Year |
Citation |
Score |
2023 |
Sharma S, Choudhary S, Kaur S, Reddy MV, Thota N, Singh A, Koul S, Khan IA, Ahmed Z, Kumar A. Piperine analog PGP-41 treatment overcomes paclitaxel resistance in NCI/ADR-RES ovarian cells by inhibition of MDR1. Chemico-Biological Interactions. 381: 110569. PMID 37244399 DOI: 10.1016/j.cbi.2023.110569 |
0.379 |
|
2018 |
Rath SK, Singh S, Kumar S, Wani NA, Rai R, Koul S, Khan IA, Sangwan PL. Synthesis of amides from (E)-3-(1-chloro-3,4-dihydronaphthalen-2-yl)acrylic acid and substituted amino acid esters as NorA efflux pump inhibitors of Staphylococcus aureus. Bioorganic & Medicinal Chemistry. PMID 30552006 DOI: 10.1016/j.bmc.2018.12.008 |
0.357 |
|
2018 |
Farooq S, Banday JA, Hussain A, Nazir M, Qurishi MA, Hamid A, Koul S. Synthesis and biological evaluation of novel osthol derivatives as potent cytotoxic agents. Medicinal Chemistry (Shariqah (United Arab Emirates)). PMID 30207222 DOI: 10.2174/1573406414666180911161047 |
0.522 |
|
2016 |
Chinthakindi PK, Singh J, Gupta S, Nargotra A, Mahajan P, Kaul A, Ahmed Z, Koul S, Sangwan PL. Synthesis of α-santonin derivatives for diminutive effect on T and B-cell proliferation and their structure activity relationships. European Journal of Medicinal Chemistry. PMID 27847171 DOI: 10.1016/j.ejmech.2016.11.018 |
0.655 |
|
2016 |
Wani NA, Singh S, Farooq S, Shankar S, Koul S, Khan IA, Rai R. Amino acid amides of piperic acid (PA) and 4-ethylpiperic acid (EPA) as NorA efflux pump inhibitors of Staphylococcus aureus. Bioorganic & Medicinal Chemistry Letters. PMID 27503686 DOI: 10.1016/j.bmcl.2016.07.062 |
0.308 |
|
2016 |
Alam MI, Alam MA, Alam O, Nargotra A, Taneja SC, Koul S. Molecular modeling and snake venom phospholipase A2 inhibition by phenolic compounds: Structure-activity relationship. European Journal of Medicinal Chemistry. 114: 209-219. PMID 26986086 DOI: 10.1016/j.ejmech.2016.03.008 |
0.351 |
|
2015 |
Khan I, Guru SK, Rath SK, Chinthakindi PK, Singh B, Koul S, Bhushan S, Sangwan PL. A novel triazole derivative of betulinic acid induces extrinsic and intrinsic apoptosis in human leukemia HL-60 cells. European Journal of Medicinal Chemistry. 108: 104-116. PMID 26629862 DOI: 10.1016/j.ejmech.2015.11.018 |
0.7 |
|
2015 |
Majeed R, Hussain A, Sangwan PL, Chinthakindi PK, Khan I, Sharma PR, Koul S, Saxena AK, Hamid A. PI3K target based novel cyano derivative of betulinic acid induces its signalling inhibition by down-regulation of pGSK3β and cyclin D1 and potentially checks cancer cell proliferation. Molecular Carcinogenesis. PMID 26013878 DOI: 10.1002/mc.22339 |
0.679 |
|
2014 |
Shakeel-u-Rehman, Masood-ur-Rahman, Tripathi VK, Singh J, Ara T, Koul S, Farooq S, Kaul A. Synthesis and biological evaluation of novel isoxazoles and triazoles linked 6-hydroxycoumarin as potent cytotoxic agents. Bioorganic & Medicinal Chemistry Letters. 24: 4243-6. PMID 25088398 DOI: 10.1016/j.bmcl.2014.07.031 |
0.441 |
|
2014 |
Farooq S, Shakeel-u-Rehman, Hussain A, Hamid A, Qurishi MA, Koul S. Click chemistry inspired synthesis and bioevaluation of novel triazolyl derivatives of osthol as potent cytotoxic agents. European Journal of Medicinal Chemistry. 84: 545-54. PMID 25062005 DOI: 10.1016/j.ejmech.2014.07.069 |
0.478 |
|
2013 |
Majeed R, Sangwan PL, Chinthakindi PK, Khan I, Dangroo NA, Thota N, Hamid A, Sharma PR, Saxena AK, Koul S. Synthesis of 3-O-propargylated betulinic acid and its 1,2,3-triazoles as potential apoptotic agents. European Journal of Medicinal Chemistry. 63: 782-92. PMID 23584541 DOI: 10.1016/j.ejmech.2013.03.028 |
0.69 |
|
2013 |
Chinthakindi PK, Sangwan PL, Farooq S, Aleti RR, Kaul A, Saxena AK, Murthy YL, Vishwakarma RA, Koul S. Diminutive effect on T and B-cell proliferation of non-cytotoxic α-santonin derived 1,2,3-triazoles: a report. European Journal of Medicinal Chemistry. 60: 365-75. PMID 23314050 DOI: 10.1016/J.Ejmech.2012.12.018 |
0.681 |
|
2012 |
Majeed R, Reddy MV, Chinthakindi PK, Sangwan PL, Hamid A, Chashoo G, Saxena AK, Koul S. Bakuchiol derivatives as novel and potent cytotoxic agents: a report. European Journal of Medicinal Chemistry. 49: 55-67. PMID 22245048 DOI: 10.1016/j.ejmech.2011.12.018 |
0.709 |
|
2011 |
Nargotra A, Sharma S, Alam MI, Ahmed Z, Bhagat A, Taneja SC, Qazi GN, Koul S. In silico identification of viper phospholipaseA2 inhibitors: validation by in vitro, in vivo studies. Journal of Molecular Modeling. 17: 3063-73. PMID 21360175 DOI: 10.1007/s00894-011-0994-7 |
0.324 |
|
2010 |
Reddy MV, Thota N, Sangwan PL, Malhotra P, Ali F, Khan IA, Chimni SS, Koul S. Novel bisstyryl derivatives of bakuchiol: targeting oral cavity pathogens. European Journal of Medicinal Chemistry. 45: 3125-34. PMID 20427099 DOI: 10.1016/J.Ejmech.2010.03.049 |
0.322 |
|
2008 |
Sangwan PL, Koul JL, Koul S, Reddy MV, Thota N, Khan IA, Kumar A, Kalia NP, Qazi GN. Piperine analogs as potent Staphylococcus aureus NorA efflux pump inhibitors. Bioorganic & Medicinal Chemistry. 16: 9847-57. PMID 18848780 DOI: 10.1016/j.bmc.2008.09.042 |
0.325 |
|
2002 |
Völkert M, Koul S, Müller GH, Lehnig M, Waldmann H. Phenylhydrazide as an enzyme-labile protecting group in peptide synthesis. The Journal of Organic Chemistry. 67: 6902-10. PMID 12353981 DOI: 10.1021/Jo0259966 |
0.397 |
|
Show low-probability matches. |