☰

Oleg Tsodikov - Publications

Affiliations: 
Chemistry University of Kentucky, Lexington, KY 
Tree Info Similar researchers PubMed Report error

52 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2023 Miller ET, Tsodikov OV, Garneau-Tsodikova S. Structural insights into the diverse prenylating capabilities of DMATS prenyltransferases. Natural Product Reports. PMID 37929638 DOI: 10.1039/d3np00036b  0.558
2023 Pang AH, Green KD, Tsodikov OV, Garneau-Tsodikova S. Discovery and development of inhibitors of acetyltransferase Eis to combat Mycobacterium tuberculosis. Methods in Enzymology. 690: 369-396. PMID 37858535 DOI: 10.1016/bs.mie.2023.06.017  0.648
2023 Thamban Chandrika N, Green KD, Spencer AC, Tsodikov OV, Garneau-Tsodikova S. Discovery and development of novel substituted monohydrazides as potent antifungal agents. Rsc Medicinal Chemistry. 14: 1351-1361. PMID 37484566 DOI: 10.1039/d3md00167a  0.531
2023 Travis S, Green KD, Thamban Chandrika N, Pang AH, Frantom PA, Tsodikov OV, Garneau-Tsodikova S, Thompson MK. Identification and analysis of small molecule inhibitors of FosB from . Rsc Medicinal Chemistry. 14: 947-956. PMID 37252104 DOI: 10.1039/d3md00113j  0.651
2023 Gelzinis JA, Szahaj MK, Bekendam RH, Wurl SE, Pantos MM, Verbetsky CA, Dufresne A, Shea M, Howard KC, Tsodikov OV, Garneau-Tsodikova S, Zwicker JI, Kennedy DR. Targeting thiol isomerase activity with zafirlukast to treat ovarian cancer from the bench to clinic. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 37: e22914. PMID 37043381 DOI: 10.1096/fj.202201952R  0.487
2023 Green KD, Thamban Chandrika N, Vu LY, Pang AH, Tsodikov OV, Garneau-Tsodikova S. Aromatic hydrazides: A potential solution for Acinetobacter baumannii infections. European Journal of Medicinal Chemistry. 249: 115165. PMID 36739749 DOI: 10.1016/j.ejmech.2023.115165  0.584
2023 Pang AH, Green KD, Punetha A, Thamban Chandrika N, Howard KC, Garneau-Tsodikova S, Tsodikov OV. Discovery and Mechanistic Analysis of Structurally Diverse Inhibitors of Acetyltransferase Eis among FDA-Approved Drugs. Biochemistry. 62: 710-721. PMID 36657084 DOI: 10.1021/acs.biochem.2c00658  0.629
2022 Travis S, Green KD, Gilbert NC, Tsodikov OV, Garneau-Tsodikova S, Thompson MK. Inhibition of Fosfomycin Resistance Protein FosB from Gram-Positive Pathogens by Phosphonoformate. Biochemistry. PMID 36525630 DOI: 10.1021/acs.biochem.2c00566  0.646
2022 Pang AH, Tsodikov OV. A Colorimetric Assay to Identify and Characterize Bacterial Primase Inhibitors. Methods in Molecular Biology (Clifton, N.J.). 2601: 283-301. PMID 36445590 DOI: 10.1007/978-1-0716-2855-3_15  0.313
2022 Pang AH, Green KD, Chandrika NT, Garzan A, Punetha A, Holbrook SYL, Willby MJ, Posey JE, Tsodikov OV, Garneau-Tsodikova S. Discovery of substituted benzyloxy-benzylamine inhibitors of acetyltransferase Eis and their anti-mycobacterial activity. European Journal of Medicinal Chemistry. 242: 114698. PMID 36037791 DOI: 10.1016/j.ejmech.2022.114698  0.663
2022 Green KD, Pang AH, Thamban Chandrika N, Garzan A, Baughn AD, Tsodikov OV, Garneau-Tsodikova S. Discovery and Optimization of 6-(1-Substituted pyrrole-2-yl)--triazine Containing Compounds as Antibacterial Agents. Acs Infectious Diseases. 8: 757-767. PMID 35239306 DOI: 10.1021/acsinfecdis.1c00450  0.59
2021 Punetha A, Green KD, Garzan A, Thamban Chandrika N, Willby MJ, Pang AH, Hou C, Holbrook SYL, Krieger K, Posey JE, Parish T, Tsodikov OV, Garneau-Tsodikova S. Structure-based design of haloperidol analogues as inhibitors of acetyltransferase Eis from to overcome kanamycin resistance. Rsc Medicinal Chemistry. 12: 1894-1909. PMID 34825186 DOI: 10.1039/d1md00239b  0.659
2021 Green KD, Punetha A, Chandrika NT, Hou C, Garneau-Tsodikova S, Tsodikov OV. Development of single-stranded DNA bisintercalating inhibitors of primase DnaG as antibiotics. Chemmedchem. PMID 33711198 DOI: 10.1002/cmdc.202100001  0.603
2020 Mori S, Garneau-Tsodikova S, Tsodikov OV. Unimodular Methylation by Adenylation-Thiolation Domains Containing an Embedded Methyltransferase. Journal of Molecular Biology. PMID 32920052 DOI: 10.1016/J.Jmb.2020.09.004  0.495
2020 Punetha A, Ngo HX, Holbrook SYL, Green KD, Willby MJ, Bonnett SA, Krieger K, Dennis EK, Posey JE, Parish T, Tsodikov OV, Garneau-Tsodikova S. Structure-Guided Optimization of Inhibitors of Acetyltransferase Eis from . Acs Chemical Biology. PMID 32421305 DOI: 10.1021/Acschembio.0C00184  0.646
2019 Thamban Chandrika N, Fosso MY, Tsodikov OV, LeVine Iii H, Garneau-Tsodikova S. Combining Chalcones with Donepezil to Inhibit Both Cholinesterases and Aβ Fibril Assembly. Molecules (Basel, Switzerland). 25. PMID 31878304 DOI: 10.3390/Molecules25010077  0.544
2019 Green KD, Punetha A, Hou C, Garneau-Tsodikova S, Tsodikov OV. Probing the Robustness of Inhibitors of Tuberculosis Aminoglycoside Resistance Enzyme Eis by Mutagenesis. Acs Infectious Diseases. PMID 31433614 DOI: 10.1021/Acsinfecdis.9B00228  0.659
2019 Mori S, Pang AH, Chandrika NT, Garneau-Tsodikova S, Tsodikov OV. Publisher Correction: Unusual substrate and halide versatility of phenolic halogenase PltM. Nature Communications. 10: 2053. PMID 31040284 DOI: 10.1038/S41467-019-09731-8  0.444
2019 Mori S, Pang AH, Thamban Chandrika N, Garneau-Tsodikova S, Tsodikov OV. Unusual substrate and halide versatility of phenolic halogenase PltM. Nature Communications. 10: 1255. PMID 30890712 DOI: 10.1038/s41467-019-09215-9  0.557
2019 Hayden RC, Hou C, Mitra P, Mandal A, Rohr J, Thorson J, Tsodikov O, Leggas M. Abstract 2954: Mithramycin analogues disrupt ETS transcription factor DNA binding Cancer Research. 79: 2954-2954. DOI: 10.1158/1538-7445.Sabcs18-2954  0.326
2018 Holbrook SYL, Gentry MS, Tsodikov OV, Garneau-Tsodikova S. Nucleoside triphosphate cosubstrates control the substrate profile and efficiency of aminoglycoside 3'--phosphotransferase type IIa. Medchemcomm. 9: 1332-1339. PMID 30151088 DOI: 10.1039/C8Md00234G  0.549
2018 Ngo HX, Green KD, Gajadeera CS, Willby MJ, Holbrook SYL, Hou C, Garzan A, Mayhoub AS, Posey JE, Tsodikov OV, Garneau-Tsodikova S. Potent 1,2,4-Triazino[5,6 b]indole-3-thioether Inhibitors of the Kanamycin Resistance Enzyme Eis from Mycobacterium tuberculosis. Acs Infectious Diseases. PMID 29601176 DOI: 10.1021/Acsinfecdis.8B00074  0.659
2018 Mori S, Pang AH, Lundy TA, Garzan A, Tsodikov OV, Garneau-Tsodikova S. Structural basis for backbone N-methylation by an interrupted adenylation domain. Nature Chemical Biology. PMID 29556104 DOI: 10.1038/S41589-018-0014-7  0.552
2018 Green KD, Biswas T, Pang AH, Willby MJ, Reed MS, Stuchlik O, Pohl J, Posey JE, Tsodikov OV, Garneau-Tsodikova S. Acetylation by Eis and Deacetylation by Rv1151c of Mycobacterium tuberculosis HupB: Biochemical and Structural Insight. Biochemistry. PMID 29345920 DOI: 10.1021/Acs.Biochem.7B01089  0.549
2017 Thamban Chandrika N, Shrestha SK, Ngo HX, Tsodikov OV, Howard KC, Garneau-Tsodikova S. Alkylated Piperazines and Piperazine-Azole Hybrids as Antifungal Agents. Journal of Medicinal Chemistry. PMID 29256601 DOI: 10.1021/Acs.Jmedchem.7B01138  0.59
2017 Mori S, Garzan A, Tsodikov OV, Garneau-Tsodikova S. Deciphering Nature's Intricate Way of N,S-Dimethylating l-Cysteine: Sequential Action of Two Bifunctional Adenylation Domains. Biochemistry. PMID 29112395 DOI: 10.1021/Acs.Biochem.7B00980  0.513
2017 Garzan A, Willby MJ, Ngo HX, Gajadeera CS, Green KD, Holbrook SY, Hou C, Posey JE, Tsodikov OV, Garneau-Tsodikova S. Combating Eis-mediated kanamycin resistance of M. tuber-culosis by novel pyrrolo[1,5-a]pyrazine-based Eis inhibitors. Acs Infectious Diseases. PMID 28192916 DOI: 10.1021/Acsinfecdis.6B00193  0.662
2017 Pang AH, Garneau-Tsodikova S, Tsodikov OV. In Vitro Assays to Identify Antibiotics Targeting DNA Metabolism. Methods in Molecular Biology (Clifton, N.J.). 1520: 175-200. PMID 27873253 DOI: 10.1007/978-1-4939-6634-9_11  0.519
2016 Garzan A, Willby MJ, Green KD, Tsodikov OV, Posey JE, Garneau-Tsodikova S. Discovery and Optimization of Two Eis Inhibitor Families as Kanamycin Adjuvants against Drug-Resistant M. tuberculosis. Acs Medicinal Chemistry Letters. 7: 1219-1221. PMID 27994767 DOI: 10.1021/Acsmedchemlett.6B00261  0.629
2016 Garzan A, Willby MJ, Green KD, Gajadeera CS, Hou C, Tsodikov OV, Posey JE, Garneau-Tsodikova S. Sulfonamide-Based Inhibitors of Aminoglycoside Acetyltransferase Eis Abolish Resistance to Kanamycin in Mycobacterium tuberculosis. Journal of Medicinal Chemistry. 59: 10619-10628. PMID 27933949 DOI: 10.1021/Acs.Jmedchem.6B01161  0.644
2016 Pang AH, Garzan A, Larsen MJ, McQuade TJ, Garneau-Tsodikova S, Tsodikov OV. Discovery of allosteric and selective inhibitors of inorganic pyrophosphatase from Mycobacterium tuberculosis. Acs Chemical Biology. PMID 27622287 DOI: 10.1021/Acschembio.6B00510  0.639
2016 Willby MJ, Green KD, Gajadeera CS, Hou C, Tsodikov OV, Posey JE, Garneau-Tsodikova S. Potent inhibitors of acetyltransferase Eis overcome kanamycin re-sistance in Mycobacterium tuberculosis. Acs Chemical Biology. PMID 27010218 DOI: 10.1021/Acschembio.6B00110  0.656
2015 Pang AH, Garneau-Tsodikova S, Tsodikov OV. Crystal structure of halogenase PltA from the pyoluteorin biosynthetic pathway. Journal of Structural Biology. PMID 26416533 DOI: 10.1016/J.Jsb.2015.09.013  0.562
2015 Pratt AC, Dewage SW, Pang AH, Biswas T, Barnard-Britson S, Cisneros GA, Tsodikov OV. Structural and computational dissection of the catalytic mechanism of the inorganic pyrophosphatase from Mycobacterium tuberculosis. Journal of Structural Biology. 192: 76-87. PMID 26296329 DOI: 10.1016/J.Jsb.2015.08.010  0.32
2015 Fosso MY, LeVine H, Green KD, Tsodikov OV, Garneau-Tsodikova S. Effects of structural modifications on the metal binding, anti-amyloid activity, and cholinesterase inhibitory activity of chalcones. Organic & Biomolecular Chemistry. 13: 9418-26. PMID 26248214 DOI: 10.1039/C5Ob01478F  0.528
2015 Tsodikov OV, Hou C, Walsh CT, Garneau-Tsodikova S. Crystal structure of O-methyltransferase CalO6 from the calicheamicin biosynthetic pathway: a case of challenging structure determination at low resolution. Bmc Structural Biology. 15: 13. PMID 26170207 DOI: 10.1186/S12900-015-0040-6  0.562
2015 Green KD, Biswas T, Chang C, Wu R, Chen W, Janes BK, Chalupska D, Gornicki P, Hanna PC, Tsodikov OV, Joachimiak A, Garneau-Tsodikova S. Biochemical and Structural Analysis of an Eis Family Aminoglycoside Acetyltransferase from Bacillus anthracis. Biochemistry. 54: 3197-206. PMID 25928210 DOI: 10.1021/Acs.Biochem.5B00244  0.612
2015 Gajadeera C, Willby MJ, Green KD, Shaul P, Fridman M, Garneau-Tsodikova S, Posey JE, Tsodikov OV. Antimycobacterial activity of DNA intercalator inhibitors of Mycobacterium tuberculosis primase DnaG. The Journal of Antibiotics. 68: 153-7. PMID 25248725 DOI: 10.1038/Ja.2014.131  0.64
2015 Tsodikov OV, Hou C, Walsh CT, Garneau-Tsodikova S. Crystal structure of O-methyltransferase CalO6 from the calicheamicin biosynthetic pathway: A case of challenging structure determination at low resolution Bmc Structural Biology. 15. DOI: 10.1186/s12900-015-0040-6  0.509
2015 Fosso MY, LeVine H, Green KD, Tsodikov OV, Garneau-Tsodikova S. Effects of structural modifications on the metal binding, anti-amyloid activity, and cholinesterase inhibitory activity of chalcones Organic and Biomolecular Chemistry. 13: 9418-9426. DOI: 10.1039/c5ob01478f  0.526
2014 Tsodikov OV, Green KD, Garneau-Tsodikova S. A random sequential mechanism of aminoglycoside acetylation by Mycobacterium tuberculosis Eis protein. Plos One. 9: e92370. PMID 24699000 DOI: 10.1371/Journal.Pone.0092370  0.619
2013 Houghton JL, Biswas T, Chen W, Tsodikov OV, Garneau-Tsodikova S. Chemical and structural insights into the regioversatility of the aminoglycoside acetyltransferase Eis. Chembiochem : a European Journal of Chemical Biology. 14: 2127-35. PMID 24106131 DOI: 10.1002/Cbic.201300359  0.64
2013 Biswas T, Green KD, Garneau-Tsodikova S, Tsodikov OV. Discovery of inhibitors of Bacillus anthracis primase DnaG. Biochemistry. 52: 6905-10. PMID 24004110 DOI: 10.1021/Bi4011286  0.602
2013 Larrouy-Maumus G, Biswas T, Hunt DM, Kelly G, Tsodikov OV, de Carvalho LP. Discovery of a glycerol 3-phosphate phosphatase reveals glycerophospholipid polar head recycling in Mycobacterium tuberculosis. Proceedings of the National Academy of Sciences of the United States of America. 110: 11320-5. PMID 23801751 DOI: 10.1073/Pnas.1221597110  0.305
2013 Houghton JL, Biswas T, Chen W, Tsodikov OV, Garneau-Tsodikova S. Cover Picture: Chemical and Structural Insights into the Regioversatility of the Aminoglycoside Acetyltransferase Eis (ChemBioChem 16/2013) Chembiochem. 14: 2061-2061. DOI: 10.1002/cbic.201390058  0.521
2012 Chen W, Green KD, Tsodikov OV, Garneau-Tsodikova S. Aminoglycoside multiacetylating activity of the enhanced intracellular survival protein from Mycobacterium smegmatis and its inhibition. Biochemistry. 51: 4959-67. PMID 22646013 DOI: 10.1021/Bi3004473  0.606
2012 Biswas T, Houghton JL, Garneau-Tsodikova S, Tsodikov OV. The structural basis for substrate versatility of chloramphenicol acetyltransferase CATI. Protein Science : a Publication of the Protein Society. 21: 520-30. PMID 22294317 DOI: 10.1002/Pro.2036  0.592
2011 Chen W, Biswas T, Porter VR, Tsodikov OV, Garneau-Tsodikova S. Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB. Proceedings of the National Academy of Sciences of the United States of America. 108: 9804-8. PMID 21628583 DOI: 10.1073/Pnas.1105379108  0.61
2010 Biswas T, Zolova OE, Lombó F, de la Calle F, Salas JA, Tsodikov OV, Garneau-Tsodikova S. A new scaffold of an old protein fold ensures binding to the bisintercalator thiocoraline. Journal of Molecular Biology. 397: 495-507. PMID 20122935 DOI: 10.1016/J.Jmb.2010.01.053  0.562
2009 Biswas T, Yi L, Aggarwal P, Wu J, Rubin JR, Stuckey JA, Woodard RW, Tsodikov OV. The tail of KdsC: conformational changes control the activity of a haloacid dehalogenase superfamily phosphatase. The Journal of Biological Chemistry. 284: 30594-603. PMID 19726684 DOI: 10.1074/Jbc.M109.012278  0.314
2009 Garneau-Tsodikova S, Shkel IA, Tsodikov OV. Exact and user-friendly kinetic analysis of the two-step rapid equilibrium Michaelis-Menten mechanism. Analytical Biochemistry. 387: 276-9. PMID 19344659 DOI: 10.1016/J.Ab.2009.01.023  0.491
2009 McQuade TJ, Shallop AD, Sheoran A, Delproposto JE, Tsodikov OV, Garneau-Tsodikova S. A nonradioactive high-throughput assay for screening and characterization of adenylation domains for nonribosomal peptide combinatorial biosynthesis. Analytical Biochemistry. 386: 244-50. PMID 19135023 DOI: 10.1016/J.Ab.2008.12.014  0.535
Show low-probability matches.