| Year |
Citation |
Score |
| 2014 |
Sidhu PS, Nassif N, McCallum MM, Teske K, Feleke B, Yuan NY, Nandhikonda P, Cook JM, Singh RK, Bikle DD, Arnold LA. Development of novel Vitamin D Receptor-Coactivator Inhibitors. Acs Medicinal Chemistry Letters. 5: 199-204. PMID 24799995 DOI: 10.1021/Ml400462J |
0.478 |
|
| 2014 |
McCallum MM, Pawlak AJ, Shadrick WR, Simeonov A, Jadhav A, Yasgar A, Maloney DJ, Arnold LA. A fluorescence-based high throughput assay for the determination of small molecule-human serum albumin protein binding. Analytical and Bioanalytical Chemistry. 406: 1867-75. PMID 24390461 DOI: 10.1007/S00216-013-7560-3 |
0.461 |
|
| 2013 |
Nandhikonda P, Yasgar A, Baranowski AM, Sidhu PS, McCallum MM, Pawlak AJ, Teske K, Feleke B, Yuan NY, Kevin C, Bikle DD, Ayers SD, Webb P, Rai G, Simeonov A, et al. Peroxisome proliferation-activated receptor δ agonist GW0742 interacts weakly with multiple nuclear receptors, including the vitamin D receptor. Biochemistry. 52: 4193-203. PMID 23713684 DOI: 10.1021/Bi400321P |
0.49 |
|
| 2013 |
McCallum MM, Nandhikonda P, Temmer JJ, Eyermann C, Simeonov A, Jadhav A, Yasgar A, Maloney D, Arnold AL. High-throughput identification of promiscuous inhibitors from screening libraries with the use of a thiol-containing fluorescent probe. Journal of Biomolecular Screening. 18: 705-13. PMID 23446699 DOI: 10.1177/1087057113476090 |
0.419 |
|
| 2012 |
Nandhikonda P, Lynt WZ, McCallum MM, Ara T, Baranowski AM, Yuan NY, Pearson D, Bikle DD, Guy RK, Arnold LA. Discovery of the first irreversible small molecule inhibitors of the interaction between the vitamin D receptor and coactivators. Journal of Medicinal Chemistry. 55: 4640-51. PMID 22563729 DOI: 10.1021/Jm300460C |
0.471 |
|
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