| Year |
Citation |
Score |
| 2025 |
You C, Wei S, Yu J, Xu G, Li H, Liu X, Wang M, Meng X, Xu Y, Yu G, Luo H, Xu B. Design and synthesis of 2-amino-4-(trifluoromethyl)pyrimidine derivatives as potential Werner-dependent antiproliferative agents. Molecular Diversity. PMID 40517347 DOI: 10.1007/s11030-025-11225-3 |
0.389 |
|
| 2025 |
Yu G, Yu J, Zhou Y, Liu K, Peng X, Xu G, Chen C, Meng X, Zeng X, Wu H, Zan N, Luo H, Xu B. Discovery of novel quinazoline derivatives containing trifluoromethyl against cell proliferation by targeting werner helicase. Molecular Diversity. PMID 40148606 DOI: 10.1007/s11030-025-11175-w |
0.609 |
|
| 2025 |
Li C, Cheng S, Yu J, Zheng Q, Yu G, Xu M, Meng X, Zeng X, Liu K, Xu B, Luo H, Xu G. Hit to lead optimization of the 4-trifluoromethylquinoline derivatives as novel SGK1 inhibitors with potent anti-prostate cancer activity. European Journal of Medicinal Chemistry. 287: 117336. PMID 39908792 DOI: 10.1016/j.ejmech.2025.117336 |
0.635 |
|
| 2024 |
Meng X, Shao X, Kuang A, Xu B, Zeng X, Kong X, Xu G, Yu G. Design, Synthesis and Biological Evaluation of Novel Trifluoromethylated Dipeptide Mimetics of Matijin-Su as Potent Anti-HBV Agents. Chemistry & Biodiversity. e202402061. PMID 39714596 DOI: 10.1002/cbdv.202402061 |
0.607 |
|
| 2024 |
Yu J, Zhou Y, Liang G, Cheng S, Wei J, Li H, Liu X, You C, Mao M, Ahmad M, Yu G, Xu B, Luo H. Quinazoline derivatives inhibit cell growth of prostate cancer as a WRN helicase dependent manner by regulating DNA damage repair and microsatellite instability. Bioorganic Chemistry. 153: 107963. PMID 39571305 DOI: 10.1016/j.bioorg.2024.107963 |
0.34 |
|
| 2024 |
Xu G, Li L, Lv M, Li C, Yu J, Zeng X, Meng X, Yu G, Liu K, Cheng S, Luo H, Xu B. Discovery of novel 4-trifluoromethyl-2-anilinoquinoline derivatives as potential anti-cancer agents targeting SGK1. Molecular Diversity. PMID 39117890 DOI: 10.1007/s11030-024-10951-4 |
0.625 |
|
| 2024 |
Li H, Yu J, Yu G, Cheng S, Wu H, Wei J, You C, Liu K, Wang M, Meng X, Xu G, Luo H, Xu B. Design and synthesis of N-aryl-2-trifluoromethyl-quinazoline-4-amine derivatives as potential Werner-dependent antiproliferative agents. Molecular Diversity. PMID 38739229 DOI: 10.1007/s11030-024-10844-6 |
0.609 |
|
| 2024 |
Chen M, Cheng S, Dai X, Yu J, Wang H, Xu B, Luo H, Xu G. Design, Synthesis, and Biological Evaluation of Novel Quinazoline Derivatives Possessing a Trifluoromethyl Moiety as Potential Antitumor Agents. Chemistry & Biodiversity. e202301776. PMID 38602834 DOI: 10.1002/cbdv.202301776 |
0.622 |
|
| 2024 |
Wang M, Yu J, Huang X, Yu G, Liang Q, Cheng S, Meng X, Xu G, Li H, Luo H, Xu B. Design, synthesis and antitumor activity of 2-substituted quinazoline-4-amine derivatives. Bioorganic & Medicinal Chemistry. 102: 117660. PMID 38442524 DOI: 10.1016/j.bmc.2024.117660 |
0.597 |
|
| 2023 |
Yu J, Wang X, Cheng S, Zeng X, Wan X, Wei S, Xu B, Luo H, Meng X. Design, synthesis and bioevaluation of novel prenylated chalcones derivatives as potential antitumor agents. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. 192: 106660. PMID 38052256 DOI: 10.1016/j.ejps.2023.106660 |
0.374 |
|
| 2023 |
Zhang S, Mo M, Lv M, Xia W, Liu K, Yu G, Yu J, Xu G, Zeng X, Cheng S, Xu B, Luo H, Meng X. Design, synthesis and bioevaluation of novel trifluoromethylquinoline derivatives as tubulin polymerization inhibitors. Future Medicinal Chemistry. PMID 37937524 DOI: 10.4155/fmc-2023-0151 |
0.614 |
|
| 2023 |
Liu K, Mo M, Yu G, Yu J, Song SM, Cheng S, Li HM, Meng XL, Zeng XP, Xu GC, Luo H, Xu BX. Discovery of novel 2-(trifluoromethyl)quinolin-4-amine derivatives as potent antitumor agents with microtubule polymerization inhibitory activity. Bioorganic Chemistry. 139: 106727. PMID 37451147 DOI: 10.1016/j.bioorg.2023.106727 |
0.634 |
|
| 2023 |
Wu H, Wang LS, Li P, Yu J, Cheng S, Yu G, Ahmad M, Meng XL, Luo H, Xu BX. Discovery of novel N-aryl-2-trifluoromethyl-quinazoline-4-amine derivatives as the inhibitors of tubulin polymerization in leukemia cells. European Journal of Medicinal Chemistry. 256: 115470. PMID 37201429 DOI: 10.1016/j.ejmech.2023.115470 |
0.447 |
|
| 2017 |
Wen Z, Zhang Y, Wang X, Zeng X, Hu Z, Liu Y, Xie Y, Liang G, Zhu J, Luo H, Xu B. Novel 3',5'-diprenylated chalcones inhibited the proliferation of cancer cells in vitro by inducing cell apoptosis and arresting cell cycle phase. European Journal of Medicinal Chemistry. 133: 227-239. PMID 28390228 DOI: 10.1016/j.ejmech.2017.03.077 |
0.4 |
|
| 2016 |
Qiu J, Xu B, Gong Q, Pan W, Liu C, Huang Z, Gu X, Liang G. Synthesis and biological evaluation of Matijin-Su derivatives as potential anti-hepatitis B virus and anti-cancer agents. Chemistry & Biodiversity. PMID 27451105 DOI: 10.1002/cbdv.201600113 |
0.312 |
|
| 2016 |
Cao D, Liu Y, Yan W, Wang C, Bai P, Wang T, Tang M, Wang X, Yang Z, Ma B, Ma L, Lei L, Wang F, Xu B, Zhou Y, et al. Design, Synthesis, and Evaluation of in Vitro and In Vivo Anticancer Activity of 4-Substituated Coumarins: A Novel Class of Potent Tubulin Polymerization Inhibitors. Journal of Medicinal Chemistry. PMID 27213819 DOI: 10.1021/acs.jmedchem.6b00158 |
0.386 |
|
| 2015 |
Unione L, Xu B, Díaz D, Martín-Santamaría S, Poveda A, Sardinha J, Rauter AP, Blériot Y, Zhang Y, Cañada FJ, Sollogoub M, Jiménez-Barbero J. Conformational Plasticity in Glycomimetics: Fluorocarbamethyl-L-idopyranosides Mimic the Intrinsic Dynamic Behaviour of Natural Idose Rings. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 10513-21. PMID 26096911 DOI: 10.1002/Chem.201501249 |
0.641 |
|
| 2014 |
Xu B, Unione L, Sardinha J, Wu S, Ethève-Quelquejeu M, Pilar Rauter A, Blériot Y, Zhang Y, Martín-Santamaría S, Díaz D, Jiménez-Barbero J, Sollogoub M. gem-Difluorocarbadisaccharides: restoring the exo-anomeric effect. Angewandte Chemie (International Ed. in English). 53: 9597-602. PMID 25044775 DOI: 10.1002/Anie.201405008 |
0.64 |
|
| 2014 |
Xu B, Wang N, Pan W, Qiu J, Cao P, Zhu M, Feng Y, Liang G. Synthesis and anti-tumor activity evaluation of Matijin-Su derivatives. Bioorganic Chemistry. 56: 34-40. PMID 24930072 DOI: 10.1016/j.bioorg.2014.05.009 |
0.372 |
|
| 2014 |
Patzel KA, Yardeni T, Le Poëc-Celic E, Leoyklang P, Dorward H, Alonzi DS, Kukushkin NV, Xu B, Zhang Y, Sollogoub M, Blériot Y, Gahl WA, Huizing M, Butters TD. Non-specific accumulation of glycosphingolipids in GNE myopathy. Journal of Inherited Metabolic Disease. 37: 297-308. PMID 24136589 DOI: 10.1007/S10545-013-9655-6 |
0.451 |
|
| 2006 |
Pan W, Zhang Y, Xu B, Cao P, Liang G. Two new naturally occurring optical polyacetylene compounds from Torricellia angulata var intermedia and the determination of their absolute configurations. Natural Product Research. 20: 1098-104. PMID 17127663 DOI: 10.1080/14786410600743951 |
0.33 |
|
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