Year |
Citation |
Score |
2021 |
Zirimwabagabo JO, Jailani ABA, Avgoustou P, Tozer MJ, Gibson KR, Glossop PA, Mills JEJ, Porter RA, Blaney P, Wang N, Skerry TM, Richards GO, Harrity JPA. Discovery of a First-In-Class Small Molecule Antagonist against the Adrenomedullin-2 Receptor: Structure-Activity Relationships and Optimization. Journal of Medicinal Chemistry. PMID 33666424 DOI: 10.1021/acs.jmedchem.0c02191 |
0.647 |
|
2020 |
Avgoustou P, Jailani ABA, Zirimwabagabo JO, Tozer MJ, Gibson KR, Glossop PA, Mills JEJ, Porter RA, Blaney P, Bungay PJ, Wang N, Shaw AP, Bigos KJA, Holmes JL, Warrington JI, et al. Discovery of a First-in-Class Potent Small Molecule Antagonist against the Adrenomedullin-2 Receptor. Acs Pharmacology & Translational Science. 3: 706-719. PMID 32832872 DOI: 10.1021/acsptsci.0c00032 |
0.642 |
|
2008 |
Clark RD, Ray NC, Williams K, Blaney P, Ward S, Crackett PH, Hurley C, Dyke HJ, Clark DE, Lockey P, Devos R, Wong M, Porres SS, Bright CP, Jenkins RE, et al. 1H-Pyrazolo[3,4-g]hexahydro-isoquinolines as selective glucocorticoid receptor antagonists with high functional activity. Bioorganic & Medicinal Chemistry Letters. 18: 1312-7. PMID 18226897 DOI: 10.1016/j.bmcl.2008.01.027 |
0.622 |
|
2007 |
Clark RD, Ray NC, Blaney P, Crackett PH, Hurley C, Williams K, Dyke HJ, Clark DE, Lockey PM, Devos R, Wong M, White A, Belanoff JK. 2-Benzenesulfonyl-8a-benzyl-hexahydro-2H-isoquinolin-6-ones as selective glucocorticoid receptor antagonists. Bioorganic & Medicinal Chemistry Letters. 17: 5704-8. PMID 17822897 DOI: 10.1016/j.bmcl.2007.07.055 |
0.628 |
|
2002 |
Blaney P, Grigg R, Sridharan V. Traceless solid-phase organic synthesis. Chemical Reviews. 102: 2607-24. PMID 12105937 DOI: 10.1021/cr0103827 |
0.5 |
|
Show low-probability matches. |