Rob Leurs

Medicinal Chemistry Vrije Universiteit Amsterdam, Amsterdam, Netherlands 
GPCRs, Histamine receptors, Chemokine receptors
"Rob Leurs"
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Wang Z, Bosma R, Kuhne S, et al. (2021) Exploring the Effect of Cyclization of Histamine H Receptor Antagonists on Ligand Binding Kinetics. Acs Omega. 6: 12755-12768
Egyed A, Kelemen ÁA, Vass M, et al. (2021) Controlling the selectivity of aminergic GPCR ligands from the extracellular vestibule. Bioorganic Chemistry. 111: 104832
Schihada H, Ma X, Zabel U, et al. (2020) Development of a conformational histamine H receptor biosensor for the synchronous screening of agonists and inverse agonists. Acs Sensors
Adlere I, Caspar B, Arimont M, et al. (2019) Modulators of CXCR4 and CXCR7/ACKR3 function. Molecular Pharmacology
van Senten JR, Bebelman MP, Fan TS, et al. (2019) The human cytomegalovirus-encoded G protein-coupled receptor UL33 exhibits oncomodulatory properties. The Journal of Biological Chemistry
Bosma R, Wang Z, Kooistra AJ, et al. (2019) Route to Prolonged Residence Time at the Histamine H Receptor: Growing from Desloratadine to Rupatadine. Journal of Medicinal Chemistry
Arimont M, Hoffmann C, de Graaf C, et al. (2019) Chemokine receptor crystal structures: what can be learnt from them? Molecular Pharmacology
Chazot P, Cowart M, Fukui H, et al. (2019) Histamine receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database Iuphar/Bps Guide to Pharmacology Cite. 2019
Adlere I, Sun S, Zarca A, et al. (2018) Structure-based exploration and pharmacological evaluation of N-substituted piperidin-4-yl-methanamine CXCR4 chemokine receptor antagonists. European Journal of Medicinal Chemistry. 162: 631-649
Vass M, Podlewska S, De Esch IJP, et al. (2018) Aminergic GPCR-ligand interactions: A chemical and structural map of receptor mutation data. Journal of Medicinal Chemistry
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