| Year |
Citation |
Score |
| 2023 |
Regni A, Bartoccini F, Piersanti G. Photoredox catalysis enabling decarboxylative radical cyclization of γ,γ-dimethylallyltryptophan (DMAT) derivatives: formal synthesis of 6,7-secoagroclavine. Beilstein Journal of Organic Chemistry. 19: 918-927. PMID 37404801 DOI: 10.3762/bjoc.19.70 |
0.43 |
|
| 2022 |
Retini M, Bartolucci S, Bartoccini F, Piersanti G. Asymmetric Alkylation of Cyclic Ketones with Dehydroalanine via H-Bond-Directing Enamine Catalysis: Straightforward Access to Enantiopure Unnatural α-Amino Acids. Chemistry (Weinheim An Der Bergstrasse, Germany). e202201994. PMID 35916657 DOI: 10.1002/chem.202201994 |
0.376 |
|
| 2021 |
Bartoccini F, Regni A, Retini M, Piersanti G. Concise catalytic asymmetric synthesis of (R)-4-amino Uhle's ketone. Organic & Biomolecular Chemistry. 19: 2932-2940. PMID 33885552 DOI: 10.1039/d1ob00353d |
0.386 |
|
| 2020 |
Linciano P, Cullia G, Borsari C, Santucci M, Ferrari S, Witt G, Gul S, Kuzikov M, Ellinger B, Santarém N, Cordeiro da Silva A, Conti P, Bolognesi ML, Roberti M, Prati F, ... ... Piersanti G, et al. Identification of a 2,4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign. European Journal of Medicinal Chemistry. 189: 112047. PMID 31982652 DOI: 10.1016/J.Ejmech.2020.112047 |
0.306 |
|
| 2020 |
Bartoccini F, Fanini F, Retini M, Piersanti G. General synthesis of unnatural 4-, 5-, 6-, and 7-bromo-d-tryptophans by means of a regioselective indole alkylation Tetrahedron Letters. 61: 151923. DOI: 10.1016/J.Tetlet.2020.151923 |
0.429 |
|
| 2020 |
Bartoccini F, Retini M, Piersanti G. C3-Alkylation of indoles and oxindoles by alcohols by means of borrowing hydrogen methodology Tetrahedron Letters. 61: 151875. DOI: 10.1016/J.Tetlet.2020.151875 |
0.301 |
|
| 2020 |
Bartoccini F, Mari M, Retini M, Galarini R, Bartolucci S, Piersanti G. Single‐Step Synthesis of Dehydroalanine Derivatives via a Brønsted Acid‐Catalyzed Multicomponent Reaction Chemistryselect. 5: 3330-3336. DOI: 10.1002/slct.202000898 |
0.658 |
|
| 2019 |
Retini M, Bartolucci S, Bartoccini F, Mari M, Piersanti G. Concise and Convergent Enantioselective Total Syntheses of (+)- and (-)-Fumimycin. The Journal of Organic Chemistry. PMID 31476858 DOI: 10.1021/Acs.Joc.9B02020 |
0.694 |
|
| 2019 |
Bartoccini F, Venturi S, Retini M, Mari M, Piersanti G. Total Synthesis of (-)-Clavicipitic Acid via γ,γ-Dimethylallyltryptophan (DMAT) and Chemoselective C-H Hydroxylation. The Journal of Organic Chemistry. PMID 31120249 DOI: 10.1021/Acs.Joc.9B00879 |
0.651 |
|
| 2019 |
Bartoccini F, Mari M, Retini M, Fraternale A, Piersanti G. Large-Scale Preparation of N-Butanoyl-l-glutathione (C4-GSH) Organic Process Research & Development. 23: 2069-2073. DOI: 10.1021/Acs.Oprd.9B00120 |
0.615 |
|
| 2018 |
Bartoccini F, Mari M, Retini M, Bartolucci S, Piersanti G. Organocatalytic Aza-Friedel-Crafts/Lactonization Domino Reaction of Naphthols and Phenols with 2-Acetamidoacrylate to Naphtho- and Benzofuranones Bearing a Quaternary Center at the C3 Position. The Journal of Organic Chemistry. PMID 30191715 DOI: 10.1021/Acs.Joc.8B01774 |
0.677 |
|
| 2018 |
Bartoccini F, Bartolucci S, Mari M, Piersanti G. A simple, modular synthesis of C4-substituted tryptophan derivatives. Organic & Biomolecular Chemistry. 14: 10095-10100. PMID 27722724 DOI: 10.1039/C6Ob01791F |
0.656 |
|
| 2018 |
Di Gregorio G, Mari M, Bartolucci S, Bartoccini F, Piersanti G. Divergent reactions of oxindoles with amino alcohols via the borrowing hydrogen process: oxindole ring opening vs. C3 alkylation Organic Chemistry Frontiers. 5: 1622-1627. DOI: 10.1039/C8Qo00184G |
0.614 |
|
| 2018 |
Ciccolini C, Mari M, Lucarini S, Mantellini F, Piersanti G, Favi G. Polycyclic Indolines by an Acid‐Mediated Intramolecular Dearomative Strategy: Reversing Indole Reactivity in the Pictet‐Spengler‐Type Reaction Advanced Synthesis & Catalysis. 360: 4060-4067. DOI: 10.1002/Adsc.201800981 |
0.623 |
|
| 2017 |
Di Gregorio G, Mari M, Bartoccini F, Piersanti G. Iron-Catalyzed Direct C3-Benzylation of Indoles with Benzyl Alcohols through Borrowing Hydrogen. The Journal of Organic Chemistry. PMID 28745505 DOI: 10.1021/Acs.Joc.7B01603 |
0.761 |
|
| 2017 |
Mantenuto S, Ciccolini C, Lucarini S, Piersanti G, Favi G, Mantellini F. Palladium(II)-Catalyzed Intramolecular Oxidative C-H/C-H Cross-Coupling Reaction of C3,N-Linked Biheterocycles: Rapid Access to Polycyclic Nitrogen Heterocycles. Organic Letters. PMID 28094964 DOI: 10.1021/Acs.Orglett.6B03775 |
0.349 |
|
| 2016 |
Bartoccini F, Cannas DM, Fini F, Piersanti G. Palladium(II)-Catalyzed Cross-Dehydrogenative Coupling (CDC) of N-Phthaloyl Dehydroalanine Esters with Simple Arenes: Stereoselective Synthesis of Z-Dehydrophenylalanine Derivatives. Organic Letters. PMID 27206072 DOI: 10.1021/Acs.Orglett.6B01255 |
0.467 |
|
| 2016 |
Formica M, Fusi V, Giorgi L, Piersanti G, Retini M, Zappia G. Neutral urea-based receptors for phosphates: synthesis and spectrophotometric studies Tetrahedron. 72: 7039-7049. DOI: 10.1016/J.Tet.2016.09.042 |
0.359 |
|
| 2016 |
Bartolucci S, Mari M, Di Gregorio G, Piersanti G. Observations concerning the synthesis of tryptamine homologues and branched tryptamine derivatives via the borrowing hydrogen process: synthesis of psilocin, bufotenin, and serotonin Tetrahedron. 72: 2233-2238. DOI: 10.1016/J.Tet.2016.03.007 |
0.678 |
|
| 2016 |
Mantenuto S, Lucarini S, De Santi M, Piersanti G, Brandi G, Favi G, Mantellini F. One-Pot Synthesis of Biheterocycles Based on Indole and Azole Scaffolds Using Tryptamines and 1,2-Diaza-1,3-dienes as Building Blocks European Journal of Organic Chemistry. 2016: 3193-3199. DOI: 10.1002/Ejoc.201600210 |
0.403 |
|
| 2016 |
Bartolucci S, Mari M, Di Gregorio G, Piersanti G. ChemInform Abstract: Observations Concerning the Synthesis of Tryptamine Homologues and Branched Tryptamine Derivatives via the Borrowing Hydrogen Process: Synthesis of Psilocin, Bufotenin, and Serotonin. Cheminform. 47. DOI: 10.1002/chin.201633131 |
0.619 |
|
| 2015 |
Pace S, Brogin G, Stasi MA, Riccioni T, Borsini F, Capocasa F, Manera F, Tallarico C, Grossi P, Vacondio F, Bassi M, Bartoccini F, Lucarini S, Piersanti G, Tarzia G, et al. Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands. Chemmedchem. PMID 25951302 DOI: 10.1002/Cmdc.201500113 |
0.567 |
|
| 2015 |
Bartolucci S, Mari M, Bedini A, Piersanti G, Spadoni G. Iridium-catalyzed direct synthesis of tryptamine derivatives from indoles: exploiting n-protected β-amino alcohols as alkylating agents. The Journal of Organic Chemistry. 80: 3217-22. PMID 25699684 DOI: 10.1021/Acs.Joc.5B00195 |
0.728 |
|
| 2015 |
Bartoccini F, Bartolucci S, Lucarini S, Piersanti G. Synthesis of boron- and silicon-containing amino acids through copper-catalysed conjugate additions to dehydroalanine derivatives European Journal of Organic Chemistry. 2015: 3352-3360. DOI: 10.1002/Ejoc.201500362 |
0.456 |
|
| 2014 |
Mari M, Lucarini S, Bartoccini F, Piersanti G, Spadoni G. Synthesis of 2-substituted tryptophans via a C3- to C2-alkyl migration. Beilstein Journal of Organic Chemistry. 10: 1991-8. PMID 25246958 DOI: 10.3762/Bjoc.10.207 |
0.733 |
|
| 2014 |
Bartoccini F, Casoli M, Mari M, Piersanti G. Synthesis of (±)-cis-clavicipitic acid by a Rh(I)-catalyzed intramolecular imine reaction. The Journal of Organic Chemistry. 79: 3255-9. PMID 24605802 DOI: 10.1021/Jo500245S |
0.71 |
|
| 2014 |
Bartoccini F, Piersanti G, Armaroli S, Cerri A, Cabri W. Development of a practical and sustainable strategy for the synthesis of ST1535 by an iron-catalyzed Kumada cross-coupling reaction Tetrahedron Letters. 55: 1376-1378. DOI: 10.1016/J.Tetlet.2014.01.030 |
0.398 |
|
| 2014 |
Mari M, Tassoni A, Lucarini S, Fanelli M, Piersanti G, Spadoni G. Brønsted acid catalyzed bisindolization of α-amido acetals: Synthesis and anticancer activity of bis(indolyl)ethanamino derivatives European Journal of Organic Chemistry. 2014: 3822-3830. DOI: 10.1002/Ejoc.201402055 |
0.736 |
|
| 2014 |
Bartoccini F, Casoli M, Mari M, Piersanti G. ChemInform Abstract: Synthesis of (.+-.)-cis-Clavicipitic Acid by a Rh(I)-Catalyzed Intramolecular Imine Reaction. Cheminform. 45: no-no. DOI: 10.1002/chin.201439134 |
0.647 |
|
| 2013 |
Mari M, Bartoccini F, Piersanti G. Synthesis of (-)-epi-indolactam V by an intramolecular Buchwald-Hartwig C-N coupling cyclization reaction. The Journal of Organic Chemistry. 78: 7727-34. PMID 23845025 DOI: 10.1021/Jo4013767 |
0.691 |
|
| 2013 |
Piersanti G, Bartoccini F, Lucarini S, Cabri W, Stasi MA, Riccioni T, Borsini F, Tarzia G, Minetti P. Synthesis and biological evaluation of metabolites of 2-n-butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535), a potent antagonist of the A2A adenosine receptor for the treatment of Parkinson's disease. Journal of Medicinal Chemistry. 56: 5456-63. PMID 23789814 DOI: 10.1021/Jm400491X |
0.626 |
|
| 2013 |
Rivara S, Piersanti G, Bartoccini F, Diamantini G, Pala D, Riccioni T, Stasi MA, Cabri W, Borsini F, Mor M, Tarzia G, Minetti P. Synthesis of (E)-8-(3-chlorostyryl)caffeine analogues leading to 9-deazaxanthine derivatives as dual A(2A) antagonists/MAO-B inhibitors. Journal of Medicinal Chemistry. 56: 1247-61. PMID 23281824 DOI: 10.1021/Jm301686S |
0.542 |
|
| 2013 |
Attanasi OA, Favi G, Giorgi G, Mantellini F, Moscatelli G, Piersanti G. Synthesis of tetrahydropyridazine amino acid derivatives by a formal [4+2] cycloaddition reaction of 1,2-diaza-1,3-dienes with dehydroalanine esters Current Organic Synthesis. 10: 803-811. DOI: 10.2174/1570179411310050011 |
0.514 |
|
| 2013 |
Lucarini S, Mari M, Piersanti G, Spadoni G. Organocatalyzed coupling of indoles with dehydroalanine esters: Synthesis of bis(indolyl)propanoates and indolacrylates Rsc Advances. 3: 19135-19143. DOI: 10.1039/C3Ra42922A |
0.77 |
|
| 2012 |
Bartoccini F, Piersanti G, Mor M, Tarzia G, Minetti P, Cabri W. Divergent synthesis of novel 9-deazaxanthine derivatives via late-stage cross-coupling reactions. Organic & Biomolecular Chemistry. 10: 8860-7. PMID 23047760 DOI: 10.1039/C2Ob26516H |
0.658 |
|
| 2012 |
Righi M, Topi F, Bartolucci S, Bedini A, Piersanti G, Spadoni G. Synthesis of tryptamine derivatives via a direct, one-pot reductive alkylation of indoles. The Journal of Organic Chemistry. 77: 6351-7. PMID 22724919 DOI: 10.1021/Jo3010028 |
0.678 |
|
| 2012 |
Bartolucci S, Bartoccini F, Righi M, Piersanti G. Direct, regioselective, and chemoselective preparation of novel boronated tryptophans by Friedel-Crafts alkylation. Organic Letters. 14: 600-3. PMID 22208950 DOI: 10.1021/Ol203216H |
0.513 |
|
| 2012 |
Lucarini S, Bartolucci S, Bedini A, Gatti G, Orlando P, Piersanti G, Spadoni G. Synthesis and configuration determination of all enantiopure stereoisomers of the melatonin receptor ligand 4-phenyl-2-propionamidotetralin using an expedient optical resolution of 4-phenyl-2-tetralone. Organic & Biomolecular Chemistry. 10: 305-13. PMID 22095411 DOI: 10.1039/C1Ob06369C |
0.634 |
|
| 2011 |
Righi M, Bedini A, Piersanti G, Romagnoli F, Spadoni G. Direct, one-pot reductive alkylation of anilines with functionalized acetals mediated by triethylsilane and TFA. Straightforward route for unsymmetrically substituted ethylenediamine. The Journal of Organic Chemistry. 76: 704-7. PMID 21175194 DOI: 10.1021/Jo102109F |
0.648 |
|
| 2011 |
Piersanti G, Retini M, Espartero JL, Madrona A, Zappia G. An efficient, economical synthesis of hydroxytyrosol and its protected forms via Baeyer-Villiger oxidation Tetrahedron Letters. 52: 4938-4940. DOI: 10.1016/J.Tetlet.2011.07.063 |
0.367 |
|
| 2011 |
Righi M, Bartoccini F, Lucarini S, Piersanti G. Organocatalytic synthesis of α-quaternary amino acid derivatives via aza-Friedel-Crafts alkylation of indoles with simple α-amidoacrylates Tetrahedron. 67: 7923-7928. DOI: 10.1016/J.Tet.2011.08.039 |
0.465 |
|
| 2010 |
Lucarini S, Bartoccini F, Battistoni F, Diamantini G, Piersanti G, Righi M, Spadoni G. A novel one-pot approach of hexahydropyrrolo[2,3-b]indole nucleus by a cascade addition/cyclization strategy: synthesis of (+/-)-esermethole. Organic Letters. 12: 3844-7. PMID 20795744 DOI: 10.1021/Ol101527J |
0.672 |
|
| 2010 |
Bartoccini F, Cabri W, Celona D, Minetti P, Piersanti G, Tarzia G. Direct B-alkyl Suzuki-Miyaura cross-coupling of 2-halopurines. Practical synthesis of ST1535, a potent adenosine A2A receptor antagonist. The Journal of Organic Chemistry. 75: 5398-401. PMID 20597521 DOI: 10.1021/Jo101027H |
0.623 |
|
| 2010 |
Lucarini S, Alessi M, Bedini A, Giorgini G, Piersanti G, Spadoni G. Diastereo- and enantioselective hydrogenation of a challenging enamide derived from 4-phenyl-2-tetralone: an appealing shortcut towards enantiopure cis-2-aminotetraline derivatives. Chemistry, An Asian Journal. 5: 550-4. PMID 20108301 DOI: 10.1002/Asia.200900441 |
0.592 |
|
| 2010 |
Piersanti G, Varrese MA, Fusi V, Giorgi L, Zappia G. Short and straightforward synthesis of 1,7-dimethyl-1,4,7,10-tetraazacyclododecane Tetrahedron Letters. 51: 3436-3438. DOI: 10.1016/J.Tetlet.2010.04.115 |
0.45 |
|
| 2010 |
Siegel DS, Piizzi G, Piersanti G, Movassaghi M. ChemInform Abstract: Enantioselective Total Synthesis of (-)-Acylfulvene (IX) and (-)-Irofulven (X). Cheminform. 41. DOI: 10.1002/chin.201017189 |
0.777 |
|
| 2010 |
Bandini E, Favi G, Martelli G, Panunzio M, Piersanti G. ChemInform Abstract: A trans-Stereoselective Synthesis of 3-Halo-4-alkyl(aryl)-NH-azetidin-2-ones. Cheminform. 31: no-no. DOI: 10.1002/chin.200030094 |
0.454 |
|
| 2009 |
Movassaghi M, Piizzi G, Siegel DS, Piersanti G. Observations in the Synthesis of the Core of the Antitumor Illudins via an Enyne Ring Closing Metathesis Cascade. Tetrahedron Letters. 50: 5489-5492. PMID 20160945 DOI: 10.1016/J.Tetlet.2009.07.102 |
0.803 |
|
| 2009 |
Siegel DS, Piizzi G, Piersanti G, Movassaghi M. Enantioselective total synthesis of (-)-acylfulvene and (-)-irofulven. The Journal of Organic Chemistry. 74: 9292-304. PMID 19938810 DOI: 10.1021/Jo901926Z |
0.802 |
|
| 2009 |
Piersanti G, Remi F, Fusi V, Formica M, Giorgi L, Zappia G. Direct preparation of unsymmetrical difunctionalized cyclen derivatives by an Ugi multicomponent reaction. Organic Letters. 11: 417-20. PMID 19090699 DOI: 10.1021/Ol802674R |
0.507 |
|
| 2009 |
Valitutti G, Duranti A, Mor M, Piersanti G, Piomelli D, Rivara S, Tontini A, Tarzia G, Traldi P. The collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activity. Journal of Mass Spectrometry : Jms. 44: 561-5. PMID 19034887 DOI: 10.1002/Jms.1524 |
0.498 |
|
| 2008 |
Angelini E, Balsamini C, Bartoccini F, Lucarini S, Piersanti G. Switchable reactivity of acylated alpha, beta-dehydroamino ester in the Friedel-Crafts alkylation of indoles by changing the Lewis acid. The Journal of Organic Chemistry. 73: 5654-7. PMID 18558761 DOI: 10.1021/Jo800881U |
0.376 |
|
| 2008 |
Mor M, Lodola A, Rivara S, Vacondio F, Duranti A, Tontini A, Sanchini S, Piersanti G, Clapper JR, King AR, Tarzia G, Piomelli D. Synthesis and quantitative structure-activity relationship of fatty acid amide hydrolase inhibitors: modulation at the N-portion of biphenyl-3-yl alkylcarbamates. Journal of Medicinal Chemistry. 51: 3487-98. PMID 18507372 DOI: 10.1021/JM801482Q |
0.597 |
|
| 2008 |
Lucarini S, Bedini A, Spadoni G, Piersanti G. An improved synthesis of cis-4-phenyl-2-propionamidotetralin (4-P-PDOT): a selective MT(2) melatonin receptor antagonist. Organic & Biomolecular Chemistry. 6: 147-50. PMID 18075659 DOI: 10.1039/B713904G |
0.611 |
|
| 2008 |
Formica M, Fusi V, Macedi E, Paoli P, Piersanti G, Rossi P, Zappia G, Orlando P. New branched macrocyclic ligand and its side-arm, two urea-based receptors for anions: Synthesis, binding studies and crystal structure New Journal of Chemistry. 32: 1204-1214. DOI: 10.1039/B719342D |
0.321 |
|
| 2007 |
Valitutti G, Duranti A, Lodola A, Mor M, Piersanti G, Piomelli D, Rivara S, Tontini A, Tarzia G, Traldi P. Correlation between energetics of collisionally activated decompositions, interaction energy and biological potency of carbamate FAAH inhibitors. Journal of Mass Spectrometry : Jms. 42: 1624-7. PMID 18085570 DOI: 10.1002/Jms.1346 |
0.496 |
|
| 2007 |
Piersanti G, Giorgi L, Bartoccini F, Tarzia G, Minetti P, Gallo G, Giorgi F, Castorina M, Ghirardi O, Carminati P. Synthesis of benzo[1,2-d;3,4-d']diimidazole and 1H-pyrazolo[4,3-b]pyridine as putative A2A receptor antagonists. Organic & Biomolecular Chemistry. 5: 2567-71. PMID 18019530 DOI: 10.1039/B707599E |
0.573 |
|
| 2007 |
Movassaghi M, Piizzi G, Siegel D, Piersanti G. Synthesis of (-)-Acylfulvene and (-)-Irofulven Synfacts. 2007: 0122-0122. DOI: 10.1055/S-2006-955761 |
0.809 |
|
| 2006 |
Tarzia G, Duranti A, Gatti G, Piersanti G, Tontini A, Rivara S, Lodola A, Plazzi PV, Mor M, Kathuria S, Piomelli D. Synthesis and structure-activity relationships of FAAH inhibitors: cyclohexylcarbamic acid biphenyl esters with chemical modulation at the proximal phenyl ring. Chemmedchem. 1: 130-9. PMID 16892344 DOI: 10.1002/Cmdc.200500017 |
0.631 |
|
| 2006 |
Movassaghi M, Piizzi G, Siegel DS, Piersanti G. Enantioselective total synthesis of (-)-acylfulvene and (-)-irofulven. Angewandte Chemie (International Ed. in English). 45: 5859-63. PMID 16888819 DOI: 10.1002/Anie.200602011 |
0.814 |
|
| 2005 |
Minetti P, Tinti MO, Carminati P, Castorina M, Di Cesare MA, Di Serio S, Gallo G, Ghirardi O, Giorgi F, Giorgi L, Piersanti G, Bartoccini F, Tarzia G. 2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization. Journal of Medicinal Chemistry. 48: 6887-96. PMID 16250647 DOI: 10.1021/Jm058018D |
0.551 |
|
| 2005 |
Phillips ST, Piersanti G, Bartlett PA. Quantifying amino acid conformational preferences and side-chain-side-chain interactions in beta-hairpins. Proceedings of the National Academy of Sciences of the United States of America. 102: 13737-42. PMID 16162669 DOI: 10.1073/Pnas.0506646102 |
0.647 |
|
| 2004 |
Phillips ST, Piersanti G, Rüth M, Gubernator N, van Lengerich B, Bartlett PA. Facile synthesis of @-tide beta-strand peptidomimetics: improved assembly in solution and on solid phase. Organic Letters. 6: 4483-5. PMID 15548056 DOI: 10.1021/Ol048262J |
0.713 |
|
| 2004 |
Mor M, Rivara S, Lodola A, Plazzi PV, Tarzia G, Duranti A, Tontini A, Piersanti G, Kathuria S, Piomelli D. Cyclohexylcarbamic acid 3'- or 4'-substituted biphenyl-3-yl esters as fatty acid amide hydrolase inhibitors: synthesis, quantitative structure-activity relationships, and molecular modeling studies. Journal of Medicinal Chemistry. 47: 4998-5008. PMID 15456244 DOI: 10.1021/Jm031140X |
0.604 |
|
| 2004 |
Lucini V, Pannacci M, Scaglione F, Fraschini F, Rivara S, Mor M, Bordi F, Plazzi PV, Spadoni G, Bedini A, Piersanti G, Diamantini G, Tarzia G. Tricyclic alkylamides as melatonin receptor ligands with antagonist or inverse agonist activity. Journal of Medicinal Chemistry. 47: 4202-12. PMID 15293992 DOI: 10.1021/Jm040768K |
0.669 |
|
| 2003 |
Spadoni G, Bedini A, Piersanti G, Mor M, Rivara S, Tarzia G. Strategies leading to MT2 selective melatonin receptor antagonists. Advances in Experimental Medicine and Biology. 527: 577-85. PMID 15206776 DOI: 10.1007/978-1-4615-0135-0_66 |
0.638 |
|
| 2003 |
Burattini S, Luchetti F, Battistelli M, Della Felice M, Papa S, Piersanti G, Tarzia G, Falcieri E. 5-(2-Ethyl-phenyl)-3-(3-methoxy-phenyl)-1H-[1,2,4]triazole (DL-111-IT) and related compounds induce apoptotic patterns in cultures of human tumor cell lines. Journal of Biological Regulators and Homeostatic Agents. 17: 348-57. PMID 15065766 |
0.475 |
|
| 2003 |
Gatti G, Piersanti G, Spadoni G. Conformation by NMR of two tetralin-based receptor ligands. Farmaco (Società Chimica Italiana : 1989). 58: 469-76. PMID 12818685 DOI: 10.1016/S0014-827X(03)00064-8 |
0.551 |
|
| 2003 |
Tarzia G, Duranti A, Tontini A, Piersanti G, Mor M, Rivara S, Plazzi PV, Park C, Kathuria S, Piomelli D. Design, synthesis, and structure-activity relationships of alkylcarbamic acid aryl esters, a new class of fatty acid amide hydrolase inhibitors. Journal of Medicinal Chemistry. 46: 2352-60. PMID 12773040 DOI: 10.1021/Jm021119G |
0.624 |
|
| 2000 |
Bandini E, Favi G, Martelli G, Panunzio M, Piersanti G. A trans-stereoselective synthesis of 3-Halo-4-alkyl(aryl)-NH-azetidin-2-ones Organic Letters. 2: 1077-9. PMID 10804558 DOI: 10.1021/Ol005633X |
0.759 |
|
| 2000 |
Bongini A, Panunzio M, Piersanti G, Bandini E, Martelli G, Spunta G, Venturini A. Stereochemical Aspects of a Two‐Step Staudinger Reaction − Asymmetric Synthesis of Chiral Azetidine‐2‐ones European Journal of Organic Chemistry. 2000: 2379-2390. DOI: 10.1002/1099-0690(200007)2000:13<2379::Aid-Ejoc2379>3.0.Co;2-F |
0.48 |
|
| 2000 |
Bongini A, Panunzio M, Piersanti G, Bandini E, Martelli G, Spunta G, Venturini A. Stereochemical aspects of a two-step staudinger reaction - asymmetric synthesis of chiral azetidine-2-ones European Journal of Organic Chemistry. 2379-2390. |
0.738 |
|
| 1999 |
Bandini E, Martelli G, Spunta G, Bongini A, Panunzio M, Piersanti G. Stereoselective synthesis of chiral 3,4,5-trisubstituted 1,5- dihydropyrrol-2-ones from azadienes Tetrahedron Asymmetry. 10: 1445-1449. DOI: 10.1016/S0957-4166(99)00130-5 |
0.774 |
|
| 1997 |
Bandini E, Martelli G, Spunta G, Bongini A, Panunzio M, Piersanti G. An efficient synthesis of the cyclic form of scalemic 2,4-di-epi-polyoxamic acid exploiting the hetero Diels-Alder approach Tetrahedron Asymmetry. 8: 3717-3718. DOI: 10.1016/S0957-4166(97)00530-2 |
0.746 |
|
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