Year |
Citation |
Score |
2016 |
Crawford TD, Tsui V, Flynn EM, Wang S, Taylor AM, Côté A, Audia JE, Beresini MH, Burdick DJ, Cummings RT, Dakin LA, Duplessis M, Good AC, Hewitt MC, Huang HR, ... ... Nasveschuk CG, et al. Diving into the water: Inducible binding conformations for BRD4, TAF1(2), BRD9, and CECR2 bromodomains. Journal of Medicinal Chemistry. PMID 27219867 DOI: 10.1021/Acs.Jmedchem.6B00264 |
0.301 |
|
2015 |
Hewitt MC, Leblanc Y, Gehling VS, Vaswani RG, Côté A, Nasveschuk CG, Taylor AM, Harmange JC, Audia JE, Pardo E, Cummings R, Joshi S, Sandy P, Mertz JA, Sims RJ, et al. Development of methyl isoxazoleazepines as inhibitors of BET. Bioorganic & Medicinal Chemistry Letters. 25: 1842-8. PMID 25851940 DOI: 10.1016/J.Bmcl.2015.03.045 |
0.326 |
|
2014 |
Vaswani RG, Albrecht BK, Audia JE, Côté A, Dakin LA, Duplessis M, Gehling VS, Harmange JC, Hewitt MC, Leblanc Y, Nasveschuk CG, Taylor AM. A practical synthesis of indoles via a Pd-catalyzed C-N ring formation. Organic Letters. 16: 4114-7. PMID 25068576 DOI: 10.1021/Ol5018118 |
0.406 |
|
2014 |
Nasveschuk CG, Gagnon A, Garapaty-Rao S, Balasubramanian S, Campbell R, Lee C, Zhao F, Bergeron L, Cummings R, Trojer P, Audia JE, Albrecht BK, Harmange JC. Discovery and Optimization of Tetramethylpiperidinyl Benzamides as Inhibitors of EZH2. Acs Medicinal Chemistry Letters. 5: 378-83. PMID 24900844 DOI: 10.1021/Ml400494B |
0.318 |
|
2012 |
Ungermannova D, Parker SJ, Nasveschuk CG, Chapnick DA, Phillips AJ, Kuchta RD, Liu X. Identification and mechanistic studies of a novel ubiquitin E1 inhibitor. Journal of Biomolecular Screening. 17: 421-34. PMID 22274912 DOI: 10.1177/1087057111433843 |
0.307 |
|
2008 |
Nasveschuk CG, Rovis T. The [1, 3] O-to-C rearrangement: opportunities for stereoselective synthesis. Organic & Biomolecular Chemistry. 6: 240-54. PMID 18174990 DOI: 10.1039/B714881J |
0.521 |
|
2008 |
Nasveschuk CG, Rovis T. A diastereoselective ring contraction of 1,3-dioxepins to 2,3,4-trisubstituted and tetrasubstituted tetrahydrofurans. The Journal of Organic Chemistry. 73: 612-7. PMID 18088144 DOI: 10.1021/Jo702071V |
0.636 |
|
2008 |
Nasveschuk CG, Rovis T. A rapid total synthesis of (±)-sylvone Synlett. 0126-0128. DOI: 10.1055/S-2007-990926 |
0.513 |
|
2008 |
Nasveschuk CG, Rovis T. ChemInform Abstract: A Rapid Total Synthesis of (.+-.)-Sylvone. Cheminform. 39. DOI: 10.1002/chin.200822206 |
0.502 |
|
2007 |
Nasveschuk CG, Frein JD, Jui NT, Rovis T. A diastereoselective intermolecular heck reaction of 1,3-dioxepins. Organic Letters. 9: 5099-102. PMID 17958436 DOI: 10.1021/Ol702294U |
0.526 |
|
2006 |
Nasveschuk CG, Jui NT, Rovis T. A modular approach to the synthesis of 2,3,4-trisubstituted tetrahydrofurans. Chemical Communications (Cambridge, England). 3119-21. PMID 16855705 DOI: 10.1039/B605438B |
0.575 |
|
2005 |
Nasveschuk CG, Rovis T. Regioselective Lewis acid-mediated [1,3] rearrangement of allylvinyl ethers. Organic Letters. 7: 2173-6. PMID 15901162 DOI: 10.1021/Ol0505151 |
0.588 |
|
2005 |
Nasveschuk CG, Rovis T. Stereoselective Lewis acid mediated [1,3] ring contraction of 2,5-dihydrooxepins as a route to polysubstituted cyclopentenes. Angewandte Chemie (International Ed. in English). 44: 3264-7. PMID 15844118 DOI: 10.1002/Anie.200500088 |
0.543 |
|
2004 |
Byers JH, DeWitt A, Nasveschuk CG, Swigor JE. Tandem radical-electrophilic annulations to pyrrole Tetrahedron Letters. 45: 6587-6590. DOI: 10.1016/J.Tetlet.2004.07.037 |
0.326 |
|
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