Year |
Citation |
Score |
2019 |
Hassell-Hart S, Runcie A, Krojer T, Doyle J, Lineham E, Ocasio CA, Neto BAD, Fedorov O, Marsh G, Maple H, Felix R, Banks R, Ciulli A, Picaud S, Filippakopoulos P, et al. Synthesis and Biological Investigation of (+)-JD1, an Organometallic BET Bromodomain Inhibitor Organometallics. 39: 408-416. DOI: 10.1021/Acs.Organomet.9B00750 |
0.302 |
|
2016 |
Ocasio CA, Rajasekaran MB, Walker S, Le Grand D, Spencer J, Pearl FM, Ward SE, Savic V, Pearl LH, Hochegger H, Oliver AW. A first generation inhibitor of human Greatwall kinase, enabled by structural and functional characterisation of a minimal kinase domain construct. Oncotarget. PMID 27563826 DOI: 10.18632/Oncotarget.11511 |
0.314 |
|
2009 |
Hyman JM, Firestone AJ, Heine VM, Zhao Y, Ocasio CA, Han K, Sun M, Rack PG, Sinha S, Wu JJ, Solow-Cordero DE, Jiang J, Rowitch DH, Chen JK. Small-molecule inhibitors reveal multiple strategies for Hedgehog pathway blockade. Proceedings of the National Academy of Sciences of the United States of America. 106: 14132-7. PMID 19666565 DOI: 10.1073/Pnas.0907134106 |
0.318 |
|
2008 |
Ocasio CA, Scanlan TS. Characterization of thyroid hormone receptor α (TRα)-specific analogs with varying inner- and outer-ring substituents Bioorganic and Medicinal Chemistry. 16: 762-770. PMID 17988877 DOI: 10.1016/J.Bmc.2007.10.040 |
0.52 |
|
2007 |
Ocasio CA, Scanlan TS. ACS Chem. Biol. 2006, 1, 585–593Correction: Design and Characterization of a Thyroid Hormone Receptor α (TRα)-Specific Agonist Acs Chemical Biology. 2: 635-635. DOI: 10.1021/Cb700167W |
0.537 |
|
2006 |
Ocasio CA, Scanlan TS. Design and characterization of a thyroid hormone receptor alpha (TRalpha)-specific agonist. Acs Chemical Biology. 1: 585-593. PMID 17168554 DOI: 10.1021/Cb600311V |
0.558 |
|
2006 |
Arnold LA, Estébanez-Perpiñá E, Togashi M, Shelat A, Ocasio CA, McReynolds AC, Nguyen P, Baxter JD, Fletterick RJ, Webb P, Guy RK. A high-throughput screening method to identify small molecule inhibitors of thyroid hormone receptor coactivator binding. Science's Stke : Signal Transduction Knowledge Environment. 2006: pl3. PMID 16804159 DOI: 10.1126/Stke.3412006Pl3 |
0.38 |
|
2005 |
Ocasio CA, Scanlan TS. Clinical prospects for new thyroid hormone analogues Current Opinion in Endocrinology and Diabetes. 12: 363-370. DOI: 10.1097/01.Med.0000177422.57988.B2 |
0.516 |
|
2002 |
Swann SL, Bergh J, Farach-Carson MC, Ocasio CA, Koh JT. Structure-based design of selective agonists for a rickets-associated mutant of the vitamin d receptor. Journal of the American Chemical Society. 124: 13795-805. PMID 12431109 DOI: 10.1021/Ja0268377 |
0.351 |
|
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