Year |
Citation |
Score |
2024 |
Gurol KC, Jursa T, Cho EJ, Fast W, Dalby KN, Smith DR, Mukhopadhyay S. PHD2 enzyme is an intracellular manganese sensor that initiates the homeostatic response against elevated manganese. Proceedings of the National Academy of Sciences of the United States of America. 121: e2402538121. PMID 38905240 DOI: 10.1073/pnas.2402538121 |
0.478 |
|
2024 |
Sammons RM, Devkota AK, Kaoud TS, Warthaka M, Cho EJ, Dalby KN. Steady State and Time-Dependent Fluorescent Peptide Assays for Protein Kinases. Current Protocols. 4: e998. PMID 38439594 DOI: 10.1002/cpz1.998 |
0.516 |
|
2024 |
Wible DJ, Parikh Z, Cho EJ, Chen MD, Jeter CR, Mukhopadhyay S, Dalby KN, Varadarajan S, Bratton SB. Unexpected inhibition of the lipid kinase PIKfyve reveals an epistatic role for p38 MAPKs in endolysosomal fission and volume control. Cell Death & Disease. 15: 80. PMID 38253602 DOI: 10.1038/s41419-024-06423-0 |
0.529 |
|
2023 |
Lee J, Guo HF, Wang S, Maghsoud Y, Vázquez-Montelongo EA, Jing Z, Sammons RM, Cho EJ, Ren P, Cisneros GA, Kurie JM, Dalby KN. Unleashing the Potential of 1,3-Diketone Analogues as Selective LH2 Inhibitors. Acs Medicinal Chemistry Letters. 14: 1396-1403. PMID 37849534 DOI: 10.1021/acsmedchemlett.3c00305 |
0.523 |
|
2023 |
Wible DJ, Parikh Z, Cho EJ, Chen MD, Mukhopadhyay S, Dalby KN, Varadarajan S, Bratton SB. Unexpected inhibition of the lipid kinase PIKfyve reveals an epistatic role for p38 MAPKs in endolysosomal fission and volume control. Biorxiv : the Preprint Server For Biology. PMID 36993747 DOI: 10.1101/2023.03.13.532495 |
0.516 |
|
2022 |
Sammons RM, Bohanon AL, Kowtha A, Dejong A, Cho EJ, Kaoud TS, Dalby KN. High-Throughput Assay for Identifying Diverse Antagonists of the Binding Interaction between the ACE2 Receptor and the Dynamic Spike Proteins of SARS-CoV-2. Acs Infectious Diseases. 8: 2259-2270. PMID 36315931 DOI: 10.1021/acsinfecdis.2c00297 |
0.515 |
|
2022 |
Li Y, Fan Y, Xu J, Huo L, Scott AW, Jin J, Yang B, Shao S, Ma L, Wang Y, Yao X, Pool Pizzi M, Sewastjanow Da Silva M, Zhang G, Zhuo L, ... Cho EJ, et al. GRK3 is a poor prognosticator and serves as a therapeutic target in advanced gastric adenocarcinoma. Journal of Experimental & Clinical Cancer Research : Cr. 41: 257. PMID 35996148 DOI: 10.1186/s13046-022-02463-6 |
0.476 |
|
2022 |
Thomas PW, Cho EJ, Bethel CR, Smisek T, Ahn YC, Schroeder JM, Thomas CA, Dalby KN, Beckham JT, Crowder MW, Bonomo RA, Fast W. Discovery of an Effective Small-Molecule Allosteric Inhibitor of New Delhi Metallo-β-lactamase (NDM). Acs Infectious Diseases. PMID 35353502 DOI: 10.1021/acsinfecdis.1c00577 |
0.537 |
|
2021 |
Cho EJ, Dalby KN. Luminescence Energy Transfer-Based Screening and Target Engagement Approaches for Chemical Biology and Drug Discovery. Slas Discovery : Advancing Life Sciences R & D. 24725552211036056. PMID 34330171 DOI: 10.1177/24725552211036056 |
0.527 |
|
2021 |
Mohiuddin IS, Wei SJ, Yang IH, Martinez GM, Yang S, Cho EJ, Dalby KN, Kang MH. Development of Cell-based High Throughput Luminescence Assay for Drug Discovery in Inhibiting OCT4-DNA-PKcs and OCT4-MK2 Interactions. Biotechnology and Bioengineering. PMID 33565603 DOI: 10.1002/bit.27712 |
0.567 |
|
2020 |
Cho EJ, Devkota AK, Stancu G, Edupunganti R, Debevec G, Giulianotti M, Houghten R, Powis G, Dalby KN. A Robust and Cost-Effective Luminescent-Based High-Throughput Assay for Fructose-1,6-Bisphosphate Aldolase A. Slas Discovery : Advancing Life Sciences R & D. 2472555220926146. PMID 32462959 DOI: 10.1177/2472555220926146 |
0.561 |
|
2020 |
Del Mundo IMA, Cho EJ, Dalby KN, Vasquez KM. A 'light-up' intercalator displacement assay for detection of triplex DNA stabilizers. Chemical Communications (Cambridge, England). PMID 31960843 DOI: 10.1039/C9Cc08817B |
0.525 |
|
2019 |
Sammons RM, Perry NA, Li Y, Cho EJ, Piserchio A, Zamora-Olivares DP, Ghose R, Kaoud TS, Debevec G, Bartholomeusz C, Gurevich VV, Iverson TM, Giulianotti M, Houghten RA, Dalby KN. A Novel Class of Common Docking Domain Inhibitors That Prevent ERK2 Activation and Substrate Phosphorylation. Acs Chemical Biology. PMID 31058487 DOI: 10.1021/Acschembio.9B00093 |
0.599 |
|
2019 |
Veloria J, Shin M, Devkota AK, Payne SM, Cho EJ, Dalby KN. Developing Colorimetric and Luminescence-Based High-Throughput Screening Platforms for Monitoring the GTPase Activity of Ferrous Iron Transport Protein B (FeoB). Slas Discovery : Advancing Life Sciences R & D. 2472555219844572. PMID 31039677 DOI: 10.1177/2472555219844572 |
0.521 |
|
2019 |
Del Mundo IMA, Cho EJ, Dalby KN, Vasquez KM. A tunable assay for modulators of genome-destabilizing DNA structures. Nucleic Acids Research. PMID 30949695 DOI: 10.1093/Nar/Gkz237 |
0.522 |
|
2018 |
Devkota AK, Veloria JR, Guo HF, Kurie JM, Cho EJ, Dalby KN. Development of a High-Throughput Lysyl Hydroxylase (LH) Assay and Identification of Small-Molecule Inhibitors against LH2. Slas Discovery : Advancing Life Sciences R & D. 2472555218817057. PMID 30589612 DOI: 10.1177/2472555218817057 |
0.565 |
|
2018 |
Veloria JR, Devkota AK, Cho EJ, Dalby KN. Development of a cost effective and robust AlphaScreen platform for application. Biotechniques. 64: 181-183. PMID 29661010 DOI: 10.2144/Btn-2018-2001 |
0.548 |
|
2017 |
Cho EJ, Devkota AK, Stancu G, Edupunganti R, Powis G, Dalby KN. A Fluorescence-Based High-Throughput Assay for the Identification of Anticancer Reagents Targeting Fructose-1,6-Bisphosphate Aldolase. Slas Discovery. 2472555217726325. PMID 28820953 DOI: 10.1177/2472555217726325 |
0.563 |
|
2017 |
Edupuganti R, Taliaferro JM, Wang Q, Xie X, Cho EJ, Vidhu F, Ren P, Anslyn EV, Bartholomeusz C, Dalby KN. Discovery of a potent inhibitor of MELK that inhibits expression of the anti-apoptotic protein Mcl-1 and TNBC cell growth. Bioorganic & Medicinal Chemistry. PMID 28351607 DOI: 10.1016/J.Bmc.2017.03.018 |
0.595 |
|
2017 |
Guo HF, Cho EJ, Devkota AK, Chen Y, Russell W, Phillips GN, Yamauchi M, Dalby KN, Kurie JM. A scalable lysyl hydroxylase 2 expression system and luciferase-based enzymatic activity assay. Archives of Biochemistry and Biophysics. PMID 28216326 DOI: 10.1016/J.Abb.2017.02.003 |
0.58 |
|
2017 |
Guo H, Tsai C, Chen Y, Terajima M, Yamauchi M, Alvarado S, Cho E, Dalby K, Phillips G, Tainer J, Kurie J. Structure-Based Drug Design Targeting a Pro-Metastatic Collagen Lysyl Hydroxylase Journal of Thoracic Oncology. 12: S1543. DOI: 10.1016/J.Jtho.2017.06.048 |
0.511 |
|
2016 |
Veloria JR, Devkota AK, Cho EJ, Dalby KN. Optimization of a Luminescence-Based High-Throughput Screening Assay for Detecting Apyrase Activity. Journal of Biomolecular Screening. PMID 27821623 DOI: 10.1177/1087057116675859 |
0.604 |
|
2016 |
Grandjean G, De Jong PR, James BP, Koh MY, Lemos R, Kingston J, Aleshin A, Bankston LA, Miller CP, Cho EJ, Edupuganti R, Devkota A, Stancu G, Liddington RC, Dalby KN, et al. Definition of a novel feed-forward mechanism for glycolysis-HIF1α signaling in hypoxic tumors highlights adolase A as a therapeutic target. Cancer Research. PMID 27261507 DOI: 10.1158/0008-5472.Can-16-0401 |
0.566 |
|
2016 |
Rycaj K, Cho EJ, Liu X, Chao HP, Liu B, Li Q, Devkota AK, Zhang D, Chen X, Moore J, Dalby KN, Tang DG. Longitudinal tracking of subpopulation dynamics and molecular changes during LNCaP cell castration and identification of inhibitors that could target the PSA-/lo castration-resistant cells. Oncotarget. PMID 26871947 DOI: 10.18632/Oncotarget.7303 |
0.571 |
|
2016 |
Tavares CD, Devkota AK, Dalby KN, Cho EJ. Application of Eukaryotic Elongation Factor-2 Kinase (eEF-2K) for Cancer Therapy: Expression, Purification, and High-Throughput Inhibitor Screening. Methods in Molecular Biology (Clifton, N.J.). 1360: 19-33. PMID 26501899 DOI: 10.1007/978-1-4939-3073-9_2 |
0.62 |
|
2015 |
Jong PRd, Grandjean GV, Devkota AK, Cho EJ, Dalby KN, Powis G. Abstract 4448: Identification of a small molecule inhibitor of aldolase A for the targeting of hypoxic cancer cells Cancer Research. 75: 4448-4448. DOI: 10.1158/1538-7445.Am2015-4448 |
0.414 |
|
2015 |
Sammons RM, Kaoud TS, Devkota AK, Cho EJ, Dalby KN. Abstract 3648: A high-throughput fluorescence anisotropy screening for discovery of inhibitors that target the D-recruitment site of ERK in vitro and in cells Cancer Research. 75: 3648-3648. DOI: 10.1158/1538-7445.Am2015-3648 |
0.444 |
|
2014 |
Devkota AK, Edupuganti R, Yan C, Shi Y, Jose J, Wang Q, Kaoud TS, Cho EJ, Ren P, Dalby KN. Reversible covalent inhibition of eEF-2K by carbonitriles. Chembiochem : a European Journal of Chemical Biology. 15: 2435-42. PMID 25224652 DOI: 10.1002/Cbic.201402321 |
0.564 |
|
2014 |
Wang Q, Park J, Devkota AK, Cho EJ, Dalby KN, Ren P. Identification and validation of novel PERK inhibitors. Journal of Chemical Information and Modeling. 54: 1467-75. PMID 24745945 DOI: 10.1021/Ci500114R |
0.599 |
|
2014 |
Devkota AK, Warthaka M, Edupuganti R, Tavares CD, Johnson WH, Ozpolat B, Cho EJ, Dalby KN. High-throughput screens for eEF-2 kinase. Journal of Biomolecular Screening. 19: 445-52. PMID 24078616 DOI: 10.1177/1087057113505204 |
0.614 |
|
2012 |
Cho EJ, Xia S, Ma LC, Robertus J, Krug RM, Anslyn EV, Montelione GT, Ellington AD. Identification of influenza virus inhibitors targeting NS1A utilizing fluorescence polarization-based high-throughput assay Journal of Biomolecular Screening. 17: 448-459. PMID 22223052 DOI: 10.1177/1087057111431488 |
0.409 |
|
2011 |
You L, Cho EJ, Leavitt J, Ma LC, Montelione GT, Anslyn EV, Krug RM, Ellington A, Robertus JD. Synthesis and evaluation of quinoxaline derivatives as potential influenza NS1A protein inhibitors. Bioorganic & Medicinal Chemistry Letters. 21: 3007-11. PMID 21478016 DOI: 10.1016/J.Bmcl.2011.03.042 |
0.32 |
|
2011 |
Zhang M, Cho EJ, Burstein G, Siegel D, Zhang Y. Selective inactivation of a human neuronal silencing phosphatase by a small molecule inhibitor Acs Chemical Biology. 6: 511-519. PMID 21348431 DOI: 10.1021/Cb100357T |
0.361 |
|
2007 |
Yang L, Fung CW, Cho EJ, Ellington AD. Real-time rolling circle amplification for protein detection. Analytical Chemistry. 79: 3320-9. PMID 17378540 DOI: 10.1021/Ac062186B |
0.316 |
|
2006 |
Cho EJ, Collett JR, Szafranska AE, Ellington AD. Optimization of aptamer microarray technology for multiple protein targets. Analytica Chimica Acta. 564: 82-90. PMID 17723365 DOI: 10.1016/J.Aca.2005.12.038 |
0.317 |
|
2005 |
Collett JR, Cho EJ, Lee JF, Levy M, Hood AJ, Wan C, Ellington AD. Functional RNA microarrays for high-throughput screening of antiprotein aptamers. Analytical Biochemistry. 338: 113-23. PMID 15707941 DOI: 10.1016/J.Ab.2004.11.027 |
0.314 |
|
2004 |
Kirby R, Cho EJ, Gehrke B, Bayer T, Park YS, Neikirk DP, McDevitt JT, Ellington AD. Aptamer-based sensor arrays for the detection and quantitation of proteins. Analytical Chemistry. 76: 4066-75. PMID 15253644 DOI: 10.1021/Ac049858N |
0.32 |
|
2003 |
Cho EJ, Tao Z, Tang Y, Tehan EC, Bright FV, Hicks WL, Gardella JA, Hard R. Tailored delivery of active keratinocyte growth factor from biodegradable polymer formulations. Journal of Biomedical Materials Research. Part A. 66: 417-24. PMID 12889013 DOI: 10.1002/Jbm.A.10598 |
0.304 |
|
2002 |
Cho EJ, Tao Z, Tang Y, Tehan EC, Bright FV, Hicks WL, Gardella JA, Hard R. Tools to rapidly produce and screen biodegradable polymer and sol-gel-derived xerogel formulations Applied Spectroscopy. 56: 1385-1389. DOI: 10.1366/00037020260377661 |
0.302 |
|
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