Year |
Citation |
Score |
2017 |
Moslin R, Gardner D, Santella J, Zhang Y, Duncia JV, Liu C, Lin J, Tokarski JS, Strnad J, Pedicord D, Chen J, Blat Y, Zupa-Fernandez A, Cheng L, Sun H, et al. Identification of imidazo[1,2-]pyridazine TYK2 pseudokinase ligands as potent and selective allosteric inhibitors of TYK2 signalling. Medchemcomm. 8: 700-712. PMID 30108788 DOI: 10.1039/C6Md00560H |
0.305 |
|
2016 |
Chupak LS, Zheng X, Hu S, Huang Y, Ding M, Lewis MA, Westphal RS, Blat Y, McClure A, Gentles RG. Structure activity relationship studies on chemically non-reactive glycine sulfonamide inhibitors of diacylglycerol lipase. Bioorganic & Medicinal Chemistry. PMID 26917221 DOI: 10.1016/J.Bmc.2016.02.006 |
0.323 |
|
2015 |
Chaudhry C, Davis J, Zhang Y, Posy S, Lei M, Shen H, Yan C, Devaux B, Zhang L, Blat Y, Metzler W, Borzilleri RM, Talbott RL. Building HTRF assays for characterization of bivalent inhibitors of an Inhibitor of Apoptosis Protein target. Analytical Biochemistry. PMID 26743718 DOI: 10.1016/J.Ab.2015.11.026 |
0.359 |
|
2015 |
Tokarski JS, Zupa-Fernandez A, Tredup JA, Pike K, Chang C, Xie D, Cheng L, Pedicord D, Muckelbauer J, Johnson SR, Wu S, Edavettal SC, Hong Y, Witmer MR, Elkin LL, ... Blat Y, et al. Tyrosine Kinase 2-mediated Signal Transduction in T Lymphocytes Is Blocked by Pharmacological Stabilization of Its Pseudokinase Domain. The Journal of Biological Chemistry. 290: 11061-74. PMID 25762719 DOI: 10.1074/Jbc.M114.619502 |
0.314 |
|
2014 |
Appiah KK, Blat Y, Robertson BJ, Pearce BC, Pedicord DL, Gentles RG, Yu XC, Mseeh F, Nguyen N, Swaffield JC, Harden DG, Westphal RS, Banks MN, O'Connell JC. Identification of small molecules that selectively inhibit diacylglycerol lipase-α activity. Journal of Biomolecular Screening. 19: 595-605. PMID 24241710 DOI: 10.1177/1087057113511111 |
0.304 |
|
2010 |
Blat Y. Non-competitive inhibition by active site binders. Chemical Biology & Drug Design. 75: 535-40. PMID 20374252 DOI: 10.1111/J.1747-0285.2010.00972.X |
0.348 |
|
2010 |
Fanslau C, Pedicord D, Nagulapalli S, Gray H, Pang S, Jayaraman L, Lippy J, Blat Y. An electrophoretic mobility shift assay for the identification and kinetic analysis of acetyl transferase inhibitors. Analytical Biochemistry. 402: 65-8. PMID 20338149 DOI: 10.1016/J.Ab.2010.03.025 |
0.321 |
|
2007 |
Sahni-Arya B, Flynn MJ, Bergeron L, Salyan ME, Pedicord DL, Golla R, Ma Z, Wang H, Seethala R, Wu SC, Li JJ, Nayeem A, Gates C, Hamann LG, Gordon DA, ... Blat Y, et al. Cofactor-specific modulation of 11beta-hydroxysteroid dehydrogenase 1 inhibitor potency. Biochimica Et Biophysica Acta. 1774: 1184-91. PMID 17707701 DOI: 10.1016/J.Bbapap.2007.07.005 |
0.303 |
|
2002 |
Blat Y, Protacio RU, Hunter N, Kleckner N. Physical and functional interactions among basic chromosome organizational features govern early steps of meiotic chiasma formation. Cell. 111: 791-802. PMID 12526806 DOI: 10.1016/S0092-8674(02)01167-4 |
0.534 |
|
2002 |
Blat Y, Meredith JE, Wang Q, Bradley JD, Thompson LA, Olson RE, Stern AM, Seiffert D. Mutations at the P1' position of Notch1 decrease intracellular domain stability rather than cleavage by gamma-secretase. Biochemical and Biophysical Research Communications. 299: 569-73. PMID 12459176 DOI: 10.1016/S0006-291X(02)02705-5 |
0.321 |
|
2002 |
Bachant J, Alcasabas A, Blat Y, Kleckner N, Elledge SJ. The SUMO-1 isopeptidase Smt4 is linked to centromeric cohesion through SUMO-1 modification of DNA topoisomerase II. Molecular Cell. 9: 1169-82. PMID 12086615 DOI: 10.1016/S1097-2765(02)00543-9 |
0.516 |
|
1999 |
Blat Y, Kleckner N. Cohesins bind to preferential sites along yeast chromosome III, with differential regulation along arms versus the centric region. Cell. 98: 249-59. PMID 10428036 DOI: 10.1016/S0092-8674(00)81019-3 |
0.52 |
|
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