen M. Polyhydroxylated indolizidine alkaloids-synthesis of dideoxycastanospermine Tetrahedron. 65: 9285-9290. DOI: 10.1016/J.Tet.2009.09.017  1
2009 Habrant D, Stewart AJW, Koskinen AMP. Towards the total synthesis of Calyculin C: preparation of the C13-C25 spirocyclic core Tetrahedron. 65: 7927-7934. DOI: 10.1016/J.Tet.2009.07.070  1
2009 Bassas O, Huuskonen J, Rissanen K, Koskinen AMP. A simple organocatalytic enantioselective synthesis of pregabalin European Journal of Organic Chemistry. 1340-1351. DOI: 10.1002/Ejoc.200801220  1
2008 Koskinen AMP, Pihko AJ. Synthesis of DEFG ring system of cneorins Arkivoc. 2008: 20-35. DOI: 10.3998/Ark.5550190.0009.H03  1
2008 Oila MJ, Tois JE, Koskinen AMP. A new application for PyOX-ligands: The asymmetric Henry reaction Letters in Organic Chemistry. 5: 11-16. DOI: 10.2174/157017808783330216  1
2008 Oila MJ, Tois JE, Koskinen AMP. Mild and efficient synthesis of 2-indole-2′-oxazolines at room temperature - A simple access to novel IndOX ligands Synthetic Communications. 38: 361-370. DOI: 10.1080/00397910701767072  1
2008 Passiniemi M, Koskinen AMP. Stereoselective total synthesis of pachastrissamine (jaspine B) Tetrahedron Letters. 49: 980-983. DOI: 10.1016/J.Tetlet.2007.12.014  1
2008 Routasalo T, Helaja J, Kavakka J, Koskinen AMP. Development of bis(2-picolyl)amine-zinc chelates for imidazole receptors European Journal of Organic Chemistry. 3190-3199. DOI: 10.1002/Ejoc.200700926  1
2007 Kumpulainen ET, Koskinen AM, Rissanen K. Total synthesis of amaminol A: establishment of the absolute stereochemistry. Organic Letters. 9: 5043-5. PMID 17956115 DOI: 10.1021/Ol7022856  1
2007 Myllymäki MJ, Saario SM, Kataja AO, Castillo-Melendez JA, Nevalainen T, Juvonen RO, Järvinen T, Koskinen AM. Design, synthesis, and in vitro evaluation of carbamate derivatives of 2-benzoxazolyl- and 2-benzothiazolyl-(3-hydroxyphenyl)-methanones as novel fatty acid amide hydrolase inhibitors. Journal of Medicinal Chemistry. 50: 4236-42. PMID 17665899 DOI: 10.1021/Jm070501W  1
2007 Andberg M, Jäntti J, Heilimo S, Pihkala P, Paananen A, Koskinen AM, Söderlund H, Linder MB. Cleavage of recombinant proteins at poly-His sequences by Co(II) and Cu(II). Protein Science : a Publication of the Protein Society. 16: 1751-61. PMID 17600148 DOI: 10.1110/Ps.072846407  1
2007 Abe AM, Sauerland SJ, Koskinen AM. Highly enantioselective conjugate addition of thiols using mild scandium triflate catalysis. The Journal of Organic Chemistry. 72: 5411-3. PMID 17550292 DOI: 10.1021/Jo070492Z  1
2007 Myllymäki MJ, Koskinen AMP. A rapid method for the preparation of 2-substituted oxazolo[4,5-b]pyridines using microwave-assisted direct condensation reactions Tetrahedron Letters. 48: 2295-2298. DOI: 10.1016/J.Tetlet.2007.01.161  1
2006 Abe AM, Helaja J, Koskinen AM. Novel crown ether and salen metal chelation driven molecular pincers. Organic Letters. 8: 4537-40. PMID 16986944 DOI: 10.1021/Ol061726O  1
2006 Parkkari T, Myllymäki M, Savinainen JR, Saario SM, Castillo-Meléndez JA, Laitinen JT, Nevalainen T, Koskinen AM, Järvinen T. Alpha-methylated derivatives of 2-arachidonoyl glycerol: synthesis, CB1 receptor activity, and enzymatic stability. Bioorganic & Medicinal Chemistry Letters. 16: 2437-40. PMID 16466915 DOI: 10.1016/J.Bmcl.2006.01.101  1
2006 Oila MJ, Koskinen AMP. Chirally modified gold nanoparticles: Nanostructured chiral ligands for catalysis Arkivoc. 2006: 76-83. DOI: 10.3998/Ark.5550190.0007.F10  1
2006 Monfray J, Koskinen AMP. Aza-Michael additons on α,β-unsaturated esters catalysed by bismuth (III) triflate in conventional chemistry and under microwave irradiation Letters in Organic Chemistry. 3: 324-327. DOI: 10.2174/157017806776114496  0.01
2006 Koskinen AMP, Laitinen RS, Oilunkaniemi R, Savilampi SK, Toivola RJ. Methyl 3,3,7,7,9-pentamethyl-1,5-dioxaspiro-[5.5]undec-8-ene-8-carboxylate Acta Crystallographica Section E: Structure Reports Online. 61: o1627-o1628. DOI: 10.1107/S1600536805013127  1
2006 Salo TM, Helaja J, Koskinen AMP. Development of Dpa-based imidazole zinc anion receptors Tetrahedron Letters. 47: 2977-2980. DOI: 10.1016/J.Tetlet.2006.02.105  1
2006 Sauerland SJK, Kiljunen E, Koskinen AMP. Enantioselective Michael additions on α,β-unsaturated N-acylated oxazolidin-2-ones using mild scandium triflate catalysis Tetrahedron Letters. 47: 1291-1293. DOI: 10.1016/J.Tetlet.2005.12.076  1
2006 Straub T, Bitterwolf TE, Weiss CA, Pakkanen TA, Koskinen AMP. Mo-Ru complexes - Highly efficient HDS catalysts: Synthesis, catalytic applications and reactivity studies Acs National Meeting Book of Abstracts. 231.  1
2005 Koskinen AM, Karisalmi K. Polyketide stereotetrads in natural products. Chemical Society Reviews. 34: 677-90. PMID 16186897 DOI: 10.1039/B417466F  1
2005 Koskinen AM, Helaja J, Kumpulainen ET, Koivisto J, Mansikkamäki H, Rissanen K. Locked conformations for proline pyrrolidine ring: synthesis and conformational analysis of cis- and trans-4-tert-butylprolines. The Journal of Organic Chemistry. 70: 6447-53. PMID 16050708 DOI: 10.1021/Jo050838A  1
2005 Straub T, Brunner M, Koskinen AMP. Model studies towards alternative cross-linking of unsaturated polyesters Letters in Organic Chemistry. 2: 74-76. DOI: 10.2174/1570178053399868  1
2005 Tois J, Vahermo M, Koskinen A. Novel and convenient synthesis of 4(1H)quinolones Tetrahedron Letters. 46: 735-737. DOI: 10.1016/J.Tetlet.2004.12.046  1
2005 Oila MJ, Tois JE, Koskinen AMP. Synthesis of a novel carboxy functionalized PyOX-ligand Tetrahedron Letters. 46: 967-969. DOI: 10.1016/J.Tetlet.2004.12.045  1
2005 Oila MJ, Tois JE, Koskinen AMP. Ligand creation via linking - A rapid and convenient method for construction of novel supported PyOX-ligands Tetrahedron. 61: 10748-10756. DOI: 10.1016/J.Tet.2005.08.073  1
2005 Pihko AJ, Koskinen AMP. Synthesis of propellane-containing natural products Tetrahedron. 61: 8769-8807. DOI: 10.1016/J.Tet.2005.06.013  1
2005 Brunner M, Nissinen M, Rissanen K, Straub T, Koskinen AMP. Diastereoselective formation of highly functionalised α-substituted amino acid derivatives via aldol addition Journal of Molecular Structure. 734: 177-182. DOI: 10.1016/J.Molstruc.2004.09.020  1
2005 Straub T, Haukka M, Brunner M, Koskinen AMP, Pakkanen TA. Synthesis and molecular structure of (η5-pentamethyl- cyclopentadienyl) (η5-cyclopentadienyl) hexacarbonyl molybdenum tungsten Journal of Organometallic Chemistry. 690: 674-677. DOI: 10.1016/J.Jorganchem.2004.10.023  1
2005 Rauhala V, Nättinen K, Rissanen K, Koskinen AMP. The reaction mechanism of spirocylization and stereoselectivity studies for the calyculin C 16-C 25 fragment European Journal of Organic Chemistry. 4119-4126. DOI: 10.1002/Ejoc.200500206  1
2005 Selkälä SA, Koskinen AMP. Preparation of bicyclo[4.3.0]nonanes by an organocatalytic intramolecular Diels-Alder reaction European Journal of Organic Chemistry. 1620-1624. DOI: 10.1002/Ejoc.200400802  1
2004 Mäntylä A, Garnier T, Rautio J, Nevalainen T, Vepsälainen J, Koskinen A, Croft SL, Järvinen T. Synthesis, in Vitro Evaluation, and Antileishmanial Activity of Water-Soluble Prodrugs of Buparvaquone Journal of Medicinal Chemistry. 47: 188-195. PMID 14695832 DOI: 10.1021/Jm030868A  1
2004 Koskinen AMP, Brunner M, Straub T, Saarenketo P, Rissanen K. Highly Diastereoselective Methylation of Five-Ring N,O-Acetals Letters in Organic Chemistry. 1: 268-270. DOI: 10.2174/1570178043400929  1
2004 Brunner M, Koskinen AMP. Biology and chemistry of sphingosine-related metabolites Current Organic Chemistry. 8: 1629-1645. DOI: 10.2174/1385272043369638  1
2004 Karisalmi K, Koskinen AMP. Studies towards the synthesis of the C(9)-C(20) lactone-dipropionate fragment of calyculin C Synthesis. 1331-1342. DOI: 10.1055/S-2004-822389  1
2004 Karisalmi K, Koskinen AMP. Stereoselective synthesis of the C 9-C 19 lactone-dipropionate fragment of calyculin C Tetrahedron Letters. 45: 8245-8248. DOI: 10.1016/J.Tetlet.2004.09.012  1
2004 Brunner M, Koskinen AMP. Highly diastereoselective aldol additions to five-ring N,O-acetals Tetrahedron Letters. 45: 3063-3065. DOI: 10.1016/J.Tetlet.2004.02.104  1
2004 Pihko AJ, Lundell K, Kanerva L, Koskinen AMP. Enantioselective synthesis of a hindered furyl substituted allyl alcohol intermediate: A case study in asymmetric synthesis Tetrahedron Asymmetry. 15: 1637-1643. DOI: 10.1016/J.Tetasy.2004.04.004  1
2004 Rauhala V, Nevalainen M, Koskinen AMP. An expedient synthesis of spiroketals: Model studies for the calyculin C 16-C 25 fragment Tetrahedron. 60: 9199-9204. DOI: 10.1016/J.Tet.2004.07.059  1
2004 Brunner M, Saarenketo P, Straub T, Rissanen K, Koskinen AMP. Stereocontrolled α-alkylation of fully protected L-serine European Journal of Organic Chemistry. 3879-3883. DOI: 10.1002/Ejoc.200400207  1
2003 Karisalmi K, Rissanen K, Koskinen AM. An enantioselective synthesis of the C(33)-C(37) fragment of Amphotericin B. Organic & Biomolecular Chemistry. 1: 3193-6. PMID 14527151 DOI: 10.1039/B305845J  1
2003 Tois J, Koskinen A. Solid-phase lithiation of 5-carboxyindoles Tetrahedron Letters. 44: 2093-2095. DOI: 10.1016/S0040-4039(03)00175-8  1
2003 Koskinen AMP, Kallatsa OA. Polyhydroxylated indolizidine alkaloids - An efficient synthesis of 1-deoxy-8,8a-di-epi-castanospermine Tetrahedron. 59: 6947-6954. DOI: 10.1016/S0040-4020(03)00918-9  1
2003 Tois J, Franzén R, Koskinen A. Synthetic approaches towards indoles on solid phase recent advances and future directions Tetrahedron. 59: 5395-5405. DOI: 10.1016/S0040-4020(03)00851-2  1
2003 Karisalmi K, Koskinen AMP, Nissinen M, Rissanen K. Model studies on a diastereoselective synthesis of the C(33)-C(37) fragment of Amphotericin B Tetrahedron. 59: 1421-1427. DOI: 10.1016/S0040-4020(03)00070-X  1
2002 Nevalainen M, Koskinen AM. Total synthesis of nor-1,6-germacradien-5-ols. The Journal of Organic Chemistry. 67: 1554-60. PMID 11871886 DOI: 10.1021/Jo016110L  1
2002 Törmäkangas OP, Saarenketo P, Koskinen AMP. Selective mixed Tishchenko reaction via substituted 1,3-dioxan-4-ols Organic Process Research and Development. 6: 125-131. DOI: 10.1021/Op0100652  1
2002 Straub T, Koskinen AMP. Catalytic oxidation of THF with homo and hetero metallic Mo/Ru complexes and molecular oxygen Inorganic Chemistry Communications. 5: 1052-1055. DOI: 10.1016/S1387-7003(02)00644-5  1
2002 Törmäkangas OP, Toivola RJ, Karvinen EK, Koskinen AMP. A short and convenient way to produce the Taxol™ A-ring utilizing the Shapiro reaction Tetrahedron. 58: 2175-2181. DOI: 10.1016/S0040-4020(02)00089-3  1
2002 Selkälä SA, Tois J, Pihko PM, Koskinen AMP. Asymmetric Organocatalytic Diels-Alder Reactions on Solid Support Advanced Synthesis and Catalysis. 344: 941-945. DOI: 10.1002/1615-4169(200210)344:9<941::Aid-Adsc941>3.0.Co;2-M  1
2002 Koskinen A, Pihko P. Laboratoriotyöt integroidaan luentoihin: Teknillisen korkeakoulun orgaanisen kemian laboratorio pyrkii Euroopan kärkiviisikkoon Kemia-Kemi/Finnish Chemical Journal. 29: 31-33.  1
2001 Nevalainen M, Koskinen AMP. Synthesis of a 10-Membered Carbocycle By Olefin Metathesis. Angewandte Chemie (International Ed. in English). 40: 4060-4062. PMID 29712259 DOI: 10.1002/1521-3757(20011105)113:21<4184::Aid-Ange4184>3.0.Co;2-R  1
2001 Nevalainen M, Koskinen AM. Synthesis of a 10-Membered Carbocycle By Olefin Metathesis Financial support has been provided by the Academy of Finland and HUT. Angewandte Chemie (International Ed. in English). 40: 4060-4062. PMID 12404492 DOI: 10.1002/1521-3773(20011105)40:21<4060::AID-ANIE4060>3.0.CO;2-8  1
2001 Nevalainen M, Kauppinen PM, Koskinen AM. Synthesis of Fmoc-protected trans-4-methylproline. The Journal of Organic Chemistry. 66: 2061-6. PMID 11300901 DOI: 10.1021/Jo005726S  1
2001 Nevalainen M, Koskinen AMP. The hydrogenation of (4R)-4-[(tert-butoxycarbonyl)amino]-2-methyl-2-penten-5-olide: A precursor of trans-4-methylproline Synlett. 640-642. DOI: 10.1055/S-2001-13380  1
2001 Törmäkangas OP, Koskinen AMP. Fast aldol-Tishchenko reaction utilizing 1,3-diol monoalcoholates as the catalysts Organic Process Research and Development. 5: 421-425. DOI: 10.1021/Op0001335  1
2001 Pihko AJ, Nicolaou KC, Koskinen AMP. An expedient synthesis of D-callipeltose Tetrahedron Asymmetry. 12: 937-942. DOI: 10.1016/S0957-4166(01)00146-X  1
2001 Selkälä SA, Alakurtti S, Koskinen AMP. Hydrogenation of 4-deoxy-β-L-threo-hex-4-enopyranosyluronic acid sodium salt attached to xylodiose or xylotriose Tetrahedron Letters. 42: 3215-3217. DOI: 10.1016/S0040-4039(01)00398-7  1
2001 Törmäkangas OP, Koskinen AMP. Monoalcoholates of 1,3-diols as effective catalysts in the Tishchenko esterification of 1,3-dioxan-4-ols Tetrahedron Letters. 42: 2743-2746. DOI: 10.1016/S0040-4039(01)00277-5  1
2001 Myllymäki VT, Lindvall MK, Koskinen AMP. Computer-assisted discovery of novel amino acid derived sulfides for enantioselective epoxidation of aldehydes Tetrahedron. 57: 4629-4635. DOI: 10.1016/S0040-4020(01)00396-9  1
2000 Koskinen PM, Koskinen AM. Total synthesis of sphingosine and its analogs. Methods in Enzymology. 311: 458-79. PMID 10563344 DOI: 10.1016/S0076-6879(00)11100-0  0.01
2000 Lajunen M, Koskinen A. Hajos–Parrish ketone: approaches toward C-ring precursors of 7-deoxytaxol Journal of the Chemical Society-Perkin Transactions 1. 1439-1443. DOI: 10.1039/A909471G  0.76
2000 Toivola RJ, Savilampi SK, Koskinen AMP. The first direct synthesis of bicyclo[4.2.0]oct-1(6)-en-7-one Tetrahedron Letters. 41: 6207-6210. DOI: 10.1016/S0040-4039(00)01009-1  1
2000 Lajunen MK, Maunula T, Koskinen AMP. Co(II) catalysed oxidation of α-pinene by molecular oxygen. Part 2 Tetrahedron. 56: 8167-8171. DOI: 10.1016/S0040-4020(00)00742-0  0.08
2000 Laitinen RH, Heikkinen V, Haukka M, Koskinen AMP, Pursiainen J. 2-Thioanisyldichlorophosphine, new starting material for the preparation of multidentate phosphine ligands: syntheses and characterization of derivatives of 2-anisyl- and 2-thioanisyldichlorophosphines Journal of Organometallic Chemistry. 598: 235-242. DOI: 10.1016/S0022-328X(99)00711-1  1
1999 Lindvall MK, Koskinen AM. Origins of Stereoselectivity in the Corey-Chaykovsky Reaction. Insights from Quantum Chemistry. The Journal of Organic Chemistry. 64: 4596-4606. PMID 11674528 DOI: 10.1021/Jo9818935  1
1999 Pihko PM, Koskinen AMP. The triumph of zinc: A short and highly efficient synthesis of the calyculin C1-C9 tetraene building block by Negishi coupling Synlett. 1966-1968. DOI: 10.1055/S-1999-2979  1
1999 Pihko PM, Koskinen AMP, Nissinen MJ, Rissanen K. Formation of stable spiro[4.4] ortho ester aminals during the synthesis of the C26-C32 oxazole fragment of calyculin C Journal of Organic Chemistry. 64: 652-654. DOI: 10.1021/Jo981674J  1
1999 Lindvall MK, Rissanen K, Hakala JML, Koskinen AMP. Novel γ-turn mimetics with a reinforced hydrogen bond Tetrahedron Letters. 40: 7427-7430. DOI: 10.1016/S0040-4039(99)01519-1  1
1998 Pihko PM, Koskinen AM. Synthesis of the C(26)-C(32) Oxazole Fragment of Calyculin C: A Test Case for Oxazole Syntheses. The Journal of Organic Chemistry. 63: 92-98. PMID 11674047 DOI: 10.1021/Jo971167M  1
1998 Heino P, Oksala O, Palkama A, Valo T, Vihavainen S, Koskinen A, Uusitalo H. Binding of CGRP Analogs and their Effect on Adenylate Cyclase Activity in Porcine Iris-Ciliary Body Journal of Ocular Pharmacology and Therapeutics. 14: 543-554. PMID 9867337 DOI: 10.1089/Jop.1998.14.543  1
1998 Otsomaa LA, Koskinen AM. Synthesis of 6-deoxyamino sugars. Fortschritte Der Chemie Organischer Naturstoffe = Progress in the Chemistry of Organic Natural Products. ProgrèS Dans La Chimie Des Substances Organiques Naturelles. 74: 197-263. PMID 9597942 DOI: 10.1007/978-3-7091-6496-9_2  1
1998 Koskinen PM, Koskinen AMP. Sphingosine, an Enigmatic Lipid: A Review of Recent Literature Syntheses Synthesis. 1998: 1075-1091. DOI: 10.1055/S-1998-4494  1
1997 Lindvall MK, Pihko PM, Koskinen AM. The binding mode of calyculin A to protein phosphatase-1. A novel spiroketal vector model. The Journal of Biological Chemistry. 272: 23312-6. PMID 9287341 DOI: 10.1074/Jbc.272.37.23312  1
1997 Kallatsa OA, Koskinen AMP. Anti-Kishi selective dihydroxylation of allylic alcohol derivatives Tetrahedron Letters. 38: 8895-8898. DOI: 10.1016/S0040-4039(97)10350-1  1
1997 Bauer U, Ho W, Koskinen AMP. A Novel Linkage For The Solid-Phase Synthesis Of Hydroxamic Acids Tetrahedron Letters. 38: 7233-7236. DOI: 10.1016/S0040-4039(97)01678-X  0.64
1997 Koskinen AMP, Schwerdtfeger J, Edmonds M. A simple route to 4-substituted-3,4-didehydroprolines. Mechanistic probes for the inhibition of prolyl-4-hydroxylase Tetrahedron Letters. 38: 5399-5402. DOI: 10.1016/S0040-4039(97)01182-9  0.64
1997 Kauppinen PM, Koskinen AMP. Studies on 1,3-Allylic Strain Control on Dihydroxylations and Hydrogenations of α-Substituted Enoates Tetrahedron Letters. 38: 3103-3106. DOI: 10.1016/S0040-4039(97)00556-X  1
1997 Koskinen AMP, Otsomaa LA. A new access to enantiomerically pure deoxy aminohexoses: Methyl 4-amino-4,6-dideoxygulopyranoside and epi-tolyposamine Tetrahedron. 53: 6473-6484. DOI: 10.1016/S0040-4020(97)00304-9  1
1996 Hakala JM, Lindvall M, Koskinen AM. Modelling constrained calcitonin gene-related peptide analogues. Protein Engineering. 9: 143-8. PMID 9005435  1
1996 Koskinen AMP, Hassila H, Harms K, Simonsen K, Liptay G, Trautwein-Fritz K, Stackhouse J, Ciglic MI, Haugg M, Trabesinger-Rüf N, Weinhold EG. Asymmetric Intramolecular Cyclopropanation. Synthesis of Conformationally Constrained Aminocyclopropane Carboxylic Acids. Acta Chemica Scandinavica. 50: 323-327. DOI: 10.3891/Acta.Chem.Scand.50-0323  0.64
1996 Toivola RJ, Koskinen AMP. A Versatile A-ring Synthesis for Taxol Synlett. 1996: 1159-1161. DOI: 10.1055/S-1996-5714  1
1996 Geffaut T, Bauer U, Airola K, Koskinen AMP. Asymmetric 1,3-dipolar cycloaddition: Synthesis of N-protected (4S)-4-hydroxy L-glutamic acid diester Tetrahedron-Asymmetry. 7: 3099-3102. DOI: 10.1016/0957-4166(96)00407-7  0.64
1995 Koskinen AMP. Asymmetry : To Make A Distinction Pure and Applied Chemistry. 67: 1031-1036. DOI: 10.1351/Pac199567071031  0.64
1995 Koskinen AMP, Valo T, Vihavainen S, Hakala JML. Synthesis of α-helix substituted analogs of calcitonin gene-related peptide Bioorganic & Medicinal Chemistry Letters. 5: 573-578. DOI: 10.1016/0960-894X(95)00078-8  1
1995 Koskinen AMP, Hassilla H, Myllymäki VT, Rissanen K. Stereocontrolled conversion of L-serine into a series of valuable unnatural α-amino acids Tetrahedron Letters. 36: 5619-5622. DOI: 10.1016/0040-4039(95)01029-H  1
1995 Karvinen EK, Koskinen AMP. A short synthesis of the A-ring of taxol Tetrahedron. 51: 7555-7560. DOI: 10.1016/0040-4020(95)00378-L  1
1994 Hakala JM, Valo T, Vihavainen S, Hermonen J, Heino P, Halme M, Koskinen AM. Constrained analogues of the calcitonin gene-related peptide. Biochemical and Biophysical Research Communications. 202: 497-503. PMID 8037754 DOI: 10.1006/bbrc.1994.1956  1
1994 Koskinen AMP, Karvinen EK, Siirilä JP. Enantioselective synthesis of the Taxol and Taxotere side chains Journal of the Chemical Society, Chemical Communications. 21-22. DOI: 10.1039/C39940000021  1
1994 Lajunen M, Koskinen AMP. Co(II)-catalysed allylic oxidation of α-pinene by molecular oxygen; synthesis of verbenone Tetrahedron Letters. 35: 4461-4464. DOI: 10.1016/S0040-4039(00)73384-3  0.64
1994 Koskinen AMP, Pihko PM. Calyculins. Asymmetric synthesis of the C26-C32 fragment Tetrahedron Letters. 35: 7417-7420. DOI: 10.1016/0040-4039(94)85330-4  1
1993 Koskinen A. Asymmetric synthesis of chiral macrocyclic ligands Pure and Applied Chemistry. 65: 1465-1470. DOI: 10.1351/Pac199365071465  0.76
1993 Koskinen AMP, Koskinen PM. Improved Horner-Wadsworth-Emmons olefination of base sensitive-γ-chiral β-ketophosphonates Synlett. 1993: 501-502. DOI: 10.1055/S-1993-22506  1
1993 Rissanen K, Huuskonen J, Koskinen A. 12,52,92,132-Tetranitro-1,5,9, 13(1,3)-tetrabenzena-3,7,11,15(1,4)-tetrapiperazinacyclo-hexadecaphane, a new host compound Journal of the Chemical Society, Chemical Communications. 771-772. DOI: 10.1039/C39930000771  1
1993 Koskinen AMP, Muñoz L, Rissanen K. Unexpected acid-catalysed rearrangement of a vinylcyclopropane derivative Journal of the Chemical Society, Chemical Communications. 491-492. DOI: 10.1039/C39930000491  1
1993 Koskinen AMP, Hassila H. Asymmetric catalysis in intramolecular cyclopropanation Journal of Organic Chemistry. 58: 4479-4480. DOI: 10.1021/Jo00068A054  0.64
1993 Koskinen AMP, Munoz L. Intramolecular cyclopropanation: stereospecific synthesis of (E)- and (Z)-1-aminocyclopropane-1-carboxylic acids Journal of Organic Chemistry. 58: 879-886. DOI: 10.1021/Jo00056A020  0.64
1993 Koskinen AMP, Koskinen PM. Synthetic studies towards amino alcohols. Diastereocontrolled reduction of α′-chiral α,β-enones. Tetrahedron Letters. 34: 6765-6768. DOI: 10.1016/S0040-4039(00)61696-9  1
1991 Gunda TE, Koskinen AMP. Carbamimidates, carbamimidothioates and related compounds. The effect of lipophilicity on the antibacterial activity European Journal of Medicinal Chemistry. 26: 449-454. DOI: 10.1016/0223-5234(91)90106-W  0.64
1990 Koskinen AMP, Muñoz L. 1-Amino-2-oxo-3-oxabicyclo[3.1.0]hexane (2,3-methanohomoserine lactone), a conformationally constrained amino acid Journal of the Chemical Society, Chemical Communications. 1373-1374. DOI: 10.1039/C39900001373  0.64
1990 Koskinen AMP, Muñoz L. Diazo transfer reactions under mildly basic conditions Journal of the Chemical Society, Chemical Communications. 652-653. DOI: 10.1039/C39900000652  0.64
1989 Sardina FJ, Howard MH, Koskinen AMP, Rapoport H. Chirospecific synthesis of nitrogen and side chain modified analogs of (+)-anatoxin Journal of Organic Chemistry. 54: 4654-4660. DOI: 10.1021/Jo00280A037  1
1989 Koskinen AMP, Rapoport H. Synthesis of 4-substituted prolines as conformationally constrained amino acid analogs Journal of Organic Chemistry. 54: 1859-1866. DOI: 10.1021/Jo00269A022  1
1987 Lounasmaa M, Karvinen E, Koskinen A, Jokela R. Novel applications of the modified polonovski reaction-IX. A new route to wenkert's enamine Tetrahedron. 43: 2135-2146. DOI: 10.1016/S0040-4020(01)86795-8  1
1986 Koskinen AMP, Lounasmaa M. 2D NMR study of ajmaline Heterocycles. 24: 331-334. DOI: 10.3987/R-1986-02-0331  0.76
1986 Lounasmaa M, Koskinen A, O'Connell J. NMR Studies of Alkaloids. Assignment of the Configuration at C(20) in Tubotaiwine (Dihydrocondylocarpine) Helvetica Chimica Acta. 69: 1343-1348. DOI: 10.1002/Hlca.19860690608  0.76
1986 Lounasmaa M, Koskinen A, O'connell J. NMR Studies of Alkaloids. Assignment of the Configuration at C(20) in Tubotaiwine (Dihydrocondylocarpine). Cheminform. 17. DOI: 10.1002/Chin.198652301  0.76
1985 Koskinen AM, Rapoport H. Synthetic and conformational studies on anatoxin-a: a potent acetylcholine agonist. Journal of Medicinal Chemistry. 28: 1301-9. PMID 4032432 DOI: 10.1002/Chin.198552240  1
1984 Lounasmaa M, Koskinen A. Modified Polonovski reaction, a versatile synthetic tool Heterocycles. 22: 1591-1612. DOI: 10.1002/Chin.198448368  0.76
1984 Koskinen A, Lounasmaa M. Tryptophan derived pyridinium salts: preparation, reductive cyanation and addition reactions Heterocycles. 22: 733-744. DOI: 10.1002/Chin.198439169  0.76
1983 Lounasmaa M, Koskinen A. 13C NMR Spectral Analysis of a-Aminonitriles Heterocycles. 20: 563. DOI: 10.3987/R-1983-04-0563  0.76
1983 Lounasmaa M, Koskinen A, somersalo P. NMR Spectroacopic Studies of Tryptophan Derivatives Heterocycles. 20: 557. DOI: 10.3987/R-1983-04-0557  0.76
1983 Koskinen A, Lounasmaa M. Mild general synthesis of 4-substituted piperidines Journal of the Chemical Society, Chemical Communications. 821-822. DOI: 10.1039/C39830000821  0.76
1983 Koskinen A, Lounasmaa M. Novel applications of the modified polonovski reaction - V1 silyl enolates as nucleophilic alkylating reagents Tetrahedron Letters. 24: 1951-1952. DOI: 10.1016/S0040-4039(00)81814-6  1
1983 Koskinen A, Lounasmaa M. Regiospecific functionalisation of carbon atoms α to heterocyclic nitrogen Tetrahedron. 39: 1627-1633. DOI: 10.1016/S0040-4020(01)88573-2  1
1983 Suortti T, Koskinen A. Necatorin, a highly mutagenic compound from Lactarius necator Phytochemistry. 22: 2873-2874. DOI: 10.1016/S0031-9422(00)97723-9  0.76
1983 Koskinen A, Lounasmaa M. Mild General Synthesis Of 4-Substituted Piperidines Cheminform. 14. DOI: 10.1002/Chin.198349228  0.76
1982 Lounasmaa M, Koskinen A. A plausible biogenetic proposal for koumine. Planta Medica. 44: 120-1. PMID 17402092 DOI: 10.1055/S-2007-971416  0.76
1982 Koskinen A, Lounasmaa M. Biogenesis of the ajmaline type alkaloids. Planta Medica. 45: 248-9. PMID 17396924 DOI: 10.1055/S-2007-971385  1
1982 Koskinen A. 13C NMR Spectroscopy of Substituted Imidazoles Heterocycles. 19: 1633. DOI: 10.3987/R-1982-09-1633  0.76
1982 Lounasmaa M, Koskinen A. On the Structure of Ajmalinol Heterocycles. 19: 851. DOI: 10.3987/R-1982-05-0851  0.76
1982 Lounasmaa M, Koskinen A. Indoloquinolizidine synthesis. Stereochemistry and mechanism of cyclisation Tetrahedron Letters. 23: 1489-1492. DOI: 10.1016/S0040-4039(00)87140-3  1
1982 Lounasmaa M, Koskinen A. Novel applications of the modified polonovski reaction. A biomimetic synthesis of quinuclidines Tetrahedron Letters. 23: 349-352. DOI: 10.1016/S0040-4039(00)86828-8  1
1982 Lounasmaa M, Koskinen A. Novel Applications Of The Modified Polonovski Reaction. Ii. Regiocontrolled Iminium Ion Formation Cheminform. 14: 2115. DOI: 10.1002/Chin.198315236  0.76
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