Rob Leurs

Medicinal Chemistry Vrije Universiteit Amsterdam, Amsterdam, Netherlands 
GPCRs, Histamine receptors, Chemokine receptors
"Rob Leurs"
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Rahman SN, McNaught-Flores DA, Huppelschoten Y, et al. (2023) Structural and Molecular Determinants for Isoform Bias at Human Histamine H Receptor Isoforms. Acs Chemical Neuroscience
Wágner G, Mocking TAM, Ma X, et al. (2022) SAR exploration of the non-imidazole histamine H receptor ligand ZEL-H16 reveals potent inverse agonism. Archiv Der Pharmazie. e2200451
Ma X, Gao M, Vischer HF, et al. (2022) A NanoBRET-Based HR Conformational Biosensor to Study Real-Time H Receptor Pharmacology in Cell Membranes and Living Cells. International Journal of Molecular Sciences. 23
Zheng Y, Wágner G, Hauwert N, et al. (2022) New Chemical Biology Tools for the Histamine Receptor Family. Current Topics in Behavioral Neurosciences
Kok ZY, Stoddart LA, Mistry SJ, et al. (2022) Optimization of Peptide Linker-Based Fluorescent Ligands for the Histamine H Receptor. Journal of Medicinal Chemistry. 65: 8258-8288
Verweij EWE, Bosma R, Gao M, et al. (2022) BRET-Based Biosensors to Measure Agonist Efficacies in Histamine H Receptor-Mediated G Protein Activation, Signaling and Interactions with GRKs and β-Arrestins. International Journal of Molecular Sciences. 23
Ma X, Verweij EWE, Siderius M, et al. (2021) Identification of TSPAN4 as Novel Histamine H Receptor Interactor. Biomolecules. 11
Ma X, Leurs R, Vischer HF. (2021) NanoLuc-Based Methods to Measure β-Arrestin2 Recruitment to G Protein-Coupled Receptors. Methods in Molecular Biology (Clifton, N.J.). 2268: 233-248
Wang Z, Bosma R, Kuhne S, et al. (2021) Exploring the Effect of Cyclization of Histamine H Receptor Antagonists on Ligand Binding Kinetics. Acs Omega. 6: 12755-12768
Ma X, Segura MA, Zarzycka B, et al. (2021) Analysis of Missense Variants in the Human Histamine Receptor Family Reveals Increased Constitutive Activity of E410K Variant in the Histamine H Receptor. International Journal of Molecular Sciences. 22
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