Rob Leurs

Medicinal Chemistry Vrije Universiteit Amsterdam, Amsterdam, Netherlands 
GPCRs, Histamine receptors, Chemokine receptors
"Rob Leurs"
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Munday JC, Kunz S, Kalejaiye TD, et al. (2020) Cloning and functional complementation of ten Schistosoma mansoni phosphodiesterases expressed in the mammalian host stages. Plos Neglected Tropical Diseases. 14: e0008447
Schihada H, Ma X, Zabel U, et al. (2020) Development of a conformational histamine H receptor biosensor for the synchronous screening of agonists and inverse agonists. Acs Sensors
Verweij EWE, Al Araaj B, Prabhata WR, et al. (2020) Differential Role of Serines and Threonines in Intracellular Loop 3 and C-Terminal Tail of the Histamine H Receptor in β-Arrestin and G Protein-Coupled Receptor Kinase Interaction, Internalization, and Signaling. Acs Pharmacology & Translational Science. 3: 321-333
Sijm M, Sterk GJ, Caljon G, et al. (2020) Structure activity relationship of phenylpyrazolones against Trypanosoma cruzi. Chemmedchem
G Salado I, Singh AK, Moreno-Cinos C, et al. (2020) Lead optimization of phthalazinone phosphodiesterase inhibitors as novel antitrypanosomal compounds. Journal of Medicinal Chemistry
Wágner G, Mocking TAM, Kooistra AJ, et al. (2019) Covalent Inhibition of the Histamine H Receptor. Molecules (Basel, Switzerland). 24
Gómez-Santacana X, de Munnik SM, Mocking TAM, et al. (2019) A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with light. Beilstein Journal of Organic Chemistry. 15: 2509-2523
Kanev GK, de Graaf C, de Esch IJP, et al. (2019) The Landscape of Atypical and Eukaryotic Protein Kinases. Trends in Pharmacological Sciences. 40: 818-832
Wágner G, Mocking T, Arimont M, et al. (2019) 4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines as high-affinity non-imidazole histamine H3 receptor agonists with in vivo central nervous system activity. Journal of Medicinal Chemistry
Adlere I, Caspar B, Arimont M, et al. (2019) Modulators of CXCR4 and CXCR7/ACKR3 function. Molecular Pharmacology
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