| Ebru D. Akten | Physical Chemistry, Plastics Technology | | 2003 | | Peter G. Schultz (post-doc) |
| Shane Atwell | | | 2001 | | Peter G. Schultz (post-doc) |
| Jun Y. Axup | | | 2008 | 2013 | Peter G. Schultz (grad student) |
| Markus Berger | | | 2001 | | Peter G. Schultz (post-doc) |
| Michael D Best | Lipid Synthesis, Liposomes, Chemistry and Physics of Lipids, Chemical Biology, Drug Delivery | | | | |
| Tony E. Boitano | Hematopoiesis | | 2005 | 2007 | Peter G. Schultz (post-doc) |
| Michael J. Bollong | | Chemistry | 2010 | 2016 | Peter G. Schultz (grad student) |
| Mohua Bose | Organic Chemistry, Biochemistry | Chemistry | 2002 | 2004 | Peter G. Schultz (post-doc) |
| Laure Bouchez | | | 2008 | 2010 | Peter G. Schultz (post-doc) |
| Achim Brinker | | | 2001 | 2003 | Peter G. Schultz (post-doc) |
| Mark Bushey | | | 2008 | | Peter G. Schultz (post-doc) |
| John Cavanagh | | | 1991 | 1994 | Mark Rance (post-doc), Peter E. Wright (research scientist) |
| Eli Chapman | organic chemistry | | 1996 | | Peter G. Schultz (research assistant) |
| Abhishek Chatterjee | Chemical Biology, Synthetic Biology | | 2013 | | Peter G. Schultz (post-doc) |
| Liangjing Chen | | | 2001 | | Peter G. Schultz (post-doc) |
| Shawn Chen | | | 2006 | | Peter G. Schultz (post-doc) |
| Susanna Chen | | | 2006 | | Peter G. Schultz (grad student) |
| Sivasankar Chinnappan | | | 2007 | 2008 | Roy A. Periana (post-doc) |
| Dong-Gyu Cho | Functional Molecular Synthesis | | 2008 | 2009 | M.G. Finn (post-doc) |
| Seihyun Choi | | | 2015 | | Peter G. Schultz (post-doc) |
| Woojin Choi | Chemical Biology | | | | |
| Joyanta Choudhury | Organometallics, Catalysis, Surface Chemistry | Chemistry | 2007 | 2008 | Roy A. Periana (post-doc) |
| Eugene Chun | | | | | Raymond C. Stevens (grad student) |
| Julie Clark | | | | | |
| Corey M. Dambacher | | Chemistry | 2006 | 2011 | Peter G. Schultz (grad student) |
| Philip E. Dawson | | | 1993 | 1996 | Stephen B. H. Kent (grad student) |
| Jonathan Day | | | 2011 | | Peter G. Schultz (post-doc) |
| Min Deng | | | | | |
| David Díaz Díaz | | | 2002 | 2005 | M.G. Finn (post-doc) |
| Anna Dubrovska | | | 2007 | 2011 | Peter G. Schultz (post-doc) |
| Scott Dunning | | | 2005 | | Peter G. Schultz (research scientist) |
| Jörg Eppinger | | | 2001 | | Peter G. Schultz (post-doc) |
| Ines Forrest | Chemical Biology, Proteomics, Drug Discovery | Chemistry | 2020 | | Christopher G. Parker (grad student) |
| Jennifer L. Furman | Bioorganic Chemistry | | 2011 | 2014 | Peter G. Schultz (post-doc) |
| Veeranjaneyulu Gannedi | Chemistry | Beckman Center for Chemical Sciences | 2022 | | Chi-Huey Wong (post-doc) |
| Varun Gauba | Organic Chemistry, General Biophysics | Chemistry | 2009 | 2012 | Peter G. Schultz (post-doc) |
| Haibo Ge | | | | | Dale L. Boger (post-doc) |
| Jeffrey Gildersleeve | | | 2003 | | Peter G. Schultz (post-doc) |
| Agi Glownia | | | 2002 | | Peter G. Schultz (research assistant) |
| Rodolfo Gonzalez | | | 2011 | | Peter G. Schultz (post-doc) |
| Jovana Grbic | | | 2007 | | Peter G. Schultz (grad student) |
| Carlos Guijas | | Chemistry | 2017 | 2020 | Gary Siuzdak (post-doc) |
| Sayam Sen Gupta | Inorganic Chemistry, Environmental Engineering, Chemical Engineering | | 2002 | 2005 | M.G. Finn (post-doc) |
| Rajkumar Halder | | | 2012 | | Peter G. Schultz (post-doc) |
| Michael A. Hanson | | | | | |
| Sarah Hanson | | | 1999 | | Peter G. Schultz (grad student) |
| Bradley Herberich | | | 2003 | | Peter G. Schultz (post-doc) |
| Simon Hilcove | | | | | Sheng Ding (grad student) |
| David Hill | | | 2014 | 2020 | Donna G. Blackmond (grad student) |
| Jordi C. J. Hintzen | Chemical biology, peptide chemistry, medicinal chemistry, protein synthesis | | 2017 | 2018 | Philip E. Dawson (research assistant) |
| Mannkyu Hong | | Chemistry | 2022 | | Peter G. Schultz (post-doc) |
| Min Kyung Hoon | | | 2015 | | Peter G. Schultz (research scientist) |
| Xiaoyi Hu | Proteomics | Chemistry | 2007 | 2011 | Peter G. Schultz (post-doc) |
| Jin-Feng Hu | | | 2002 | | Peter G. Schultz (post-doc) |
| Qihong Huang | Pesticide Biotechnology | | 2001 | 2005 | Peter G. Schultz (post-doc) |
| Chunhui Huang | | Chemistry | 2012 | 2014 | Peter G. Schultz (post-doc) |
| Woo-Young Hur | | | 2004 | | Peter G. Schultz (grad student) |
| Ben Hutchins | | | 2009 | | Peter G. Schultz (post-doc) |
| Appaso M Jadhav | Organic Chemistry, Medicinal Chemistry, Proteomics | | | | |
| Valer Jeso | | | 2004 | 2009 | K. C. Nicolaou (grad student) |
| Fanyi Jiang | | | 2001 | | Peter G. Schultz (post-doc) |
| Mingchao Kang | Chemical Biology | Chemistry | 2008 | 2013 | Peter G. Schultz (grad student) |
| Akira Kawamura | | | 2003 | | Peter G. Schultz (post-doc) |
| Stephanie Kazane | | | | | |
| Chanhyuk Kim | | | 2008 | | Peter G. Schultz (research scientist) |
| Jong-Man Kim | | | 2012 | | Peter G. Schultz (post-doc) |
| Atsushi Kimishima | Synthetic Organic Chemistry | | | | Kim David Janda (post-doc) |
| Douglas J. Kojetin | Nuclear receptors, NMR spectroscopy, Structural biology | | 2009 | 2010 | Thomas P Burris (post-doc) |
| Luke L. Lairson | | Chemistry | 2007 | 2009 | Peter G. Schultz (post-doc) |
| Jongkook Lee | Pharmaceutical chemistry | Chemistry | 2004 | 2007 | Peter G. Schultz (post-doc) |
| Jae Wook Lee | | | 2007 | | Peter G. Schultz (post-doc) |
| Jing Li | Drug Discovery | Chemistry | 2000 | 2001 | Peter G. Schultz (post-doc) |
| Han Li | | | 2013 | | Peter G. Schultz (post-doc) |
| Qing Lin | chemical biology | Chemistry | 2000 | 2003 | Peter G. Schultz (post-doc) |
| Jun Liu | | | 2002 | | Peter G. Schultz (post-doc) |
| Zilei Liu | Immunology, Click chemistry, carbohydrate chemistry | | | | |
| Hendrik Luesch | | | 2002 | 2005 | Peter G. Schultz (post-doc) |
| Felix Marr | | | 2006 | | Peter G. Schultz (post-doc) |
| Kevin W. Martin | | | 2014 | | Peter G. Schultz (post-doc) |
| Casey J. N. Mathison | | | | | |
| Eric Meggers | Organic Chemistry, Inorganic Chemistry, Chemical Biology, Catalysis | | 1999 | 2002 | Peter G. Schultz (post-doc) |
| Ryan A. Mehl | Barton Professor of Chemistry | | 2004 | | Peter G. Schultz (post-doc) |
| Mauro Mileni | | | | | |
| Rebecca L. Miller | | | | | Raymond C. Stevens (grad student) |
| Karthik Nadendla | | Chemistry | | | Lucas J. Leman (grad student) |
| Advait Nagle | | | 2004 | | Peter G. Schultz (post-doc) |
| Tae-gyu Nam | | | 2008 | | Peter G. Schultz (post-doc) |
| Anthony Ogawa | | | 1998 | | Peter G. Schultz (post-doc) |
| Toshihide Okajima | | | 1999 | | Peter G. Schultz (post-doc) |
| Barun Okram | | | 2004 | | Peter G. Schultz (post-doc) |
| Kevin Oldenburg | | | 1996 | | Peter G. Schultz (post-doc) |
| Takanori Otomo | | | | | Michael K. Rosen (post-doc) |
| Nitin T. Patil | Synthetic organic chemistry, organo-catalysis | | 2006 | 2008 | K. C. Nicolaou (post-doc) |
| Joshua Payette | | | 2010 | 2012 | Peter G. Schultz (post-doc) |
| Roshan Perera | Bio-inorganic, bio-physical, and bio-organic chemistry; spectroscopy and mechanisms of action of dioxygen- and peroxide-activating heme iron enzymes and model systems; cytochrome P-450; magnetic circular dichroism spectroscopy | | 2005 | | Peter G. Schultz (post-doc) |
| Frank Peters | | | 2006 | | Peter G. Schultz (grad student) |
| Hank Michael Petrassi | | | 2001 | | Peter G. Schultz (post-doc) |
| John P. Pezacki | | | 2001 | | Peter G. Schultz (research scientist) |
| Joshua G. Pierce | Organic Synthesis, Chemical Microbiology | | | | |
| Christoph Rader | | | | | |
| Mark Rance | structure and dynamics of biomolecules | | | | |
| Adam R. Renslo | Biochemistry, Organic Chemistry, Parasitology Biology | | 1998 | 2000 | Julius Rebek, Jr. (post-doc) |
| Rainer Riedl | | | | | |
| Amit Sagi | | | 2009 | | Peter G. Schultz (post-doc) |
| Stephen Santoro | | | 1999 | | Peter G. Schultz (post-doc) |
| Petri Saviranta | | | 2002 | | Peter G. Schultz (post-doc) |
| Stefan Schiller | | | 2003 | 2008 | Peter G. Schultz (post-doc) |
| Peter G. Schultz | | | | | |
| Urs Schwitter | | | 2004 | | Peter G. Schultz (post-doc) |
| Joan-Emma Shea | Physical Chemistry, Theory & Computation, Biochemistry & Biophysics, Biomedical Sciences, Biology-Inspired Chemistry & Physics, Structural Chemistry, Spectroscopy & Advanced Analysis | | 1997 | 2000 | Charles L. Brooks (post-doc), José Nelson Onuchic (post-doc) |
| Jana Shen | Computational Chemistry and Biophysics, Drug and Material Design | | 2003 | 2007 | Charles L. Brooks (post-doc) |
| Weijun Shen | drug discovery, peptide engineering, cell biology, high throughput screening, | | 2007 | 2009 | Peter G. Schultz (post-doc) |
| Jiayin Shen | | | 2014 | | Peter G. Schultz (post-doc) |
| Injae Shin | | | 1995 | 1998 | Peter G. Schultz (post-doc) |
| Shoji Shinichiro | | | 2009 | 2011 | Peter G. Schultz (post-doc) |
| Eric E. Simanek | Organic Chemistry, Biochemistry | | | | Chi-Huey Wong (post-doc) |
| Fai Yiu Siu | | | | | Raymond C. Stevens (post-doc) |
| Vaughn Smider | | | 2006 | | Peter G. Schultz (research scientist) |
| Kristen Smith | | | 2009 | 2010 | Peter G. Schultz (research scientist) |
| Scott A. Snyder | total synthesis of natural products | | | | |
| Thereza Amélia Soares | | Department of Integrative Structural and Computational Biology | 1997 | 1998 | Arthur Olson (grad student) |
| Ryan L. Stowe | Chemistry Education Research | | | | |
| Steven J. Sucheck | Organic Chemistry | Chemistry | | | Chi-Huey Wong (post-doc) |
| Daniel Summerer | Chemical Biology | Chemistry | 2004 | 2006 | Peter G. Schultz (post-doc) |
| Sophie Sun | | | 2008 | | Peter G. Schultz (grad student) |
| Lubica Supekova | | | 1998 | | Peter G. Schultz (research scientist) |
| Eunju Lee Tae | | | 1999 | | Peter G. Schultz (post-doc) |
| Nobuyuki Tamaoki | | | 1995 | 1996 | M. Reza Ghadiri (post-doc) |
| Feng Tian | | | 2000 | | Peter G. Schultz (post-doc) |
| Meng-Lin Tsao | | | 2009 | | Peter G. Schultz (post-doc) |
| Jim Turner | | | 2004 | | Peter G. Schultz (post-doc) |
| Daniel Wacker | | | | | Raymond C. Stevens (grad student) |
| Jingxin Wang | Chemical Biology | | 2014 | 2019 | Peter G. Schultz (post-doc) |
| Feng Wang | | | 2010 | | Peter G. Schultz (research scientist) |
| Yan Wang | | | 2014 | | Peter G. Schultz (post-doc) |
| Danling Wang | | | 2014 | | Peter G. Schultz (research scientist) |
| Tsung-Shing Wang | molecular mechanisms of various antibiotics | | 2011 | | Peter G. Schultz (post-doc) |
| Weidong Wang | | | 2006 | | Peter G. Schultz (post-doc) |
| Jan Wang | | | 2007 | 2008 | Peter G. Schultz (post-doc) |
| Peng George Wang | Glycoscience | | | 1994 | Chi-Huey Wong (post-doc) |
| Chong Wang | | | | | Raymond C. Stevens (grad student) |
| Jie Wang | Organic Chemistry | Department of Chemistry | 2015 | 2018 | Phil S. Baran (grad student) |
| Masaki Warashina | | | 2003 | | Peter G. Schultz (post-doc) |
| Michael P. Washburn | | | | | John Yates III (research scientist) |
| Coran Watanabe | Organic Chemistry | | 1999 | | Peter G. Schultz (post-doc) |
| Aaron Willingham | | | 2002 | | Peter G. Schultz (post-doc) |
| Carrie M. Wilmot | Biochemistry | | 1989 | 1992 | Ian A. Wilson (post-doc) |
| Luke Wiseman | | | | | |
| Krista Witte | | | 1997 | | Peter G. Schultz (post-doc) |
| Chi-Huey Wong | organic chemistry | | | | |
| Xu Wu | lipid biochemistry, chemical biology, developmental biology and cancer | | 2001 | 2004 | Peter G. Schultz (grad student) |
| Gang Xia | | | 1999 | | Peter G. Schultz (post-doc) |
| Han Xiao | | | 2010 | 2015 | Peter G. Schultz (grad student) |
| Wen Xiong | | | | | Sheng Ding (research scientist) |
| Fei Xu | | | | | Raymond C. Stevens (grad student) |
| Jiong Yang | organic synthesis | Chemistry | 2003 | 2004 | Peter G. Schultz (post-doc) |
| Shuyuan Yao | | | 2004 | | Sheng Ding (post-doc), Peter G. Schultz (post-doc) |
| Mengchun Ye | | | | | |
| Seungwan Yoon | | | 2004 | | Peter G. Schultz (post-doc) |
| Doug Young | | | 2009 | 2011 | Peter G. Schultz (post-doc) |
| Douglas Young | | | 2009 | | Peter G. Schultz (post-doc) |
| Fanwen Zeng | | | 1997 | | Peter G. Schultz (post-doc) |
| Qisheng Zhang | Lipid signaling, Small GTPase, Chemical Biology | | 2004 | | Peter G. Schultz (post-doc) |
| Lianxing Zheng | RNA Biology | | 2001 | 2004 | Peter G. Schultz (post-doc) |
| De-Min Zhou | | | 1999 | | Peter G. Schultz (post-doc) |
| Nicole Zimmerman | | | 2002 | | Peter G. Schultz (post-doc) |