| Year |
Citation |
Score |
| 2024 |
Gazzillo E, Colarusso E, Giordano A, Chini MG, Potenza M, Hofstetter RK, Iorizzi M, Werz O, Lauro G, Bifulco G. Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH). Chempluschem. e202400234. PMID 38753468 DOI: 10.1002/cplu.202400234 |
0.76 |
|
| 2024 |
De Vita S, Colarusso E, Chini MG, Bifulco G, Lauro G. PharmaCore: The Automatic Generation of 3D Structure-Based Pharmacophore Models from Protein/Ligand Complexes. Journal of Chemical Information and Modeling. PMID 38728062 DOI: 10.1021/acs.jcim.3c01920 |
0.712 |
|
| 2024 |
Colarusso E, Chini MG, Bifulco G, Lauro G, Giordano A. Identification and Development of BRD9 Chemical Probes. Pharmaceuticals (Basel, Switzerland). 17. PMID 38543178 DOI: 10.3390/ph17030392 |
0.692 |
|
| 2024 |
Samukha V, Fantasma F, D'Urso G, Caprari C, De Felice V, Saviano G, Lauro G, Casapullo A, Chini MG, Bifulco G, Iorizzi M. NMR Metabolomics and Chemometrics of Commercial Varieties of L. Seeds from Italy and In Vitro Antioxidant and Antifungal Activity. Plants (Basel, Switzerland). 13. PMID 38256780 DOI: 10.3390/plants13020227 |
0.646 |
|
| 2024 |
Capuano A, D'Urso G, Aliberti M, Ruggiero D, Terracciano S, Festa C, Tosco A, Chini MG, Lauro G, Bifulco G, Casapullo A. Chemoproteomics Reveals USP5 (Ubiquitin Carboxyl-Terminal Hydrolase 5) as Promising Target of the Marine Polyketide Gracilioether A. Marine Drugs. 22. PMID 38248666 DOI: 10.3390/md22010041 |
0.709 |
|
| 2024 |
Ciaglia T, Vestuto V, Di Sarno V, Musella S, Smaldone G, Di Matteo F, Napolitano V, Miranda MR, Pepe G, Basilicata MG, Novi S, Capolupo I, Bifulco G, Campiglia P, Gomez-Monterrey I, ... ... Lauro G, et al. Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterization. European Journal of Medicinal Chemistry. 266: 116128. PMID 38232463 DOI: 10.1016/j.ejmech.2024.116128 |
0.566 |
|
| 2023 |
De Vita S, Meninno S, Capasso L, Colarusso E, Chini MG, Lauro G, Rinaldi R, De Cicco A, Sian V, Terracciano S, Nebbioso A, Lattanzi A, Bifulco G. 2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines. Bioorganic & Medicinal Chemistry. 93: 117444. PMID 37611334 DOI: 10.1016/j.bmc.2023.117444 |
0.729 |
|
| 2023 |
Gazzillo E, Pierri M, Colarusso E, Chini MG, Ferraro MG, Piccolo M, Irace C, Bruno I, Bifulco G, Terracciano S, Lauro G. Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9. Bioorganic Chemistry. 139: 106677. PMID 37352721 DOI: 10.1016/j.bioorg.2023.106677 |
0.763 |
|
| 2023 |
Rogati F, Maioli C, Lauro G, Caprioglio D, Imperio D, Del Grosso E, Botta B, Mannina L, Bifulco G, Ingallina C, Minassi A. A Classic Photochemical Approach Inducing an Unexpected Rearrangement: Exploring the Photoreactivity of Pentacyclic Triterpenic Acids. Journal of Natural Products. PMID 37036806 DOI: 10.1021/acs.jnatprod.3c00067 |
0.49 |
|
| 2023 |
De Vita S, Chini MG, Bifulco G, Lauro G. Target identification by structure-based computational approaches: Recent advances and perspectives. Bioorganic & Medicinal Chemistry Letters. 83: 129171. PMID 36739998 DOI: 10.1016/j.bmcl.2023.129171 |
0.702 |
|
| 2022 |
Potenza M, Giordano A, Chini MG, Saviano A, Kretzer C, Raucci F, Russo M, Lauro G, Terracciano S, Bruno I, Iorizzi M, Hofstetter RK, Pace S, Maione F, Werz O, et al. Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E and Leukotriene Biosynthesis Inhibitors. Acs Medicinal Chemistry Letters. 14: 26-34. PMID 36655121 DOI: 10.1021/acsmedchemlett.2c00343 |
0.784 |
|
| 2022 |
Colarusso E, Ceccacci S, Monti MC, Gazzillo E, Giordano A, Chini MG, Ferraro MG, Piccolo M, Ruggiero D, Irace C, Terracciano S, Bruno I, Bifulco G, Lauro G. Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders. European Journal of Medicinal Chemistry. 247: 115018. PMID 36577218 DOI: 10.1016/j.ejmech.2022.115018 |
0.745 |
|
| 2022 |
Kılınc H, Masullo M, Lauro G, D'Urso G, Alankus O, Bifulco G, Piacente S. Scabiosa atropurpurea: A rich source of iridoids with α-glucosidase inhibitory activity evaluated by in vitro and in silico studies. Phytochemistry. 205: 113471. PMID 36241054 DOI: 10.1016/j.phytochem.2022.113471 |
0.527 |
|
| 2022 |
Micco SD, Lauro G, Bifulco G. Extensive molecular dynamics simulations disclosed the stability of mPGES-1 enzyme and the structural role of glutathione (GSH) cofactor. Molecular Informatics. PMID 36075865 DOI: 10.1002/minf.202200140 |
0.737 |
|
| 2022 |
De Vita S, Finamore C, Chini MG, Saviano G, De Felice V, De Marino S, Lauro G, Casapullo A, Fantasma F, Trombetta F, Bifulco G, Iorizzi M. Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches. Plants (Basel, Switzerland). 11. PMID 35807623 DOI: 10.3390/plants11131671 |
0.645 |
|
| 2022 |
Gazzillo E, Terracciano S, Ruggiero D, Potenza M, Chini MG, Lauro G, Fischer K, Hofstetter RK, Giordano A, Werz O, Bruno I, Bifulco G. Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation. Molecules (Basel, Switzerland). 27. PMID 35744994 DOI: 10.3390/molecules27123866 |
0.798 |
|
| 2022 |
Di Sarno V, Giovannelli P, Medina-Peris A, Ciaglia T, Di Donato M, Musella S, Lauro G, Vestuto V, Smaldone G, Di Matteo F, Bifulco G, Castoria G, Migliaccio A, Fernandez-Carvajal A, Campiglia P, et al. New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models. European Journal of Medicinal Chemistry. 238: 114435. PMID 35598411 DOI: 10.1016/j.ejmech.2022.114435 |
0.509 |
|
| 2022 |
Masullo M, Lauro G, Cerulli A, Bifulco G, Piacente S. : A Source of Diarylheptanoids With α-Glucosidase Inhibitory Activity Evaluated by and Studies. Frontiers in Plant Science. 13: 805660. PMID 35237285 DOI: 10.3389/fpls.2022.805660 |
0.499 |
|
| 2022 |
Ruggiero D, Terracciano S, Lauro G, Pecoraro M, Franceschelli S, Bifulco G, Bruno I. Structural Refinement of 2,4-Thiazolidinedione Derivatives as New Anticancer Agents Able to Modulate the BAG3 Protein. Molecules (Basel, Switzerland). 27. PMID 35163936 DOI: 10.3390/molecules27030665 |
0.559 |
|
| 2022 |
Saviano A, De Vita S, Chini MG, Marigliano N, Lauro G, Casillo GM, Raucci F, Iorizzi M, Hofstetter RK, Fischer K, Koeberle A, Werz O, Maione F, Bifulco G. In Silico, In Vitro, and In Vivo Analysis of Tanshinone IIA and Cryptotanshinone from as Modulators of Cyclooxygenase-2/mPGES-1/Endothelial Prostaglandin EP3 Pathway. Biomolecules. 12. PMID 35053247 DOI: 10.3390/biom12010099 |
0.677 |
|
| 2022 |
Pierri M, Gazzillo E, Chini MG, Ferraro MG, Piccolo M, Maione F, Irace C, Bifulco G, Bruno I, Terracciano S, Lauro G. Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders. Bioorganic Chemistry. 118: 105480. PMID 34823196 DOI: 10.1016/j.bioorg.2021.105480 |
0.752 |
|
| 2021 |
De Vita S, Chini MG, Bifulco G, Lauro G. Insights into the Ligand Binding to Bromodomain-Containing Protein 9 (BRD9): A Guide to the Selection of Potential Binders by Computational Methods. Molecules (Basel, Switzerland). 26. PMID 34885774 DOI: 10.3390/molecules26237192 |
0.688 |
|
| 2021 |
De Vita S, Chini MG, Saviano G, Finamore C, Festa C, Lauro G, De Marino S, Russo R, Avagliano C, Casapullo A, Calignano A, Bifulco G, Iorizzi M. Biological Profile of Two L. Metabolites Using Computational Approaches and In Vitro Tests. Biomolecules. 11. PMID 34680124 DOI: 10.3390/biom11101490 |
0.675 |
|
| 2021 |
Di Sarno V, Lauro G, Musella S, Ciaglia T, Vestuto V, Sala M, Scala MC, Smaldone G, Di Matteo F, Novi S, Tecce MF, Moltedo O, Bifulco G, Campiglia P, Gomez-Monterrey IM, et al. Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization. European Journal of Medicinal Chemistry. 226: 113863. PMID 34571172 DOI: 10.1016/j.ejmech.2021.113863 |
0.578 |
|
| 2021 |
Potenza M, Cavalluzzi MM, Milani G, Lauro G, Carino A, Roselli R, Fiorucci S, Zampella A, Pierri CL, Lentini G, Bifulco G. Inverse Virtual Screening for the rapid re-evaluation of the presumed biological safe profile of natural products. The case of steviol from Stevia rebaudiana glycosides on farnesoid X receptor (FXR). Bioorganic Chemistry. 111: 104897. PMID 33901797 DOI: 10.1016/j.bioorg.2021.104897 |
0.8 |
|
| 2021 |
Masullo M, Lauro G, Cerulli A, Kontek B, Olas B, Bifulco G, Piacente S, Pizza C. Giffonins, Antioxidant Diarylheptanoids from , and Their Ability to Prevent Oxidative Changes in Human Plasma Proteins. Journal of Natural Products. PMID 33616390 DOI: 10.1021/acs.jnatprod.0c01251 |
0.455 |
|
| 2020 |
De Vita S, Chini MG, Lauro G, Bifulco G. Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19). Rsc Advances. 10: 40867-40875. PMID 35519188 DOI: 10.1039/d0ra09010g |
0.738 |
|
| 2020 |
Farooq S, Qayum A, Nalli Y, Lauro G, Chini MG, Bifulco G, Chaubey A, Singh SK, Riyaz-Ul-Hassan S, Ali A. Discovery of a Secalonic Acid Derivative from , an Endophyte of Mill., Triggers Apoptosis in MDA-MB-231 Triple Negative Breast Cancer Cells. Acs Omega. 5: 24296-24310. PMID 33015446 DOI: 10.1021/acsomega.0c02505 |
0.667 |
|
| 2020 |
Bertamino A, Ostacolo C, Medina A, Di Sarno V, Lauro G, Ciaglia T, Vestuto V, Pepe G, Basilicata MG, Musella S, Smaldone G, Cristiano C, Gonzalez-Rodriguez S, Fernandez-Carvajal A, Bifulco G, et al. Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their In Vitro Characterization and In Vivo Analgesic Activities. Journal of Medicinal Chemistry. PMID 32787109 DOI: 10.1021/Acs.Jmedchem.0C00816 |
0.486 |
|
| 2020 |
Nemati F, Salehi P, Bararjanian M, Hadian N, Mohebbi M, Lauro G, Ruggiero D, Terracciano S, Bifulco G, Bruno I. Discovery of noscapine derivatives as potential β-tubulin inhibitors. Bioorganic & Medicinal Chemistry Letters. 30: 127489. PMID 32784088 DOI: 10.1016/J.Bmcl.2020.127489 |
0.562 |
|
| 2020 |
Lauro G, Terracciano S, Cantone V, Ruggiero D, Fischer K, Pace S, Werz O, Bruno I, Bifulco G. A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors. Chemmedchem. PMID 32022480 DOI: 10.1002/Cmdc.201900694 |
0.603 |
|
| 2020 |
Lauro G, Das P, Riccio R, Reddy DS, Bifulco G. DFT/NMR approach for the configuration assignment of groups of stereoisomers by the combination and comparison of experimental and predicted sets of data. The Journal of Organic Chemistry. PMID 31961156 DOI: 10.1021/Acs.Joc.9B03129 |
0.597 |
|
| 2019 |
De Vita S, Lauro G, Ruggiero D, Terracciano S, Riccio R, Bifulco G. Protein Preparation Automatic Protocol for High-Throughput Inverse Virtual Screening: Accelerating the Target Identification by Computational Methods. Journal of Chemical Information and Modeling. PMID 31593460 DOI: 10.1021/Acs.Jcim.9B00428 |
0.708 |
|
| 2019 |
Nalli Y, Jan S, Lauro G, Ur Rasool J, Lone WI, Sarkar AR, Banday J, Bifulco G, Laatsch H, Syed SH, Ali A. Isolation, Synthesis And Structure Determination Of Cannabidiol Derivatives And Their Cytotoxic Activities. Natural Product Research. 1-10. PMID 31282748 DOI: 10.1080/14786419.2019.1638381 |
0.575 |
|
| 2019 |
Sun P, Cai FY, Lauro G, Tang H, Su L, Wang HL, Li HH, Mándi A, Kurtán T, Riccio R, Bifulco G, Zhang W. Immunomodulatory Biscembranoids and Assignment of Their Relative and Absolute Configurations: Data Set Modulation in the Density Functional Theory/Nuclear Magnetic Resonance Approach. Journal of Natural Products. PMID 30957492 DOI: 10.1021/Acs.Jnatprod.8B01037 |
0.61 |
|
| 2019 |
Ostacolo C, Di Sarno V, Lauro G, Pepe G, Musella S, Ciaglia T, Vestuto V, Autore G, Bifulco G, Marzocco S, Campiglia P, Gomez-Monterrey IM, Bertamino A. Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach. European Journal of Medicinal Chemistry. 167: 61-75. PMID 30763817 DOI: 10.1016/J.Ejmech.2019.01.066 |
0.567 |
|
| 2018 |
Lauro G, Cantone V, Potenza M, Fischer K, Koeberle A, Werz O, Riccio R, Bifulco G. Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol. Medchemcomm. 9: 2028-2036. PMID 30746063 DOI: 10.1039/C8Md00497H |
0.806 |
|
| 2018 |
Jachak GR, Athawale PR, Agarwal H, Barthwal MK, Lauro G, Bifulco G, Reddy DS. Total synthesis of the potent anti-inflammatory natural product solomonamide A along with structural revision and biological activity evaluation. Organic & Biomolecular Chemistry. PMID 30478463 DOI: 10.1039/C8Ob02713G |
0.5 |
|
| 2018 |
Khalfaoui A, Chini MG, Bouheroum M, Belaabed S, Lauro G, Terracciano S, Vaccaro MC, Bruno I, Benayache S, Mancini I, Bifulco G. Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells. Journal of Natural Products. PMID 30063349 DOI: 10.1021/Acs.Jnatprod.8B00234 |
0.714 |
|
| 2018 |
Terracciano S, Lauro G, Russo A, Vaccaro MC, Vassallo A, De Marco M, Ranieri B, Rosati A, Turco MC, Riccio R, Bifulco G, Bruno I. Discovery and synthesis of the first selective BAG domain modulator of BAG3 as an attractive candidate for the development of a new class of chemotherapeutics. Chemical Communications (Cambridge, England). PMID 29926854 DOI: 10.1039/C8Cc03399D |
0.621 |
|
| 2017 |
Bertamino A, Lauro G, Ostacolo C, Di Sarno V, Musella S, Ciaglia T, Campiglia P, Bifulco G, Gomez-Monterrey IM. Ring-Fused Cyclic Aminals from Tetrahydro-β-carboline-Based Dipeptide Compounds. The Journal of Organic Chemistry. 82: 12014-12027. PMID 29091729 DOI: 10.1021/Acs.Joc.7B01656 |
0.448 |
|
| 2017 |
Proto MC, Fiore D, Piscopo C, Franceschelli S, Bizzarro V, Laezza C, Lauro G, Feoli A, Tosco A, Bifulco G, Sbardella G, Bifulco M, Gazzerro P. Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer. Scientific Reports. 7: 11678. PMID 28916833 DOI: 10.1038/S41598-017-11688-X |
0.4 |
|
| 2017 |
Liu HB, Lauro G, O'Connor RD, Lohith K, Kelly M, Colin P, Bifulco G, Bewley CA. Tulongicin, an Antibacterial Tri-Indole Alkaloid from a Deep-Water Topsentia sp. Sponge. Journal of Natural Products. PMID 28837335 DOI: 10.1021/Acs.Jnatprod.7B00452 |
0.475 |
|
| 2017 |
Cerulli A, Lauro G, Masullo M, Cantone V, Olas B, Kontek B, Nazzaro F, Bifulco G, Piacente S. Cyclic Diarylheptanoids from Corylus avellana Green Leafy Covers: Determination of Their Absolute Configurations and Evaluation of Their Antioxidant and Antimicrobial Activities. Journal of Natural Products. 80: 1703-1713. PMID 28520428 DOI: 10.1021/Acs.Jnatprod.6B00703 |
0.493 |
|
| 2017 |
Dardic D, Lauro G, Bifulco G, Laboudie P, Sakhaii P, Bauer A, Vilcinskas A, Hammann PE, Plaza A. Svetamycins A-G, Unusual Piperazic Acid-Containing Peptides from Streptomyces sp. The Journal of Organic Chemistry. PMID 28489377 DOI: 10.1021/Acs.Joc.7B00228 |
0.433 |
|
| 2017 |
Li J, Li C, Riccio R, Lauro G, Bifulco G, Li TJ, Tang H, Zhuang CL, Ma H, Sun P, Zhang W. Chemistry and Selective Tumor Cell Growth Inhibitory Activity of Polyketides from the South China Sea Sponge Plakortis sp. Marine Drugs. 15. PMID 28467388 DOI: 10.3390/Md15050129 |
0.668 |
|
| 2016 |
Sun P, Yu Q, Li J, Riccio R, Lauro G, Bifulco G, Kurtán T, Mándi A, Tang H, Li TJ, Zhuang CL, Gerwick WH, Zhang W. Bissubvilides A and B, Cembrane-Capnosane Heterodimers from the Soft Coral Sarcophyton subviride. Journal of Natural Products. PMID 27704808 DOI: 10.1021/Acs.Jnatprod.6B00453 |
0.61 |
|
| 2016 |
Lauro G, Manfra M, Pedatella S, Fischer K, Cantone V, Terracciano S, Bertamino A, Ostacolo C, Gomez-Monterrey I, De Nisco M, Riccio R, Novellino E, Werz O, Campiglia P, Bifulco G. Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening. European Journal of Medicinal Chemistry. 125: 278-287. PMID 27688183 DOI: 10.1016/J.Ejmech.2016.09.042 |
0.678 |
|
| 2016 |
Abbas Bukhari SN, Lauro G, Jantan I, Chee CF, Amjad MW, Bifulco G, Sher H, Abdullah I, Rahman NA. Anti-inflammatory trends of new benzimidazole derivatives. Future Medicinal Chemistry. PMID 27654499 DOI: 10.4155/Fmc-2016-0062 |
0.435 |
|
| 2016 |
Lauro G, Tortorella P, Bertamino A, Ostacolo C, Koeberle A, Fischer K, Bruno I, Terracciano S, Gomez-Monterrey IM, Tauro M, Loiodice F, Novellino E, Riccio R, Werz O, Campiglia P, et al. Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme. Chemmedchem. PMID 26915684 DOI: 10.1002/Cmdc.201500598 |
0.699 |
|
| 2015 |
Masullo M, Cantone V, Cerulli A, Lauro G, Messano F, Russo GL, Pizza C, Bifulco G, Piacente S. Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni". Journal of Natural Products. PMID 26606246 DOI: 10.1021/Acs.Jnatprod.5B00695 |
0.474 |
|
| 2015 |
Picaud S, Strocchia M, Terracciano S, Lauro G, Mendez J, Daniels DL, Riccio R, Bifulco G, Bruno I, Filippakopoulos P. 9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain. Journal of Medicinal Chemistry. 58: 2718-36. PMID 25703523 DOI: 10.1021/Jm501893K |
0.679 |
|
| 2015 |
Terracciano S, Lauro G, Strocchia M, Fischer K, Werz O, Riccio R, Bruno I, Bifulco G. Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors. Acs Medicinal Chemistry Letters. 6: 187-91. PMID 25699159 DOI: 10.1021/Ml500433J |
0.671 |
|
| 2014 |
Scrima M, Lauro G, Grimaldi M, Di Marino S, Tosco A, Picardi P, Gazzerro P, Riccio R, Novellino E, Bifulco M, Bifulco G, D'Ursi AM. Structural evidence of N6-isopentenyladenosine as a new ligand of farnesyl pyrophosphate synthase. Journal of Medicinal Chemistry. 57: 7798-803. PMID 25184810 DOI: 10.1021/Jm500869X |
0.692 |
|
| 2014 |
Nadmid S, Plaza A, Lauro G, Garcia R, Bifulco G, Müller R. Hyalachelins A-C, unusual siderophores isolated from the terrestrial myxobacterium Hyalangium minutum. Organic Letters. 16: 4130-3. PMID 25058569 DOI: 10.1021/Ol501826A |
0.438 |
|
| 2014 |
Bukhari SN, Lauro G, Jantan I, Bifulco G, Amjad MW. Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A₂, cyclooxygenases, lipoxygenase and proinflammatory cytokines. Bioorganic & Medicinal Chemistry. 22: 4151-61. PMID 24938495 DOI: 10.1016/J.Bmc.2014.05.052 |
0.533 |
|
| 2014 |
Lauro G, Strocchia M, Terracciano S, Bruno I, Fischer K, Pergola C, Werz O, Riccio R, Bifulco G. Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E₂ synthase-1 enzyme (mPGES-1). European Journal of Medicinal Chemistry. 80: 407-15. PMID 24794772 DOI: 10.1016/J.Ejmech.2014.04.061 |
0.68 |
|
| 2014 |
Gong J, Sun P, Jiang N, Riccio R, Lauro G, Bifulco G, Li TJ, Gerwick WH, Zhang W. New steroids with a rearranged skeleton as (h)P300 inhibitors from the sponge Theonella swinhoei. Organic Letters. 16: 2224-7. PMID 24694058 DOI: 10.1021/Ol5007345 |
0.666 |
|
| 2013 |
Festa C, D'Amore C, Renga B, Lauro G, De Marino S, D'Auria MV, Bifulco G, Zampella A, Fiorucci S. Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists Marine Drugs. 11: 2314-2327. PMID 23820629 DOI: 10.3390/Md11072314 |
0.547 |
|
| 2013 |
Dal Piaz F, Cotugno R, Lepore L, Vassallo A, Malafronte N, Lauro G, Bifulco G, Belisario MA, De Tommasi N. Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells. Journal of Proteomics. 82: 14-26. PMID 23416714 DOI: 10.1016/J.Jprot.2013.01.030 |
0.504 |
|
| 2012 |
Festa C, Lauro G, De Marino S, D'Auria MV, Monti MC, Casapullo A, D'Amore C, Renga B, Mencarelli A, Petek S, Bifulco G, Fiorucci S, Zampella A. Plakilactones from the marine sponge Plakinastrella mamillaris. discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ Journal of Medicinal Chemistry. 55: 8303-8317. PMID 22934537 DOI: 10.1021/Jm300911G |
0.49 |
|
| 2012 |
Sepe V, Ummarino R, D'Auria MV, Lauro G, Bifulco G, D'Amore C, Renga B, Fiorucci S, Zampella A. Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist. Organic & Biomolecular Chemistry. 10: 6350-62. PMID 22733410 DOI: 10.1039/C2Ob25800E |
0.474 |
|
| 2012 |
Lauro G, Masullo M, Piacente S, Riccio R, Bifulco G. Inverse Virtual Screening allows the discovery of the biological activity of natural compounds. Bioorganic & Medicinal Chemistry. 20: 3596-602. PMID 22537682 DOI: 10.1016/J.Bmc.2012.03.072 |
0.707 |
|
| 2012 |
Cheruku P, Plaza A, Lauro G, Keffer J, Lloyd JR, Bifulco G, Bewley CA. Discovery and synthesis of namalide reveals a new anabaenopeptin scaffold and peptidase inhibitor. Journal of Medicinal Chemistry. 55: 735-42. PMID 22168797 DOI: 10.1021/Jm201238P |
0.523 |
|
| 2011 |
Lauro G, Romano A, Riccio R, Bifulco G. Inverse virtual screening of antitumor targets: pilot study on a small database of natural bioactive compounds. Journal of Natural Products. 74: 1401-7. PMID 21542600 DOI: 10.1021/Np100935S |
0.702 |
|
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