| Year |
Citation |
Score |
| 2023 |
Liu C, Voskressensky LG, Van der Eycken E. Recent Advances in the Synthesis of Peptidomimetics via Ugi Reactions. Chemistry (Weinheim An Der Bergstrasse, Germany). e202303597. PMID 38123521 DOI: 10.1002/chem.202303597 |
0.362 |
|
| 2023 |
Liu C, Van der Eycken J, Van der Eycken E. Transition Metal-Free N-S Bond Cleavage and C-N Bond Activation of Ugi-Adducts for Rapid Preparation of Primary Amides and α-Ketoamides. Chemistry (Weinheim An Der Bergstrasse, Germany). e202301541. PMID 37410246 DOI: 10.1002/chem.202301541 |
0.64 |
|
| 2023 |
Vázquez-Amaya LY, Dootselaere B, Ojeda-Carralero GM, Pillitteri S, Van der Eycken J, Van der Eycken EV, Sharma UK. Light-Driven Four-Component Reaction with Boronic Acid Derivatives as Alkylating Agents: An Amine/Imine-Mediated Activation Approach. Organic Letters. PMID 37249484 DOI: 10.1021/acs.orglett.3c01020 |
0.675 |
|
| 2023 |
Tang X, Song L, Van der Eycken EV. Post-Ugi Cyclizations Towards Polycyclic N-Heterocycles. Chemical Record (New York, N.Y.). e202300095. PMID 37218998 DOI: 10.1002/tcr.202300095 |
0.4 |
|
| 2023 |
Xu X, Zhong L, Feng H, Van der Eycken EV. Application of Metal-Free Dearomatization Reaction as a Sustainable Strategy to Direct Access Complex Cyclic Compounds. Chemical Record (New York, N.Y.). e202300101. PMID 37132130 DOI: 10.1002/tcr.202300101 |
0.477 |
|
| 2023 |
Song L, Lv Z, Li Y, Zhang K, Van der Eycken EV, Cai L. Construction of Peptide-Isoquinolone Conjugates via Rh(III)-Catalyzed C-H Activation/Annulation. Organic Letters. 25: 2996-3000. PMID 37129283 DOI: 10.1021/acs.orglett.3c00766 |
0.343 |
|
| 2023 |
Song L, Cai L, Gong L, Van der Eycken EV. Photoinduced copper-catalyzed enantioselective coupling reactions. Chemical Society Reviews. PMID 36916421 DOI: 10.1039/d2cs00734g |
0.474 |
|
| 2023 |
Vis C, Schuurmans J, Aouizerate B, Atipei Craggs M, Batterham P, Bührmann L, Calear A, Cerga Pashoja A, Christensen H, Dozeman E, Duedal Pedersen C, Ebert DD, Etzelmueller A, Fanaj N, Finch TL, ... ... Van der Eycken E, et al. Effectiveness of Self-guided Tailored Implementation Strategies in Integrating and Embedding Internet-Based Cognitive Behavioral Therapy in Routine Mental Health Care: Results of a Multicenter Stepped-Wedge Cluster Randomized Trial. Journal of Medical Internet Research. 25: e41532. PMID 36735287 DOI: 10.2196/41532 |
0.23 |
|
| 2023 |
Tang X, Ding S, Song L, Van der Eycken EV. Transition metal-catalyzed C-H activation/annulation approaches to isoindolo[2,1-b]isoquinolin-5(7H)-ones. Chemical Record (New York, N.Y.). e202200255. PMID 36646518 DOI: 10.1002/tcr.202200255 |
0.414 |
|
| 2022 |
Chen S, Pillitteri S, Fron E, Van Meervelt L, Van der Eycken EV, Sharma UK. Visible-Light-Induced Cascade Difunctionalization of Indoles Enabled by the Synergy of Photoredox and Photoexcited Ketones: Direct Access to Alkylated Pyrrolophenanthridones. Organic Letters. 24: 9386-9391. PMID 36525615 DOI: 10.1021/acs.orglett.2c03697 |
0.451 |
|
| 2022 |
Liu C, Bolognani A, Song L, Van Meervelt L, Peshkov VA, Van der Eycken EV. Gold(I)-Catalyzed Intramolecular Bicyclization: Divergent Construction of Quinazolinone and Ampakine Analogues. Organic Letters. PMID 36374298 DOI: 10.1021/acs.orglett.2c03547 |
0.741 |
|
| 2022 |
Xie Y, Huang L, Feng H, Qi Y, Van der Eycken EV, Feng H. Regio- and Chemoselective Copper-Catalyzed Formal [2+2+2] Cycloaddition of Primary Amines with Arylacetylenes to 2,4,5-Trisubstituted Pyridines. Organic Letters. 24: 6346-6350. PMID 36005451 DOI: 10.1021/acs.orglett.2c02606 |
0.504 |
|
| 2022 |
Song L, Cai L, Van der Eycken EV. Microwave-Assisted Post-Ugi Reactions for the Synthesis of Polycycles. Molecules (Basel, Switzerland). 27. PMID 35630582 DOI: 10.3390/molecules27103105 |
0.468 |
|
| 2022 |
Oliva M, Martens F, Van der Eycken EV, Sharma UK. A continuous-flow protocol for photoredox-catalyzed multicomponent Petasis reaction. Star Protocols. 3: 101162. PMID 35535166 DOI: 10.1016/j.xpro.2022.101162 |
0.442 |
|
| 2022 |
Coppola GA, Pillitteri S, Van der Eycken EV, You SL, Sharma UK. Multicomponent reactions and photo/electrochemistry join forces: atom economy meets energy efficiency. Chemical Society Reviews. 51: 2313-2382. PMID 35244107 DOI: 10.1039/d1cs00510c |
0.442 |
|
| 2022 |
Chen S, Van Meervelt L, Van der Eycken EV, Sharma UK. Visible-Light-Driven Palladium-Catalyzed Radical Tandem Dearomatization of Indoles with Unactivated Alkenes. Organic Letters. 24: 1213-1218. PMID 35107015 DOI: 10.1021/acs.orglett.1c04390 |
0.399 |
|
| 2022 |
Xu X, Feng H, Zhang X, Song L, Van Meervelt L, Van der Eycken J, Harvey JN, Van der Eycken EV. Pd-Catalyzed Ring Restructuring of Oxazolidines with Alkenes Leading to Fused Polycyclic Indolizines. Organic Letters. 24: 1232-1236. PMID 35099981 DOI: 10.1021/acs.orglett.2c00007 |
0.764 |
|
| 2021 |
Song L, Manno R, Ranjan P, Sebastian V, Irusta S, Mallada R, Van Meervelt L, Santamaria J, Van der Eycken EV. Preparation of Cu cluster catalysts by simultaneous cooling-microwave heating: application in radical cascade annulation. Nanoscale Advances. 3: 1087-1095. PMID 36133300 DOI: 10.1039/d0na00980f |
0.343 |
|
| 2021 |
Liu C, Zhao R, Song L, Li Z, Tian G, He Y, Van Meervelt L, Peshkov VA, Van der Eycken EV. Palladium-catalyzed post-Ugi arylative dearomatization/Michael addition cascade towards plicamine analogues. Organic & Biomolecular Chemistry. PMID 34730164 DOI: 10.1039/d1ob01805a |
0.75 |
|
| 2021 |
Oliva M, Ranjan P, Pillitteri S, Coppola GA, Messina M, Van der Eycken EV, Sharma UK. Photoredox-catalyzed multicomponent Petasis reaction in batch and continuous flow with alkyl boronic acids. Iscience. 24: 103134. PMID 34632333 DOI: 10.1016/j.isci.2021.103134 |
0.474 |
|
| 2021 |
Aleti RR, Festa AA, Voskressensky LG, Van der Eycken EV. Synthetic Strategies in the Preparation of Phenanthridinones. Molecules (Basel, Switzerland). 26. PMID 34577030 DOI: 10.3390/molecules26185560 |
0.509 |
|
| 2021 |
Xu X, Feng H, Van der Eycken EV. Microwave-Assisted Palladium-Catalyzed Reductive Cyclization/Ring-Opening/Aromatization Cascade of Oxazolidines to Isoquinolines. Organic Letters. PMID 34379418 DOI: 10.1021/acs.orglett.1c02416 |
0.513 |
|
| 2021 |
Liu C, Song L, Van Meervelt L, Peshkov VA, Li Z, Van der Eycken EV. Palladium-Catalyzed Arylative Dearomatization and Subsequent Aromatization/Dearomatization/Aza-Michael Addition: Access to Zephycarinatine and Zephygranditine Skeletons. Organic Letters. PMID 34115493 DOI: 10.1021/acs.orglett.1c01590 |
0.74 |
|
| 2021 |
Coppola GA, Onsea J, Moriarty TF, Nehrbass D, Constant C, Zeiter S, Aktan MK, Braem A, Van der Eycken EV, Steenackers HP, Metsemakers WJ. An Improved 2-Aminoimidazole Based Anti-Biofilm Coating for Orthopedic Implants: Activity, Stability, and Biocompatibility. Frontiers in Microbiology. 12: 658521. PMID 33967997 DOI: 10.3389/fmicb.2021.658521 |
0.228 |
|
| 2021 |
Xu X, Feng H, Van der Eycken EV. Microwave-Assisted Cu(I)-Catalyzed Synthesis of Unsymmetrical 1,4-Diamino-2-butynes via Cross-A-Coupling/Decarboxylative A-Coupling. The Journal of Organic Chemistry. PMID 33890472 DOI: 10.1021/acs.joc.1c00537 |
0.445 |
|
| 2021 |
Jacobs L, Meesters J, Parijs I, Hooyberghs G, Van der Eycken EV, Lories B, Steenackers HP. 2-Aminoimidazoles as potent inhibitors of contaminating brewery biofilms. Biofouling. 1-17. PMID 33573402 DOI: 10.1080/08927014.2021.1874366 |
0.265 |
|
| 2021 |
Rivera DG, Ricardo MG, Vasco AV, Wessjohann LA, Van der Eycken EV. On-resin multicomponent protocols for biopolymer assembly and derivatization. Nature Protocols. PMID 33473197 DOI: 10.1038/s41596-020-00445-6 |
0.602 |
|
| 2020 |
Song L, Zhang X, Tang X, Van Meervelt L, Van der Eycken J, Harvey JN, Van der Eycken EV. Ruthenium-catalyzed cascade C-H activation/annulation of -alkoxybenzamides: reaction development and mechanistic insight. Chemical Science. 11: 11562-11569. PMID 34094402 DOI: 10.1039/d0sc04434b |
0.748 |
|
| 2020 |
He Y, Song L, Liu C, Wu D, Li Z, Van Meervelt L, Van der Eycken EV. Access to Polycyclic Azepino[5,4,3-]indoles via a Gold-Catalyzed Post-Ugi Dearomatization Cascade. The Journal of Organic Chemistry. PMID 33200934 DOI: 10.1021/acs.joc.0c01972 |
0.479 |
|
| 2020 |
Chen S, Ranjan P, Voskressensky LG, Van der Eycken EV, Sharma UK. Recent Developments in Transition-Metal Catalyzed Direct C-H Alkenylation, Alkylation, and Alkynylation of Azoles. Molecules (Basel, Switzerland). 25. PMID 33121108 DOI: 10.3390/molecules25214970 |
0.418 |
|
| 2020 |
Bührmann L, Schuurmans J, Ruwaard J, Fleuren M, Etzelmüller A, Piera-Jiménez J, Finch T, Rapley T, Potthoff S, Aouizerate B, Batterham PJ, Calear A, Christensen H, Pedersen CD, Ebert DD, ... Van der Eycken E, et al. Tailored implementation of internet-based cognitive behavioural therapy in the multinational context of the ImpleMentAll project: a study protocol for a stepped wedge cluster randomized trial. Trials. 21: 893. PMID 33115545 DOI: 10.1186/s13063-020-04686-4 |
0.207 |
|
| 2020 |
Sharma UK, Ranjan P, Van der Eycken EV, You SL. Sequential and direct multicomponent reaction (MCR)-based dearomatization strategies. Chemical Society Reviews. PMID 33079105 DOI: 10.1039/d0cs00128g |
0.4 |
|
| 2020 |
Tian G, Song L, Li Z, Robeyns K, Van Meervelt L, Van der Eycken EV. A Gold(I)-Catalyzed Hydroamination/Cycloisomerization Cascade: Concise Synthesis of (±)-seco-Antofine and (±)-Septicine. Organic Letters. PMID 33050695 DOI: 10.1021/acs.orglett.0c03062 |
0.368 |
|
| 2020 |
Kumar P, Dutta S, Kumar S, Bahadur V, Van der Eycken EV, Vimaleswaran KS, Parmar VS, Singh BK. Aldehydes: magnificent acyl equivalents for direct acylation. Organic & Biomolecular Chemistry. PMID 33000845 DOI: 10.1039/d0ob01458c |
0.693 |
|
| 2020 |
Sokolova EA, Festa AA, Subramani K, Rybakov VB, Varlamov AV, Voskressensky LG, Van der Eycken EV. Microwave-Assisted Synthesis of Fluorescent Pyrido[2,3-]indolizines from Alkylpyridinium Salts and Enaminones. Molecules (Basel, Switzerland). 25. PMID 32899473 DOI: 10.3390/molecules25184059 |
0.402 |
|
| 2020 |
Reguera L, Cano A, Rodríguez-Hernández J, Rivera DG, Van der Eycken EV, Ramírez-Rosales D, Reguera E. CuCu and Ag-isocyanobenzoates as novel 1D semiconducting coordination oligomers. Dalton Transactions (Cambridge, England : 2003). PMID 32851997 DOI: 10.1039/d0dt02461a |
0.572 |
|
| 2020 |
Song L, Tian G, Van Meervelt L, Van der Eycken EV. Synthesis of Pyrrolo[1,2-]isoquinolines via Gold(I)-Catalyzed Cyclization/Enyne Cycloisomerization/1,2-Migration Cascade. Organic Letters. PMID 32806156 DOI: 10.1021/acs.orglett.0c02310 |
0.473 |
|
| 2020 |
Van der Eycken E, Song L. Transition Metal-Catalyzed Intermolecular Cascade C-H Activation/Annulation Processes for the Synthesis of Polycycles. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 32530508 DOI: 10.1002/chem.202002110 |
0.515 |
|
| 2020 |
Chen S, Ranjan P, Ramkumar N, Meervelt LV, Van der Eycken EV, Sharma UK. Ligand Enabled Palladium-Catalysed Through-Space C-H Bond Activation via a Carbopalladation/1,4-Pd Migration/C-H Functionalization Sequence. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 32497367 DOI: 10.1002/chem.202001582 |
0.422 |
|
| 2020 |
Song L, Claessen S, Van der Eycken EV. Pyridine-Enabled C-N Bond Activation for the Rapid Construction of Amides and 4-Pyridylglyoxamides by Cooperative Palladium/Copper Catalysis. The Journal of Organic Chemistry. PMID 32441517 DOI: 10.1021/acs.joc.0c00845 |
0.413 |
|
| 2020 |
Rivera DG, Ojeda-Carralero GM, Reguera L, Van der Eycken EV. Peptide macrocyclization by transition metal catalysis. Chemical Society Reviews. PMID 32142086 DOI: 10.1039/c9cs00366e |
0.63 |
|
| 2020 |
Dieltjens L, Appermans K, Lissens M, Lories B, Kim W, Van der Eycken EV, Foster KR, Steenackers HP. Inhibiting bacterial cooperation is an evolutionarily robust anti-biofilm strategy. Nature Communications. 11: 107. PMID 31919364 DOI: 10.1038/s41467-019-13660-x |
0.21 |
|
| 2019 |
Storozhenko OA, Festa AA, Detistova GI, Rybakov VB, Varlamov AV, Van der Eycken EV, Voskressensky LG. Photoredox-Catalyzed Hydrosulfonylation of Arylallenes. The Journal of Organic Chemistry. PMID 31874037 DOI: 10.1021/acs.joc.9b02960 |
0.451 |
|
| 2019 |
Ojeda GM, Ranjan P, Fedoseev P, Amable L, Sharma UK, Rivera DG, Van der Eycken EV. Combining the Ugi-azide multicomponent reaction and rhodium(III)-catalyzed annulation for the synthesis of tetrazole-isoquinolone/pyridone hybrids. Beilstein Journal of Organic Chemistry. 15: 2447-2457. PMID 31666879 DOI: 10.3762/bjoc.15.237 |
0.722 |
|
| 2019 |
He Y, Narmon T, Wu D, Li Z, Van Meervelt L, Van der Eycken EV. A gold-triggered dearomative spirocarbocyclization/Diels-Alder reaction cascade towards diverse bridged N-heterocycles. Organic & Biomolecular Chemistry. PMID 31663568 DOI: 10.1039/c9ob01967g |
0.477 |
|
| 2019 |
Li H, Feng H, Zhang J, Van der Eycken EV, Huang L. Synthetic Access to Secondary Propargylamines via Copper-Catalyzed Oxidative Deamination-Alkynylation Cascade. The Journal of Organic Chemistry. PMID 31347364 DOI: 10.1021/acs.joc.9b01431 |
0.427 |
|
| 2019 |
Murlykina MV, Kolomiets OV, Kornet MM, Sakhno YI, Desenko SM, Dyakonenko VV, Shishkina SV, Brazhko OA, Musatov VI, Tsygankov AV, Van der Eycken EV, Chebanov VA. Doebner-type pyrazolopyridine carboxylic acids in an Ugi four-component reaction. Beilstein Journal of Organic Chemistry. 15: 1281-1288. PMID 31293676 DOI: 10.3762/bjoc.15.126 |
0.815 |
|
| 2019 |
Festa AA, Voskressensky LG, Van der Eycken EV. Visible light-mediated chemistry of indoles and related heterocycles. Chemical Society Reviews. PMID 31268435 DOI: 10.1039/c8cs00790j |
0.373 |
|
| 2019 |
He Y, Wu D, Li Z, Robeyns K, Van Meervelt L, Van der Eycken EV. Facile construction of diverse polyheterocyclic scaffolds via gold-catalysed dearomative spirocyclization/1,6-addition cascade. Organic & Biomolecular Chemistry. PMID 31194210 DOI: 10.1039/c9ob01299k |
0.402 |
|
| 2019 |
He Y, Liu Z, Wu D, Li Z, Robeyns K, Van Meervelt L, Van der Eycken EV. Modular Access to Diverse Bridged Indole Alkaloid Mimics via a Gold-Triggered Cascade Dearomative Spirocarbocyclization/[4 + 2] Cycloaddition Sequence. Organic Letters. PMID 31184165 DOI: 10.1021/acs.orglett.9b01296 |
0.466 |
|
| 2019 |
Lipson VV, Pavlovska TL, Svetlichnaya NV, Poryvai AA, Gorobets NY, Van der Eycken EV, Konovalova IS, Shiskina SV, Borisov AV, Musatov VI, Mazepa AV. Novel (2-amino-4-arylimidazolyl)propanoic acids and pyrrolo[1,2-]imidazoles via the domino reactions of 2-amino-4-arylimidazoles with carbonyl and methylene active compounds. Beilstein Journal of Organic Chemistry. 15: 1032-1045. PMID 31164941 DOI: 10.3762/bjoc.15.101 |
0.382 |
|
| 2019 |
Golantsov NE, Nguyen HM, Golubenkova AS, Varlamov AV, Van der Eycken EV, Voskressensky LG. Three-Component Reaction of 3-Arylidene-3-Indolium Salts, Isocyanides, and Alcohols. Frontiers in Chemistry. 7: 345. PMID 31157211 DOI: 10.3389/fchem.2019.00345 |
0.411 |
|
| 2019 |
Van der Eycken E, Song L, Tian G. Chemo- and Regioselective Catalyst-Controlled Carbocyclization of Alkynyl Ketones: Rapid Synthesis of 1-Indanones and 1-Naphthols. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 31017698 DOI: 10.1002/chem.201901860 |
0.373 |
|
| 2019 |
Song L, Tian G, Van der Eycken J, Van der Eycken EV. Intramolecular cascade annulation triggered by rhodium(III)-catalyzed sequential C(sp)-H activation and C(sp)-H amination. Beilstein Journal of Organic Chemistry. 15: 571-576. PMID 30873242 DOI: 10.3762/bjoc.15.52 |
0.691 |
|
| 2019 |
Xiong H, Li Y, Qian B, Wei R, Van der Eycken EV, Bao H. Iron(II)-Catalyzed Heck-Type Coupling of Vinylarenes with Alkyl Iodides. Organic Letters. PMID 30668128 DOI: 10.1021/Acs.Orglett.8B04024 |
0.357 |
|
| 2018 |
Peeters E, Hooyberghs G, Robijns S, De Weerdt A, Kucharíková S, Tournu H, Braem A, Čeh K, Majdič G, Španič T, Pogorevc E, Claes B, Dovgan B, Girandon L, Impellizzeri F, ... ... Van der Eycken E, et al. An antibiofilm coating of 5-aryl-2-aminoimidazole covalently attached to a titanium surface. Journal of Biomedical Materials Research. Part B, Applied Biomaterials. PMID 30549192 DOI: 10.1002/Jbm.B.34283 |
0.251 |
|
| 2018 |
Bariwal J, Kaur R, Voskressensky LG, Van der Eycken EV. Post-Ugi Cyclization for the Construction of Diverse Heterocyclic Compounds: Recent Updates. Frontiers in Chemistry. 6: 557. PMID 30525022 DOI: 10.3389/Fchem.2018.00557 |
0.751 |
|
| 2018 |
Ranjan P, Ojeda GM, Sharma UK, Van der Eycken E. Metal-Free Dearomatization: Direct access to Spiroindol(en)ines in Batch and Continuous-Flow. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 30507048 DOI: 10.1002/chem.201805945 |
0.424 |
|
| 2018 |
Ilya E, Kulikova L, Van der Eycken EV, Voskressensky L. Recent Advances in Phthalan and Coumaran Chemistry. Chemistryopen. 7: 914-929. PMID 30498677 DOI: 10.1002/open.201800184 |
0.318 |
|
| 2018 |
Sharma UK, Tian G, Voskressensky LG, Van der Eycken EV. Gold-catalyzed post-MCR transformations towards complex (poly)heterocycles. Drug Discovery Today. Technologies. 29: 61-69. PMID 30471675 DOI: 10.1016/j.ddtec.2018.08.003 |
0.396 |
|
| 2018 |
Ramkumar N, Van Meervelt L, Van der Eycken EV. Iron-Catalyzed Three-Component Reaction: Synthesis of Fluoroalkylated 2 H-Azirines. Organic Letters. PMID 30461283 DOI: 10.1021/acs.orglett.8b03324 |
0.459 |
|
| 2018 |
Titov AA, Samavati R, Alexandrova EV, Borisova TN, Dang Thi TA, Nguyen VT, Le TA, Varlamov AV, Van der Eycken EV, Voskressensky LG. Synthesis of 1-(-methoxyphenyl)tetrazolyl-Substituted 1,2,3,4-Tetrahydroisoquinolines and Their Transformations Involving Activated Alkynes. Molecules (Basel, Switzerland). 23. PMID 30453635 DOI: 10.3390/molecules23113010 |
0.414 |
|
| 2018 |
Du X, Huang J, Nechaev AA, Yao R, Gong J, Van der Eycken EV, Pereshivko OP, Peshkov VA. Gold-catalyzed post-Ugi alkyne hydroarylation for the synthesis of 2-quinolones. Beilstein Journal of Organic Chemistry. 14: 2572-2579. PMID 30410618 DOI: 10.3762/Bjoc.14.234 |
0.747 |
|
| 2018 |
Nechaev AA, Van Hecke K, Zaman M, Kashtanov S, Ungur L, Pereshivko OP, Peshkov VA, Van der Eycken EV. Gold-Catalyzed Post-Ugi Ipso-Cyclization with Switchable Diastereoselectivity. The Journal of Organic Chemistry. PMID 29966417 DOI: 10.1021/Acs.Joc.8B00953 |
0.723 |
|
| 2018 |
Festa AA, Zalte RR, Golantsov NE, Varlamov AV, Van der Eycken EV, Voskressensky LG. DBU-Catalyzed Alkyne-Imidate Cyclization towards 1-Alkoxypyrazino[1,2-a]indole Synthesis. The Journal of Organic Chemistry. PMID 29944827 DOI: 10.1021/acs.joc.8b01279 |
0.44 |
|
| 2018 |
Mishra NM, Stolarzewicz I, Cannaerts D, Schuermans J, Lavigne R, Looz Y, Landuyt B, Schoofs L, Schols D, Paeshuyse J, Hickenbotham P, Clokie M, Luyten W, Van der Eycken EV, Briers Y. Iterative Chemical Engineering of Vancomycin Leads to Novel Vancomycin Analogs With a High Therapeutic Index. Frontiers in Microbiology. 9: 1175. PMID 29930540 DOI: 10.3389/fmicb.2018.01175 |
0.249 |
|
| 2018 |
Bariwal J, Voskressensky LG, Van der Eycken EV. Recent advances in spirocyclization of indole derivatives. Chemical Society Reviews. PMID 29632917 DOI: 10.1039/C7Cs00508C |
0.723 |
|
| 2018 |
Fedoseev P, Coppola G, Ojeda GM, Van der Eycken EV. Synthesis of spiroindolenines by intramolecular ipso-iodocyclization of indol ynones. Chemical Communications (Cambridge, England). 54: 3625-3628. PMID 29577155 DOI: 10.1039/c8cc01474d |
0.439 |
|
| 2018 |
Peshkov VA, Pereshivko OP, Nechaev AA, Peshkov AA, Van der Eycken EV. Reactions of secondary propargylamines with heteroallenes for the synthesis of diverse heterocycles. Chemical Society Reviews. PMID 29546891 DOI: 10.1039/C7Cs00065K |
0.722 |
|
| 2018 |
Trang TTT, Dieltjens L, Hooyberghs G, Waldrant K, Ermolat'ev DS, Van der Eycken EV, Steenackers HPL. Enhancing the anti-biofilm activity of 5-aryl-2-aminoimidazoles through nature inspired dimerisation. Bioorganic & Medicinal Chemistry. PMID 29449125 DOI: 10.1016/j.bmc.2018.01.005 |
0.341 |
|
| 2017 |
Van der Eycken E, He Y, Li Z, Robeyns K, Van Meervelt L. A Gold-Catalyzed Domino Cyclization Enabling Rapid Construction of Diverse Polyheterocyclic Frameworks. Angewandte Chemie (International Ed. in English). PMID 29144011 DOI: 10.1002/anie.201710592 |
0.494 |
|
| 2017 |
Lima F, Sharma UK, Grunenberg L, Saha D, Johannsen S, Sedelmeier J, Van der Eycken EV, Ley SV. A Lewis Base Catalysis Approach for the Photoredox Activation of Boronic Acids and Esters. Angewandte Chemie (International Ed. in English). PMID 29024307 DOI: 10.1002/Anie.201709690 |
0.741 |
|
| 2017 |
Song L, Tian G, He Y, Van der Eycken EV. Rhodium(iii)-catalyzed intramolecular annulation through C-H activation: concise synthesis of rosettacin and oxypalmatime. Chemical Communications (Cambridge, England). PMID 28956561 DOI: 10.1039/c7cc06860c |
0.536 |
|
| 2017 |
Singh S, Butani HH, Vachhani DD, Shah A, Van der Eycken EV. Ruthenium-catalysed one-pot regio- and diastereoselective synthesis of pyrrolo[1,2-a]indoles via cascade C-H functionalization/annulation. Chemical Communications (Cambridge, England). PMID 28920982 DOI: 10.1039/C7Cc06276A |
0.796 |
|
| 2017 |
Murlykina MV, Kornet MN, Desenko SM, Shishkina SV, Shishkin OV, Brazhko AA, Musatov VI, Van der Eycken EV, Chebanov VA. New tricks of well-known aminoazoles in isocyanide-based multicomponent reactions and antibacterial activity of the compounds synthesized. Beilstein Journal of Organic Chemistry. 13: 1050-1063. PMID 28684984 DOI: 10.3762/bjoc.13.104 |
0.436 |
|
| 2017 |
Gill RK, Kumar V, Robijns SCA, Steenackers HPL, Van der Eycken EV, Bariwal J. Polysubstituted 2-aminoimidazoles as anti-biofilm and antiproliferative agents: Discovery of potent lead. European Journal of Medicinal Chemistry. 138: 152-169. PMID 28667872 DOI: 10.1016/J.Ejmech.2017.06.043 |
0.689 |
|
| 2017 |
He Y, Li Z, Tian G, Song L, Van Meervelt L, Van der Eycken EV. Gold-catalyzed diastereoselective domino dearomatization/ipso-cyclization/aza-Michael sequence: a facile access to diverse fused azaspiro tetracyclic scaffolds. Chemical Communications (Cambridge, England). PMID 28569296 DOI: 10.1039/c7cc03152a |
0.49 |
|
| 2017 |
Fedoseev P, Van der Eycken E. Temperature switchable Brønsted acid-promoted selective syntheses of spiro-indolenines and quinolines. Chemical Communications (Cambridge, England). 53: 7732-7735. PMID 28492644 DOI: 10.1039/c7cc02580g |
0.362 |
|
| 2017 |
Tian G, Fedoseev P, Van der Eycken E. Hypervalent Iodine(III)-Mediated Cascade Cyclization of Propargylguanidines and Total Syntheses of Kealiinines B and C. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28263005 DOI: 10.1002/chem.201700934 |
0.418 |
|
| 2017 |
Claes B, Boudewijns T, Muchez L, Hooyberghs G, Van der Eycken EV, Vanderleyden J, Steenackers HP, De Vos DE. Smart Metal-Organic Framework Coatings: Triggered Antibiofilm Compound Release. Acs Applied Materials & Interfaces. 9: 4440-4449. PMID 28081368 DOI: 10.1021/acsami.6b14152 |
0.263 |
|
| 2016 |
Sutens B, Swusten T, Zhong K, Jochum JK, Van Bael MJ, Van der Eycken EV, Brullot W, Bloemen M, Verbiest T. Tunability of Size and Magnetic Moment of Iron Oxide Nanoparticles Synthesized by Forced Hydrolysis. Materials (Basel, Switzerland). 9. PMID 28773675 DOI: 10.3390/ma9070554 |
0.232 |
|
| 2016 |
Peeters E, Hooyberghs G, Robijns S, Waldrant K, De Weerdt A, Delattin N, Liebens V, Kucharíková S, Tournu H, Verstraeten N, Dovgan B, Girandon L, Fröhlich M, De Brucker K, Van Dijck P, ... ... Van der Eycken E, et al. Modulation of the Substitution Pattern of 5-Aryl-2-Aminoimidazoles Allows Fine-Tuning of Their Antibiofilm Activity Spectrum and Toxicity. Antimicrobial Agents and Chemotherapy. 60: 6483-6497. PMID 27550355 DOI: 10.1128/Aac.00035-16 |
0.332 |
|
| 2016 |
Sharma PK, Balwani S, Mathur D, Malhotra S, Singh BK, Prasad AK, Len C, Van der Eycken EV, Ghosh B, Richards NG, Parmar VS. Synthesis and anti-inflammatory activity evaluation of novel triazolyl-isatin hybrids. Journal of Enzyme Inhibition and Medicinal Chemistry. 31: 1520-6. PMID 27146339 DOI: 10.3109/14756366.2016.1151015 |
0.504 |
|
| 2016 |
Zhao Y, Li Z, Sharma UK, Sharma N, Song G, Van der Eycken EV. Copper-catalyzed alkylarylation of activated alkenes using isocyanides as the alkyl source: an efficient radical access to 3,3-dialkylated oxindoles. Chemical Communications (Cambridge, England). PMID 27086905 DOI: 10.1039/c6cc02024k |
0.465 |
|
| 2016 |
Li Z, Sharma N, Sharma UK, Jacobs J, Van Meervelt L, Van der Eycken EV. Ligand-controlled product selectivity in palladium-catalyzed domino post-Ugi construction of (spiro)polyheterocycles. Chemical Communications (Cambridge, England). PMID 26964634 DOI: 10.1039/c6cc00784h |
0.349 |
|
| 2016 |
Zhao Y, Sharma N, Sharma UK, Li Z, Song G, Van Der Eycken E. Microwave-Assisted Copper-Catalyzed Oxidative Cyclization of Acrylamides with Non-Activated Ketones. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 26868308 DOI: 10.1002/chem.201504776 |
0.46 |
|
| 2015 |
Sharma UK, Sharma N, Kumar Y, Singh BK, Van Der Eycken E. Domino carbopalladation/C-H functionalization sequence: an expedient synthesis of bis-heteroaryls via transient alkyl/vinyl palladium species capture. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 26584957 DOI: 10.1002/chem.201503708 |
0.509 |
|
| 2015 |
Kumar A, Singh S, Sharma SK, Parmar VS, Van der Eycken EV. Gold-Catalyzed Cyclization Processes: Pivotal Avenues for Organic Synthesis. Chemical Record (New York, N.Y.). PMID 26554536 DOI: 10.1002/tcr.201500230 |
0.588 |
|
| 2015 |
Vachhani DD, Butani HH, Sharma N, Bhoya UC, Shah AK, Van der Eycken EV. Domino Heck/borylation sequence towards indolinone-3-methyl boronic esters: trapping of the σ-alkylpalladium intermediate with boron. Chemical Communications (Cambridge, England). 51: 14862-5. PMID 26300449 DOI: 10.1039/c5cc05193b |
0.793 |
|
| 2015 |
Mishra NM, Briers Y, Lamberigts C, Steenackers H, Robijns S, Landuyt B, Vanderleyden J, Schoofs L, Lavigne R, Luyten W, Van der Eycken EV. Evaluation of the antibacterial and antibiofilm activities of novel CRAMP-vancomycin conjugates with diverse linkers. Organic & Biomolecular Chemistry. 13: 7477-86. PMID 26068402 DOI: 10.1039/c5ob00830a |
0.305 |
|
| 2015 |
Peshkov AA, Peshkov VA, Pereshivko OP, Van Hecke K, Kumar R, Van der Eycken EV. Heck-Suzuki Tandem Reaction for the Synthesis of 3-Benzazepines. The Journal of Organic Chemistry. 80: 6598-608. PMID 25996648 DOI: 10.1021/Acs.Joc.5B00670 |
0.747 |
|
| 2015 |
Kumar S, Malhotra S, Prasad AK, Van der Eycken EV, Bracke ME, Stetler-Stevenson WG, Parmar VS, Ghosh B. Anti-inflammatory and antioxidant properties of Piper species: a perspective from screening to molecular mechanisms. Current Topics in Medicinal Chemistry. 15: 886-93. PMID 25697561 |
0.447 |
|
| 2015 |
Sharma UK, Sharma N, Xu J, Song G, Van der Eycken EV. Pd-catalyzed Csp(2) -H functionalization of heteroarenes via isocyanide insertion: concise synthesis of di-(hetero)aryl ketones and di-(hetero)aryl alkylamines. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 4908-12. PMID 25663081 DOI: 10.1002/chem.201406562 |
0.5 |
|
| 2015 |
Sharma UK, Sharma N, Vachhani DD, Van der Eycken EV. Metal-mediated post-Ugi transformations for the construction of diverse heterocyclic scaffolds. Chemical Society Reviews. 44: 1836-60. PMID 25652577 DOI: 10.1039/c4cs00253a |
0.744 |
|
| 2014 |
Steenackers H, Dubey A, Robijns S, Ermolat'ev D, Delattin N, Dovgan B, Girandon L, Fröhlich M, De Brucker K, Cammue BP, Thevissen K, Balzarini J, Van der Eycken EV, Vanderleyden J. Evaluation of the toxicity of 5-aryl-2-aminoimidazole-based biofilm inhibitors against eukaryotic cell lines, bone cells and the nematode Caenorhabditis elegans. Molecules (Basel, Switzerland). 19: 16707-23. PMID 25325155 DOI: 10.3390/Molecules191016707 |
0.314 |
|
| 2014 |
Ambasana PA, Vachhani DD, Galli M, Jacobs J, Van Meervelt L, Shah AK, Van der Eycken EV. Solvent switchable cycloaddition: a (one-pot) metal-free approach towards N-substituted benzo[e]- or [f]isoindolones via C(sp(2))-H functionalization. Organic & Biomolecular Chemistry. 12: 8861-5. PMID 25257733 DOI: 10.1039/c4ob01644k |
0.767 |
|
| 2014 |
Peshkov VA, Peshkov AA, Pereshivko OP, Van Hecke K, Zamigaylo LL, Van der Eycken EV, Gorobets NY. Three-component reaction of a 2-aminoazine, a 2-oxoaldehyde, and a cyclic 1,3-dicarbonyl compound for the synthesis of imidazo[1,2-a]azine derivatives. Acs Combinatorial Science. 16: 535-42. PMID 25170540 DOI: 10.1021/Co5000695 |
0.727 |
|
| 2014 |
Sharma N, Li Z, Sharma UK, Van der Eycken EV. Facile access to functionalized spiro[indoline-3,2'-pyrrole]-2,5'-diones via post-Ugi domino Buchwald-Hartwig/Michael reaction. Organic Letters. 16: 3884-7. PMID 25029554 DOI: 10.1021/ol5019079 |
0.47 |
|
| 2014 |
Kumar Y, Bahadur V, Singh AK, Parmar VS, Van der Eycken EV, Singh BK. Microwave-assisted Cu(I)-catalyzed, three-component synthesis of 2-(4-((1-phenyl-1H-1,2,3-triazol-4-yl)methoxy)phenyl)-1H-benzo[d]imidazoles. Beilstein Journal of Organic Chemistry. 10: 1413-20. PMID 24991296 DOI: 10.3762/bjoc.10.145 |
0.548 |
|
| 2014 |
Steenackers H, Ermolat'ev D, Trang TT, Savalia B, Sharma UK, De Weerdt A, Shah A, Vanderleyden J, Van der Eycken EV. Microwave-assisted one-pot synthesis and anti-biofilm activity of 2-amino-1H-imidazole/triazole conjugates. Organic & Biomolecular Chemistry. 12: 3671-8. PMID 24763714 DOI: 10.1039/C3Ob42282H |
0.662 |
|
| 2014 |
Pereshivko OP, Peshkov VA, Peshkov AA, Jacobs J, Van Meervelt L, Van der Eycken EV. Unexpected regio- and chemoselectivity of cationic gold-catalyzed cycloisomerizations of propargylureas: access to tetrasubstituted 3,4-dihydropyrimidin-2(1H)-ones. Organic & Biomolecular Chemistry. 12: 1741-50. PMID 24492944 DOI: 10.1039/C3Ob42221F |
0.749 |
|
| 2013 |
Kumar A, Vachhani DD, Modha SG, Sharma SK, Parmar VS, Van der Eycken EV. Post-Ugi gold-catalyzed diastereoselective domino cyclization for the synthesis of diversely substituted spiroindolines. Beilstein Journal of Organic Chemistry. 9: 2097-102. PMID 24204421 DOI: 10.3762/Bjoc.9.246 |
0.818 |
|
| 2013 |
Bariwal J, Van der Eycken E. C-N bond forming cross-coupling reactions: an overview. Chemical Society Reviews. 42: 9283-303. PMID 24077333 DOI: 10.1039/C3Cs60228A |
0.732 |
|
| 2013 |
Cavalluzzo C, Christ F, Voet A, Sharma A, Singh BK, Zhang KY, Lescrinier E, De Maeyer M, Debyser Z, Van der Eycken E. Identification of small peptides inhibiting the integrase-LEDGF/p75 interaction through targeting the cellular co-factor. Journal of Peptide Science : An Official Publication of the European Peptide Society. 19: 651-8. PMID 24014475 DOI: 10.1002/Psc.2543 |
0.237 |
|
| 2013 |
Vachhani DD, Galli M, Jacobs J, Van Meervelt L, Van der Eycken EV. Synthesis of (spiro)cyclopentapyridinones via C(sp3)-H functionalization: a post-Ugi gold-catalyzed regioselective tandem cyclization. Chemical Communications (Cambridge, England). 49: 7171-3. PMID 23831954 DOI: 10.1039/c3cc43418d |
0.776 |
|
| 2013 |
Kumar A, Li Z, Sharma SK, Parmar VS, Van der Eycken EV. Switching the regioselectivity via indium(III) and gold(I) catalysis: a post-Ugi intramolecular hydroarylation to azepino- and azocino-[c,d]indolones. Chemical Communications (Cambridge, England). 49: 6803-5. PMID 23783807 DOI: 10.1039/c3cc42704h |
0.54 |
|
| 2013 |
Kumar R, Ermolat'ev DS, Van der Eycken EV. Synthesis of differentially substituted 2-aminoimidazolidines via a microwave-assisted tandem Staudinger/aza-Wittig cyclization. The Journal of Organic Chemistry. 78: 5737-43. PMID 23641751 DOI: 10.1021/jo400481b |
0.459 |
|
| 2013 |
Kumar A, Li Z, Sharma SK, Parmar VS, Van der Eycken EV. An expedient route to imidazo[1,4]diazepin-7-ones via a post-Ugi gold-catalyzed heteroannulation. Organic Letters. 15: 1874-7. PMID 23544989 DOI: 10.1021/ol400526a |
0.58 |
|
| 2013 |
Modha SG, Mehta VP, Van der Eycken EV. Transition metal-catalyzed C-C bond formation via C-S bond cleavage: an overview. Chemical Society Reviews. 42: 5042-55. PMID 23467811 DOI: 10.1039/C3Cs60041F |
0.787 |
|
| 2013 |
Vachhani DD, Sharma A, Van der Eycken E. Copper-catalyzed direct secondary and tertiary C-H alkylation of azoles through a heteroarene-amine-aldehyde/ketone coupling reaction. Angewandte Chemie (International Ed. in English). 52: 2547-50. PMID 23341157 DOI: 10.1002/Anie.201209312 |
0.835 |
|
| 2013 |
Sharma A, Vacchani D, Van der Eycken E. Developments in direct C-H arylation of (hetero)arenes under microwave irradiation. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 1158-68. PMID 23293098 DOI: 10.1002/Chem.201201868 |
0.686 |
|
| 2013 |
Pitta E, Geronikaki A, Surmava S, Eleftheriou P, Mehta VP, Van der Eycken EV. Synthesis and HIV-1 RT inhibitory action of novel (4/6-substituted benzo[d]thiazol -2-yl)thiazolidin-4-ones. Divergence from the non-competitive inhibition mechanism. Journal of Enzyme Inhibition and Medicinal Chemistry. 28: 113-22. PMID 22380777 DOI: 10.3109/14756366.2011.636362 |
0.29 |
|
| 2012 |
Modha SG, Kumar A, Vachhani DD, Sharma SK, Parmar VS, Van der Eycken EV. Gold(I) and platinum(II) switch: a post-Ugi intramolecular hydroarylation to pyrrolopyridinones and pyrroloazepinones. Chemical Communications (Cambridge, England). 48: 10916-8. PMID 23032641 DOI: 10.1039/C2Cc35900F |
0.798 |
|
| 2012 |
Vachhani DD, Sharma A, Van der Eycken E. Pd/Cu-catalyzed C-H arylation of 1,3,4-thiadiazoles with (hetero)aryl iodides, bromides, and triflates. The Journal of Organic Chemistry. 77: 8768-74. PMID 22957511 DOI: 10.1021/Jo301401Q |
0.806 |
|
| 2012 |
Modha SG, Kumar A, Vachhani DD, Jacobs J, Sharma SK, Parmar VS, Van Meervelt L, Van der Eycken EV. A diversity-oriented approach to spiroindolines: post-Ugi gold-catalyzed diastereoselective domino cyclization. Angewandte Chemie (International Ed. in English). 51: 9572-5. PMID 22907654 DOI: 10.1002/Anie.201205052 |
0.819 |
|
| 2012 |
Modha SG, Vachhani DD, Jacobs J, Van Meervelt L, Van der Eycken EV. A concise route to indoloazocines via a sequential Ugi-gold-catalyzed intramolecular hydroarylation. Chemical Communications (Cambridge, England). 48: 6550-2. PMID 22622200 DOI: 10.1039/C2Cc32586A |
0.826 |
|
| 2012 |
Feng H, Ermolat'ev DS, Song G, Van der Eycken EV. Synthesis of symmetric 1,4-diamino-2-butynes via a Cu(I)-catalyzed one-pot A3-coupling/decarboxylative coupling of a propiolic acid, an aldehyde, and an amine. The Journal of Organic Chemistry. 77: 5149-54. PMID 22563934 DOI: 10.1021/jo300562j |
0.43 |
|
| 2012 |
Feng H, Ermolat'ev DS, Song G, Van der Eycken EV. Regioselective Cu(I)-catalyzed tandem A3-coupling/decarboxylative coupling to 3-amino-1,4-enynes. Organic Letters. 14: 1942-5. PMID 22455453 DOI: 10.1021/ol3006612 |
0.477 |
|
| 2012 |
Peshkov VA, Pereshivko OP, Van der Eycken EV. A walk around the A3-coupling. Chemical Society Reviews. 41: 3790-807. PMID 22422343 DOI: 10.1039/C2Cs15356D |
0.714 |
|
| 2012 |
Sharma A, Vachhani D, Van der Eycken E. Direct heteroarylation of tautomerizable heterocycles into unsymmetrical and symmetrical biheterocycles via Pd/Cu-catalyzed phosphonium coupling. Organic Letters. 14: 1854-7. PMID 22416815 DOI: 10.1021/Ol300455E |
0.786 |
|
| 2012 |
Kumar S, Reddy L CS, Kumar Y, Kumar A, Singh BK, Kumar V, Malhotra S, Pandey MK, Jain R, Thimmulappa R, Sharma SK, Prasad AK, Biswal S, Van der Eycken E, DePass AL, et al. Arylalkyl ketones, benzophenones, desoxybenzoins and chalcones inhibit TNF-α induced expression of ICAM-1: structure-activity analysis. Archiv Der Pharmazie. 345: 368-77. PMID 22190402 DOI: 10.1002/Ardp.201100279 |
0.567 |
|
| 2012 |
Sharma A, Appukkuttan P, Van der Eycken E. Microwave-assisted synthesis of medium-sized heterocycles. Chemical Communications (Cambridge, England). 48: 1623-37. PMID 22031184 DOI: 10.1039/C1Cc15238F |
0.655 |
|
| 2011 |
Kumar S, Singh BK, Arya P, Malhotra S, Thimmulappa R, Prasad AK, Van der Eycken E, Olsen CE, DePass AL, Biswal S, Parmar VS, Ghosh B. Novel natural product-based cinnamates and their thio and thiono analogs as potent inhibitors of cell adhesion molecules on human endothelial cells. European Journal of Medicinal Chemistry. 46: 5498-511. PMID 21955679 DOI: 10.1016/J.Ejmech.2011.09.008 |
0.488 |
|
| 2011 |
Feng H, Ermolat'ev DS, Song G, Van der Eycken EV. Microwave-assisted decarboxylative three-component coupling of a 2-oxoacetic acid, an amine, and an alkyne. The Journal of Organic Chemistry. 76: 7608-13. PMID 21823621 DOI: 10.1021/jo2013725 |
0.413 |
|
| 2011 |
Mehta VP, Van der Eycken EV. Microwave-assisted C-C bond forming cross-coupling reactions: an overview. Chemical Society Reviews. 40: 4925-36. PMID 21717007 DOI: 10.1039/c1cs15094d |
0.44 |
|
| 2011 |
Peshkov VA, Pereshivko OP, Sharma S, Meganathan T, Parmar VS, Ermolat'ev DS, Van der Eycken EV. Tetrasubstituted 2-imidazolones via Ag(I)-catalyzed cycloisomerization of propargylic ureas. The Journal of Organic Chemistry. 76: 5867-72. PMID 21639124 DOI: 10.1021/Jo200789T |
0.75 |
|
| 2011 |
Steenackers HP, Ermolat'ev DS, Savaliya B, Weerdt AD, Coster DD, Shah A, Van der Eycken EV, De Vos DE, Vanderleyden J, De Keersmaecker SC. Structure-activity relationship of 2-hydroxy-2-aryl-2,3-dihydro-imidazo[1,2-a]pyrimidinium salts and 2N-substituted 4(5)-aryl-2-amino-1H-imidazoles as inhibitors of biofilm formation by Salmonella Typhimurium and Pseudomonas aeruginosa. Bioorganic & Medicinal Chemistry. 19: 3462-73. PMID 21550812 DOI: 10.1016/J.Bmc.2011.04.026 |
0.627 |
|
| 2011 |
Mehta VP, Sharma Ak, Modha SG, Sharma S, Meganathan T, Parmar VS, Van der Eycken E. N-heterocyclic carbene catalyzed aroylation of 3,5-dichloro-2(1H)-pyrazinones. The Journal of Organic Chemistry. 76: 2920-5. PMID 21405078 DOI: 10.1021/Jo200155N |
0.799 |
|
| 2011 |
Mehta VP, Modha SG, Ruijter E, Van Hecke K, Van Meervelt L, Pannecouque C, Balzarini J, Orru RV, Van der Eycken E. A microwave-assisted diastereoselective multicomponent reaction to access dibenzo[c,e]azepinones: synthesis and biological evaluation. The Journal of Organic Chemistry. 76: 2828-39. PMID 21391618 DOI: 10.1021/Jo200251Q |
0.78 |
|
| 2011 |
Modha SG, Trivedi JC, Mehta VP, Ermolat'ev DS, Van der Eycken EV. An expeditious route toward pyrazine-containing nucleoside analogues. The Journal of Organic Chemistry. 76: 846-56. PMID 21214232 DOI: 10.1021/Jo102089H |
0.788 |
|
| 2011 |
Steenackers HP, Ermolat'ev DS, Savaliya B, De Weerdt A, De Coster D, Shah A, Van der Eycken EV, De Vos DE, Vanderleyden J, De Keersmaecker SC. Structure-activity relationship of 4(5)-aryl-2-amino-1H-imidazoles, N1-substituted 2-aminoimidazoles and imidazo[1,2-a]pyrimidinium salts as inhibitors of biofilm formation by Salmonella typhimurium and Pseudomonas aeruginosa. Journal of Medicinal Chemistry. 54: 472-84. PMID 21174477 DOI: 10.1021/Jm1011148 |
0.637 |
|
| 2010 |
Ermolat'ev DS, Bariwal JB, Steenackers HP, De Keersmaecker SC, Van der Eycken EV. Concise and diversity-oriented route toward polysubstituted 2-aminoimidazole alkaloids and their analogues. Angewandte Chemie (International Ed. in English). 49: 9465-8. PMID 20963737 DOI: 10.1002/anie.201004256 |
0.696 |
|
| 2010 |
Ermolat'ev DS, Savaliya B, Shah A, Van der Eycken E. One-pot microwave-assisted protocol for the synthesis of substituted 2-amino-1H-imidazoles. Molecular Diversity. 15: 491-6. PMID 20740313 DOI: 10.1007/S11030-010-9270-5 |
0.664 |
|
| 2010 |
Bariwal JB, Ermolat'ev DS, Glasnov TN, Van Hecke K, Mehta VP, Van Meervelt L, Kappe CO, Van der Eycken EV. Diversity-oriented synthesis of dibenzoazocines and dibenzoazepines via a microwave-assisted intramolecular A(3)-coupling reaction. Organic Letters. 12: 2774-7. PMID 20481446 DOI: 10.1021/ol1008729 |
0.77 |
|
| 2010 |
Pereshivko OP, Peshkov VA, Van der Eycken EV. Unprecedented Cu(I)-catalyzed microwave-assisted three-component coupling of a ketone, an alkyne, and a primary amine. Organic Letters. 12: 2638-41. PMID 20441203 DOI: 10.1021/Ol1008312 |
0.698 |
|
| 2010 |
Appukkuttan P, Mehta VP, Van der Eycken EV. Microwave-assisted cycloaddition reactions. Chemical Society Reviews. 39: 1467-77. PMID 20419202 DOI: 10.1039/b815717k |
0.441 |
|
| 2010 |
Kappe CO, Van der Eycken E. Click chemistry under non-classical reaction conditions. Chemical Society Reviews. 39: 1280-90. PMID 20309486 DOI: 10.1039/b901973c |
0.406 |
|
| 2010 |
Bariwal JB, Ermolat'ev DS, Van der Eycken EV. Efficient microwave-assisted synthesis of secondary alkylpropargylamines by using A3-coupling with primary aliphatic amines. Chemistry (Weinheim An Der Bergstrasse, Germany). 16: 3281-4. PMID 20162654 DOI: 10.1002/chem.200903143 |
0.711 |
|
| 2010 |
Modha SG, Mehta VP, Ermolat'ev D, Balzarini J, Van Hecke K, Van Meervelt L, Van der Eycken E. Microwave-assisted synthesis of a novel class of imidazolylthiazolidin-4-ones and evaluation of its biological activities. Molecular Diversity. 14: 767-76. PMID 20084456 DOI: 10.1007/S11030-009-9221-1 |
0.751 |
|
| 2010 |
Mehta VP, Modha SG, Van der Eycken EV. Microwave-assisted palladium-catalyzed phosphonium coupling of 2(1H)-pyrazinones. The Journal of Organic Chemistry. 75: 976-9. PMID 20039626 DOI: 10.1021/Jo9024754 |
0.794 |
|
| 2010 |
Claerhout S, Duchène T, Tourwé D, Van der Eycken EV. Development of a new microwave-assisted cleavable backbone amide linker (BAL): a comparative study. Organic & Biomolecular Chemistry. 8: 60-5. PMID 20024133 DOI: 10.1039/b919365k |
0.311 |
|
| 2009 |
Mehta VP, Modha SG, Van der Eycken E. Mild room-temperature palladium-catalyzed C3-arylation of 2(1H)-pyrazinones via a desulfitative Kumada-type cross-coupling reaction. The Journal of Organic Chemistry. 74: 6870-3. PMID 19650631 DOI: 10.1021/Jo901327Y |
0.795 |
|
| 2009 |
Donets PA, Van Hecke K, Van Meervelt L, Van der Eycken EV. Efficient synthesis of the indoloazocine framework via intramolecular alkyne carbocyclization. Organic Letters. 11: 3618-21. PMID 19610606 DOI: 10.1021/ol901356h |
0.5 |
|
| 2009 |
Dolka C, Van Hecke K, Van Meervelt L, Tsoungas PG, Van der Eycken EV, Varvounis G. Novel thermal and microwave-assisted facile route to naphthalen-2(1H)-ones via an oxidative alkoxylation-ring-opening protocol. Organic Letters. 11: 2964-7. PMID 19586060 DOI: 10.1021/ol9008574 |
0.415 |
|
| 2009 |
François IE, Cammue BP, Bresseleers S, Fleuren H, Hoornaert G, Mehta VP, Modha SG, Van der Eycken EV, Thevissen K. Synthesis and fungicidal activity of 3,5-dichloropyrazin-2(1H)-one derivatives. Bioorganic & Medicinal Chemistry Letters. 19: 4064-6. PMID 19556127 DOI: 10.1016/J.Bmcl.2009.06.024 |
0.756 |
|
| 2008 |
Mont N, Mehta VP, Appukkuttan P, Beryozkina T, Toppet S, Van Hecke K, Van Meervelt L, Voet A, DeMaeyer M, Van der Eycken E. Diversity oriented microwave-assisted synthesis of (-)-steganacin aza-analogues. The Journal of Organic Chemistry. 73: 7509-16. PMID 18754579 DOI: 10.1021/jo801290j |
0.5 |
|
| 2008 |
Ermolat'ev DS, Van der Eycken EV. A divergent synthesis of substituted 2-aminoimidazoles from 2-aminopyrimidines. The Journal of Organic Chemistry. 73: 6691-7. PMID 18656979 DOI: 10.1021/jo8008758 |
0.471 |
|
| 2008 |
Claerhout S, Ermolat'ev DS, Van der Eycken EV. A new colorimetric test for solid-phase amines and thiols. Journal of Combinatorial Chemistry. 10: 580-5. PMID 18543976 DOI: 10.1021/cc800031y |
0.232 |
|
| 2008 |
Mehta VP, Sharma A, Van der Eycken E. The first palladium-catalyzed desulfitative Sonogashira-type cross-coupling of (hetero)aryl thioethers with terminal alkynes. Organic Letters. 10: 1147-50. PMID 18284248 DOI: 10.1021/ol800054b |
0.624 |
|
| 2007 |
Appukkuttan P, Dehaen W, Van der Eycken E. Suzuki-Miyaura and Stille reactions as key steps in the synthesis of diversely functionalized Amaryllidaceae alkaloid analogs bearing a 5,6,7,8-tetrahydrobenzo[c,e]azocine skeleton. Combinatorial Chemistry & High Throughput Screening. 10: 790-801. PMID 18478960 DOI: 10.2174/138620707783018513 |
0.518 |
|
| 2007 |
Singh BK, Mehta VP, Parmar VS, Van der Eycken E. Palladium-catalyzed copper(I)-mediated cross-coupling of arylboronic acids and 2(1H)-pyrazinones facilitated by microwave irradiation with simultaneous cooling. Organic & Biomolecular Chemistry. 5: 2962-5. PMID 17728862 DOI: 10.1039/b704389a |
0.567 |
|
| 2007 |
Donets PA, Van der Eycken EV. Efficient synthesis of the 3-benzazepine framework via intramolecular Heck reductive cyclization. Organic Letters. 9: 3017-20. PMID 17608431 DOI: 10.1021/ol071079g |
0.491 |
|
| 2007 |
Appukkuttan P, Dehaen W, Van der Eycken E. Microwave-assisted transition-metal-catalyzed synthesis of N-shifted and ring-expanded buflavine analogues. Chemistry (Weinheim An Der Bergstrasse, Germany). 13: 6452-60. PMID 17508369 DOI: 10.1002/chem.200700177 |
0.452 |
|
| 2007 |
Kumar S, Singh BK, Pandey AK, Kumar A, Sharma SK, Raj HG, Prasad AK, Van der Eycken E, Parmar VS, Ghosh B. A chromone analog inhibits TNF-alpha induced expression of cell adhesion molecules on human endothelial cells via blocking NF-kappaB activation. Bioorganic & Medicinal Chemistry. 15: 2952-62. PMID 17321745 DOI: 10.1016/j.bmc.2007.02.004 |
0.464 |
|
| 2007 |
Kumar A, Singh BK, Sharma NK, Gyanda K, Jain SK, Tyagi YK, Baghel AS, Pandey M, Sharma SK, Prasad AK, Jain SC, Rastogi RC, Raj HG, Watterson AC, Van der Eycken E, et al. Specificities of acetoxy derivatives of coumarins, biscoumarins, chromones, flavones, isoflavones and xanthones for acetoxy drug: protein transacetylase. European Journal of Medicinal Chemistry. 42: 447-55. PMID 17182154 DOI: 10.1016/J.Ejmech.2006.09.008 |
0.615 |
|
| 2006 |
Ermolat'ev DS, Babaev EV, Van der Eycken EV. Efficient one-pot, two-step, microwave-assisted procedure for the synthesis of polysubstituted 2-aminoimidazoles. Organic Letters. 8: 5781-4. PMID 17134271 DOI: 10.1021/ol062421c |
0.463 |
|
| 2006 |
Ermolat'ev DS, Giménez VN, Babaev EV, Van der Eycken E. Efficient Pd(0)-mediated microwave-assisted arylation of 2-substituted imidazo[1,2-a]pyrimidines. Journal of Combinatorial Chemistry. 8: 659-63. PMID 16961403 DOI: 10.1021/CC060031B |
0.448 |
|
| 2006 |
Singh BK, Appukkuttan P, Claerhout S, Parmar VS, Van der Eycken E. Copper(II)-mediated cross-coupling of arylboronic acids and 2(1H)-pyrazinones facilitated by microwave irradiation with simultaneous cooling. Organic Letters. 8: 1863-6. PMID 16623570 DOI: 10.1021/ol060422z |
0.59 |
|
| 2006 |
Beryozkina T, Appukkuttan P, Mont N, Van der Eycken E. Microwave-enhanced synthesis of new (-)-steganacin and (-)-steganone aza analogues. Organic Letters. 8: 487-90. PMID 16435866 DOI: 10.1021/ol052766f |
0.495 |
|
| 2005 |
Appukkuttan P, Dehaen W, Van der Eycken E. Microwave-enhanced synthesis of N-shifted buflavine analogues via a Suzuki-ring-closing metathesis protocol. Organic Letters. 7: 2723-6. PMID 15957931 DOI: 10.1021/ol050806+ |
0.489 |
|
| 2005 |
Kaval N, Ermolat'ev D, Appukkuttan P, Dehaen W, Kappe CO, Van Der Eycken E. The application of "click chemistry" for the decoration of 2(1H)-pyrazinone scaffold: Generation of templates Journal of Combinatorial Chemistry. 7: 490-502. PMID 15877478 DOI: 10.1021/cc0498377 |
0.431 |
|
| 2005 |
Kaval N, Dehaen W, Van Der Eycken E. Solid-phase synthesis of the 2(1H)-pyrazinone scaffold: A new approach toward diversely substituted heterocycles Journal of Combinatorial Chemistry. 7: 90-95. PMID 15638486 DOI: 10.1021/cc049882e |
0.502 |
|
| 2004 |
Appukkuttan P, Dehaen W, Fokin VV, Van der Eycken E. A microwave-assisted click chemistry synthesis of 1,4-disubstituted 1,2,3-triazoles via a copper(I)-catalyzed three-component reaction. Organic Letters. 6: 4223-5. PMID 15524448 DOI: 10.1021/Ol048341V |
0.455 |
|
| 2004 |
Kaval N, Dehaen W, Kappe CO, Van der Eycken E. The effect of pressure on microwave-enhanced Diels-Alder reactions. A case study. Organic & Biomolecular Chemistry. 2: 154-6. PMID 14737635 DOI: 10.1039/b315150f |
0.4 |
|
| 2004 |
Kaval N, Dehaen W, Kappe CO, Van der Eycken E. The effect of pressure on microwave-enhanced Diels-Alder reactions. A case study Organic and Biomolecular Chemistry. 2: 154-156. DOI: 10.1039/b315150f |
0.367 |
|
| 2003 |
Kaval N, Bisztray K, Dehaen W, Kappe CO, Van Der Eycken E. Microwave-enhanced transition metal-catalyzed decoration of 2(1H)-pyrazinone scaffolds Molecular Diversity. 7: 125-133. PMID 14870841 DOI: 10.1023/B:MODI.0000006807.43408.d5 |
0.549 |
|
| 2002 |
Van Der Eycken E, Appukkuttan P, De Borggraeve W, Dehaen W, Dallinger D, Kappe CO. High-speed microwave-promoted hetero-Diels-Alder reactions of 2(1H)-pyrazinones in ionic liquid doped solvents. The Journal of Organic Chemistry. 67: 7904-7. PMID 12398527 DOI: 10.1021/JO0263216 |
0.397 |
|
| 2001 |
Vízvárdi K, Desmet K, Luyten I, Sandra P, Hoornaert G, Van der Eycken E. Asymmetric induction in intramolecular meta photocycloaddition: cyclodextrin-mediated solid-phase photochemistry of various phenoxyalkenes. Organic Letters. 3: 1173-5. PMID 11348187 DOI: 10.1021/Ol0156345 |
0.343 |
|
| 2000 |
Van der Eycken E, Terryn N, Goeman JL, Carlens G, Nerinckx W, Claeyssens M, Van der Eycken J, Van Montagu M, Brito-Arias M, Engler G. Sudan-β-D-glucuronides and their use for the histochemical localization of β-glucuronidase activity in transgenic plants Plant Cell Reports. 19: 966-970. DOI: 10.1007/s002990000219 |
0.557 |
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