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Joseph J. Barchi - Publications

Affiliations: 
National Cancer Institute, Rockville, MD, United States 
Area:
Chemical Biology
Website:
http://ccr.cancer.gov/staff/staff.asp?profileid=6281

43 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2023 Barchi JJ, De Meo C, Mootoo DR. Editorial: Tribute to Professor Bert Fraser-Reid. Carbohydrate Research. 108795. PMID 37002031 DOI: 10.1016/j.carres.2023.108795  0.475
2017 Gibadullin R, Farnsworth DW, Barchi JJ, Gildersleeve JC. GalNAc-Tyrosine Is a Ligand of Plant Lectins, Antibodies, and Human and Murine Macrophage Galactose-Type Lectins. Acs Chemical Biology. PMID 28644609 DOI: 10.1021/Acschembio.7B00471  0.323
2013 Mallajosyula SS, Adams KM, Barchi JJ, MacKerell AD. Conformational determinants of the activity of antiproliferative factor glycopeptide. Journal of Chemical Information and Modeling. 53: 1127-37. PMID 23627670 DOI: 10.1021/Ci400147S  0.336
2012 Zhang Y, Muthana SM, Farnsworth D, Ludek O, Adams K, Barchi JJ, Gildersleeve JC. Enhanced epimerization of glycosylated amino acids during solid-phase peptide synthesis Journal of the American Chemical Society. 134: 6316-6325. PMID 22390544 DOI: 10.1021/Ja212188R  0.321
2011 Johannessen L, Remsberg J, Gaponenko V, Adams KM, Barchi JJ, Tarasov SG, Jiang S, Tarasova NI. Peptide structure stabilization by membrane anchoring and its general applicability to the development of potent cell-permeable inhibitors. Chembiochem : a European Journal of Chemical Biology. 12: 914-21. PMID 21365731 DOI: 10.1002/Cbic.201000563  0.318
2010 Kaczmarek P, Tocci GM, Keay SK, Adams KM, Zhang CO, Koch KR, Grkovic D, Guo L, Michejda CJ, Barchi JJ. Structure-Activity Studies on Antiproliferative Factor (APF) Glycooctapeptide Derivatives. Acs Medicinal Chemistry Letters. 1: 390-4. PMID 24900223 DOI: 10.1021/Ml100087A  0.34
2009 Saavedra JE, Davies KM, Barchi JJ, Keefer LK. Unexpected Incorporation of Bromine at a Non-anomeric Position during the Synthesis of an O-Glycosylated Diazeniumdiolate. Organic Preparations and Procedures International. 41: 143-147. PMID 20354584 DOI: 10.1080/00304940902801968  0.34
2009 Barchi JJ, Kaczmarek P. Short and sweet: Evolution of a small glycopeptide from a bladder disorder to an anticancer lead Molecular Interventions. 9: 14-17. PMID 19299659 DOI: 10.1124/Mi.9.1.5  0.303
2008 Kaczmarek P, Keay SK, Tocci GM, Koch KR, Zhang CO, Barchi JJ, Grkovic D, Guo L, Michejda CJ. Structure-activity relationship studies for the peptide portion of the bladder epithelial cell antiproliferative factor from interstitial cystitis patients Journal of Medicinal Chemistry. 51: 5974-5983. PMID 18788730 DOI: 10.1021/Jm8002763  0.351
2008 Barchi JJ, Karki RG, Nicklaus MC, Siddiqui MA, George C, Mikhailopulo IA, Marquez VE. Comprehensive structural studies of 2′,3′-difluorinated nucleosides: Comparison of theory, solution, and solid state Journal of the American Chemical Society. 130: 9048-9057. PMID 18558684 DOI: 10.1021/Ja800964G  0.322
2008 Garg H, Francella N, Tony KA, Augustine LA, Barchi JJ, Fantini J, Puri A, Mootoo DR, Blumenthal R. Glycoside analogs of β-galactosylceramide, a novel class of small molecule antiviral agents that inhibit HIV-1 entry Antiviral Research. 80: 54-61. PMID 18538869 DOI: 10.1016/J.Antiviral.2008.04.004  0.546
2006 Furrer J, Luy B, Basrur V, Roberts DD, Barchi JJ. Conformational analysis of an α3β1 integrin-binding peptide from thrombospondin-1: Implications for antiangiogenic drug design Journal of Medicinal Chemistry. 49: 6324-6333. PMID 17034138 DOI: 10.1021/Jm060833L  0.328
2006 Deng J, Kelley JA, Barchi JJ, Sanchez T, Dayam R, Pommier Y, Neamati N. Mining the NCI antiviral compounds for HIV-1 integrase inhibitors Bioorganic and Medicinal Chemistry. 14: 3785-3792. PMID 16460953 DOI: 10.1016/J.Bmc.2006.01.040  0.335
2005 Oishi S, Karki RG, Shi ZD, Worthy KM, Bindu L, Chertov O, Esposito D, Frank P, Gillette WK, Maderia M, Hartley J, Nicklaus MC, Barchi JJ, Fisher RJ, Burke TR. Evaluation of macrocyclic Grb2 SH2 domain-binding peptide mimetics prepared by ring-closing metathesis of C-terminal allylglycines with an N-terminal β-vinyl-substituted phosphotyrosyl mimetic Bioorganic and Medicinal Chemistry. 13: 2431-2438. PMID 15755645 DOI: 10.1016/J.Bmc.2005.01.052  0.323
2004 Keay SK, Szekely Z, Conrads TP, Veenstra TD, Barchi JJ, Zhang CO, Koch KR, Michejda CJ. An antiproliferative factor from interstitial cystitis patients is a frizzled 8 protein-related sialoglycopeptide Proceedings of the National Academy of Sciences of the United States of America. 101: 11803-11808. PMID 15282374 DOI: 10.1073/Pnas.0404509101  0.303
2004 Marquez VE, Ben-Kasus T, Barchi JJ, Green KM, Nicklaus MC, Agbaria R. Experimental and Structural Evidence that Herpes 1 Kinase and Cellular DNA Polymerase(s) Discriminate on the Basis of Sugar Pucker Journal of the American Chemical Society. 126: 543-549. PMID 14719951 DOI: 10.1021/Ja037929E  0.311
2003 Svarovsky SA, Barchi JJ. Highly efficient preparation of tumor antigen-containing glycopeptide building blocks from novel pentenyl glycosides Carbohydrate Research. 338: 1925-1935. PMID 14499569 DOI: 10.1016/S0008-6215(03)00323-9  0.304
2003 Choi Y, George C, Comin MJ, Barchi JJ, Kim HS, Jacobson KA, Balzarini J, Mitsuya H, Boyer PL, Hughes SH, Marquez VE. A conformationally locked analogue of the anti-HIV agent stavudine. An important correlation between pseudorotation and maximum amplitude. Journal of Medicinal Chemistry. 46: 3292-9. PMID 12852759 DOI: 10.1021/Jm030116G  0.311
2002 Nacro K, Lee J, Barchi JJ, Lewin NE, Blumberg PM, Marquez VE. Conformationally constrained analogues of diacylglycerol (DAG). Part 19: Asymmetric syntheses of (3R)- and (3S)-3-hydroxy-4,4-disubstituted heptono-1,4-lactones as protein kinase C (PK-C) ligands with increased hydrophilicity Tetrahedron. 58: 5335-5345. DOI: 10.1016/S0040-4020(02)00477-5  0.307
2000 Chen IJ, Neamati N, Nicklaus MC, Orr A, Anderson L, Barchi JJ, Kelley JA, Pommier Y, MacKerell AD. Identification of HIV-1 integrase inhibitors via three-dimensional database searching using ASV and HIV-1 integrases as targets. Bioorganic & Medicinal Chemistry. 8: 2385-98. PMID 11058033 DOI: 10.1016/S0968-0896(00)00180-2  0.313
2000 Mu L, Sarafianos SG, Nicklaus MC, Russ P, Siddiqui MA, Ford J, Mitsuya H, Le R, Kodama E, Meier C, Knispel T, Anderson L, Barchi JJ, Marquez VE. Interactions of conformationally biased north and south 2'-fluoro-2',3'-dideoxynucleoside 5'-triphosphates with the active site of HIV-1 reverse transcriptase Biochemistry. 39: 11205-11215. PMID 10985766 DOI: 10.1021/Bi001090N  0.308
2000 Ford H, Dai F, Mu L, Siddiqui MA, Nicklaus MC, Anderson L, Marquez VE, Barchi JJ. Adenosine deaminase prefers a distinct sugar ring conformation for binding and catalysis: Kinetic and structural studies Biochemistry. 39: 2581-2592. PMID 10704207 DOI: 10.1021/Bi992112C  0.319
1998 Sharma P, Barchi JJ, Huang X, Amin ND, Jaffe H, Pant HC. Site-specific phosphorylation of Lys-Ser-Pro repeat peptides from neurofilament H by cyclin-dependent kinase 5: structural basis for substrate recognition. Biochemistry. 37: 4759-66. PMID 9537991 DOI: 10.1021/Bi972746O  0.315
1998 Marquez VE, Ezzitouni A, Russ P, Siddiqui MA, Ford H, Feldman RJ, Mitsuya H, George C, Barchi JJ. HIV-1 reverse transcriptase can discriminate between two conformationally locked carbocyclic AZT triphosphate analogues Journal of the American Chemical Society. 120: 2780-2789. DOI: 10.1021/Ja973535+  0.326
1997 Huang X, Barchi JJ, Lung FDT, Roller PP, Nara PL, Muschik J, Garrity RR. Glycosylation affects both the three-dimensional structure and antibody binding properties of the HIV-1(IIIB) GP120 peptide RP135 Biochemistry. 36: 10846-10856. PMID 9312273 DOI: 10.1021/Bi9703655  0.35
1997 Barchi JJ, Jeong LS, Siddiqui MA, Marquez VE. Conformational analysis of the complete series of 2' and 3' monofluorinated dideoxyuridines Journal of Biochemical and Biophysical Methods. 34: 11-29. PMID 9089381 DOI: 10.1016/S0165-022X(96)00032-2  0.301
1997 Buolamwini JK, Barchi JJ. Solution NMR conformational analysis of the potent equilibrative sensitive (ES) nucleoside transporter inhibitor, S6-(4- nitrobenzyl)mercaptopurine riboside (NBMPR) Nucleosides and Nucleotides. 16: 2101-2110. DOI: 10.1080/07328319708002561  0.323
1996 Huang X, Smith MC, Berzofsky JA, Barchi JJ. Structural comparison of a 15 residue peptide from the V3 loop of HIV-1(IIIB) and an O-glycosylated analogue Febs Letters. 393: 280-286. PMID 8814305 DOI: 10.1016/0014-5793(96)00912-X  0.334
1996 Barchi JJ, Nomizu M, Otaka A, Roller PP, Burke TR. Conformational analysis of cyclic hexapeptides designed as constrained ligands for the SH2 domain of the p85 subunit of phosphatidylinositol-3-OH kinase Biopolymers. 38: 191-208. PMID 8589253 DOI: 10.1002/(Sici)1097-0282(199602)38:2<191::Aid-Bip6>3.0.Co;2-Q  0.352
1995 Kazanietz MG, Barchi JJ, Omichinski JG, Blumberg PM. Low affinity binding of phorbol esters to protein kinase C and its recombinant cysteine-rich region in the absence of phospholipids Journal of Biological Chemistry. 270: 14679-14684. PMID 7782331 DOI: 10.1074/Jbc.270.24.14679  0.304
1995 Burke TR, Barchi JJ, George C, Wolf G, Shoelson SE, Yan X. Conformationally constrained phosphotyrosyl mimetics designed as monomeric Src homology 2 domain inhibitors. Journal of Medicinal Chemistry. 38: 1386-96. PMID 7537333 DOI: 10.1021/Jm00008A017  0.314
1994 Rodriguez JB, Marquez VE, Nicklaus MC, Mitsuya H, Barchi JJ. Conformationally locked nucleoside analogues. Synthesis of dideoxycarbocyclic nucleoside analogues structurally related to neplanocin C Journal of Medicinal Chemistry. 37: 3389-3399. PMID 7932567 DOI: 10.1021/Jm00046A024  0.383
1994 Gharehbaghi K, Paull KD, Kelley JA, Barchi JJ, Marquez VE, Cooney DA, Monks A, Scudiero D, Krohn K, Jayaram HN. Cytotoxicity and characterization of an active metabolite of benzamide riboside, a novel inhibitor of IMP dehydrogenase International Journal of Cancer. 56: 892-899. PMID 7907081 DOI: 10.1002/Ijc.2910560623  0.302
1994 Siddiqui MA, Marquez VE, Driscoll JS, Barchi JJ. A diastereoselective synthesis of (S,S)-α-fluoro-2,2-dimethyl-1,3-dioxolane-4-propanoic acid methyl ester, a key intermediate for the preparation of anti-HIV effective fluorodideoxynucleosides Tetrahedron Letters. 35: 3263-3266. DOI: 10.1016/S0040-4039(00)76880-8  0.302
1993 Bodenteich M, Marquez VE, Barchi JJ, Hallows WH, Goldstein BM, Driscoll JS. Synthesis of carbocyclic analogs of 1-.beta.-D-psicofuranosyl nucleosides. psico-Cyclopentenyladenosine (psicoplanocin A) and psico-cyclopentenylcytosine Journal of Organic Chemistry. 58: 6009-6015. DOI: 10.1021/Jo00074A030  0.312
1993 Rodriguez JB, Marquez VE, Nicklaus MC, Barchi JJ. Synthesis of cyclopropane-fused dideoxycarbocyclic nucleosides structurally related to neplanocin C Tetrahedron Letters. 34: 6233-6236. DOI: 10.1016/S0040-4039(00)73718-X  0.326
1992 Siddiqui MA, Driscoll JS, Marquez VE, Roth JS, Shirasaka T, Mitsuya H, Barchi JJ, Kelley JA. Chemistry and anti-HIV properties of 2′-fluoro-2′,3′-dideoxyarabinofuranosylpyrimidines Journal of Medicinal Chemistry. 35: 2195-2201. PMID 1351945 DOI: 10.1021/Jm00090A008  0.322
1991 Barchi JJ, Marquez VE, Driscoll JS, Ford H, Mitsuya H, Shirasaka T, Aoki S, Kelley JA. Potential anti-AIDS drugs. Lipophilic, adenosine deaminase-activated prodrugs. Journal of Medicinal Chemistry. 34: 1647-55. PMID 2033591 DOI: 10.1021/Jm00109A018  0.316
1985 Moore RE, Barchi JJ, Bartolini G. Use of borate complexation in assigning relative stereochemistry of acyclic polyhydroxylated compounds Journal of Organic Chemistry. 50: 374-379. DOI: 10.1021/Jo00203A017  0.395
1985 Ainslie RD, Barchi JJ, Kuniyoshi M, Moore RE, Mynderse JS. Structure of malyngamide C Journal of Organic Chemistry. 50: 2859-2862. DOI: 10.1002/Chin.198551327  0.413
1984 Barchi JJ, Moore RE, Patterson GML. Acutiphycin and 20,21-didehydroacutiphycin, new antineoplastic agents from the cyanophyte Oscillatoria acutissima Journal of the American Chemical Society. 106: 8193-8197. DOI: 10.1021/Ja00338A031  0.383
1982 Moore R, Bartolini G, Barchi J, Bothner-By A, Dadok J, Ford J. Additions & Corrections: Absolute Stereochemistry of Palytoxin Journal of the American Chemical Society. 104: 5572-5572. DOI: 10.1021/Ja00384A600  0.33
1982 Moore RE, Bartolini G, Barchi J, Bothner-By AA, Dadok J, Ford J. Absolute stereochemistry of palytoxin Journal of the American Chemical Society. 104: 3776-3779. DOI: 10.1021/Ja00377A064  0.345
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