Rob Leurs

Affiliations: 
Medicinal Chemistry Vrije Universiteit Amsterdam, Amsterdam, Netherlands 
Area:
GPCRs, Histamine receptors, Chemokine receptors
Website:
http://www.chem.vu.nl/en/research/division-of-medicinal-chemistry/index.asp
Google:
"Rob Leurs"
Mean distance: 13.53
 
SNBCP
BETA: Related publications

Publications

You can help our author matching system! If you notice any publications incorrectly attributed to this author, please sign in and mark matches as correct or incorrect.

Wang Z, Bosma R, Kuhne S, et al. (2021) Exploring the Effect of Cyclization of Histamine H Receptor Antagonists on Ligand Binding Kinetics. Acs Omega. 6: 12755-12768
Egyed A, Kelemen ÁA, Vass M, et al. (2021) Controlling the selectivity of aminergic GPCR ligands from the extracellular vestibule. Bioorganic Chemistry. 111: 104832
Schihada H, Ma X, Zabel U, et al. (2020) Development of a conformational histamine H receptor biosensor for the synchronous screening of agonists and inverse agonists. Acs Sensors
Adlere I, Caspar B, Arimont M, et al. (2019) Modulators of CXCR4 and CXCR7/ACKR3 function. Molecular Pharmacology
van Senten JR, Bebelman MP, Fan TS, et al. (2019) The human cytomegalovirus-encoded G protein-coupled receptor UL33 exhibits oncomodulatory properties. The Journal of Biological Chemistry
Bosma R, Wang Z, Kooistra AJ, et al. (2019) Route to Prolonged Residence Time at the Histamine H Receptor: Growing from Desloratadine to Rupatadine. Journal of Medicinal Chemistry
Arimont M, Hoffmann C, de Graaf C, et al. (2019) Chemokine receptor crystal structures: what can be learnt from them? Molecular Pharmacology
Chazot P, Cowart M, Fukui H, et al. (2019) Histamine receptors (version 2019.4) in the IUPHAR/BPS Guide to Pharmacology Database Iuphar/Bps Guide to Pharmacology Cite. 2019
Adlere I, Sun S, Zarca A, et al. (2018) Structure-based exploration and pharmacological evaluation of N-substituted piperidin-4-yl-methanamine CXCR4 chemokine receptor antagonists. European Journal of Medicinal Chemistry. 162: 631-649
Vass M, Podlewska S, De Esch IJP, et al. (2018) Aminergic GPCR-ligand interactions: A chemical and structural map of receptor mutation data. Journal of Medicinal Chemistry
See more...