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Sarang S. Kulkarni, Ph.D. - Publications

Affiliations: 
2009 Chemistry Purdue University, West Lafayette, IN, United States 
Area:
HIV-1 protease inhibitors
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22 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2016 Lad NP, Kulkarni S, Sharma R, Mascarenhas M, Kulkarni MR, Pandit SS. Piperlongumine derived cyclic sulfonamides (sultams): Synthesis and in vitro exploration for therapeutic potential against HeLa cancer cell lines. European Journal of Medicinal Chemistry. 126: 870-878. PMID 27987486 DOI: 10.1016/J.Ejmech.2016.12.022  0.52
2016 Chaube MA, Sarpe VA, Jana S, Kulkarni SS. First total synthesis of trehalose containing tetrasaccharides from Mycobacterium smegmatis. Organic & Biomolecular Chemistry. PMID 27035801 DOI: 10.1039/C6Ob00412A  0.33
2014 Sarpe VA, Kulkarni SS. Expeditious synthesis of Mycobacterium tuberculosis sulfolipids SL-1 and Ac2SGL analogues. Organic Letters. 16: 5732-5. PMID 25322198 DOI: 10.1021/ol5027987  0.315
2014 Sanapala SR, Kulkarni SS. Chemical synthesis of asparagine-linked archaeal N-glycan from Methanothermus fervidus. Chemistry (Weinheim An Der Bergstrasse, Germany). 20: 3578-83. PMID 24616211 DOI: 10.1002/chem.201304950  0.301
2013 Emmadi M, Kulkarni SS. Expeditious synthesis of bacterial, rare sugar building blocks to access the prokaryotic glycome. Organic & Biomolecular Chemistry. 11: 3098-102. PMID 23563627 DOI: 10.1039/C3Ob40615F  0.312
2013 Kulkarni SS, Hu X, Manetsch R. A simple base-mediated amidation of aldehydes with azides. Chemical Communications (Cambridge, England). 49: 1193-5. PMID 23287824 DOI: 10.1039/C2Cc37289D  0.341
2013 Patil SM, Kulkarni S, Mascarenhas M, Sharma R, Roopan SM, Roychowdhury A. DMSO-POCl3: A reagent for methylthiolation of imidazo[1,2-a]pyridines and other imidazo-fused heterocycles Tetrahedron. 69: 8255-8262. DOI: 10.1016/J.Tet.2013.07.017  0.349
2012 McCarthy JG, Eisman EB, Kulkarni S, Gerwick L, Gerwick WH, Wipf P, Sherman DH, Smith JL. Structural basis of functional group activation by sulfotransferases in complex metabolic pathways. Acs Chemical Biology. 7: 1994-2003. PMID 22991895 DOI: 10.1021/Cb300385M  0.322
2012 Ghosh AK, Pandey S, Gangarajula S, Kulkarni S, Xu X, Rao KV, Huang X, Tang J. Structure-based design, synthesis, and biological evaluation of dihydroquinazoline-derived potent β-secretase inhibitors. Bioorganic & Medicinal Chemistry Letters. 22: 5460-5. PMID 22863204 DOI: 10.1016/J.Bmcl.2012.07.043  0.6
2011 Sarpe VA, Kulkarni SS. Synthesis of maradolipid. The Journal of Organic Chemistry. 76: 6866-70. PMID 21739985 DOI: 10.1021/jo200979n  0.357
2010 Tojo Y, Koh Y, Amano M, Aoki M, Das D, Kulkarni S, Anderson DD, Ghosh AK, Mitsuya H. Novel protease inhibitors (PIs) containing macrocyclic components and 3(R),3a(S),6a(R)-bis-tetrahydrofuranylurethane that are potent against multi-PI-resistant HIV-1 variants in vitro. Antimicrobial Agents and Chemotherapy. 54: 3460-70. PMID 20439612 DOI: 10.1128/Aac.01766-09  0.423
2010 Schombs M, Park FE, Du W, Kulkarni SS, Gervay-Hague J. One-pot syntheses of immunostimulatory glycolipids. The Journal of Organic Chemistry. 75: 4891-8. PMID 20387787 DOI: 10.1021/Jo100366V  0.342
2010 Ghosh AK, Shurrush K, Kulkarni S. Synthesis of (-)-Tetrahydrolipstatin Synfacts. 2010: 6-6. DOI: 10.1055/S-0029-1218402  0.697
2009 Ghosh AK, Kulkarni S, Anderson DD, Hong L, Baldridge A, Wang YF, Chumanevich AA, Kovalevsky AY, Tojo Y, Amano M, Koh Y, Tang J, Weber IT, Mitsuya H. Design, synthesis, protein-ligand X-ray structure, and biological evaluation of a series of novel macrocyclic human immunodeficiency virus-1 protease inhibitors to combat drug resistance. Journal of Medicinal Chemistry. 52: 7689-705. PMID 19746963 DOI: 10.1021/Jm900695W  0.557
2009 Ghosh AK, Shurrush K, Kulkarni S. Asymmetric synthesis of anti-aldol segments via a nonaldol route: synthetic applications to statines and (-)-tetrahydrolipstatin. The Journal of Organic Chemistry. 74: 4508-18. PMID 19438217 DOI: 10.1021/Jo900642F  0.708
2008 Ghosh AK, Kulkarni SS, Xu CX, Shurrush K. Asymmetric multi-component reactions: convenient access to acyclic stereocenters and functionalized cyclopentenoids. Tetrahedron, Asymmetry. 19: 1020-1026. PMID 21954322 DOI: 10.1016/J.Tetasy.2008.04.005  0.688
2008 Ghosh AK, Kulkarni S. Enantioselective total synthesis of (+)-largazole, a potent inhibitor of histone deacetylase. Organic Letters. 10: 3907-9. PMID 18662003 DOI: 10.1021/Ol8014623  0.606
2008 Ghosh AK, Kumaragurubaran N, Hong L, Kulkarni S, Xu X, Miller HB, Reddy DS, Weerasena V, Turner R, Chang W, Koelsch G, Tang J. Potent memapsin 2 (beta-secretase) inhibitors: design, synthesis, protein-ligand X-ray structure, and in vivo evaluation. Bioorganic & Medicinal Chemistry Letters. 18: 1031-6. PMID 18180160 DOI: 10.1016/J.Bmcl.2007.12.028  0.576
2007 Ghosh AK, Kumaragurubaran N, Hong L, Kulkarni SS, Xu X, Chang W, Weerasena V, Turner R, Koelsch G, Bilcer G, Tang J. Design, synthesis, and X-ray structure of potent memapsin 2 (beta-secretase) inhibitors with isophthalamide derivatives as the P2-P3-ligands. Journal of Medicinal Chemistry. 50: 2399-407. PMID 17432843 DOI: 10.1021/Jm061338S  0.596
2007 Ghosh AK, Kulkarni S, Xu CX, Fanwick PE. Asymmetric multicomponent reactions: diastereoselective synthesis of substituted pyrrolidines and prolines. Organic Letters. 8: 4509-11. PMID 16986937 DOI: 10.1021/Ol061672I  0.593
2006 Ghosh A, Kulkarni S, Xu C, Fanwick P. Diastereoselective Synthesis of Pyrrolidines and Prolines Synfacts. 2006: 1245-1245. DOI: 10.1055/S-2006-955639  0.64
2005 Ghosh AK, Xu CX, Kulkarni SS, Wink D. TiCl4-promoted multicomponent reaction: a new entry to functionalized alpha-amino acids. Organic Letters. 7: 7-10. PMID 15624964 DOI: 10.1021/Ol048302J  0.517
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