| Year |
Citation |
Score |
| 2023 |
Helal MA, Chittiboyina AG, Avery MA. Structure-based design of novel melanin-concentrating hormone receptor-1 ligands based on saturated nitrogen-containing heterocycles. Bioorganic & Medicinal Chemistry Letters. 84: 129194. PMID 36813053 DOI: 10.1016/j.bmcl.2023.129194 |
0.545 |
|
| 2020 |
Kochanowska-Karamyan AJ, Araujo HC, Zhang X, El-Alfy A, Carvalho P, Avery MA, Holmbo SD, Magolan J, Hamann MT. Isolation and Synthesis of Veranamine, an Antidepressant Lead from the Marine Sponge . Journal of Natural Products. PMID 32227883 DOI: 10.1021/Acs.Jnatprod.9B01107 |
0.428 |
|
| 2019 |
Helal MA, Chittiboyina AG, Avery MA. Identification of a new small molecule chemotype of Melanin Concentrating Hormone Receptor-1 antagonists using pharmacophore-based virtual screening. Bioorganic & Medicinal Chemistry Letters. 126741. PMID 31678007 DOI: 10.1016/J.Bmcl.2019.126741 |
0.624 |
|
| 2019 |
Zou Y, Wang X, Sims J, Wang B, Pandey P, Welsh C, Stone RS, Avery MA, Doerksen RJ, Ferreira D, Anklin C, Valeriote FA, Kelly M, Hamann MT. Computationally-Assisted Discovery and Assignment of a Highly Strained and PANC-1 Selective Alkaloid from Alaska's Deep Ocean. Journal of the American Chemical Society. PMID 30758203 DOI: 10.1021/Jacs.8B11403 |
0.307 |
|
| 2017 |
Bacherikov VA, Chittiboyina AG, Avery MA. Design, synthesis and biological evaluation of peptidomimetic n-substituted cbz-4-hyp-hpa-amides as novel inhibitors of plasmodium falciparum. Chemistry & Biodiversity. PMID 28498611 DOI: 10.1002/Cbdv.201700037 |
0.672 |
|
| 2017 |
Avery BA, Pabbisetty D, Li L, Sharma A, Gundluru MK, Chittiboyina AG, Williamson JS, Avery MA. A pharmacokinetic comparison of homodimer ARB-92 and heterodimer ARB-89: novel, potent antimalarial candidates derived from 7β-hydroxyartemisinin Journal of Pharmaceutical Investigation. 48: 585-593. DOI: 10.1007/S40005-017-0352-6 |
0.379 |
|
| 2014 |
Avery MA, Choudhry SC, Dhingra OP, Gray BD, Kang MC, Kuo SC, Vedananda TR, White JD, Whittle AJ. Total synthesis of macrodiolide ionophores aplasmomycin A and boromycin via double ring contraction. Organic & Biomolecular Chemistry. 12: 9116-32. PMID 25096282 DOI: 10.1039/c4ob01017e |
0.403 |
|
| 2014 |
Yang J, Liang Q, Wang M, Jeffries C, Smithson D, Tu Y, Boulos N, Jacob MR, Shelat AA, Wu Y, Ravu RR, Gilbertson R, Avery MA, Khan IA, Walker LA, et al. UPLC-MS-ELSD-PDA as a powerful dereplication tool to facilitate compound identification from small-molecule natural product libraries. Journal of Natural Products. 77: 902-9. PMID 24617915 DOI: 10.1021/Np4009706 |
0.595 |
|
| 2014 |
Weldon DJ, Shah F, Chittiboyina AG, Sheri A, Chada RR, Gut J, Rosenthal PJ, Shivakumar D, Sherman W, Desai P, Jung JC, Avery MA. Synthesis, biological evaluation, hydration site thermodynamics, and chemical reactivity analysis of α-keto substituted peptidomimetics for the inhibition of Plasmodium falciparum. Bioorganic & Medicinal Chemistry Letters. 24: 1274-9. PMID 24507921 DOI: 10.1016/J.Bmcl.2014.01.062 |
0.819 |
|
| 2014 |
Porta EO, Carvalho PB, Avery MA, Tekwani BL, Labadie GR. Click chemistry decoration of amino sterols as promising strategy to developed new leishmanicidal drugs. Steroids. 79: 28-36. PMID 24200958 DOI: 10.1016/J.Steroids.2013.10.010 |
0.789 |
|
| 2013 |
Chittiboyina AG, Peddikotla P, Avery MA, Khan IA. Directed hydrogenation of acyclic homoallylic alcohols: enantioselective syntheses of (+)- and (-)-laurenditerpenol. The Journal of Organic Chemistry. 78: 9223-32. PMID 23985032 DOI: 10.1021/Jo401461X |
0.628 |
|
| 2013 |
Wu Y, Rodenburg DL, Ibrahim MA, McChesney JD, Avery MA. Stevioside methanol tetra-solvate. Acta Crystallographica. Section E, Structure Reports Online. 69: o410-1. PMID 23476589 DOI: 10.1107/S1600536813003954 |
0.524 |
|
| 2013 |
Peddikotla P, Chittiboyina A, Avery M, Khan I. Enantioselective Synthesis of (-)-Laurenditerpenol Planta Medica. 79: 46. DOI: 10.1055/S-0033-1336488 |
0.318 |
|
| 2012 |
Helal MA, Avery MA. Combined receptor-based and ligand-based approach to delineate the mode of binding of guaianolide-endoperoxides to PfATP6. Bioorganic & Medicinal Chemistry Letters. 22: 5410-4. PMID 22877631 DOI: 10.1016/J.Bmcl.2012.07.053 |
0.318 |
|
| 2012 |
Pabbisetty D, Illendula A, Muraleedharan KM, Chittiboyina AG, Williamson JS, Avery MA, Avery BA. Determination of antimalarial compound, ARB-89 (7β-hydroxy-artemisinin carbamate) in rat serum by UPLC/MS/MS and its application in pharmacokinetics. Journal of Chromatography. B, Analytical Technologies in the Biomedical and Life Sciences. 889: 123-9. PMID 22365535 DOI: 10.1016/J.Jchromb.2012.02.007 |
0.601 |
|
| 2012 |
Shah F, Gut J, Legac J, Shivakumar D, Sherman W, Rosenthal PJ, Avery MA. Computer-aided drug design of falcipain inhibitors: virtual screening, structure-activity relationships, hydration site thermodynamics, and reactivity analysis. Journal of Chemical Information and Modeling. 52: 696-710. PMID 22332946 DOI: 10.1021/Ci2005516 |
0.362 |
|
| 2011 |
Mukherjee P, Shah F, Desai P, Avery M. Inhibitors of SARS-3CLpro: virtual screening, biological evaluation, and molecular dynamics simulation studies. Journal of Chemical Information and Modeling. 51: 1376-92. PMID 21604711 DOI: 10.1021/Ci1004916 |
0.596 |
|
| 2011 |
Shah F, Mukherjee P, Gut J, Legac J, Rosenthal PJ, Tekwani BL, Avery MA. Identification of novel malarial cysteine protease inhibitors using structure-based virtual screening of a focused cysteine protease inhibitor library. Journal of Chemical Information and Modeling. 51: 852-64. PMID 21428453 DOI: 10.1021/Ci200029Y |
0.628 |
|
| 2011 |
Helal MA, Chittiboyina AG, Avery MA. New insights into the binding mode of melanin concentrating hormone receptor-1 antagonists: homology modeling and explicit membrane molecular dynamics simulation study. Journal of Chemical Information and Modeling. 51: 635-46. PMID 21370821 DOI: 10.1021/Ci100355C |
0.581 |
|
| 2011 |
Ahmed R, Ali Z, Wu Y, Kulkarni S, Avery MA, Choudhary MI, Khan IA. Chemical characterization of a commercial Commiphora wightii resin sample and chemical profiling to assess for authenticity. Planta Medica. 77: 945-50. PMID 21240842 DOI: 10.1055/S-0030-1250674 |
0.683 |
|
| 2011 |
Ghiano DG, Carvalho PB, Tekwani BL, Avery MA, Labadie G. Parallel solution synthesis of lavendustin analogs as antileishmanial agents Arkivoc. 2011. DOI: 10.3998/Ark.5550190.0012.725 |
0.793 |
|
| 2011 |
Shah F, Wu Y, Gut J, Pedduri Y, Legac J, Rosenthal PJ, Avery MA. Design, synthesis and biological evaluation of novel benzothiazole and triazole analogs as falcipain inhibitors Medchemcomm. 2: 1201. DOI: 10.1039/C1Md00129A |
0.633 |
|
| 2011 |
Hammond NL, Choi SR, Carvalho P, Liu H, Khan S, Avery MA. Synthesis and biological evaluation of a novel anti-malarial lead Medicinal Chemistry Research. 20: 401-407. DOI: 10.1007/S00044-010-9325-2 |
0.784 |
|
| 2010 |
Na BK, Bae YA, Zo YG, Choe Y, Kim SH, Desai PV, Avery MA, Craik CS, Kim TS, Rosenthal PJ, Kong Y. Biochemical properties of a novel cysteine protease of Plasmodium vivax, vivapain-4. Plos Neglected Tropical Diseases. 4: e849. PMID 20967286 DOI: 10.1371/Journal.Pntd.0000849 |
0.301 |
|
| 2010 |
Sun L, Shah F, Helal MA, Wu Y, Pedduri Y, Chittiboyina AG, Gut J, Rosenthal PJ, Avery MA. Design, synthesis, and development of novel guaianolide-endoperoxides as potential antimalarial agents. Journal of Medicinal Chemistry. 53: 7864-8. PMID 20945914 DOI: 10.1021/Jm1006462 |
0.79 |
|
| 2010 |
Battu SK, Repka MA, Maddineni S, Chittiboyina AG, Avery MA, Majumdar S. Physicochemical characterization of berberine chloride: a perspective in the development of a solution dosage form for oral delivery. Aaps Pharmscitech. 11: 1466-75. PMID 20842541 DOI: 10.1208/S12249-010-9520-Y |
0.574 |
|
| 2010 |
Mukherjee P, Desai P, Zhou YD, Avery M. Targeting the BH3 domain mediated protein-protein interaction of Bcl-xL through virtual screening. Journal of Chemical Information and Modeling. 50: 906-23. PMID 20392095 DOI: 10.1021/Ci1000373 |
0.573 |
|
| 2010 |
Shah F, Mukherjee P, Desai P, Avery M. Computational approaches for the discovery of cysteine protease inhibitors against malaria and SARS. Current Computer-Aided Drug Design. 6: 1-23. PMID 20370692 DOI: 10.2174/157340910790980142 |
0.604 |
|
| 2010 |
Kulkarni SJ, Pedduri Y, Chittiboyina AG, Avery MA. Asymmetric total synthesis of the caspase-1 inhibitor (-)-berkeleyamide A. The Journal of Organic Chemistry. 75: 3113-6. PMID 20356061 DOI: 10.1021/Jo1001033 |
0.718 |
|
| 2010 |
Upadhye SB, Kulkarni SJ, Majumdar S, Avery MA, Gul W, ElSohly MA, Repka MA. Preparation and characterization of inclusion complexes of a hemisuccinate ester prodrug of delta9-tetrahydrocannabinol with modified beta-cyclodextrins. Aaps Pharmscitech. 11: 509-17. PMID 20333489 DOI: 10.1208/S12249-010-9401-4 |
0.562 |
|
| 2010 |
Zeng F, Wang W, Wu Y, Dey M, Ye M, Avery MA, Khan IA, Guo DA. Two prenylated and C-methylated flavonoids from Tripterygium wilfordii. Planta Medica. 76: 1596-9. PMID 20309799 DOI: 10.1055/S-0029-1241017 |
0.573 |
|
| 2010 |
Mizuno CS, Chittiboyina AG, Shah FH, Patny A, Kurtz TW, Pershadsingh HA, Speth RC, Karamyan VT, Carvalho PB, Avery MA. Design, synthesis, and docking studies of novel benzimidazoles for the treatment of metabolic syndrome. Journal of Medicinal Chemistry. 53: 1076-85. PMID 20073471 DOI: 10.1021/Jm901272D |
0.78 |
|
| 2010 |
Avery MA, Chittiboyina AG. Anti‐Inflammatory Glucocorticoids Burger's Medicinal Chemistry and Drug Discovery. 35-152. DOI: 10.1002/0471266949.Bmc192 |
0.319 |
|
| 2009 |
Hammond N, Carvalho P, Wu Y, Avery MA. 3,3',5,5'-Tetra-nitro-biphen-yl. Acta Crystallographica. Section E, Structure Reports Online. 65: o1052-3. PMID 21583870 DOI: 10.1107/S1600536809011088 |
0.771 |
|
| 2009 |
Pradhan A, Tripathi AK, Desai PV, Mukherjee PK, Avery MA, Walker LA, Tekwani BL. Structure and function of Plasmodium falciparum malate dehydrogenase: role of critical amino acids in co-substrate binding pocket. Biochimie. 91: 1509-17. PMID 19772885 DOI: 10.1016/J.Biochi.2009.09.005 |
0.562 |
|
| 2009 |
Shah F, Zhang SQ, Kandhari SP, Mukherjee P, Chittiboyina A, Avery MA, Avery BA. In vitro erythrocytic uptake studies of artemisinin and selected derivatives using LC-MS and 2D-QSAR analysis of uptake in parasitized erythrocytes. Bioorganic & Medicinal Chemistry. 17: 5325-31. PMID 19497754 DOI: 10.1016/J.Bmc.2009.05.026 |
0.711 |
|
| 2009 |
Muraleedharan KM, Avery MA. Progress in the development of peroxide-based anti-parasitic agents. Drug Discovery Today. 14: 793-803. PMID 19477287 DOI: 10.1016/J.Drudis.2009.05.008 |
0.375 |
|
| 2009 |
Pradhan A, Mukherjee P, Tripathi AK, Avery MA, Walker LA, Tekwani BL. Analysis of quaternary structure of a [LDH-like] malate dehydrogenase of Plasmodium falciparum with oligomeric mutants. Molecular and Cellular Biochemistry. 325: 141-8. PMID 19184366 DOI: 10.1007/S11010-009-0028-2 |
0.57 |
|
| 2009 |
Zhang SQ, Vinnakota H, Jung JC, Carvalho P, Chittiboyina AG, Avery MA, Avery BA. Determination of a novel epothilone D analog (AV-EPO-106) in human plasma using ultra-performance liquid chromatography-tandem mass spectrometry. Biomedical Chromatography : Bmc. 23: 302-7. PMID 18800336 DOI: 10.1002/Bmc.1114 |
0.556 |
|
| 2009 |
Mizuno CS, Chittiboyina AG, Patny A, Kurtz TW, Pershadsingh HA, Speth RC, Karamyan VT, Avery MA. Design, synthesis, and docking studies of telmisartan analogs for the treatment of metabolic syndrome Medicinal Chemistry Research. 18: 611-628. DOI: 10.1007/S00044-008-9153-9 |
0.725 |
|
| 2009 |
Chittiboyina AG, Mizuno CS, Desai PV, Patny A, Kurtz TW, Pershadsingh HA, Speth RC, Karamyan V, Avery MA. Design, synthesis, and docking studies of novel telmisartan-glitazone hybrid analogs for the treatment of metabolic syndrome Medicinal Chemistry Research. 18: 589-610. DOI: 10.1007/S00044-008-9152-X |
0.715 |
|
| 2008 |
Gul W, Carvalho P, Berberich DW, Avery MA, Elsohly MA. (6aR,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tetra-hydro-6H-benzo[c]-chromen-1-yl 4-methyl-benzene-sulfonate. Acta Crystallographica. Section E, Structure Reports Online. 64: o1686. PMID 21201675 DOI: 10.1107/S1600536808022010 |
0.306 |
|
| 2008 |
Carvalho PB, Liu B, Wu Y, Williamson JS, Avery MA. 7β-Hydroxy-artemisinin. Acta Crystallographica. Section E, Structure Reports Online. 64: o395-6. PMID 21201424 DOI: 10.1107/S1600536808000251 |
0.534 |
|
| 2008 |
Li Z, Watkins EB, Liu H, Chittiboyina AG, Carvalho PB, Avery MA. 1,3-Diaxially substituted trans-decalins: potential nonsteroidal human progesterone receptor inhibitors. The Journal of Organic Chemistry. 73: 7764-7. PMID 18771323 DOI: 10.1021/Jo800947M |
0.705 |
|
| 2008 |
Rando DG, Avery MA, Tekwani BL, Khan SI, Ferreira EI. Antileishmanial activity screening of 5-nitro-2-heterocyclic benzylidene hydrazides. Bioorganic & Medicinal Chemistry. 16: 6724-31. PMID 18571927 DOI: 10.1016/J.Bmc.2008.05.076 |
0.432 |
|
| 2008 |
Taranto AG, Carvalho P, Avery MA. QM/QM studies for Michael reaction in coronavirus main protease (3CL Pro). Journal of Molecular Graphics & Modelling. 27: 275-85. PMID 18567519 DOI: 10.1016/J.Jmgm.2008.05.002 |
0.349 |
|
| 2008 |
Srivastava A, Mukherjee P, Desai PV, Avery MA, Tekwani BL. Structural analysis of farnesyl pyrophosphate synthase from parasitic protozoa, a potential chemotherapeutic target. Infectious Disorders Drug Targets. 8: 16-30. PMID 18473904 DOI: 10.2174/187152608784139587 |
0.584 |
|
| 2008 |
Mukherjee P, Desai PV, Srivastava A, Tekwani BL, Avery MA. Probing the structures of leishmanial farnesyl pyrophosphate synthases: homology modeling and docking studies. Journal of Chemical Information and Modeling. 48: 1026-40. PMID 18419114 DOI: 10.1021/Ci700355Z |
0.575 |
|
| 2008 |
Mukherjee P, Pradhan A, Shah F, Tekwani BL, Avery MA. Structural insights into the Plasmodium falciparum histone deacetylase 1 (PfHDAC-1): A novel target for the development of antimalarial therapy. Bioorganic & Medicinal Chemistry. 16: 5254-65. PMID 18362073 DOI: 10.1016/J.Bmc.2008.03.005 |
0.592 |
|
| 2008 |
Mukherjee P, Desai P, Ross L, White EL, Avery MA. Structure-based virtual screening against SARS-3CL(pro) to identify novel non-peptidic hits. Bioorganic & Medicinal Chemistry. 16: 4138-49. PMID 18343121 DOI: 10.1016/J.Bmc.2008.01.011 |
0.605 |
|
| 2008 |
Mizuno CS, Ma G, Khan S, Patny A, Avery MA, Rimando AM. Design, synthesis, biological evaluation and docking studies of pterostilbene analogs inside PPARalpha. Bioorganic & Medicinal Chemistry. 16: 3800-8. PMID 18272370 DOI: 10.1016/J.Bmc.2008.01.051 |
0.741 |
|
| 2008 |
Choi SR, Mukherjee P, Avery MA. The fight against drug-resistant malaria: novel plasmodial targets and antimalarial drugs. Current Medicinal Chemistry. 15: 161-71. PMID 18220771 DOI: 10.2174/092986708783330575 |
0.69 |
|
| 2008 |
Mizuno CS, Chittiboyina AG, Kurtz TW, Pershadsingh HA, Avery MA. Type 2 diabetes and oral antihyperglycemic drugs. Current Medicinal Chemistry. 15: 61-74. PMID 18220763 DOI: 10.2174/092986708783330656 |
0.748 |
|
| 2008 |
Sayed KA, Khalil AA, Yousaf M, Labadie G, Kumar GM, Franzblau SG, Mayer AM, Avery MA, Hamann MT. Semisynthetic studies on the manzamine alkaloids. Journal of Natural Products. 71: 300-8. PMID 18198837 DOI: 10.1021/Np0703702 |
0.645 |
|
| 2008 |
Oh S, Moon H, Jung J, Avery MA. Convenient Synthesis and Evaluation of Biological Activity of Benzyl (2S)-2-[(R)-1-hydroxy-2-oxo-(1-phenethyl)prop-3-ylcarbamoyl]- 4-oxopiperidine- (or -4-oxopyrrolidine)-1-carboxylate as Novel Histone Deacetylase Inhibitors Zeitschrift FüR Naturforschung B. 63: 1300-1304. DOI: 10.1515/Znb-2008-1108 |
0.437 |
|
| 2008 |
Oh S, Jung J, Avery MA. A Simple Synthesis of 4-Substituted 2-(3-Hydroxy-2-oxo-1-phenethylpropylcarbamoyl) pyrrolidine-1-carboxylic Acid Benzyl Esters as Novel Cysteine Protease Inhibitors Zeitschrift FüR Naturforschung B. 63: 210-216. DOI: 10.1515/Znb-2008-0215 |
0.365 |
|
| 2008 |
Zhang SQ, Chittiboyina AG, Kulkarni SJ, Avery MA, Avery BA. LC determination of a novel synthetic thiazolidinedione (BP-1107) in rat plasma and its application to a pharmacokinetic study Chromatographia. 68: 551-555. DOI: 10.1365/S10337-008-0745-9 |
0.534 |
|
| 2007 |
Chittiboyina AG, Kumar GM, Carvalho PB, Liu Y, Zhou YD, Nagle DG, Avery MA. Total synthesis and absolute configuration of laurenditerpenol: a hypoxia inducible factor-1 activation inhibitor. Journal of Medicinal Chemistry. 50: 6299-302. PMID 18004798 DOI: 10.1021/Jm7011062 |
0.599 |
|
| 2007 |
Singh N, Avery MA, McCurdy CR. Toward Mycobacterium tuberculosis DXR inhibitor design: homology modeling and molecular dynamics simulations. Journal of Computer-Aided Molecular Design. 21: 511-22. PMID 17874041 DOI: 10.1007/S10822-007-9132-0 |
0.336 |
|
| 2007 |
Oh S, Moon HI, Son IH, Jung JC, Avery MA. Synthesis of sulfonamides and evaluation of their histone deacetylase (HDAC) activity. Molecules (Basel, Switzerland). 12: 1125-35. PMID 17873846 DOI: 10.3390/12051125 |
0.413 |
|
| 2007 |
Choi SR, Pradhan A, Hammond NL, Chittiboyina AG, Tekwani BL, Avery MA. Design, synthesis, and biological evaluation of Plasmodium falciparum lactate dehydrogenase inhibitors. Journal of Medicinal Chemistry. 50: 3841-50. PMID 17636950 DOI: 10.1021/Jm070336K |
0.808 |
|
| 2007 |
Singh N, Chevé G, Avery MA, McCurdy CR. Targeting the methyl erythritol phosphate (MEP) pathway for novel antimalarial, antibacterial and herbicidal drug discovery: inhibition of 1-deoxy-D-xylulose-5-phosphate reductoisomerase (DXR) enzyme. Current Pharmaceutical Design. 13: 1161-77. PMID 17430177 DOI: 10.2174/138161207780618939 |
0.357 |
|
| 2007 |
Choi SR, Beeler AB, Pradhan A, Watkins EB, Rimoldi JM, Tekwani B, Avery MA. Generation of oxamic acid libraries: antimalarials and inhibitors of Plasmodium falciparum lactate dehydrogenase. Journal of Combinatorial Chemistry. 9: 292-300. PMID 17316052 DOI: 10.1021/Cc060110N |
0.636 |
|
| 2006 |
Menon RB, Kannoth MM, Tekwani BL, Gut J, Rosenthal PJ, Avery MA. A new library of C-16 modified artemisinin analogs and evaluation of their anti-parasitic activities. Combinatorial Chemistry & High Throughput Screening. 9: 729-41. PMID 17168678 DOI: 10.2174/138620706779026051 |
0.431 |
|
| 2006 |
Patny A, Desai PV, Avery MA. Ligand-supported homology modeling of the human angiotensin II type 1 (AT(1)) receptor: insights into the molecular determinants of telmisartan binding. Proteins. 65: 824-42. PMID 17034041 DOI: 10.1002/Prot.21196 |
0.307 |
|
| 2006 |
Chittiboyina AG, Venkatraman MS, Mizuno CS, Desai PV, Patny A, Benson SC, Ho CI, Kurtz TW, Pershadsingh HA, Avery MA. Design and synthesis of the first generation of dithiolane thiazolidinedione- and phenylacetic acid-based PPARgamma agonists. Journal of Medicinal Chemistry. 49: 4072-84. PMID 16821769 DOI: 10.1021/Jm0510880 |
0.794 |
|
| 2006 |
Patny A, Desai PV, Avery MA. Homology modeling of G-protein-coupled receptors and implications in drug design. Current Medicinal Chemistry. 13: 1667-91. PMID 16787212 DOI: 10.2174/092986706777442002 |
0.329 |
|
| 2006 |
Singh N, Chevé G, Avery MA, McCurdy CR. Comparative protein modeling of 1-deoxy-D-xylulose-5-phosphate reductoisomerase enzyme from Plasmodium falciparum: a potential target for antimalarial drug discovery. Journal of Chemical Information and Modeling. 46: 1360-70. PMID 16711755 DOI: 10.1021/Ci050523W |
0.346 |
|
| 2006 |
Mora FD, Jones DK, Desai PV, Patny A, Avery MA, Feller DR, Smillie T, Zhou YD, Nagle DG. Bioassay for the identification of natural product-based activators of peroxisome proliferator-activated receptor-gamma (PPARgamma): the marine sponge metabolite psammaplin A activates PPARgamma and induces apoptosis in human breast tumor cells. Journal of Natural Products. 69: 547-52. PMID 16643023 DOI: 10.1021/Np050397Q |
0.318 |
|
| 2006 |
Desai PV, Patny A, Gut J, Rosenthal PJ, Tekwani B, Srivastava A, Avery M. Identification of novel parasitic cysteine protease inhibitors by use of virtual screening. 2. The available chemical directory. Journal of Medicinal Chemistry. 49: 1576-84. PMID 16509575 DOI: 10.1021/Jm0505765 |
0.439 |
|
| 2006 |
Bashyal B, Desai P, Rao KV, Hamann MT, Avery BA, Reed JK, Avery MA. Terpenes from Eunicea laciniata and Plexaurella nutans Journal of Chemical Research-S. 2006: 165-167. DOI: 10.3184/030823406776330729 |
0.325 |
|
| 2006 |
Tumuluri VS, Kemper MS, Sheri A, Choi SR, Lewis IR, Avery MA, Avery BA. Use of Raman spectroscopy to characterize hydrogenation reactions Organic Process Research and Development. 10: 927-933. DOI: 10.1021/Op0600355 |
0.525 |
|
| 2006 |
Jung J, Avery MA. An efficient synthesis of cyclic urethanes from Boc-protected amino acids through a metal triflate-catalyzed intramolecular diazocarbonyl insertion reaction Tetrahedron Letters. 47: 7969-7972. DOI: 10.1016/J.Tetlet.2006.08.111 |
0.304 |
|
| 2006 |
Jung J, Avery MA. Diastereoselective synthesis of (2S,5S)- and (2S,5R)-N-benzyloxycarbonyl-5-hydroxypipecolic acids from trans-4-hydroxy-l-proline Tetrahedron-Asymmetry. 17: 2479-2486. DOI: 10.1016/J.Tetasy.2006.07.035 |
0.32 |
|
| 2006 |
Watkins EB, Chittiboyina AG, Avery MA. Recent Developments in the Syntheses of the Epothilones and Related Analogues European Journal of Organic Chemistry. 2006: 4071-4084. DOI: 10.1002/Ejoc.200600149 |
0.385 |
|
| 2005 |
Bhagavathula N, Nerusu KC, Reddy M, Ellis CN, Chittiboyina A, Avery M, Pershadsingh HA, Kurtz TW, Varani J. BP-1107 [{2-[4-(2,4-dioxo-thiazolidin-5-ylmethyl)-phenoxy]-ethyl}-methyl-amide]: a novel synthetic thiazolidinedione that inhibits epidermal hyperplasia in psoriatic skin-severe-combined immunodeficient mouse transplants after topical application. The Journal of Pharmacology and Experimental Therapeutics. 315: 996-1004. PMID 16109743 DOI: 10.1124/Jpet.105.091066 |
0.589 |
|
| 2005 |
Watkins EB, Chittiboyina AG, Jung JC, Avery MA. The epothilones and related analogues-a review of their syntheses and anti-cancer activities. Current Pharmaceutical Design. 11: 1615-53. PMID 15892666 DOI: 10.2174/1381612053764742 |
0.626 |
|
| 2005 |
Burk O, Arnold KA, Nussler AK, Schaeffeler E, Efimova E, Avery BA, Avery MA, Fromm MF, Eichelbaum M. Antimalarial artemisinin drugs induce cytochrome P450 and MDR1 expression by activation of xenosensors pregnane X receptor and constitutive androstane receptor. Molecular Pharmacology. 67: 1954-65. PMID 15761118 DOI: 10.1124/Mol.104.009019 |
0.329 |
|
| 2005 |
Desai PV, Avery MA. Structural characterization of vivapain-2 and vivapain-3, cysteine proteases from Plasmodium vivax: comparative protein modeling and docking studies. Journal of Biomolecular Structure & Dynamics. 21: 781-90. PMID 15107000 DOI: 10.1080/07391102.2004.10506968 |
0.369 |
|
| 2005 |
Labadie GR, Carvalho PB, Batra S, Choi S, Khan SI, Tekwani BL, Avery MA. Solid-Supported Parallel Synthesis of Hydroxybenzylamine Libraries Possessing Antileishmial Activity Medicinal Chemistry Research. 14: 332-346. DOI: 10.1007/S00044-006-0142-6 |
0.767 |
|
| 2005 |
Goud PM, Sheri A, Desai PV, Watkins EB, Tekwani B, Sabnis Y, Gut J, Rosenthal PJ, Avery MA. Design, Synthesis and Evaluation of Trisubstituted Thiazoles Targeting Plasmodium Falciparum Cysteine Proteases Medicinal Chemistry Research. 14: 74-105. DOI: 10.1007/S00044-005-0126-Y |
0.765 |
|
| 2004 |
Sawant SS, Sylvester PW, Avery MA, Desai P, Youssef DT, El Sayed KA. Bioactive rearranged and halogenated semisynthetic derivatives of the marine natural product sarcophine. Journal of Natural Products. 67: 2017-23. PMID 15620244 DOI: 10.1021/Np0497393 |
0.338 |
|
| 2004 |
Jung JC, Kache R, Vines KK, Zheng YS, Bijoy P, Valluri M, Avery MA. Total syntheses of epothilones B and d. The Journal of Organic Chemistry. 69: 9269-84. PMID 15609966 DOI: 10.1021/Jo048742O |
0.312 |
|
| 2004 |
Desai PV, Patny A, Sabnis Y, Tekwani B, Gut J, Rosenthal P, Srivastava A, Avery M. Identification of novel parasitic cysteine protease inhibitors using virtual screening. 1. The ChemBridge database. Journal of Medicinal Chemistry. 47: 6609-15. PMID 15588096 DOI: 10.1021/Jm0493717 |
0.77 |
|
| 2004 |
McLuskey K, Gibellini F, Carvalho P, Avery MA, Hunter WN. Inhibition of Leishmania major pteridine reductase by 2,4,6-triaminoquinazoline: structure of the NADPH ternary complex. Acta Crystallographica. Section D, Biological Crystallography. 60: 1780-5. PMID 15388924 DOI: 10.1107/S0907444904018955 |
0.362 |
|
| 2004 |
Parshikov IA, Muraleedharan KM, Miriyala B, Avery MA, Williamson JS. Hydroxylation of 10-deoxoartemisinin by Cunninghamella elegans. Journal of Natural Products. 67: 1595-7. PMID 15387669 DOI: 10.1021/Np040089C |
0.311 |
|
| 2004 |
Tripathi AK, Desai PV, Pradhan A, Khan SI, Avery MA, Walker LA, Tekwani BL. An alpha-proteobacterial type malate dehydrogenase may complement LDH function in Plasmodium falciparum. Cloning and biochemical characterization of the enzyme. European Journal of Biochemistry / Febs. 271: 3488-502. PMID 15317584 DOI: 10.1111/J.1432-1033.2004.04281.X |
0.338 |
|
| 2004 |
Venkatraman MS, Chittiboyina A, Meingassner J, Ho CI, Varani J, Ellis CN, Avery MA, Pershadsingh HA, Kurtz TW, Benson SC. Alpha-Lipoic acid-based PPARgamma agonists for treating inflammatory skin diseases. Archives of Dermatological Research. 296: 97-104. PMID 15221328 DOI: 10.1007/S00403-004-0480-5 |
0.618 |
|
| 2004 |
Benson SC, Pershadsingh HA, Ho CI, Chittiboyina A, Desai P, Pravenec M, Qi N, Wang J, Avery MA, Kurtz TW. Identification of telmisartan as a unique angiotensin II receptor antagonist with selective PPARgamma-modulating activity. Hypertension. 43: 993-1002. PMID 15007034 DOI: 10.1161/01.Hyp.0000123072.34629.57 |
0.582 |
|
| 2004 |
Bhagavathula N, Nerusu KC, Lal A, Ellis CN, Chittiboyina A, Avery MA, Ho CI, Benson SC, Pershadsingh HA, Kurtz TW, Varani J. Rosiglitazone inhibits proliferation, motility, and matrix metalloproteinase production in keratinocytes. The Journal of Investigative Dermatology. 122: 130-9. PMID 14962101 DOI: 10.1046/J.0022-202X.2003.22111.X |
0.568 |
|
| 2004 |
Labadie GR, Choi SR, Avery MA. Diamine derivatives with antiparasitic activities. Bioorganic & Medicinal Chemistry Letters. 14: 615-9. PMID 14741254 DOI: 10.1016/J.Bmcl.2003.11.055 |
0.765 |
|
| 2004 |
Parshikov IA, Muraleedharan KM, Avery MA, Williamson JS. Transformation of artemisinin by Cunninghamella elegans. Applied Microbiology and Biotechnology. 64: 782-6. PMID 14735322 DOI: 10.1007/S00253-003-1524-Z |
0.305 |
|
| 2004 |
Chittiboyina AG, Reddy CR, Watkins EB, Avery MA. First synthesis of antimalarial Machaeriols A and B Tetrahedron Letters. 45: 1689-1691. DOI: 10.1016/J.Tetlet.2003.12.107 |
0.359 |
|
| 2003 |
Peng J, Hu JF, Kazi AB, Li Z, Avery M, Peraud O, Hill RT, Franzblau SG, Zhang F, Schinazi RF, Wirtz SS, Tharnish P, Kelly M, Wahyuono S, Hamann MT. Manadomanzamines A and B: a novel alkaloid ring system with potent activity against mycobacteria and HIV-1. Journal of the American Chemical Society. 125: 13382-6. PMID 14583033 DOI: 10.1021/Ja030087Z |
0.482 |
|
| 2003 |
Avery MA, Muraleedharan KM, Desai PV, Bandyopadhyaya AK, Furtado MM, Tekwani BL. Structure-activity relationships of the antimalarial agent artemisinin. 8. design, synthesis, and CoMFA studies toward the development of artemisinin-based drugs against leishmaniasis and malaria. Journal of Medicinal Chemistry. 46: 4244-58. PMID 13678403 DOI: 10.1021/Jm030181Q |
0.445 |
|
| 2003 |
Batra S, Sabnis YA, Rosenthal PJ, Avery MA. Structure-based approach to falcipain-2 inhibitors: synthesis and biological evaluation of 1,6,7-trisubstituted dihydroisoquinolines and isoquinolines. Bioorganic & Medicinal Chemistry. 11: 2293-9. PMID 12713840 DOI: 10.1016/S0968-0896(03)00117-2 |
0.778 |
|
| 2003 |
Sabnis YA, Desai PV, Rosenthal PJ, Avery MA. Probing the structure of falcipain-3, a cysteine protease from Plasmodium falciparum: comparative protein modeling and docking studies. Protein Science : a Publication of the Protein Society. 12: 501-9. PMID 12592020 DOI: 10.1110/Ps.0228103 |
0.755 |
|
| 2003 |
Illapakurthy AC, Sabnis YA, Avery BA, Avery MA, Wyandt CM. Interaction of artemisinin and its related compounds with hydroxypropyl-beta-cyclodextrin in solution state: experimental and molecular-modeling studies. Journal of Pharmaceutical Sciences. 92: 649-55. PMID 12587126 DOI: 10.1002/Jps.10319 |
0.734 |
|
| 2003 |
Muri EMF, Mishra H, Avery MA, Williamson JS. Design and Synthesis of Heterocyclic Hydroxamic Acid Derivatives as Inhibitors of Helicobacter pylori Urease Synthetic Communications. 33: 1977-1995. DOI: 10.1081/Scc-120021024 |
0.367 |
|
| 2003 |
Avery MA, Woolfrey JR. Anti-Inflammatory Steroids Burger's Medicinal Chemistry and Drug Discovery. 747-854. DOI: 10.1002/0471266949.Bmc056 |
0.74 |
|
| 2002 |
Mineno T, Stanford KM, Walker LA, Avery MA. Solution-phase parallel synthesis of an isoflavone library for the discovery of novel antigiardial agents. Combinatorial Chemistry & High Throughput Screening. 5: 481-7. PMID 12470277 DOI: 10.2174/1386207023330138 |
0.726 |
|
| 2002 |
El Sayed KA, Yousaf M, Hamann MT, Avery MA, Kelly M, Wipf P. Microbial and chemical transformation studies of the bioactive marine sesquiterpenes (S)-(+)-curcuphenol and -curcudiol isolated from a deep reef collection of the Jamaican sponge Didiscus oxeata. Journal of Natural Products. 65: 1547-53. PMID 12444675 DOI: 10.1021/Np020213X |
0.325 |
|
| 2002 |
Lima PC, Avery MA, Tekwani BL, de Alves HM, Barreiro EJ, Fraga CA. Synthesis and biological evaluation of new imidazo[1,2-a]pyridine derivatives designed as mefloquine analogues. Farmaco (Societã Chimica Italiana : 1989). 57: 825-32. PMID 12420878 DOI: 10.1016/S0014-827X(02)01304-6 |
0.462 |
|
| 2002 |
Jaradat MS, Noonan DJ, Wu B, Avery MA, Feller DR, Jardat MS. Pseudolaric acid analogs as a new class of peroxisome proliferator-activated receptor agonists. Planta Medica. 68: 667-71. PMID 12221584 DOI: 10.1055/S-2002-33785 |
0.337 |
|
| 2002 |
Avery MA, Alvim-Gaston M, Vroman JA, Wu B, Ager A, Peters W, Robinson BL, Charman W. Structure-activity relationships of the antimalarial agent artemisinin. 7. Direct modification of (+)-artemisinin and in vivo antimalarial screening of new, potential preclinical antimalarial candidates. Journal of Medicinal Chemistry. 45: 4321-35. PMID 12213073 DOI: 10.1021/Jm020142Z |
0.463 |
|
| 2002 |
Sabnis Y, Rosenthal PJ, Desai P, Avery MA. Homology modeling of falcipain-2: validation, de novo ligand design and synthesis of novel inhibitors. Journal of Biomolecular Structure & Dynamics. 19: 765-74. PMID 11922834 DOI: 10.1080/07391102.2002.10506783 |
0.763 |
|
| 2002 |
Avery MA, Alvim-Gaston M, Rodrigues CR, Barreiro EJ, Cohen FE, Sabnis YA, Woolfrey JR. Structure-activity relationships of the antimalarial agent artemisinin. 6. The development of predictive in vitro potency models using CoMFA and HQSAR methodologies. Journal of Medicinal Chemistry. 45: 292-303. PMID 11784134 DOI: 10.1021/Jm0100234 |
0.799 |
|
| 2002 |
Vyas N, Avery BA, Avery MA, Wyandt CM. Carrier-mediated partitioning of artemisinin into Plasmodium falciparum-infected erythrocytes. Antimicrobial Agents and Chemotherapy. 46: 105-9. PMID 11751119 DOI: 10.1128/Aac.46.1.105-109.2002 |
0.302 |
|
| 2002 |
Jung JC, Watkins EB, Avery MA. Efficient Synthesis Of 4-Ethoxycarbonyl Pyrazolin-5-One Derivatives Synthetic Communications. 32: 3767-3777. DOI: 10.1081/Scc-120015395 |
0.338 |
|
| 2002 |
Mineno T, Choi S, Avery MA. A Mild Deprotection of Trichloroethyl Carbamates Using Indium Metal Synlett. 2002: 883-886. DOI: 10.1055/S-2002-31919 |
0.719 |
|
| 2002 |
Wu B, Karle JM, Watkins EB, Avery MA. Toward the total synthesis of pseudolaric acid B. Preparation of a key intermediate by degradation and its use in the reassembly of the natural product Tetrahedron Letters. 43: 4095-4098. DOI: 10.1016/S0040-4039(02)00596-8 |
0.318 |
|
| 2002 |
El Sayed KA, Orabi KY, Dunbar DC, Hamann MT, Avery MA, Sabnis YA, Mossa JS, El-Feraly FS. Transformation of lactone to lactam in sarcophine and antimalarial activity of the resulting N-substituted azasarcophines Tetrahedron. 58: 3699-3708. DOI: 10.1016/S0040-4020(02)00330-7 |
0.745 |
|
| 2002 |
Jung J, Watkins EB, Avery MA. Synthesis of 3-substituted and 3,4-disubstituted pyrazolin-5-ones Tetrahedron. 58: 3639-3646. DOI: 10.1016/S0040-4020(02)00306-X |
0.337 |
|
| 2001 |
Hindupur RM, Panicker B, Valluri M, Avery MA. Total synthesis of epothilone A Tetrahedron Letters. 42: 7341-7344. DOI: 10.1016/S0040-4039(01)01585-4 |
0.321 |
|
| 2001 |
Valluri M, Mineno T, Hindupur RM, Avery MA. Indium-mediated chemoselective deprotection of trichloroethoxycarbonyl and trichloroacetyl groups Tetrahedron Letters. 42: 7153-7154. DOI: 10.1016/S0040-4039(01)01489-7 |
0.645 |
|
| 2000 |
Valluri M, Hindupur RM, Bijoy P, Labadie G, Jung J, Avery MA. Total synthesis of epothilone B. Organic Letters. 3: 3607-3609. PMID 11700093 DOI: 10.1021/Ol016173Q |
0.639 |
|
| 2000 |
Khan IA, Avery MA, Burandt CL, Goins DK, Mikell JR, Nash TE, Azadegan A, Walker LA. Antigiardial activity of isoflavones from Dalbergia frutescens bark. Journal of Natural Products. 63: 1414-6. PMID 11076565 DOI: 10.1021/Np000010D |
0.379 |
|
| 2000 |
Panicker B, Karle JM, Avery MA. An unusual reversal of stereoselectivity in a boron mediated aldol reaction: Enantioselective synthesis of the C1-C6 segment of the epothilones Tetrahedron. 56: 7859-7868. DOI: 10.1016/S0040-4020(00)00708-0 |
0.316 |
|
| 1999 |
Avery BA, Venkatesh KK, Avery MA. Rapid determination of artemisinin and related analogues using high-performance liquid chromatography and an evaporative light scattering detector. Journal of Chromatography. B, Biomedical Sciences and Applications. 730: 71-80. PMID 10437674 DOI: 10.1016/S0378-4347(99)00185-1 |
0.35 |
|
| 1999 |
Bhattacharyya S, Neidigh KA, Avery MA, Williamson JS. Selective Monoalkylation of Ammonia: A High Throughput Synthesis of Primary Amines Synlett. 1999: 1781-1783. DOI: 10.1055/S-1999-2946 |
0.302 |
|
| 1999 |
Dayan FE, Hernández A, Allen SN, Moraes RM, Vroman JA, Avery MA, Duke SO. Comparative phytotoxicity of artemisinin and several sesquiterpene analogues Phytochemistry. 50: 607-614. DOI: 10.1016/S0031-9422(98)00568-8 |
0.366 |
|
| 1998 |
Woolfrey JR, Avery MA, Doweyko AM. Comparison of 3D quantitative structure-activity relationship methods: analysis of the in vitro antimalarial activity of 154 artemisinin analogues by hypothetical active-site lattice and comparative molecular field analysis. Journal of Computer-Aided Molecular Design. 12: 165-81. PMID 9690175 DOI: 10.1023/A:1007967517859 |
0.756 |
|
| 1998 |
Johnson T, Khan IA, Avery MA, Grant J, Meshnick SR. Quantitative Structure-Activity Relationship Studies of a Series of Sulfa Drugs as Inhibitors of Pneumocystis carinii Dihydropteroate Synthetase Antimicrobial Agents and Chemotherapy. 42: 1454-1458. DOI: 10.1128/Aac.42.6.1454 |
0.388 |
|
| 1998 |
Neidigh KA, Avery MA, Williamson JS, Bhattacharyya S. Facile preparation of N-methyl secondary amines by titanium(IV) isopropoxide-mediated reductive amination of carbonyl compounds Journal of the Chemical Society-Perkin Transactions 1. 2527-2532. DOI: 10.1039/A803703E |
0.36 |
|
| 1998 |
Bijoy P, Avery MA. Synthetic Studies Directed Towards Epothilone A : Enantioselective Synthesis Of A C7 - C15 Carboxaldehyde Segment Tetrahedron Letters. 39: 209-212. DOI: 10.1016/S0040-4039(97)10527-5 |
0.307 |
|
| 1997 |
Vroman JA, Khan IA, Avery MA. Copper(I) Catalyzed Conjugate Addition of Grignard Reagents to Acrylic Acids: Homologation of Artemisinic Acid and Subsequent Conversion to 9-Substituted Artemisinin Analogs Tetrahedron Letters. 38: 6173-6176. DOI: 10.1016/S0040-4039(97)01428-7 |
0.307 |
|
| 1996 |
Meshnick SR, Jefford CW, Posner GH, Avery MA, Peters W. Second-generation antimalarial endoperoxides. Parasitology Today (Personal Ed.). 12: 79-82. PMID 15275260 DOI: 10.1016/0169-4758(96)80660-0 |
0.424 |
|
| 1996 |
Avery MA, Mehrotra S, Johnson TL, Bonk JD, Vroman JA, Miller R. Structure-activity relationships of the antimalarial agent artemisinin. 5. Analogs of 10-deoxoartemisinin substituted at C-3 and C-9. Journal of Medicinal Chemistry. 39: 4149-55. PMID 8863791 DOI: 10.1021/Jm9603577 |
0.388 |
|
| 1996 |
Avery MA, Mehrotra S, Bonk JD, Vroman JA, Goins DK, Miller R. Structure-activity relationships of the antimalarial agent artemisinin. 4. Effect of substitution at C-3. Journal of Medicinal Chemistry. 39: 2900-6. PMID 8709124 DOI: 10.1021/jm960200e |
0.322 |
|
| 1995 |
Avery MA, Bonk JD, Chong WK, Mehrotra S, Miller R, Milhous W, Goins DK, Venkatesan S, Wyandt C, Khan I. Structure-activity relationships of the antimalarial agent artemisinin. 2. Effect of heteroatom substitution at O-11: synthesis and bioassay of N-alkyl-11-aza-9-desmethylartemisinins. Journal of Medicinal Chemistry. 38: 5038-44. PMID 8544180 DOI: 10.1021/Jm00026A011 |
0.733 |
|
| 1995 |
Avery MA, Fan P, Karle JM, Miller R, Goins K. Replacement of the nonperoxidic trioxane oxygen atom of artemisinin by carbon: Total synthesis of (+)-13-carbaartemisinin and related structures Tetrahedron Letters. 36: 3965-3968. DOI: 10.1016/0040-4039(95)00689-A |
0.315 |
|
| 1994 |
Lillie BM, Avery MA. The protection of ketones and aldehydes as 4-trimethylsilylmethyl-1,3-dioxolanes Tetrahedron Letters. 35: 969-972. DOI: 10.1016/S0040-4039(00)79941-2 |
0.397 |
|
| 1994 |
Avery MA, Gao F, Chong WKM, Hendrickson TF, Inman WD, Crews P. Synthesis, conformational analysis, and antimalarial activity of tricyclic analogs of artemisinin Tetrahedron. 50: 957-972. DOI: 10.1016/S0040-4020(01)80810-3 |
0.315 |
|
| 1993 |
Avery MA, Gao F, Chong WK, Mehrotra S, Milhous WK. Structure-activity relationships of the antimalarial agent artemisinin. 1. Synthesis and comparative molecular field analysis of C-9 analogs of artemisinin and 10-deoxoartemisinin. Journal of Medicinal Chemistry. 36: 4264-75. PMID 8277509 DOI: 10.1021/Jm00078A017 |
0.743 |
|
| 1990 |
Avery MA, Detre G, Yasuda D, Chao WR, Tanabe M, Crowe D, Peters R, Chong WK. Synthesis and antiinflammatory activity of novel 12 beta-substituted analogues of betamethasone. Journal of Medicinal Chemistry. 33: 1852-8. PMID 2362263 DOI: 10.1021/Jm00169A004 |
0.686 |
|
| 1990 |
Avery MA, Tanabe M, Crowe DF, Detre G, Peters RH, Chong WK. Synthesis and testing of 17a beta-hydroxy-7 alpha-methyl-D-homoestra-4,16-dien-3-one: a highly potent orally active androgen. Steroids. 55: 59-64. PMID 2326828 DOI: 10.1016/0039-128X(90)90025-7 |
0.687 |
|
| 1990 |
Avery MA, Chong WKM, Bupp JE. Tricyclic analogues of artemisinin: synthesis and antimalarial activity of (+)-4,5-secoartemisinin and (–)-5-nor-4,5-secoartemisinin Journal of the Chemical Society, Chemical Communications. 1487-1489. DOI: 10.1039/C39900001487 |
0.405 |
|
| 1990 |
Avery MA, Chong WKM, Detre G. Synthesis of (+)-8a,9-secoartemisinin and related analogs Tetrahedron Letters. 31: 1799-1802. DOI: 10.1016/S0040-4039(00)98789-6 |
0.359 |
|
| 1989 |
Peters RH, Crowe DF, Avery MA, Chong WK, Tanabe M. 11 beta-nitrate estrane analogues: potent estrogens. Journal of Medicinal Chemistry. 32: 2306-10. PMID 2795603 DOI: 10.1021/Jm00130A014 |
0.678 |
|
| 1989 |
Peters RH, Crowe DF, Avery MA, Chong WK, Tanabe M. 17-Desoxy estrogen analogues. Journal of Medicinal Chemistry. 32: 1642-52. PMID 2738897 DOI: 10.1021/Jm00127A040 |
0.717 |
|
| 1989 |
Avery MA, Jennings-White C, Chong WKM. Simplified analogs of the antimalarial artemisinin: synthesis of 6,9-desmethylartemisinin Journal of Organic Chemistry. 54: 1792-1795. DOI: 10.1021/Jo00269A009 |
0.367 |
|
| 1989 |
White JD, Avery MA, Choudhry SC, Dhingra OP, Gray BD, Kang MC, Kuo SC, Whittle AJ. Total synthesis of boromycin Journal of the American Chemical Society. 111: 790-792. DOI: 10.1021/Ja00184A088 |
0.476 |
|
| 1988 |
Peters RH, Crowe DF, Avery MA, Chong WK, Tanabe M. Analogues of [(triethylsilyl)ethynyl]estradiol as potential antifertility agents. Journal of Medicinal Chemistry. 31: 572-6. PMID 3346872 DOI: 10.1021/Jm00398A014 |
0.716 |
|
| 1988 |
Minagawa K, Furuta T, Kasuya Y, Fujino A, Avery MA, Tanabe M. Total synthesis of cortisol: application to selective deuteriation at C-1 and C-19 Journal of the Chemical Society-Perkin Transactions 1. 587-591. DOI: 10.1039/P19880000587 |
0.324 |
|
| 1987 |
Peters RH, Crowe DF, Tanabe M, Avery MA, Chong WK. Steroidal silicon side-chain analogues as potential antifertility agents. Journal of Medicinal Chemistry. 30: 646-52. PMID 3560158 DOI: 10.1021/Jm00387A011 |
0.712 |
|
| 1987 |
Avery MA, Jennings-White C, Chong WKM. The Total synthesis of (+)-artemisinin and (+)-9-desmethyltemesinin Tetrahedron Letters. 28: 4629-4632. DOI: 10.1016/S0040-4039(00)96582-1 |
0.316 |
|
| 1985 |
Reitz AB, Avery MA, Rosenkranz RP, Verlander MS, Melmon KL, Hoffman BB, Akita Y, Castagnoli N, Goodman M. Conjugates of catecholamines. 6. Synthesis and beta-adrenergic activity of N-(hydroxyalkyl)catecholamine derivatives. Journal of Medicinal Chemistry. 28: 642-7. PMID 2859373 DOI: 10.1021/Jm50001A018 |
0.558 |
|
| 1985 |
REITZ AB, AVERY MA, ROSENKRANZ RP, VERLANDER MS, MELMON KL, HOFFMAN BB, AKITA Y, CASTAGNOLI N, GOODMAN M. ChemInform Abstract: CONJUGATES OF CATECHOLAMINES. 6. SYNTHESIS AND β-ADRENERGIC ACTIVITY OF N-(HYDROXYALKYL)CATECHOLAMINE DERIVATIVES Chemischer Informationsdienst. 16. DOI: 10.1002/Chin.198534180 |
0.31 |
|
| 1984 |
WHITE JD, AVERY MA, CHOUDHRY SC, DHINGRA OP, KANG M, WHITTLE AJ. ChemInform Abstract: STEREOCONTROLLED SYNTHESIS OF THE C(1)-C(17) HALF OF BOROMYCIN Chemischer Informationsdienst. 15. DOI: 10.1002/Chin.198404338 |
0.433 |
|
| 1983 |
White JD, Avery MA, Choudhry SC, Dhingra OP, Kang MC, Whittle AJ. Stereocontrolled synthesis of the C(1)-C(17) half of boromycin Journal of the American Chemical Society. 105: 6517-6518. DOI: 10.1021/Ja00359A041 |
0.429 |
|
| 1981 |
Avery M, Verlander M, Goodman M. Correction. Synthesis of 6-Aminoisproterenol Journal of Organic Chemistry. 46: 5459-5459. DOI: 10.1021/Jo00339A603 |
0.462 |
|
| 1981 |
Reitz A, Avery MA, Verlander MS, Goodman M. Synthesis of ring-alkylated isoproterenol derivatives Journal of Organic Chemistry. 13: 4859-4863. DOI: 10.1021/Jo00337A007 |
0.502 |
|
| 1981 |
White JD, Ruppert JF, Avery MA, Torii S, Nokami J. Spiroannelation via intramolecular ketocarbenoid addition. Stereocontrolled synthesis of (-)-acorenone B and (.+-.)-.alpha.-chamigrene Journal of the American Chemical Society. 103: 1813-1821. DOI: 10.1021/Ja00397A040 |
0.445 |
|
| 1980 |
Avery MA, Verlander MS, Goodman M. Synthesis of 6-aminoisoproterenol Journal of Organic Chemistry. 11: 2750-2753. DOI: 10.1021/Jo01302A003 |
0.479 |
|
| 1977 |
RUPPERT JF, AVERY MA, WHITE JD. ChemInform Abstract: SYNTHESIS OF (-)-ACORENONE B Chemischer Informationsdienst. 8: no-no. DOI: 10.1002/Chin.197714349 |
0.448 |
|
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