William C. Pomerantz - Publications

Chemistry University of Minnesota, Twin Cities, Minneapolis, MN 
Chemical Biology; Organic Chemistry; Physical Chemistry

49 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2020 Ycas PD, Zahid H, Chan A, Olson NM, Johnson JA, Talluri SK, Schonbrunn E, Pomerantz WCK. New inhibitors for the BPTF bromodomain enabled by structural biology and biophysical assay development. Organic & Biomolecular Chemistry. PMID 32588860 DOI: 10.1039/d0ob00506a  1
2020 Pandey AK, Kirberger SE, Johnson JA, Kimbrough JR, Partridge DKD, Pomerantz WCK. Correction to "Efficient Synthesis of 1,4-Thiazepanones and 1,4-Thiazepanes as 3D-Fragments for Screening Libraries". Organic Letters. PMID 32543202 DOI: 10.1021/acs.orglett.0c01848  1
2020 Olson N, Kroc S, Johnson J, Zahid H, Ycas PD, Chan A, Kimbrough J, Kalra P, Schönbrunn E, Pomerantz WCK. NMR Analyses of Acetylated H2A.Z Isoforms Identify Differential Binding Interactions with the Bromodomain of the NURF Nucleosome Remodeling Complex. Biochemistry. PMID 32356653 DOI: 10.1021/acs.biochem.0c00159  1
2020 Pandey AK, Kirberger SE, Johnson JA, Kimbrough JR, Partridge DKD, Pomerantz WCK. Efficient Synthesis of 1,4-Thiazepanones and 1,4-Thiazepanes as 3D Fragments for Screening Libraries. Organic Letters. PMID 32347732 DOI: 10.1021/acs.orglett.0c01230  1
2019 Johnson JA, Nicolaou CA, Kirberger SE, Pandey AK, Hu H, Pomerantz WCK. Evaluating the Advantages of Using 3D-Enriched Fragments for Targeting BET Bromodomains. Acs Medicinal Chemistry Letters. 10: 1648-1654. PMID 31857841 DOI: 10.1021/acsmedchemlett.9b00414  1
2019 Ycas PD, Wagner N, Olsen NM, Fu R, Pomerantz WCK. 2-Fluorotyrosine is a valuable but understudied amino acid for protein-observed F NMR. Journal of Biomolecular Nmr. PMID 31760571 DOI: 10.1007/s10858-019-00290-0  1
2019 Kirberger SE, Ycas PD, Johnson JA, Chen C, Ciccone MF, Woo RWL, Urick AK, Zahid H, Shi K, Aihara H, McAllister SD, Kashani-Sabet M, Shi J, Dickson A, Dos Santos CO, ... Pomerantz WCK, et al. Selectivity, ligand deconstruction, and cellular activity analysis of a BPTF bromodomain inhibitor. Organic & Biomolecular Chemistry. PMID 30706071 DOI: 10.1039/c8ob02599a  1
2018 Paulson CN, Guan X, Ayoub AM, Chan A, Karim RM, Pomerantz WCK, Schönbrunn E, Georg GI, Hawkinson JE. Design, Synthesis, and Characterization of a Fluorescence Polarization Pan-BET Bromodomain Probe. Acs Medicinal Chemistry Letters. 9: 1223-1229. PMID 30613330 DOI: 10.1021/acsmedchemlett.8b00380  1
2018 Divakaran A, Talluri SK, Ayoub AM, Mishra N, Cui H, Widen JC, Berndt N, Zhu JY, Carlson AS, Topczewski JJ, Schönbrunn E, Harki DA, Pomerantz WCK. Molecular Basis for the N-Terminal Bromodomain and Extra Terminal (BET) Family Selectivity of a Dual Kinase-Bromodomain Inhibitor. Journal of Medicinal Chemistry. PMID 30253095 DOI: 10.1021/acs.jmedchem.8b01248  1
2018 Gee CT, Arntson KE, Koleski EJ, Staebell RL, Pomerantz WCK. Dual Labeling of the CBP/p300 KIX Domain for F NMR Leads to Identification of a New Small-Molecule Binding Site. Chembiochem : a European Journal of Chemical Biology. PMID 29430847 DOI: 10.1002/cbic.201700686  1
2017 Perell GT, Mishra NK, Sudhamalla B, Ycas PD, Islam K, Pomerantz WCK. Specific Acetylation Patterns of H2A.Z Form Transient Interactions with the BPTF Bromodomain. Biochemistry. PMID 28771339 DOI: 10.1021/acs.biochem.7b00648  1
2017 Ayoub AM, Hawk LML, Herzig RJ, Jiang J, Wisniewski AJ, Gee CT, Zhao P, Zhu JY, Berndt N, Offei-Addo NK, Scott TG, Qi J, Bradner JE, Ward TR, Schönbrunn E, ... ... Pomerantz WCK, et al. Correction to BET Bromodomain Inhibitors with One-Step Synthesis Discovered from Virtual Screen. Journal of Medicinal Chemistry. PMID 28696689 DOI: 10.1021/acs.jmedchem.7b00943  1
2017 Perell GT, Staebell RL, Hairani M, Cembran A, Pomerantz WCK. Tuning Sulfur Oxidation States on Thioether-Bridged Peptide Macrocycles for Modulation of Protein Interactions. Chembiochem : a European Journal of Chemical Biology. PMID 28631349 DOI: 10.1002/cbic.201700222  1
2017 Frey WD, Chaudhry A, Slepicka PF, Ouellette AM, Kirberger SE, Pomerantz WCK, Hannon GJ, Dos Santos CO. BPTF Maintains Chromatin Accessibility and the Self-Renewal Capacity of Mammary Gland Stem Cells. Stem Cell Reports. PMID 28579392 DOI: 10.1016/j.stemcr.2017.04.031  1
2017 Ayoub AM, Hawk LML, Herzig RJ, Jiang J, Wisniewski AJ, Gee CT, Zhao P, Zhu JY, Berndt N, Offei-Addo NK, Scott TG, Qi J, Bradner JE, Ward TR, Schönbrunn E, ... ... Pomerantz WCK, et al. BET Bromodomain Inhibitors With One-step Synthesis Discovered from Virtual Screen. Journal of Medicinal Chemistry. PMID 28535045 DOI: 10.1021/acs.jmedchem.6b01336  1
2017 Lee AL, Gee CT, Weegman BP, Einstein SA, Juelfs AR, Ring HL, Hurley KR, Egger SM, Swindlehurst G, Garwood MG, Pomerantz WCK, Haynes CL. Oxygen Sensing with Perfluorocarbon-Loaded Ultraporous Mesostructured Silica Nanoparticles. Acs Nano. PMID 28505422 DOI: 10.1021/acsnano.7b01006  1
2017 Kuriki Y, Komatsu T, Ycas PD, Coulup SK, Carlson EJ, Pomerantz WC. Meeting Proceedings ICBS2016-Translating the Power of Chemical Biology to Clinical Advances. Acs Chemical Biology. PMID 28303709 DOI: 10.1021/acschembio.7b00205  1
2016 Hawk LML, Gee CT, Urick AK, Hu H, Pomerantz WCK. Paramagnetic relaxation enhancement for protein-observed (19)F NMR as an enabling approach for efficient fragment screening. Rsc Advances. 6: 95715-95721. PMID 28496971 DOI: 10.1039/C6RA21226C  1
2016 Urick AK, Calle Jiménez LP, Espinosa JF, Hu H, Pomerantz WC. Protein-Observed Fluorine NMR is a Complementary Ligand Discovery Method to 1H CPMG Ligand-Observed NMR. Acs Chemical Biology. PMID 27627661 DOI: 10.1021/acschembio.6b00730  1
2016 Lewis AK, Dunleavy KM, Senkow TL, Her C, Horn BT, Jersett MA, Mahling R, McCarthy MR, Perell GT, Valley CC, Karim CB, Gao J, Pomerantz WC, Thomas DD, Cembran A, et al. Oxidation increases the strength of the methionine-aromatic interaction. Nature Chemical Biology. PMID 27547920 DOI: 10.1038/nchembio.2159  1
2016 Gee CT, Arntson KE, Urick AK, Mishra NK, Hawk LM, Wisniewski AJ, Pomerantz WC. Protein-observed (19)F-NMR for fragment screening, affinity quantification and druggability assessment. Nature Protocols. 11: 1414-27. PMID 27414758 DOI: 10.1038/nprot.2016.079  1
2016 Isley Iii WC, Urick AK, Pomerantz WC, Cramer CJ. Prediction of (19)F NMR Chemical Shifts in Labeled Proteins: Computational Protocol and Case Study. Molecular Pharmaceutics. PMID 27218275 DOI: 10.1021/acs.molpharmaceut.6b00137  1
2016 Mishra NK, Urick AK, Ember SW, Schönbrunn E, Pomerantz WC. Correction to Letter: Fluorinated Aromatic Amino Acids Are Sensitive (19)F NMR Probes for Bromodomain-Ligand Interactions. Acs Chemical Biology. PMID 26836633 DOI: 10.1021/acschembio.6b00049  1
2015 Arntson KE, Pomerantz WC. Protein-Observed Fluorine NMR: A Bioorthogonal Approach for Small Molecule Discovery. Journal of Medicinal Chemistry. PMID 26599421 DOI: 10.1021/acs.jmedchem.5b01447  1
2015 Urick AK, Hawk LM, Cassel MK, Mishra NK, Liu S, Adhikari N, Zhang W, Dos Santos CO, Hall JL, Pomerantz WC. Dual screening of BPTF and Brd4 using protein-observed fluorine NMR uncovers new bromodomain probe molecules. Acs Chemical Biology. PMID 26158404 DOI: 10.1021/acschembio.5b00483  0.96
2015 Gee CT, Koleski EJ, Pomerantz WC. Fragment screening and druggability assessment for the CBP/p300 KIX domain through protein-observed 19F NMR spectroscopy. Angewandte Chemie (International Ed. in English). 54: 3735-9. PMID 25651535 DOI: 10.1002/anie.201411658  1
2014 Mishra NK, Urick AK, Ember SW, Schönbrunn E, Pomerantz WC. Fluorinated aromatic amino acids are sensitive 19F NMR probes for bromodomain-ligand interactions. Acs Chemical Biology. 9: 2755-60. PMID 25290579 DOI: 10.1021/cb5007344  0.96
2014 Lodge JM, Rettenmaier TJ, Wells JA, Pomerantz WC, Mapp AK. FP Tethering: a screening technique to rapidly identify compounds that disrupt protein-protein interactions. Medchemcomm. 5: 370-375. PMID 24795804 DOI: 10.1039/C3MD00356F  0.96
2013 Wang N, Majmudar CY, Pomerantz WC, Gagnon JK, Sadowsky JD, Meagher JL, Johnson TK, Stuckey JA, Brooks CL, Wells JA, Mapp AK. Ordering a dynamic protein via a small-molecule stabilizer. Journal of the American Chemical Society. 135: 3363-6. PMID 23384013 DOI: 10.1021/ja3122334  0.96
2012 Majmudar CY, Højfeldt JW, Arevang CJ, Pomerantz WC, Gagnon JK, Schultz PJ, Cesa LC, Doss CH, Rowe SP, Vásquez V, Tamayo-Castillo G, Cierpicki T, Brooks CL, Sherman DH, Mapp AK. Sekikaic acid and lobaric acid target a dynamic interface of the coactivator CBP/p300. Angewandte Chemie (International Ed. in English). 51: 11258-62. PMID 23042634 DOI: 10.1002/anie.201206815  0.96
2012 Pomerantz WC, Wang N, Lipinski AK, Wang R, Cierpicki T, Mapp AK. Profiling the dynamic interfaces of fluorinated transcription complexes for ligand discovery and characterization. Acs Chemical Biology. 7: 1345-50. PMID 22725662 DOI: 10.1021/cb3002733  0.96
2011 Pomerantz WC, Yuwono VM, Drake R, Hartgerink JD, Abbott NL, Gellman SH. Lyotropic liquid crystals formed from ACHC-rich β-peptides. Journal of the American Chemical Society. 133: 13604-13. PMID 21815636 DOI: 10.1021/ja204874h  0.96
2011 Thiele CM, Pomerantz WC, Abbott NL, Gellman SH. Lyotropic liquid crystalline phases from helical β-peptides as alignment media. Chemical Communications (Cambridge, England). 47: 502-4. PMID 20972503 DOI: 10.1039/c0cc02123g  0.96
2011 Bates CA, Pomerantz WC, Mapp AK. Transcriptional tools: Small molecules for modulating CBP KIX-dependent transcriptional activators. Biopolymers. 95: 17-23. PMID 20882601 DOI: 10.1002/bip.21548  0.96
2009 Pomerantz WC, Hadley EB, Fry CG, Gellman SH. In situ monitoring of backbone thioester exchange by 19F NMR. Chembiochem : a European Journal of Chemical Biology. 10: 2177-81. PMID 19644993 DOI: 10.1002/cbic.200900380  0.96
2009 Bao L, Gorin MA, Zhang M, Ventura AC, Pomerantz WC, Merajver SD, Teknos TN, Mapp AK, Pan Q. Preclinical development of a bifunctional cancer cell homing, PKCepsilon inhibitory peptide for the treatment of head and neck cancer. Cancer Research. 69: 5829-34. PMID 19567682 DOI: 10.1158/0008-5472.CAN-08-3465  0.96
2009 Karlsson AJ, Pomerantz WC, Neilsen KJ, Gellman SH, Palecek SP. Effect of sequence and structural properties on 14-helical beta-peptide activity against Candida albicans planktonic cells and biofilms. Acs Chemical Biology. 4: 567-79. PMID 19518070 DOI: 10.1021/cb900093r  0.96
2009 Müller MM, Windsor MA, Pomerantz WC, Gellman SH, Hilvert D. A rationally designed aldolase foldamer. Angewandte Chemie (International Ed. in English). 48: 922-5. PMID 19090515 DOI: 10.1002/anie.200804996  0.96
2008 Pizzey CL, Pomerantz WC, Sung BJ, Yuwono VM, Gellman SH, Hartgerink JD, Yethiraj A, Abbott NL. Characterization of nanofibers formed by self-assembly of beta-peptide oligomers using small angle x-ray scattering. The Journal of Chemical Physics. 129: 095103. PMID 19044891 DOI: 10.1063/1.2955745  0.96
2008 Vaz E, Pomerantz WC, Geyer M, Gellman SH, Brunsveld L. Comparison of design strategies for promotion of beta-peptide 14-helix stability in water. Chembiochem : a European Journal of Chemical Biology. 9: 2254-9. PMID 18756554 DOI: 10.1002/cbic.200800355  0.96
2008 Pomerantz WC, Grygiel TL, Lai JR, Gellman SH. Distinctive circular dichroism signature for 14-helix-bundle formation by beta-peptides. Organic Letters. 10: 1799-802. PMID 18396884 DOI: 10.1021/ol800622e  0.96
2008 Pomerantz WC, Yuwono VM, Pizzey CL, Hartgerink JD, Abbott NL, Gellman SH. Nanofibers and lyotropic liquid crystals from a class of self-assembling beta-peptides. Angewandte Chemie (International Ed. in English). 47: 1241-4. PMID 18183558 DOI: 10.1002/anie.200704372  0.96
2007 Chi Y, English EP, Pomerantz WC, Horne WS, Joyce LA, Alexander LR, Fleming WS, Hopkins EA, Gellman SH. Practical synthesis of enantiomerically pure beta2-amino acids via proline-catalyzed diastereoselective aminomethylation of aldehydes. Journal of the American Chemical Society. 129: 6050-5. PMID 17439122 DOI: 10.1021/ja070063i  0.96
2007 Lee MR, Raguse TL, Schinnerl M, Pomerantz WC, Wang X, Wipf P, Gellman SH. Origins of the high 14-helix propensity of cyclohexyl-rigidified residues in beta-peptides. Organic Letters. 9: 1801-4. PMID 17394351 DOI: 10.1021/ol070511r  0.96
2007 Pomerantz WC, Cadwell KD, Hsu YJ, Gellman SH, Abbott NL. Sequence dependent behavior of amphiphilic β-peptides on gold surfaces Chemistry of Materials. 19: 4436-4441. DOI: 10.1021/cm070265d  0.96
2006 Karlsson AJ, Pomerantz WC, Weisblum B, Gellman SH, Palecek SP. Antifungal activity from 14-helical beta-peptides. Journal of the American Chemical Society. 128: 12630-1. PMID 17002340 DOI: 10.1021/ja064630y  0.96
2006 Pomerantz WC, Abbott NL, Gellman SH. Lyotropic liquid crystals from designed helical beta-peptides. Journal of the American Chemical Society. 128: 8730-1. PMID 16819857 DOI: 10.1021/ja062412z  0.96
2005 Moonen NN, Pomerantz WC, Gist R, Boudon C, Gisselbrecht JP, Kawai T, Kishioka A, Gross M, Irie M, Diederich F. Donor-substituted cyanoethynylethenes: pi-conjugation and band-gap tuning in strong charge-transfer chromophores. Chemistry (Weinheim An Der Bergstrasse, Germany). 11: 3325-41. PMID 15798969 DOI: 10.1002/chem.200500082  0.96
2002 Koch HF, Pomerantz WC, Ruggles EL, Van Laren M, Van Roon AM. Comparing isotope effects and rates for the methanolic sodium methoxide reactions of 9-r-fluorene to those for p-CF3C6H4CHClR (R = CH2Cl, CH2F and CF3) Collection of Czechoslovak Chemical Communications. 67: 1505-1516. DOI: 10.1135/cccc20021505  0.96
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