Year |
Citation |
Score |
2018 |
Michaelides MR, Kluge A, Patane M, Van Drie JH, Wang C, Hansen TM, Risi RM, Mantei R, Hertel C, Karukurichi K, Nesterov A, McElligott D, de Vries P, Langston JW, Cole PA, et al. Discovery of Spiro Oxazolidinediones as Selective, Orally Bioavailable Inhibitors of p300/CBP Histone Acetyltransferases. Acs Medicinal Chemistry Letters. 9: 28-33. PMID 29348807 DOI: 10.1021/Acsmedchemlett.7B00395 |
0.337 |
|
2017 |
Lasko LM, Jakob CG, Edalji RP, Qiu W, Montgomery D, Digiammarino EL, Hansen TM, Risi RM, Frey R, Manaves V, Shaw B, Algire M, Hessler P, Lam LT, Uziel T, ... ... Karukurichi K, et al. Discovery of a selective catalytic p300/CBP inhibitor that targets lineage-specific tumours. Nature. PMID 28953875 DOI: 10.1038/Nature24028 |
0.309 |
|
2015 |
Karukurichi KR, Fei X, Swyka RA, Broussy S, Shen W, Dey S, Roy SK, Berkowitz DB. Mini-ISES identifies promising carbafructopyranose-based salens for asymmetric catalysis: Tuning ligand shape via the anomeric effect. Science Advances. 1. PMID 26501130 DOI: 10.1126/Sciadv.1500066 |
0.638 |
|
2014 |
Wang Y, Kavran JM, Chen Z, Karukurichi KR, Leahy DJ, Cole PA. Regulation of S-adenosylhomocysteine hydrolase by lysine acetylation. The Journal of Biological Chemistry. 289: 31361-72. PMID 25248746 DOI: 10.1074/Jbc.M114.597153 |
0.379 |
|
2011 |
Karukurichi KR, Cole PA. Probing the reaction coordinate of the p300/CBP histone acetyltransferase with bisubstrate analogs. Bioorganic Chemistry. 39: 42-7. PMID 21111442 DOI: 10.1016/J.Bioorg.2010.10.004 |
0.311 |
|
2010 |
Karukurichi KR, Wang L, Uzasci L, Manlandro CM, Wang Q, Cole PA. Analysis of p300/CBP histone acetyltransferase regulation using circular permutation and semisynthesis. Journal of the American Chemical Society. 132: 1222-3. PMID 20063892 DOI: 10.1021/Ja909466D |
0.309 |
|
2009 |
Berkowitz DB, Karukurichi KR, De La Salud-Bea R, Maiti G, McFadden JM, Morris ML. Stereoselective synthesis of quaternary, α-vinyl amino acids and their α-(2'Z-fluoro)vinyl congeners: Promising candidates for PLP enzyme inactivation Acs Symposium Series. 1009: 288-303. DOI: 10.1021/bk-2009-1009.ch018 |
0.788 |
|
2008 |
Berkowitz DB, Karukurichi KR, de la Salud-Bea R, Nelson DL, McCune CD. Use of Fluorinated Functionality in Enzyme Inhibitor Development: Mechanistic and Analytical Advantages. Journal of Fluorine Chemistry. 129: 731-742. PMID 19727327 DOI: 10.1016/J.Jfluchem.2008.05.016 |
0.634 |
|
2007 |
Karukurichi KR, de la Salud-Bea R, Jahng WJ, Berkowitz DB. Examination of the new alpha-(2'Z-fluoro)vinyl trigger with lysine decarboxylase: the absolute stereochemistry dictates the reaction course. Journal of the American Chemical Society. 129: 258-9. PMID 17212389 DOI: 10.1021/Ja067240K |
0.71 |
|
2006 |
Berkowitz DB, Charette BD, Karukurichi KR, McFadden JM. α-Vinylic Amino Acids: Occurrence, Asymmetric Synthesis and Biochemical Mechanisms. Tetrahedron, Asymmetry. 17: 869-882. PMID 29977107 DOI: 10.1016/J.Tetasy.2006.02.026 |
0.784 |
|
2006 |
Berkowitz DB, Charette BD, Karukurichi KR, McFadden JM. α-Vinylic amino acids: occurrence, asymmetric synthesis, and biochemical mechanisms Tetrahedron Asymmetry. 17: 869-882. DOI: 10.1016/j.tetasy.2006.02.026 |
0.787 |
|
2005 |
Dey S, Karukurichi KR, Shen W, Berkowitz DB. Double-cuvette ISES: in situ estimation of enantioselectivity and relative rate for catalyst screening. Journal of the American Chemical Society. 127: 8610-1. PMID 15954763 DOI: 10.1021/Ja052010B |
0.753 |
|
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