Benita S. Katzenellenbogen - Publications

Affiliations: 
University of Illinois, Urbana-Champaign, Urbana-Champaign, IL 
Area:
Cell Biology, Molecular Biology, Biochemistry

285 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2018 Sharma A, Toy W, Guillen VS, Sharma N, Min J, Carlson KE, Mayne CG, Lin S, Sabio M, Greene G, Katzenellenbogen BS, Chandarlapaty S, Katzenellenbogen JA. Antagonists for Constitutively Active Mutant Estrogen Receptors: Insights into the Roles of Antiestrogen-Core and Side-Chain. Acs Chemical Biology. PMID 30404440 DOI: 10.1021/acschembio.8b00877  0.56
2018 Selvaraj UM, Zuurbier K, Whoolery C, Plautz EJ, Chambliss KL, Kong X, Zhang S, Kim SH, Katzenellenbogen BS, Katzenellenbogen JA, Mineo C, Shaul PW, Stowe AM. Selective Non-nuclear Estrogen Receptor Activation Decreases Stroke Severity and Promotes Functional Recovery in Female Mice. Endocrinology. PMID 30256928 DOI: 10.1210/en.2018-00600  0.56
2018 Katzenellenbogen JA, Mayne CG, Katzenellenbogen BS, Greene GL, Chandarlapaty S. Publisher Correction: Structural underpinnings of oestrogen receptor mutations in endocrine therapy resistance. Nature Reviews. Cancer. PMID 30185950 DOI: 10.1038/s41568-018-0053-0  0.56
2018 Wang L, Guillen VS, Sharma N, Flessa K, Min J, Carlson KE, Toy W, Braqi S, Katzenellenbogen BS, Katzenellenbogen JA, Chandarlapaty S, Sharma A. New Class of Selective Estrogen Receptor Degraders (SERDs): Expanding the Toolbox of PROTAC Degrons. Acs Medicinal Chemistry Letters. 9: 803-808. PMID 30128071 DOI: 10.1021/acsmedchemlett.8b00106  0.56
2018 Guivarc'h E, Buscato M, Guihot AL, Favre J, Vessières E, Grimaud L, Wakim J, Melhem NJ, Zahreddine R, Adlanmerini M, Loufrani L, Knauf C, Katzenellenbogen JA, Katzenellenbogen BS, Foidart JM, et al. Predominant Role of Nuclear Versus Membrane Estrogen Receptor α in Arterial Protection: Implications for Estrogen Receptor α Modulation in Cardiovascular Prevention/Safety. Journal of the American Heart Association. 7. PMID 29959137 DOI: 10.1161/JAHA.118.008950  0.56
2018 Katzenellenbogen JA, Mayne CG, Katzenellenbogen BS, Greene GL, Chandarlapaty S. Structural underpinnings of oestrogen receptor mutations in endocrine therapy resistance. Nature Reviews. Cancer. PMID 29662238 DOI: 10.1038/s41568-018-0001-z  0.56
2018 Vinel A, Coudert AE, Buscato M, Valera MC, Agnès O, Katzenellenbogen JA, Katzenellenbogen BS, Berdal A, Babajko S, Arnal JF, Fontaine C. Respective role of membrane and nuclear estrogen receptor (ER) α in the mandible of growing mice: implications for ERα modulation. Journal of Bone and Mineral Research : the Official Journal of the American Society For Bone and Mineral Research. PMID 29624728 DOI: 10.1002/jbmr.3434  0.56
2018 Miranda CL, Johnson LA, de Montgolfier O, Elias VD, Ullrich LS, Hay JJ, Paraiso IL, Choi J, Reed RL, Revel JS, Kioussi C, Bobe G, Iwaniec UT, Turner RT, Katzenellenbogen BS, et al. Non-estrogenic Xanthohumol Derivatives Mitigate Insulin Resistance and Cognitive Impairment in High-Fat Diet-induced Obese Mice. Scientific Reports. 8: 613. PMID 29330372 DOI: 10.1038/s41598-017-18992-6  0.56
2017 Katzenellenbogen BS, Zhao Y, Laws MJ, Sanabria Guillen V, Ziegler Y, Min J, Sharma A, Kim SH, Chu D, Park BH, Oesterreich S, Mao C, Shapiro DJ, Nettles KW, Katzenellenbogen JA. Structurally novel antiestrogens elicit differential responses from constitutively active mutant estrogen receptors in breast cancer cells and tumors. Cancer Research. PMID 28904064 DOI: 10.1158/0008-5472.CAN-17-1265  0.56
2017 Min J, Guillen VS, Sharma A, Zhao Y, Ziegler Y, Gong P, Mayne CG, Srinivasan S, Kim SH, Carlson KE, Nettles KW, Katzenellenbogen BS, Katzenellenbogen JA. Adamantyl Antiestrogens with Novel Side Chains Reveal a Spectrum of Activities in Suppressing Estrogen Receptor (ER)-Mediated Activities in Breast Cancer Cells. Journal of Medicinal Chemistry. PMID 28657320 DOI: 10.1021/acs.jmedchem.7b00585  0.56
2017 Lu W, Katzenellenbogen BS. Estrogen Receptor-β Modulation of the ERα-p53 Loop Regulating Gene Expression, Proliferation, and Apoptosis in Breast Cancer. Hormones & Cancer. PMID 28577282 DOI: 10.1007/s12672-017-0298-1  0.32
2017 Srinivasan S, Nwachukwu JC, Bruno NE, Dharmarajan V, Goswami D, Kastrati I, Novick S, Nowak J, Cavett V, Zhou HB, Boonmuen N, Zhao Y, Min J, Frasor J, Katzenellenbogen BS, et al. Corrigendum: Full antagonism of the estrogen receptor without a prototypical ligand side chain. Nature Chemical Biology. 13: 691. PMID 28514424 DOI: 10.1038/nchembio0617-691c  0.56
2017 Srinivasan S, Nwachukwu JC, Bruno NE, Dharmarajan V, Goswami D, Kastrati I, Novick S, Nowak J, Cavett V, Zhou HB, Boonmuen N, Zhao Y, Min J, Frasor J, Katzenellenbogen BS, et al. Erratum: Full antagonism of the estrogen receptor without a prototypical ligand side chain. Nature Chemical Biology. 13: 691. PMID 28514419 DOI: 10.1038/nchembio0617-691b  0.56
2017 Menazza S, Sun J, Appachi S, Chambliss KL, Kim SH, Aponte A, Khan S, Katzenellenbogen JA, Katzenellenbogen BS, Shaul PW, Murphy E. Non-nuclear estrogen receptor alpha activation in endothelium reduces cardiac ischemia-reperfusion injury in mice. Journal of Molecular and Cellular Cardiology. PMID 28457941 DOI: 10.1016/j.yjmcc.2017.04.004  0.56
2017 Madak-Erdogan Z, Charn TH, Jiang Y, Liu ET, Katzenellenbogen JA, Katzenellenbogen BS. Integrative genomics of gene and metabolic regulation by estrogen receptors α and β, and their coregulators. Molecular Systems Biology. 13: 929. PMID 28442489  0.56
2017 Christenson JL, Butterfield KT, Spoelstra NS, Norris JD, Josan JS, Pollock JA, McDonnell DP, Katzenellenbogen BS, Katzenellenbogen JA, Richer JK. MMTV-PyMT and Derived Met-1 Mouse Mammary Tumor Cells as Models for Studying the Role of the Androgen Receptor in Triple-Negative Breast Cancer Progression. Hormones & Cancer. PMID 28194662 DOI: 10.1007/s12672-017-0285-6  0.56
2016 Srinivasan S, Nwachukwu JC, Bruno NE, Dharmarajan V, Goswami D, Kastrati I, Novick S, Nowak J, Cavett V, Zhou HB, Boonmuen N, Zhao Y, Min J, Frasor J, Katzenellenbogen BS, et al. Full antagonism of the estrogen receptor without a prototypical ligand side chain. Nature Chemical Biology. PMID 27870835 DOI: 10.1038/nchembio.2236  0.56
2016 Chambliss KL, Barrera J, Umetani M, Umetani J, Kim SH, Madak-Erdogan Z, Huang L, Katzenellenbogen BS, Katzenellenbogen JA, Mineo C, Shaul PW. Non-Nuclear Estrogen Receptor Activation Improves Hepatic Steatosis in Female Mice. Endocrinology. en20151629. PMID 27552247 DOI: 10.1210/en.2015-1629  0.56
2016 Gong P, Madak-Erdogan Z, Flaws JA, Shapiro DJ, Katzenellenbogen JA, Katzenellenbogen BS. Estrogen receptor-α and aryl hydrocarbon receptor involvement in the actions of botanical estrogens in target cells. Molecular and Cellular Endocrinology. PMID 27543265 DOI: 10.1016/j.mce.2016.08.025  0.64
2016 Madak-Erdogan Z, Kim SH, Gong P, Zhao YC, Zhang H, Chambliss KL, Carlson KE, Mayne CG, Shaul PW, Korach KS, Katzenellenbogen JA, Katzenellenbogen BS. Design of pathway preferential estrogens that provide beneficial metabolic and vascular effects without stimulating reproductive tissues. Science Signaling. 9: ra53. PMID 27221711 DOI: 10.1126/scisignal.aad8170  0.64
2016 Katzenellenbogen BS, Katzenellenbogen JA, Madak-Erdogan Z, VanHook AM. Science Signaling podcast for 24 May 2016: Designer estrogens. Science Signaling. 9: pc12. PMID 27221709 DOI: 10.1126/scisignal.aag1040  0.56
2016 Bhatt S, Stender JD, Joshi S, Wu G, Katzenellenbogen BS. OCT-4: a novel estrogen receptor-α collaborator that promotes tamoxifen resistance in breast cancer cells. Oncogene. PMID 27065334 DOI: 10.1038/onc.2016.105  0.56
2016 Fanning SW, Mayne CG, Dharmarajan V, Carlson KE, Martin TA, Novick SJ, Toy W, Green B, Panchamukhi S, Katzenellenbogen BS, Tajkhorshid E, Griffin PR, Shen Y, Chandarlapaty S, Katzenellenbogen JA, et al. Estrogen receptor alpha somatic mutations Y537S and D538G confer breast cancer endocrine resistance by stabilizing the activating function-2 binding conformation. Elife. 5. PMID 26836308 DOI: 10.7554/eLife.12792  0.56
2015 Madak-Erdogan Z, Gong P, Katzenellenbogen BS. Differential Utilization of Nuclear and Extranuclear Receptor Signaling Pathways in the Actions of Estrogens, SERMs, and a Tissue-Selective Estrogen Complex (TSEC). The Journal of Steroid Biochemistry and Molecular Biology. PMID 26689478 DOI: 10.1016/j.jsbmb.2015.12.008  0.64
2015 Aumsuwan P, Khan SI, Khan IA, Ali Z, Avula B, Walker LA, Shariat-Madar Z, Helferich WG, Katzenellenbogen BS, Dasmahapatra AK. The anticancer potential of steroidal saponin, dioscin, isolated from wild yam (Dioscorea villosa) root extract in invasive human breast cancer cell line MDA-MB-231 in vitro. Archives of Biochemistry and Biophysics. PMID 26682631 DOI: 10.1016/j.abb.2015.12.001  0.32
2015 Zhao Y, Chen Y, Kuang Y, Bagchi MK, Taylor RN, Katzenellenbogen JA, Katzenellenbogen BS. Multiple Beneficial Roles of Repressor of Estrogen Receptor Activity (REA) in Suppressing the Progression of Endometriosis. Endocrinology. en20151324. PMID 26653759 DOI: 10.1210/en.2015-1324  0.64
2015 Boonmuen N, Gong P, Ali Z, Chittiboyina AG, Khan I, Doerge DR, Helferich WG, Carlson KE, Martin T, Piyachaturawat P, Katzenellenbogen JA, Katzenellenbogen BS. Licorice Root Components in Dietary Supplements are Selective Estrogen Receptor Modulators with a Spectrum of Estrogenic and Anti-Estrogenic Activities. Steroids. PMID 26631549 DOI: 10.1016/j.steroids.2015.11.006  0.64
2015 Madak-Erdogan Z, Gong P, Zhao YC, Xu L, Wrobel KU, Hartman JA, Wang M, Cam A, Iwaniec UT, Turner RT, Twaddle NC, Doerge DR, Khan IA, Katzenellenbogen JA, Katzenellenbogen BS, et al. Dietary licorice root supplementation reduces diet-induced weight gain, lipid deposition, and hepatic steatosis in ovariectomized mice without stimulating reproductive tissues and mammary gland. Molecular Nutrition & Food Research. PMID 26555669 DOI: 10.1002/mnfr.201500445  0.56
2015 Smirnova NF, Fontaine C, Buscato M, Lupieri A, Vinel A, Valera MC, Guillaume M, Malet N, Foidart JM, Raymond-Letron I, Lenfant F, Gourdy P, Katzenellenbogen BS, Katzenellenbogen JA, Laffargue M, et al. The Activation Function-1 of Estrogen Receptor Alpha Prevents Arterial Neointima Development Through a Direct Effect on Smooth Muscle Cells. Circulation Research. 117: 770-8. PMID 26316608 DOI: 10.1161/CIRCRESAHA.115.306416  0.56
2015 Valéra MC, Fontaine C, Lenfant F, Cabou C, Guillaume M, Smirnova N, Kim SH, Chambon P, Katzenellenbogen JA, Katzenellenbogen BS, Payrastre B, Arnal JF. Protective Hematopoietic Effect of Estrogens in a Mouse Model of Thrombosis: Respective Roles of Nuclear Versus Membrane Estrogen Receptor α. Endocrinology. 156: 4293-301. PMID 26280130 DOI: 10.1210/en.2015-1522  0.56
2015 Kim SH, Madak-Erdogan Z, Bae SC, Carlson KE, Mayne CG, Granick S, Katzenellenbogen BS, Katzenellenbogen JA. Ligand Accessibility and Bioactivity of a Hormone-Dendrimer Conjugate Depend on pH and pH History. Journal of the American Chemical Society. PMID 26186415 DOI: 10.1021/jacs.5b05952  0.56
2015 Zhao Y, Gong P, Chen Y, Nwachukwu JC, Srinivasan S, Ko C, Bagchi MK, Taylor RN, Korach KS, Nettles KW, Katzenellenbogen JA, Katzenellenbogen BS. Dual suppression of estrogenic and inflammatory activities for targeting of endometriosis. Science Translational Medicine. 7: 271ra9. PMID 25609169 DOI: 10.1126/scitranslmed.3010626  0.64
2015 Paterni I, Bertini S, Granchi C, Tuccinardi T, Macchia M, Martinelli A, Caligiuri I, Toffoli G, Rizzolio F, Carlson KE, Katzenellenbogen BS, Katzenellenbogen JA, Minutolo F. Highly selective salicylketoxime-based estrogen receptor β agonists display antiproliferative activities in a glioma model. Journal of Medicinal Chemistry. 58: 1184-94. PMID 25559213 DOI: 10.1021/jm501829f  0.64
2015 Aumsuwan P, Khan SI, Khan IA, Avula B, Walker LA, Helferich WG, Katzenellenbogen BS, Dasmahapatra AK. Evaluation of wild yam (Dioscorea villosa) root extract as a potential epigenetic agent in breast cancer cells. In Vitro Cellular & Developmental Biology. Animal. 51: 59-71. PMID 25148825 DOI: 10.1007/s11626-014-9807-5  0.64
2014 Gong P, Madak-Erdogan Z, Li J, Cheng J, Greenlief CM, Helferich W, Katzenellenbogen JA, Katzenellenbogen BS. Transcriptomic analysis identifies gene networks regulated by estrogen receptor α (ERα) and ERβ that control distinct effects of different botanical estrogens. Nuclear Receptor Signaling. 12: e001. PMID 25363786 DOI: 10.1621/nrs.12001  0.56
2014 Abot A, Fontaine C, Buscato M, Solinhac R, Flouriot G, Fabre A, Drougard A, Rajan S, Laine M, Milon A, Muller I, Henrion D, Adlanmerini M, Valéra MC, Gompel A, ... ... Katzenellenbogen BS, et al. The uterine and vascular actions of estetrol delineate a distinctive profile of estrogen receptor α modulation, uncoupling nuclear and membrane activation. Embo Molecular Medicine. 6: 1328-46. PMID 25214462 DOI: 10.15252/emmm.201404112  0.64
2014 Bergamaschi A, Madak-Erdogan Z, Kim YJ, Choi YL, Lu H, Katzenellenbogen BS. The forkhead transcription factor FOXM1 promotes endocrine resistance and invasiveness in estrogen receptor-positive breast cancer by expansion of stem-like cancer cells. Breast Cancer Research : Bcr. 16: 436. PMID 25213081 DOI: 10.1186/s13058-014-0436-4  0.52
2014 Holton SE, Bergamaschi A, Katzenellenbogen BS, Bhargava R. Integration of molecular profiling and chemical imaging to elucidate fibroblast-microenvironment impact on cancer cell phenotype and endocrine resistance in breast cancer. Plos One. 9: e96878. PMID 24816718 DOI: 10.1371/journal.pone.0096878  0.64
2014 Mir M, Bergamaschi A, Katzenellenbogen BS, Popescu G. Highly sensitive quantitative imaging for monitoring single cancer cell growth kinetics and drug response. Plos One. 9: e89000. PMID 24558461 DOI: 10.1371/journal.pone.0089000  0.64
2014 Madak-Erdogan Z, Ventrella R, Petry L, Katzenellenbogen BS. Novel roles for ERK5 and cofilin as critical mediators linking ERα-driven transcription, actin reorganization, and invasiveness in breast cancer. Molecular Cancer Research : McR. 12: 714-27. PMID 24505128 DOI: 10.1158/1541-7786.MCR-13-0588  0.52
2014 Clark S, Rainville J, Zhao X, Katzenellenbogen BS, Pfaff D, Vasudevan N. Estrogen receptor-mediated transcription involves the activation of multiple kinase pathways in neuroblastoma cells Journal of Steroid Biochemistry and Molecular Biology. 139: 45-53. PMID 24121066 DOI: 10.1016/j.jsbmb.2013.09.010  0.64
2013 Jiang Y, Gong P, Madak-Erdogan Z, Martin T, Jeyakumar M, Carlson K, Khan I, Smillie TJ, Chittiboyina AG, Rotte SC, Helferich WG, Katzenellenbogen JA, Katzenellenbogen BS. Mechanisms enforcing the estrogen receptor β selectivity of botanical estrogens. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 27: 4406-18. PMID 23882126 DOI: 10.1096/fj.13-234617  0.64
2013 Madak-Erdogan Z, Charn TH, Jiang Y, Liu ET, Katzenellenbogen JA, Katzenellenbogen BS. Integrative genomics of gene and metabolic regulation by estrogen receptors α and β, and their coregulators. Molecular Systems Biology. 9: 676. PMID 23774759 DOI: 10.1038/msb.2013.28  0.64
2013 Bartell SM, Han L, Kim HN, Kim SH, Katzenellenbogen JA, Katzenellenbogen BS, Chambliss KL, Shaul PW, Roberson PK, Weinstein RS, Jilka RL, Almeida M, Manolagas SC. Non-nuclear-initiated actions of the estrogen receptor protect cortical bone mass. Molecular Endocrinology (Baltimore, Md.). 27: 649-56. PMID 23443267 DOI: 10.1210/me.2012-1368  0.64
2013 Bergamaschi A, Frasor J, Borgen K, Stanculescu A, Johnson P, Rowland K, Wiley EL, Katzenellenbogen BS. 14-3-3ζ as a predictor of early time to recurrence and distant metastasis in hormone receptor-positive and -negative breast cancers. Breast Cancer Research and Treatment. 137: 689-96. PMID 23271328 DOI: 10.1007/s10549-012-2390-0  0.64
2013 Kim K, Madak-Erdogan Z, Ventrella R, Katzenellenbogen BS. A MicroRNA196a2* and TP63 circuit regulated by estrogen receptor-α and ERK2 that controls breast cancer proliferation and invasiveness properties. Hormones & Cancer. 4: 78-91. PMID 23250869 DOI: 10.1007/s12672-012-0129-3  0.52
2012 Park S, Yoon S, Zhao Y, Park SE, Liao L, Xu J, Lydon JP, DeMayo FJ, O'Malley BW, Bagchi MK, Katzenellenbogen BS. Uterine development and fertility are dependent on gene dosage of the nuclear receptor coregulator REA. Endocrinology. 153: 3982-94. PMID 22585830 DOI: 10.1210/en.2012-1044  0.32
2012 Bhatt S, Xiao Z, Meng Z, Katzenellenbogen BS. Phosphorylation by p38 mitogen-activated protein kinase promotes estrogen receptor α turnover and functional activity via the SCF(Skp2) proteasomal complex. Molecular and Cellular Biology. 32: 1928-43. PMID 22431515 DOI: 10.1128/MCB.06561-11  0.64
2012 Madak-Erdogan Z, Katzenellenbogen BS. Aryl hydrocarbon receptor modulation of estrogen receptor α-mediated gene regulation by a multimeric chromatin complex involving the two receptors and the coregulator RIP140. Toxicological Sciences : An Official Journal of the Society of Toxicology. 125: 401-11. PMID 22071320 DOI: 10.1093/toxsci/kfr300  0.64
2012 Stossi F, Madak-Erdoǧan Z, Katzenellenbogen BS. Macrophage-elicited loss of estrogen receptor-α in breast cancer cells via involvement of MAPK and c-Jun at the ESR1 genomic locus Oncogene. 31: 1825-1834. PMID 21860415 DOI: 10.1038/onc.2011.370  0.64
2012 Bergamaschi A, Katzenellenbogen BS. Tamoxifen downregulation of miR-451 increases 14-3-3ζ and promotes breast cancer cell survival and endocrine resistance Oncogene. 31: 39-47. PMID 21666713 DOI: 10.1038/onc.2011.223  0.64
2011 Stender JD, Stossi F, Funk CC, Charn TH, Barnett DH, Katzenellenbogen BS. The estrogen-regulated transcription factor PITX1 coordinates gene-specific regulation by estrogen receptor-alpha in breast cancer cells. Molecular Endocrinology (Baltimore, Md.). 25: 1699-709. PMID 21868451 DOI: 10.1210/me.2011-0102  0.64
2011 Bergamaschi A, Christensen BL, Katzenellenbogen BS. Reversal of endocrine resistance in breast cancer: interrelationships among 14-3-3ζ, FOXM1, and a gene signature associated with mitosis. Breast Cancer Research : Bcr. 13: R70. PMID 21707964 DOI: 10.1186/bcr2913  0.64
2011 Madak-Erdogan Z, Lupien M, Stossi F, Brown M, Katzenellenbogen BS. Genomic collaboration of estrogen receptor alpha and extracellular signal-regulated kinase 2 in regulating gene and proliferation programs. Molecular and Cellular Biology. 31: 226-36. PMID 20956553 DOI: 10.1128/MCB.00821-10  0.52
2011 Minutolo F, Macchia M, Katzenellenbogen BS, Katzenellenbogen JA. Estrogen receptor β ligands: recent advances and biomedical applications. Medicinal Research Reviews. 31: 364-442. PMID 19967775 DOI: 10.1002/med.20186  0.64
2010 Santollo J, Katzenellenbogen BS, Katzenellenbogen JA, Eckel LA. Activation of ERα is necessary for estradiol's anorexigenic effect in female rats. Hormones and Behavior. 58: 872-7. PMID 20807534 DOI: 10.1016/j.yhbeh.2010.08.012  0.64
2010 Wong WP, Tiano JP, Liu S, Hewitt SC, Le May C, Dalle S, Katzenellenbogen JA, Katzenellenbogen BS, Korach KS, Mauvais-Jarvis F. Extranuclear estrogen receptor-alpha stimulates NeuroD1 binding to the insulin promoter and favors insulin synthesis. Proceedings of the National Academy of Sciences of the United States of America. 107: 13057-62. PMID 20616010 DOI: 10.1073/pnas.0914501107  0.64
2010 Chambliss KL, Wu Q, Oltmann S, Konaniah ES, Umetani M, Korach KS, Thomas GD, Mineo C, Yuhanna IS, Kim SH, Madak-Erdogan Z, Maggi A, Dineen SP, Roland CL, Hui DY, ... ... Katzenellenbogen BS, et al. Non-nuclear estrogen receptor alpha signaling promotes cardiovascular protection but not uterine or breast cancer growth in mice. The Journal of Clinical Investigation. 120: 2319-30. PMID 20577047 DOI: 10.1172/JCI38291  0.64
2010 Stender JD, Kim K, Charn TH, Komm B, Chang KC, Kraus WL, Benner C, Glass CK, Katzenellenbogen BS. Genome-wide analysis of estrogen receptor alpha DNA binding and tethering mechanisms identifies Runx1 as a novel tethering factor in receptor-mediated transcriptional activation. Molecular and Cellular Biology. 30: 3943-55. PMID 20547749 DOI: 10.1128/MCB.00118-10  0.64
2010 Kieser KJ, Kim DW, Carlson KE, Katzenellenbogen BS, Katzenellenbogen JA. Characterization of the pharmacophore properties of novel selective estrogen receptor downregulators (SERDs). Journal of Medicinal Chemistry. 53: 3320-9. PMID 20334372 DOI: 10.1021/jm100047k  0.64
2010 Charn TH, Liu ET, Chang EC, Lee YK, Katzenellenbogen JA, Katzenellenbogen BS. Genome-wide dynamics of chromatin binding of estrogen receptors alpha and beta: mutual restriction and competitive site selection. Molecular Endocrinology (Baltimore, Md.). 24: 47-59. PMID 19897598 DOI: 10.1210/me.2009-0252  0.64
2009 Waibel M, Kieser KJ, Carlson KE, Stossi F, Katzenellenbogen BS, Katzenellenbogen JA. Phenethyl pyridines with non-polar internal substituents as selective ligands for estrogen receptor beta. European Journal of Medicinal Chemistry. 44: 3560-70. PMID 19394116 DOI: 10.1016/j.ejmech.2009.03.013  0.64
2009 Waibel M, De Angelis M, Stossi F, Kieser KJ, Carlson KE, Katzenellenbogen BS, Katzenellenbogen JA. Bibenzyl- and stilbene-core compounds with non-polar linker atom substituents as selective ligands for estrogen receptor beta. European Journal of Medicinal Chemistry. 44: 3412-24. PMID 19286283 DOI: 10.1016/j.ejmech.2009.02.006  0.64
2009 Stossi F, Madak-Erdogan Z, Katzenellenbogen BS. Estrogen receptor alpha represses transcription of early target genes via p300 and CtBP1. Molecular and Cellular Biology. 29: 1749-59. PMID 19188451 DOI: 10.1128/MCB.01476-08  0.64
2009 Achari Y, Lu T, Katzenellenbogen BS, Hart DA. Distinct roles for AF-1 and -2 of ER-alpha in regulation of MMP-13 promoter activity. Biochimica Et Biophysica Acta. 1792: 211-20. PMID 19185056 DOI: 10.1016/j.bbadis.2009.01.002  0.64
2009 Zhou HB, Carlson KE, Stossi F, Katzenellenbogen BS, Katzenellenbogen JA. Analogs of methyl-piperidinopyrazole (MPP): antiestrogens with estrogen receptor alpha selective activity. Bioorganic & Medicinal Chemistry Letters. 19: 108-10. PMID 19014882 DOI: 10.1016/j.bmcl.2008.11.006  0.64
2009 Sengupta S, Schiff R, Katzenellenbogen BS. Post-transcriptional regulation of chemokine receptor CXCR4 by estrogen in HER2 overexpressing, estrogen receptor-positive breast cancer cells. Breast Cancer Research and Treatment. 117: 243-51. PMID 18807177 DOI: 10.1007/s10549-008-0186-z  0.64
2008 Sheng S, Barnett DH, Katzenellenbogen BS. Differential estradiol and selective estrogen receptor modulator (SERM) regulation of Keratin 13 gene expression and its underlying mechanism in breast cancer cells. Molecular and Cellular Endocrinology. 296: 1-9. PMID 18951949 DOI: 10.1016/j.mce.2008.09.022  0.64
2008 Madak-Erdogan Z, Kieser KJ, Kim SH, Komm B, Katzenellenbogen JA, Katzenellenbogen BS. Nuclear and extranuclear pathway inputs in the regulation of global gene expression by estrogen receptors. Molecular Endocrinology (Baltimore, Md.). 22: 2116-27. PMID 18617595 DOI: 10.1210/me.2008-0059  0.64
2008 Alyea RA, Laurence SE, Kim SH, Katzenellenbogen BS, Katzenellenbogen JA, Watson CS. The roles of membrane estrogen receptor subtypes in modulating dopamine transporters in PC-12 cells. Journal of Neurochemistry. 106: 1525-33. PMID 18489713 DOI: 10.1111/j.1471-4159.2008.05491.x  0.64
2008 Barnett DH, Sheng S, Charn TH, Waheed A, Sly WS, Lin CY, Liu ET, Katzenellenbogen BS. Estrogen receptor regulation of carbonic anhydrase XII through a distal enhancer in breast cancer. Cancer Research. 68: 3505-15. PMID 18451179 DOI: 10.1158/0008-5472.CAN-07-6151  0.64
2008 Paulmurugan R, Tamrazi A, Katzenellenbogen JA, Katzenellenbogen BS, Gambhir SS. A human estrogen receptor (ER)alpha mutation with differential responsiveness to nonsteroidal ligands: novel approaches for studying mechanism of ER action. Molecular Endocrinology (Baltimore, Md.). 22: 1552-64. PMID 18451095 DOI: 10.1210/me.2007-0570  0.64
2008 Nettles KW, Bruning JB, Gil G, Nowak J, Sharma SK, Hahm JB, Kulp K, Hochberg RB, Zhou H, Katzenellenbogen JA, Katzenellenbogen BS, Kim Y, Joachmiak A, Greene GL. NFkappaB selectivity of estrogen receptor ligands revealed by comparative crystallographic analyses. Nature Chemical Biology. 4: 241-7. PMID 18344977 DOI: 10.1038/nchembio.76  0.64
2008 Minutolo F, Bellini R, Bertini S, Carboni I, Lapucci A, Pistolesi L, Prota G, Rapposelli S, Solati F, Tuccinardi T, Martinelli A, Stossi F, Carlson KE, Katzenellenbogen BS, Katzenellenbogen JA, et al. Monoaryl-substituted salicylaldoximes as ligands for estrogen receptor beta. Journal of Medicinal Chemistry. 51: 1344-51. PMID 18269232 DOI: 10.1021/jm701396g  0.64
2008 Chang EC, Charn TH, Park SH, Helferich WG, Komm B, Katzenellenbogen JA, Katzenellenbogen BS. Estrogen Receptors alpha and beta as determinants of gene expression: influence of ligand, dose, and chromatin binding. Molecular Endocrinology (Baltimore, Md.). 22: 1032-43. PMID 18258689 DOI: 10.1210/me.2007-0356  0.64
2007 Zhou HB, Nettles KW, Bruning JB, Kim Y, Joachimiak A, Sharma S, Carlson KE, Stossi F, Katzenellenbogen BS, Greene GL, Katzenellenbogen JA. Elemental Isomerism: A Boron-Nitrogen Surrogate for a Carbon-Carbon Double Bond Increases the Chemical Diversity of Estrogen Receptor Ligands Chemistry and Biology. 14: 659-669. PMID 17584613 DOI: 10.1016/j.chembiol.2007.04.009  0.64
2007 Stender JD, Frasor J, Komm B, Chang KC, Kraus WL, Katzenellenbogen BS. Estrogen-regulated gene networks in human breast cancer cells: involvement of E2F1 in the regulation of cell proliferation. Molecular Endocrinology (Baltimore, Md.). 21: 2112-23. PMID 17550982 DOI: 10.1210/me.2006-0474  0.64
2007 Lin CY, Vega VB, Thomsen JS, Zhang T, Kong SL, Xie M, Chiu KP, Lipovich L, Barnett DH, Stossi F, Yeo A, George J, Kuznetsov VA, Lee YK, Charn TH, ... ... Katzenellenbogen BS, et al. Whole-genome cartography of estrogen receptor alpha binding sites. Plos Genetics. 3: e87. PMID 17542648 DOI: 10.1371/journal.pgen.0030087  0.64
2007 Gowri PM, Sengupta S, Bertera S, Katzenellenbogen BS. Lipin1 regulation by estrogen in uterus and liver: implications for diabetes and fertility. Endocrinology. 148: 3685-93. PMID 17463059 DOI: 10.1210/en.2006-1728  0.64
2007 Zhou HB, Sheng S, Compton DR, Kim Y, Joachimiak A, Sharma S, Carlson KE, Katzenellenbogen BS, Nettles KW, Greene GL, Katzenellenbogen JA. Structure-guided optimization of estrogen receptor binding affinity and antagonist potency of pyrazolopyrimidines with basic side chains. Journal of Medicinal Chemistry. 50: 399-403. PMID 17228884 DOI: 10.1021/jm061035y  0.64
2006 Katzenellenbogen BS. In memoriam: Jack Gorski (1931-2006). Molecular Endocrinology (Baltimore, Md.). 20: 2611-2. PMID 17065652 DOI: 10.1210/mend.20.11.5432  0.64
2006 Mussi P, Liao L, Park SE, Ciana P, Maggi A, Katzenellenbogen BS, Xu J, O'Malley BW. Haploinsufficiency of the corepressor of estrogen receptor activity (REA) enhances estrogen receptor function in the mammary gland. Proceedings of the National Academy of Sciences of the United States of America. 103: 16716-21. PMID 17065319 DOI: 10.1073/pnas.0607768103  0.32
2006 Likhite VS, Stossi F, Kim K, Katzenellenbogen BS, Katzenellenbogen JA. Kinase-specific phosphorylation of the estrogen receptor changes receptor interactions with ligand, deoxyribonucleic acid, and coregulators associated with alterations in estrogen and tamoxifen activity. Molecular Endocrinology (Baltimore, Md.). 20: 3120-32. PMID 16945990 DOI: 10.1210/me.2006-0068  0.64
2006 Frasor J, Chang EC, Komm B, Lin CY, Vega VB, Liu ET, Miller LD, Smeds J, Bergh J, Katzenellenbogen BS. Gene expression preferentially regulated by tamoxifen in breast cancer cells and correlations with clinical outcome. Cancer Research. 66: 7334-40. PMID 16849584 DOI: 10.1158/0008-5472.CAN-05-4269  0.56
2006 Chang EC, Frasor J, Komm B, Katzenellenbogen BS. Impact of estrogen receptor beta on gene networks regulated by estrogen receptor alpha in breast cancer cells. Endocrinology. 147: 4831-42. PMID 16809442 DOI: 10.1210/en.2006-0563  0.64
2006 Harrington WR, Sengupta S, Katzenellenbogen BS. Estrogen regulation of the glucuronidation enzyme UGT2B15 in estrogen receptor-positive breast cancer cells. Endocrinology. 147: 3843-50. PMID 16690804 DOI: 10.1210/en.2006-0358  0.64
2006 Stossi F, Likhite VS, Katzenellenbogen JA, Katzenellenbogen BS. Estrogen-occupied estrogen receptor represses cyclin G2 gene expression and recruits a repressor complex at the cyclin G2 promoter. The Journal of Biological Chemistry. 281: 16272-8. PMID 16608856 DOI: 10.1074/jbc.M513405200  0.64
2006 Harrington WR, Kim SH, Funk CC, Madak-Erdogan Z, Schiff R, Katzenellenbogen JA, Katzenellenbogen BS. Estrogen dendrimer conjugates that preferentially activate extranuclear, nongenomic versus genomic pathways of estrogen action. Molecular Endocrinology (Baltimore, Md.). 20: 491-502. PMID 16306086 DOI: 10.1210/me.2005-0186  0.64
2006 Mishra RG, Stanczyk FZ, Burry KA, Oparil S, Katzenellenbogen BS, Nealen ML, Katzenellenbogen JA, Hermsmeyer RK. Metabolite ligands of estrogen receptor-beta reduce primate coronary hyperreactivity. American Journal of Physiology. Heart and Circulatory Physiology. 290: H295-303. PMID 16199482 DOI: 10.1152/ajpheart.00468.2005  0.64
2005 Zhou HB, Comninos JS, Stossi F, Katzenellenbogen BS, Katzenellenbogen JA. Synthesis and evaluation of estrogen receptor ligands with bridged oxabicyclic cores containing a diarylethylene motif: estrogen antagonists of unusual structure. Journal of Medicinal Chemistry. 48: 7261-74. PMID 16279785 DOI: 10.1021/jm0506773  0.64
2005 Frasor J, Danes JM, Funk CC, Katzenellenbogen BS. Estrogen down-regulation of the corepressor N-CoR: mechanism and implications for estrogen derepression of N-CoR-regulated genes. Proceedings of the National Academy of Sciences of the United States of America. 102: 13153-7. PMID 16141343 DOI: 10.1073/pnas.0502782102  0.64
2005 De Angelis M, Stossi F, Waibel M, Katzenellenbogen BS, Katzenellenbogen JA. Isocoumarins as estrogen receptor beta selective ligands: Isomers of isoflavone phytoestrogens and their metabolites. Bioorganic & Medicinal Chemistry. 13: 6529-42. PMID 16099659 DOI: 10.1016/j.bmc.2005.07.014  0.64
2005 Wang C, Fan S, Li Z, Fu M, Rao M, Ma Y, Lisanti MP, Albanese C, Katzenellenbogen BS, Kushner PJ, Weber B, Rosen EM, Pestell RG. Cyclin D1 antagonizes BRCA1 repression of estrogen receptor alpha activity. Cancer Research. 65: 6557-67. PMID 16061635 DOI: 10.1158/0008-5472.CAN-05-0486  0.64
2005 Rai D, Frolova A, Frasor J, Carpenter AE, Katzenellenbogen BS. Distinctive actions of membrane-targeted versus nuclear localized estrogen receptors in breast cancer cells. Molecular Endocrinology (Baltimore, Md.). 19: 1606-17. PMID 15831524 DOI: 10.1210/me.2004-0468  0.64
2005 De Angelis M, Stossi F, Carlson KA, Katzenellenbogen BS, Katzenellenbogen JA. Indazole estrogens: highly selective ligands for the estrogen receptor beta. Journal of Medicinal Chemistry. 48: 1132-44. PMID 15715479 DOI: 10.1021/jm049223g  0.64
2005 Park SE, Xu J, Frolova A, Liao L, O'Malley BW, Katzenellenbogen BS. Genetic deletion of the repressor of estrogen receptor activity (REA) enhances the response to estrogen in target tissues in vivo. Molecular and Cellular Biology. 25: 1989-99. PMID 15713652 DOI: 10.1128/MCB.25.5.1989-1999.2005  0.64
2004 Compton DR, Sheng S, Carlson KE, Rebacz NA, Lee IY, Katzenellenbogen BS, Katzenellenbogen JA. Pyrazolo[1,5-a]pyrimidines: estrogen receptor ligands possessing estrogen receptor beta antagonist activity. Journal of Medicinal Chemistry. 47: 5872-93. PMID 15537344 DOI: 10.1021/jm049631k  0.64
2004 Chen Z, Katzenellenbogen BS, Katzenellenbogen JA, Zhao H. Directed evolution of human estrogen receptor variants with significantly enhanced androgen specificity and affinity. The Journal of Biological Chemistry. 279: 33855-64. PMID 15159406 DOI: 10.1074/jbc.M402118200  0.64
2004 Katzenellenbogen BS, Frasor J. Therapeutic targeting in the estrogen receptor hormonal pathway. Seminars in Oncology. 31: 28-38. PMID 15052541  0.64
2004 Stossi F, Barnett DH, Frasor J, Komm B, Lyttle CR, Katzenellenbogen BS. Transcriptional profiling of estrogen-regulated gene expression via estrogen receptor (ER) alpha or ERbeta in human osteosarcoma cells: distinct and common target genes for these receptors. Endocrinology. 145: 3473-86. PMID 15033914 DOI: 10.1210/en.2003-1682  0.64
2004 Tsai HW, Katzenellenbogen JA, Katzenellenbogen BS, Shupnik MA. Protein kinase A activation of estrogen receptor α transcription does not require proteasome activity and protects the receptor from ligand-mediated degradation Endocrinology. 145: 2730-2738. PMID 15033909 DOI: 10.1210/en.2003-1470  0.64
2004 Acevedo ML, Lee KC, Stender JD, Katzenellenbogen BS, Kraus WL. Selective recognition of distinct classes of coactivators by a ligand-inducible activation domain. Molecular Cell. 13: 725-38. PMID 15023342 DOI: 10.1016/S1097-2765(04)00121-2  0.64
2004 Muthyala RS, Ju YH, Sheng S, Williams LD, Doerge DR, Katzenellenbogen BS, Helferich WG, Katzenellenbogen JA. Equol, a natural estrogenic metabolite from soy isoflavones: convenient preparation and resolution of R- and S-equols and their differing binding and biological activity through estrogen receptors alpha and beta. Bioorganic & Medicinal Chemistry. 12: 1559-67. PMID 15018930 DOI: 10.1016/j.bmc.2003.11.035  0.64
2004 Frasor J, Stossi F, Danes JM, Komm B, Lyttle CR, Katzenellenbogen BS. Selective estrogen receptor modulators: discrimination of agonistic versus antagonistic activities by gene expression profiling in breast cancer cells. Cancer Research. 64: 1522-33. PMID 14973112  0.36
2004 Nettles KW, Sun J, Radek JT, Sheng S, Rodriguez AL, Katzenellenbogen JA, Katzenellenbogen BS, Greene GL. Allosteric Control of Ligand Selectivity between Estrogen Receptors α and β: Implications for Other Nuclear Receptors Molecular Cell. 13: 317-327. PMID 14967140 DOI: 10.1016/S1097-2765(04)00054-1  0.64
2003 Frasor J, Danes JM, Komm B, Chang KC, Lyttle CR, Katzenellenbogen BS. Profiling of estrogen up- and down-regulated gene expression in human breast cancer cells: insights into gene networks and pathways underlying estrogenic control of proliferation and cell phenotype. Endocrinology. 144: 4562-74. PMID 12959972 DOI: 10.1210/en.2003-0567  0.36
2003 Minutolo F, Antonello M, Bertini S, Ortore G, Placanica G, Rapposelli S, Sheng S, Carlson KE, Katzenellenbogen BS, Katzenellenbogen JA, Macchia M. Novel estrogen receptor ligands based on an anthranylaldoxime structure: Role of the phenol-type pseudocycle in the binding process Journal of Medicinal Chemistry. 46: 4032-4042. PMID 12954056 DOI: 10.1021/jm0308390  0.64
2003 Harrington WR, Sheng S, Barnett DH, Petz LN, Katzenellenbogen JA, Katzenellenbogen BS. Activities of estrogen receptor alpha- and beta-selective ligands at diverse estrogen responsive gene sites mediating transactivation or transrepression. Molecular and Cellular Endocrinology. 206: 13-22. PMID 12943986 DOI: 10.1016/S0303-7207(03)00255-7  0.64
2003 Martini PG, Katzenellenbogen BS. Modulation of estrogen receptor activity by selective coregulators. The Journal of Steroid Biochemistry and Molecular Biology. 85: 117-22. PMID 12943695 DOI: 10.1016/S0960-0760(03)00207-3  0.64
2003 Frasor J, Barnett DH, Danes JM, Hess R, Parlow AF, Katzenellenbogen BS. Response-specific and ligand dose-dependent modulation of estrogen receptor (ER) alpha activity by ERbeta in the uterus. Endocrinology. 144: 3159-66. PMID 12810572 DOI: 10.1210/en.2002-0143  0.64
2003 Muthyala RS, Sheng S, Carlson KE, Katzenellenbogen BS, Katzenellenbogen JA. Bridged bicyclic cores containing a 1,1-diarylethylene motif are high-affinity subtype-selective ligands for the estrogen receptor Journal of Medicinal Chemistry. 46: 1589-1602. PMID 12699377 DOI: 10.1021/jm0204800  0.64
2003 Sun J, Katzenellenbogen JA, Zhao H, Katzenellenbogen BS. DNA shuffling method for generating estrogen receptor α and β chimeras in yeast Biotechniques. 34: 278-288. PMID 12613251  0.64
2003 Sun J, Baudry J, Katzenellenbogen JA, Katzenellenbogen BS. Molecular basis for the subtype discrimination of the estrogen receptor-β-selective ligand, diarylpropionitrile Molecular Endocrinology. 17: 247-258. PMID 12554752 DOI: 10.1210/me.2002-0341  0.64
2003 Ghosh U, Ganessunker D, Sattigeri VJ, Carlson KE, Mortensen DJ, Katzenellenbogen BS, Katzenellenbogen JA. Estrogenic diazenes: heterocyclic non-steroidal estrogens of unusual structure with selectivity for estrogen receptor subtypes. Bioorganic & Medicinal Chemistry. 11: 629-57. PMID 12538029  0.56
2003 Rajendran RR, Nye AC, Frasor J, Balsara RD, Martini PG, Katzenellenbogen BS. Regulation of nuclear receptor transcriptional activity by a novel DEAD box RNA helicase (DP97). The Journal of Biological Chemistry. 278: 4628-38. PMID 12466272 DOI: 10.1074/jbc.M210066200  0.64
2003 Katzenellenbogen JA, Muthyala R, Katzenellenbogen BS. Nature of the ligand-binding pocket of estrogen receptor α and β: The search for subtype-selective ligands and implications for the prediction of estrogenic activity Pure and Applied Chemistry. 75: 2397-2403.  0.64
2002 Sun J, Huang YR, Harrington WR, Sheng S, Katzenellenbogen JA, Katzenellenbogen BS. Antagonists Selective for Estrogen Receptor α. Endocrinology. 143: 941-947. PMID 28201446 DOI: 10.1210/endo.143.3.8704  0.6
2002 Harris HA, Katzenellenbogen JA, Katzenellenbogen BS. Characterization of the biological roles of the estrogen receptors, ERα and ERβ, in estrogen target tissues in vivo through the use of an ERα-selective ligand Endocrinology. 143: 4172-4177. PMID 12399409 DOI: 10.1210/en.2002-220403  0.64
2002 Ediger TR, Park SE, Katzenellenbogen BS. Estrogen receptor inducibility of the human Na+/H+ exchanger regulatory factor/ezrin-radixin-moesin binding protein 50 (NHE-RF/EBP50) gene involving multiple half-estrogen response elements. Molecular Endocrinology (Baltimore, Md.). 16: 1828-39. PMID 12145337 DOI: 10.1210/me.2001-0290  0.64
2002 Nye AC, Rajendran RR, Stenoien DL, Mancini MA, Katzenellenbogen BS, Belmont AS. Alteration of large-scale chromatin structure by estrogen receptor. Molecular and Cellular Biology. 22: 3437-49. PMID 11971975 DOI: 10.1128/MCB.22.10.3437-3449.2002  0.64
2002 Shiau AK, Barstad D, Radek JT, Meyers MJ, Nettles KW, Katzenellenbogen BS, Katzenellenbogen JA, Agard DA, Greene GL. Structural characterization of a subtype-selective ligand reveals a novel mode of estrogen receptor antagonism. Nature Structural Biology. 9: 359-64. PMID 11953755 DOI: 10.1038/nsb787  0.64
2002 Katzenellenbogen BS, Katzenellenbogen JA. Defining the "S" in SERMs Science. 295: 2380-2381. PMID 11923515 DOI: 10.1126/science.1070442  0.64
2002 Rickard DJ, Waters KM, Ruesink TJ, Khosla S, Katzenellenbogen JA, Katzenellenbogen BS, Riggs BL, Spelsberg TC. Estrogen receptor isoform-specific induction of progesterone receptors in human osteoblasts Journal of Bone and Mineral Research. 17: 580-592. PMID 11918216  0.64
2002 Kowalski AA, Graddy LG, Vale-Cruz DS, Choi I, Katzenellenbogen BS, Simmen FA, Simmen RC. Molecular cloning of porcine estrogen receptor-beta complementary DNAs and developmental expression in periimplantation embryos. Biology of Reproduction. 66: 760-9. PMID 11870084  0.64
2002 Sun J, Huang YR, Harrington WR, Sheng S, Katzenellenbogen JA, Katzenellenbogen BS. Antagonists selective for estrogen receptor alpha. Endocrinology. 143: 941-7. PMID 11861516 DOI: 10.1210/endo.143.3.8704  0.6
2001 Mortensen DS, Rodriguez AL, Sun J, Katzenellenbogen BS, Katzenellenbogen JA. Furans with basic side chains: synthesis and biological evaluation of a novel series of antagonists with selectivity for the estrogen receptor alpha. Bioorganic & Medicinal Chemistry Letters. 11: 2521-4. PMID 11549460 DOI: 10.1016/S0960-894X(01)00488-7  0.64
2001 Martini PG, Katzenellenbogen BS. Regulation of prothymosin alpha gene expression by estrogen in estrogen receptor-containing breast cancer cells via upstream half-palindromic estrogen response element motifs. Endocrinology. 142: 3493-501. PMID 11459795 DOI: 10.1210/endo.142.8.8314  0.64
2001 Lazennec G, Thomas JA, Katzenellenbogen BS. Involvement of cyclic AMP response element binding protein (CREB) and estrogen receptor phosphorylation in the synergistic activation of the estrogen receptor by estradiol and protein kinase activators Journal of Steroid Biochemistry and Molecular Biology. 77: 193-203. PMID 11457657 DOI: 10.1016/S0960-0760(01)00060-7  0.64
2001 Tedesco R, Thomas JA, Katzenellenbogen BS, Katzenellenbogen JA. The estrogen receptor: a structure-based approach to the design of new specific hormone-receptor combinations. Chemistry & Biology. 8: 277-87. PMID 11306352 DOI: 10.1016/S1074-5521(01)00006-0  0.64
2000 Kraichely DM, Sun J, Katzenellenbogen JA, Katzenellenbogen BS. Conformational Changes and Coactivator Recruitment by Novel Ligands for Estrogen Receptor-α and Estrogen Receptor-β: Correlations with Biological Character and Distinct Differences among SRC Coactivator Family Members. Endocrinology. 141: 3534-3545. PMID 28200959 DOI: 10.1210/endo.141.10.7698  0.56
2000 Katzenellenbogen BS, Katzenellenbogen JA. Estrogen receptor alpha and estrogen receptor beta: Regulation by selective estrogen receptor modulators and importance in breast cancer Breast Cancer Research. 2: 335-344. PMID 11250726 DOI: 10.1186/bcr78  0.64
2000 Choi I, Gudas LJ, Katzenellenbogen BS. Regulation of keratin 19 gene expression by estrogen in human breast cancer cells and identification of the estrogen responsive gene region Molecular and Cellular Endocrinology. 164: 225-237. PMID 11026574 DOI: 10.1016/S0303-7207(00)00197-0  0.64
2000 Kraichely DM, Sun J, Katzenellenbogen JA, Katzenellenbogen BS. Conformational changes and coactivator recruitment by novel ligands for estrogen receptor-α and estrogen receptor-β: Correlations with biological character and distinct differences among SRC coactivator family members Endocrinology. 141: 3534-3545. PMID 11014206  0.64
2000 Stauffer SR, Sun J, Katzenellenbogen BS, Katzenellenbogen JA. Acyclic amides as estrogen receptor ligands: Synthesis, binding, activity and receptor interaction Bioorganic and Medicinal Chemistry. 8: 1293-1316. PMID 10896109 DOI: 10.1016/S0968-0896(00)00075-4  0.64
2000 Stoica A, Katzenellenbogen BS, Martin MB. Activation of estrogen receptor-alpha by the heavy metal cadmium. Molecular Endocrinology (Baltimore, Md.). 14: 545-53. PMID 10770491 DOI: 10.1210/mend.14.4.0441  0.64
2000 Katzenellenbogen BS. Mechanisms of action and cross-talk between estrogen receptor and progesterone receptor pathways Journal of the Society For Gynecologic Investigation. 7. PMID 10732327  0.64
1999 Sun J, Meyers MJ, Fink BE, Rajendran R, Katzenellenbogen JA, Katzenellenbogen BS. Novel Ligands that Function as Selective Estrogens or Antiestrogens for Estrogen Receptor-α or Estrogen Receptor-β. Endocrinology. 140: 800-804. PMID 28204395 DOI: 10.1210/endo.140.2.6480  0.56
1999 Ediger TR, Kraus WL, Weinman EJ, Katzenellenbogen BS. Estrogen Receptor Regulation of the Na+/H+ Exchanger Regulatory Factor. Endocrinology. 140: 2976-2982. PMID 28200751 DOI: 10.1210/endo.140.7.6885  0.52
1999 Gee AC, Carlson KE, Martini PG, Katzenellenbogen BS, Katzenellenbogen JA. Coactivator peptides have a differential stabilizing effect on the binding of estrogens and antiestrogens with the estrogen receptor. Molecular Endocrinology (Baltimore, Md.). 13: 1912-23. PMID 10551784 DOI: 10.1210/mend.13.11.0373  0.64
1999 Meyers MJ, Sun J, Carlson KE, Katzenellenbogen BS, Katzenellenbogen JA. Estrogen receptor subtype-selective ligands: asymmetric synthesis and biological evaluation of cis- and trans-5,11-dialkyl- 5,6,11, 12-tetrahydrochrysenes. Journal of Medicinal Chemistry. 42: 2456-68. PMID 10395487 DOI: 10.1021/jm990101b  0.64
1999 Lazennec G, Alcorn JL, Katzenellenbogen BS. Adenovirus-mediated delivery of a dominant negative estrogen receptor gene abrogates estrogen-stimulated gene expression and breast cancer cell proliferation Molecular Endocrinology. 13: 969-980. PMID 10379895  0.64
1999 Lazennec G, Katzenellenbogen BS. Expression of human estrogen receptor using an efficient adenoviral gene delivery system is able to restore hormone-dependent features to estrogen receptor-negative breast carcinoma cells Molecular and Cellular Endocrinology. 149: 93-105. PMID 10375022 DOI: 10.1016/S0303-7207(98)00254-8  0.64
1998 McInerney EM, Weis KE, Sun J, Mosselman S, Katzenellenbogen BS. Transcription Activation by the Human Estrogen Receptor Subtypeβ (ERβ) Studied with ERβ and ERα Receptor Chimeras* *This work was supported by NIH Grants CA-18119 and CA-60514 (to B.S.K.). Endocrinology. 139: 4513-4522. PMID 28200456 DOI: 10.1210/endo.139.11.6298  0.4
1998 Montano MM, Jaiswal AK, Katzenellenbogen BS. Transcriptional regulation of the human quinone reductase gene by antiestrogen-liganded estrogen receptor-α and estrogen receptor-β Journal of Biological Chemistry. 273: 25443-25449. PMID 9738013 DOI: 10.1074/jbc.273.39.25443  0.64
1998 Ekena K, Katzenellenbogen JA, Katzenellenbogen BS. Determinants of ligand specificity of estrogen receptor-α: Estrogen versus androgen discrimination Journal of Biological Chemistry. 273: 693-699. PMID 9422719 DOI: 10.1074/jbc.273.2.693  0.64
1997 Kraus WL, Weis KE, Katzenellenbogen BS. Determinants for the repression of estrogen receptor transcriptional activity by ligand-occupied progestin receptors. The Journal of Steroid Biochemistry and Molecular Biology. 63: 175-88. PMID 9459183 DOI: 10.1016/S0960-0760(97)00089-7  0.64
1997 Carlson KE, Choi I, Gee A, Katzenellenbogen BS, Katzenellenbogen JA. Altered ligand binding properties and enhanced stability of a constitutively active estrogen receptor: Evidence that an open pocket conformation is required for ligand interaction Biochemistry. 36: 14897-14905. PMID 9398213 DOI: 10.1021/bi971746l  0.64
1997 Montano MM, Katzenellenbogen BS. The quinone reductase gene: A unique estrogen receptor-regulated gene that is activated by antiestrogens Proceedings of the National Academy of Sciences of the United States of America. 94: 2581-2586. PMID 9122238 DOI: 10.1073/pnas.94.6.2581  0.64
1997 Montano MM, Kraus WL, Katzenellenbogen BS. Identification of a novel transferable cis element in the promoter of an estrogen-responsive gene that modulates sensitivity to hormone and antihormone Molecular Endocrinology. 11: 330-341. PMID 9058379 DOI: 10.1210/me.11.3.330  0.64
1997 Katzenellenbogen BS, Korach KS. Editorial: A new actor in the estrogen receptor drama - Enter ER-β Endocrinology. 138: 861-862. PMID 9048583 DOI: 10.1210/en.138.3.861  0.64
1997 Ekena K, Weis KE, Katzenellenbogen JA, Katzenellenbogen BS. Different residues of the human estrogen receptor are involved in the recognition of structurally diverse estrogens and antiestrogens. The Journal of Biological Chemistry. 272: 5069-75. PMID 9030571 DOI: 10.1074/jbc.272.8.5069  0.64
1996 Herman ME, Katzenellenbogen BS. Response-specific antiestrogen resistance in a newly characterized MCF-7 human breast cancer cell line resulting from long-term exposure to trans-hydroxytamoxifen Journal of Steroid Biochemistry and Molecular Biology. 59: 121-134. PMID 9010327 DOI: 10.1016/S0960-0760(96)00114-8  0.64
1996 McInerney EM, Ince BA, Shapiro DJ, Katzenellenbogen BS. A transcriptionally active estrogen receptor mutant is a novel type of dominant negative inhibitor of estrogen action Molecular Endocrinology. 10: 1519-1526. PMID 8961262 DOI: 10.1210/me.10.12.1519  0.64
1996 Katzenellenbogen JA, O'Malley BW, Katzenellenbogen BS. Tripartite steroid hormone receptor pharmacology: Interaction with multiple effector sites as a basis for the cell- and promoter-specific action of these hormones Molecular Endocrinology. 10: 119-131. PMID 8825552 DOI: 10.1210/me.10.2.119  0.64
1996 Mcinerney EM, Tsai MJ, O'Malley BW, Katzenellenbogen BS. Analysis of estrogen receptor transcriptional enhancement by a nuclear hormone receptor coactivator Proceedings of the National Academy of Sciences of the United States of America. 93: 10069-10073. PMID 8816752 DOI: 10.1073/pnas.93.19.10069  0.64
1996 Katzenellenbogen JA, Katzenellenbogen BS. Nuclear hormone receptors: Ligand-activated regulators of transcription and diverse cell responses Chemistry and Biology. 3: 529-536. PMID 8807884 DOI: 10.1016/S1074-5521(96)90143-X  0.64
1996 McInerney EM, Katzenellenbogen BS. Different regions in activation function-1 of the human estrogen receptor required for antiestrogen- and estradiol-dependent transcription activation Journal of Biological Chemistry. 271: 24172-24178. PMID 8798658 DOI: 10.1074/jbc.271.39.24172  0.64
1996 Katzenellenbogen BS. Estrogen receptors: Bioactivities and interactions with cell signaling pathways Biology of Reproduction. 54: 287-293. PMID 8788178 DOI: 10.1095/biolreprod54.2.287  0.64
1996 Ekena K, Weis KE, Katzenellenbogen JA, Katzenellenbogen BS. Identification of amino acids in the hormone binding domain of the human estrogen receptor important in estrogen binding. The Journal of Biological Chemistry. 271: 20053-9. PMID 8702724 DOI: 10.1074/jbc.271.33.20053  0.64
1995 Kraus WL, Mcinerney EM, Katzenellenbogen BS. Ligand-dependent, transcriptionally productive association of the amino- and carboxyl-terminal regions of a steroid hormone nuclear receptor Proceedings of the National Academy of Sciences of the United States of America. 92: 12314-12318. PMID 8618892 DOI: 10.1073/pnas.92.26.12314  0.64
1995 Schodin DJ, Zhuang Y, Shapiro DJ, Katzenellenbogen BS. Analysis of mechanisms that determine dominant negative estrogen receptor effectiveness Journal of Biological Chemistry. 270: 31163-31171. PMID 8537380 DOI: 10.1074/jbc.270.52.31163  0.64
1995 Kraus WL, Weis KE, Katzenellenbogen BS. Inhibitory cross-talk between steroid hormone receptors: differential targeting of estrogen receptor in the repression of its transcriptional activity by agonist- and antagonist-occupied progestin receptors. Molecular and Cellular Biology. 15: 1847-57. PMID 7891678  0.64
1995 Zhuang Y, Katzenellenbogen BS, Shapiro DJ. Estrogen receptor mutants which do not bind 17β-estradiol dimerize and bind to the estrogen response element in vivo Molecular Endocrinology. 9: 457-466. PMID 7659089  0.64
1995 Ince BA, Schodin DJ, Shapiro DJ, Katzenellenbogen BS. Repression of endogenous estrogen receptor activity in MCF-7 human breast cancer cells by dominant negative estrogen receptors Endocrinology. 136: 3194-3199. PMID 7628351  0.64
1995 Montano MM, Muller V, Trobaugh A, Katzenellenbogen BS. The carboxy-terminal F domain of the human estrogen receptor: Role in the transcriptional activity of the receptor and the effectiveness of antiestrogens as estrogen antagonists Molecular Endocrinology. 9: 814-825. PMID 7476965  0.64
1994 Le Goff P, Montano MM, Schodin DJ, Katzenellenbogen BS. Phosphorylation of the human estrogen receptor: Identification of hormone-regulated sites and examination of their influence on transcriptional activity Journal of Biological Chemistry. 269: 4458-4466. PMID 8308015  0.64
1994 Aronica SM, Kraus WL, Katzenellenbogen BS. Estrogen action via the cAMP signaling pathway: Stimulation of adenylate cyclase and cAMP-regulated gene transcription Proceedings of the National Academy of Sciences of the United States of America. 91: 8517-8521. PMID 8078914  0.64
1994 Bergmann KE, Wooge CH, Carlson KE, Katzenellenbogen BS, Katzenellenbogen JA. Bivalent ligands as probes of estrogen receptor action Journal of Steroid Biochemistry and Molecular Biology. 49: 139-152. PMID 8031710 DOI: 10.1016/0960-0760(94)90004-3  0.64
1994 Kraus WL, Montano MM, Katzenellenbogen BS. Identification of multiple, widely spaced estrogen-responsive regions in the rat progesterone receptor gene Molecular Endocrinology. 8: 952-969. PMID 7997237 DOI: 10.1210/me.8.8.952  0.64
1994 Herman ME, Katzenellenbogen BS. Alterations in Transforming Growth Factor-α and -β Production and Cell Responsiveness during the Progression of MCF-7 Human Breast Cancer Cells to Estrogen-Autonomous Growth Cancer Research. 54: 5867-5874. PMID 7954416  0.64
1994 Ince BA, Montano MM, Katzenellenbogen BS. Activation of transcriptionally inactive human estrogen receptors by cyclic adenosine 3′,5′-monophosphate and ligands including antiestrogens Molecular Endocrinology. 8: 1397-1406. PMID 7531820  0.64
1994 Fujimoto N, Katzenellenbogen BS. Alteration in the agonist/antagonist balance of antiestrogens by activation of protein kinase A signaling pathways in breast cancer cells: Antiestrogen selectivity and promoter dependence Molecular Endocrinology. 8: 296-304. PMID 7517003 DOI: 10.1210/me.8.3.296  0.64
1994 Cho H, Aronica SM, Katzenellenbogen BS. Regulation of progesterone receptor gene expression in MCF-7 breast cancer cells: A comparison of the effects of cyclic adenosine 3',5'-monophosphate, estradiol, insulin-like growth factor-I, and serum factors Endocrinology. 134: 658-664. PMID 7507831 DOI: 10.1210/en.134.2.658  0.64
1993 Kraus WL, Katzenellenbogen BS. Regulation of progesterone receptor gene expression and growth in the rat uterus: Modulation of estrogen actions by progesterone and sex steroid hormone antagonists Endocrinology. 132: 2371-2379. PMID 8504742  0.64
1993 Pakdel F, Goff PL, Katzenellenbogen BS. An assessment of the role of domain F and pest sequences in estrogen receptor half-life and bioactivity Journal of Steroid Biochemistry and Molecular Biology. 46: 663-672. PMID 8274400 DOI: 10.1016/0960-0760(93)90307-I  0.64
1993 Wrenn CK, Katzenellenbogen BS. Structure-function analysis of the hormone binding domain of the human estrogen receptor by region-specific mutagenesis and phenotypic screening in yeast Journal of Biological Chemistry. 268: 24089-24098. PMID 8226955  0.64
1993 Lee Kraus W, Montano MM, Katzenellenbogen BS. Cloning of the rat progesterone receptor gene 5′-region and identification of two functionally distinct promoters Molecular Endocrinology. 7: 1603-1616. PMID 8145766  0.64
1993 Pakdel F, Reese JC, Katzenellenbogen BS. Identification of charged residues in an N-terminal portion of the hormone-binding domain of the human estrogen receptor important in transcriptional activity of the receptor Molecular Endocrinology. 7: 1408-1417. PMID 8114756  0.64
1993 Aronica SM, Katzenellenbogen BS. Stimulation of estrogen receptor-mediated transcription and alteration in the phosphorylation state of the rat uterine estrogen receptor by estrogen, cyclic adenosine monophosphate, and insulin-like growth factor-I Molecular Endocrinology. 7: 743-752. PMID 7689695 DOI: 10.1210/me.7.6.743  0.64
1993 Cho H, Katzenellenbogen BS. Synergistic activation of estrogen receptor-mediated transcription by estradiol and protein kinase activators Molecular Endocrinology. 7: 441-452. PMID 7683375 DOI: 10.1210/me.7.3.441  0.64
1992 Pakdel F, Katzenellenbogen BS. Human estrogen receptor mutants with altered estrogen and antiestrogen ligand discrimination Journal of Biological Chemistry. 267: 3429-3437. PMID 1737796  0.64
1992 Reese JC, Katzenellenbogen BS. Characterization of a temperature-sensitive mutation in the hormone binding domain of the human estrogen receptor: Studies in cell extracts and intact cells and their implications for hormone-dependent transcriptional activation Journal of Biological Chemistry. 267: 9868-9873. PMID 1577818  0.64
1992 Reese JC, Wooge CH, Katzenellenbogen BS. Identification of two cysteines closely positioned in the ligand-binding pocket of the human estrogen receptor: Roles in ligand binding and transcriptional activation Molecular Endocrinology. 6: 2160-2166. PMID 1491695  0.64
1992 Reese JC, Katzenellenbogen BS. Examination of the DNA-Binding Ability of Estrogen Receptor in Whole Cells: Implications for Hormone-Independent Transactivation and the Actions of Antiestrogens Molecular and Cellular Biology. 12: 4531-4538. PMID 1406642  0.64
1992 Read LD, Katzenellenbogen BS. Characterization and regulation of estrogen and progesterone receptors in breast cancer Cancer Treatment and Research. 61: 277-299. PMID 1360237  0.64
1991 Reese JC, Katzenellenbogen BS. Mutagenesis of cysteines in the hormone binding domain of the human estrogen receptor: Alterations in binding and transcriptional activation by covalently and reversibly attaching ligands Journal of Biological Chemistry. 266: 10880-10888. PMID 2040605  0.64
1991 Katzenellenbogen BS. Antiestrogen resistance: Mechanisms by which breast cancer cells undermine the effectiveness of endocrine therapy Journal of the National Cancer Institute. 83: 1434-1435. PMID 1920488 DOI: 10.1093/jnci/83.20.1434  0.64
1991 Reese JC, Katzenellenbogen BS. Differential DNA-binding abilites of estrogen receptor occupied with two classes of antiestrogens: Studies using human estrogen receptor overexpressed in mammalian cells Nucleic Acids Research. 19: 6595-6602. PMID 1754396 DOI: 10.1093/nar/19.23.6595  0.64
1991 Cho H, Ng PA, Katzenellenbogen BS. Differential regulation of gene expression by estrogen in estrogen growth- independent and -dependent MCF-7 human breast cancer cell sublines Molecular Endocrinology. 5: 1323-1330. PMID 1722871  0.64
1991 Aronica SM, Katzenellenbogen BS. Progesterone receptor regulation in uterine cells: Stimulation by estrogen, cyclic adenosine 3',5'-monophosphate, and insulin-like growth factor I and suppression by antiestrogens and protein kinase inhibitors Endocrinology. 128: 2045-2052. PMID 1706263  0.64
1990 Katzenellenbogen BS, Nardulli AM, Read LD. Estrogen regulation of proliferation and hormonal modulation of estrogen and progesterone receptor biosynthesis and degradation in target cells Progress in Clinical and Biological Research. 322: 201-211. PMID 2406733  0.64
1990 Katzenellenbogen BS. A tribute to Jack Gorski: estrogen receptor model builder and scientific friend to many Progress in Clinical and Biological Research. 322: 1-16. PMID 2406727  0.64
1990 Katzenellenbogen BS, Norman MJ. Multihormonal regulation of the progesterone receptor in MCF-7 human breast cancer cells: Interrelationships among insulin/insulin-like growth factor-I, serum, and estrogen Endocrinology. 126: 891-898. PMID 2404751  0.64
1990 Wrenn CK, Katzenellenbogen BS. Cross-linking of estrogen receptor to chromatin in intact MCF-7 human breast cancer cells: Optimization and effect of ligand Molecular Endocrinology. 4: 1647-1654. PMID 2280770  0.64
1990 Read LD, Keith D, Slamon DJ, Katzenellenbogen BS. Hormonal Modulation of HER-2/neu Protooncogene Messenger Ribonucleic Acid and pl85 Protein Expression in Human Breast Cancer Cell Lines Cancer Research. 50: 3947-3951. PMID 1972345  0.64
1989 Harlow KW, Smith DN, Katzenellenbogen JA, Greene GL, Katzenellenbogen BS. Identification of cysteine 530 as the covalent attachment site of an affinity-labeling estrogen (ketononestrol aziridine) and antiestrogen (tamoxifen aziridine) in the human estrogen receptor. The Journal of Biological Chemistry. 264: 17476-85. PMID 2793867  0.64
1989 Read LD, Greene GL, Katzenellenbogen BS. Regulation of estrogen receptor messenger ribonucleic acid and protein levels in human breast cancer cell lines by sex steroid hormones, their antagonists, and growth factors. Molecular Endocrinology (Baltimore, Md.). 3: 295-304. PMID 2785242 DOI: 10.1210/mend-3-2-295  0.64
1988 Bindal RD, Carlson KE, Katzenellenbogen BS, Katzenellenbogen JA. Lipophilic impurities, not phenolsulfonphthalein, account for the estrogenic activity in commercial preparations of phenol red Journal of Steroid Biochemistry. 31: 287-293. PMID 3419159 DOI: 10.1016/0022-4731(88)90352-4  0.64
1988 Nardulli AM, Katzenellenbogen BS. Progesterone receptor regulation in T47D human breast cancer cells: Analysis by density labeling of progesterone receptor synthesis and degradation and their modulation by progestin Endocrinology. 122: 1532-1540. PMID 3345726  0.64
1988 Nardulli AM, Greene GL, O'Malley BW, Katzenellenbogen BS. Regulation of progesterone receptor messenger ribonucleic acid and protein levels in MCF-7 cells by estradiol: analysis of estrogen's effect on progesterone receptor synthesis and degradation. Endocrinology. 122: 935-44. PMID 3342760 DOI: 10.1210/endo-122-3-935  0.64
1988 Elliston JF, Katzenellenbogen BS. Comparative analysis of estrogen receptors covalently labeled with an estrogen and an antiestrogen in several estrogen target cells as studied by limited proteolysis Journal of Steroid Biochemistry. 29: 559-569. PMID 3290576 DOI: 10.1016/0022-4731(88)90152-5  0.64
1988 Weaver CA, Springer PA, Katzenellenbogen BS. Regulation of pS2 gene expression by affinity labeling and reversibly binding estrogens and antiestrogens: comparison of effects on the native gene and on pS2-chloramphenicol acetyltransferase fusion genes transfected into MCF-7 human breast cancer cells. Molecular Endocrinology (Baltimore, Md.). 2: 936-45. PMID 2460749 DOI: 10.1210/mend-2-10-936  0.64
1987 Sheen YY, Katzenellenbogen BS. Antiestrogen stimulation of the production of a 37,000 molecular weight secreted protein and estrogen stimulation of the production of a 32,000 molecular weight secreted protein in MCF-7 human breast cancer cells Endocrinology. 120: 1140-1151. PMID 3803313  0.64
1987 Katzenellenbogen BS, Kendra KL, Norman MJ, Berthois Y. Proliferation, Hormonal Responsiveness, and Estrogen Receptor Content of MCF-7 Human Breast Cancer Cells Grown in the Short-Term and Long-Term Absence of Estrogens Cancer Research. 47: 4355-4360. PMID 3607768  0.64
1987 Elliston JF, Zablocki JA, Katzenellenbogen BS, Katzenellenbogen JA. Ketononestrol aziridine, an agonistic estrogen receptor affinity label: Study of its bioactivity and estrogen receptor covalent labeling Endocrinology. 121: 667-676. PMID 3595536  0.64
1987 Kendra KL, Katzenellenbogen BS. An evaluation of the involvement of polyamines in modulating MCF-7 human breast cancer cell proliferation and progesterone receptor levels by estrogen and antiestrogen Journal of Steroid Biochemistry. 28: 123-128. PMID 3114562 DOI: 10.1016/0022-4731(87)90367-0  0.64
1987 Zablocki JA, Katzenellenbogen JA, Carlson KE, Norman MJ, Katzenellenbogen BS. Estrogenic affinity labels: Synthesis, irreversible receptor binding, and bioactivity of aziridine-substituted hexestrol derivatives Journal of Medicinal Chemistry. 30: 829-838. PMID 3033242  0.64
1987 Toney TW, Katzenellenbogen BS. An evaluation of the interactions of antiestrogens with pituitary and striatal dopamine receptors Journal of Receptors and Signal Transduction. 7: 695-712. PMID 2958626 DOI: 10.3109/10799898709056780  0.64
1986 Mullick A, Katzenellenbogen BS. Antiprogestin-receptor complexes: Differences in the interaction of the antiprogestin RU38,486 and the progestin R5020 with the progesterone receptor of human breast cancer cells Biochemical and Biophysical Research Communications. 135: 90-97. PMID 3954780 DOI: 10.1016/0006-291X(86)90946-0  0.64
1986 Reiner GCA, Katzenellenbogen BS. Characterization of Estrogen and Progesterone Receptors and the Dissociated Regulation of Growth and Progesterone Receptor Stimulation by Estrogen in MDA–MB–134 Human Breast Cancer Cells Cancer Research. 46: 1124-1131. PMID 3943090  0.64
1986 Toney TW, Katzenellenbogen BS. Antiestrogen action in the medial basal hypothalamus and pituitary of immature female rats: Insights concerning relationships among estrogen, dopamine, and prolactin Endocrinology. 119: 2661-2669. PMID 3780547  0.64
1986 Mullick A, Katzenellenbogen BS. Progesterone receptor synthesis and degradation in MCF-7 human breast cancer cells as studied by dense amino acid incorporation. Evidence for a non-hormone binding receptor precursor Journal of Biological Chemistry. 261: 13236-13243. PMID 3759961  0.64
1986 Wei LL, Katzenellenbogen BS, Robertson DW, Simpson DM, Katzenellenbogen JA. Nitrosourea and nitrosocarbamate derivatives of the antiestrogen tamoxifen as potential estrogen receptor-mediated cytotoxic agents in human breast cancer cells Breast Cancer Research and Treatment. 7: 77-90. PMID 3719114 DOI: 10.1007/BF01806792  0.64
1986 Nardulli AM, Katzenellenbogen BS. Dynamics of estrogen receptor turnover in uterine cells in vitro and in uteri in vivo Endocrinology. 119: 2038-2046. PMID 3533520  0.64
1986 Berthois Y, Katzenellenbogen JA, Katzenellenbogen BS. Phenol red in tissue culture media is a weak estrogen: Implications concerning the study of estrogen-responsive cells in culture Proceedings of the National Academy of Sciences of the United States of America. 83: 2496-2500. PMID 3458212  0.64
1986 Salituro FG, Carlson KE, Elliston JF, Katzenellenbogen BS, Katzenellenbogen JA. [125I]Iododesethyl tamoxifen aziridine: Synthesis and covalent labeling of the estrogen receptor with an iodine-labeled affinity label Steroids. 48: 287-313. PMID 3445283 DOI: 10.1016/0039-128X(86)90017-6  0.64
1986 Katzenellenbogen JA, Scheeline A, Mullick A, Katzenellenbogen BS. Derivation and analysis of a lag-decay model for protein turnover involving a biosynthetic precursor Journal of Biological Chemistry. 261: 13244-13246.  0.64
1985 Sheen YY, Ruh TS, Mangel WF, Katzenellenbogen BS. Antiestrogenic Potency and Binding Characteristics of the Triphenylethylene H1285 in MCF-7 Human Breast Cancer Cells Cancer Research. 45: 4192-4199. PMID 4040807  0.64
1985 Katzenellenbogen BS, Miller MA, Mullick A, Sheen YY. Antiestrogen action in breast cancer cells: Modulation of proliferation and protein synthesis, and interaction with estrogen receptors and additional antiestrogen binding sites Breast Cancer Research and Treatment. 5: 231-243. PMID 4027393 DOI: 10.1007/BF01806018  0.64
1985 Sheen YY, Simpson DM, Katzenellenbogen BS. An evaluation of the role of antiestrogen-binding sites in mediating the growth modulatory effects of antiestrogens: Studies using t-butylphenoxyethyl diethylamine, a compound lacking affinity for the estrogen receptor Endocrinology. 117: 561-564. PMID 4017947  0.64
1985 Miller MA, Mullick A, Greene GL, Katzenellenbogen BS. Characterization of the subunit nature of nuclear estrogen receptors by chemical cross-linking and dense amino acid labeling Endocrinology. 117: 515-522. PMID 4017945  0.64
1985 Katzenellenbogen JA, Carlson KE, Katzenellenbogen BS. Facile geometric isomerization of phenolic non-steroidal estrogens and antiestrogens: Limitations to the interpretation of experiments characterizing the activity of individual isomers Journal of Steroid Biochemistry. 22: 589-596. PMID 4010284 DOI: 10.1016/0022-4731(85)90210-9  0.64
1985 Wei LL, Mangel WF, Katzenellenbogen BS. Biological activities of tamoxifen aziridine, an antiestrogen-based affinity label for the estrogen receptor, in vivo and in vitro Journal of Steroid Biochemistry. 23: 875-881. PMID 3937947 DOI: 10.1016/0022-4731(85)90042-1  0.64
1985 Reiner GCA, Katzenellenbogen BS. Dissociated regulation of growth and progesterone receptor stimulation by estrogen in MDA-MB-134 human breast cancer cells Proceedings of the American Association For Cancer Research 0.64
1984 Monsma FJ, Katzenellenbogen BS, Miller MA, Ziegler YS, Katzenellenbogen JA. Characterization of the estrogen receptor and its dynamics in MCF-7 human breast cancer cells using a covalently attaching antiestrogen. Endocrinology. 115: 143-53. PMID 6734512 DOI: 10.1210/endo-115-1-143  0.64
1984 Katzenellenbogen BS. Biology and receptor interactions of estriol and estriol derivatives in vitro and in vivo Journal of Steroid Biochemistry. 20: 1033-1037. PMID 6727348 DOI: 10.1016/0022-4731(84)90015-3  0.64
1984 Eckert RL, Mullick A, Rorke EA, Katzenellenbogen BS. Estrogen receptor synthesis and turnover in MCF-7 breast cancer cells measured by a density shift technique Endocrinology. 114: 629-637. PMID 6690295  0.64
1984 Miller MA, Greene GL, Katzenellenbogen BS. Estrogen receptor transformation in MCF-7 breast cancer cells: Characterization by immunochemical and sedimentation analyses Endocrinology. 114: 296-298. PMID 6690275  0.64
1984 Reiner GCA, Katzenellenbogen BS, Bindal RD, Katzenellenbogen JA. Biological Activity and Receptor Binding of a Strongly Interacting Estrogen in Human Breast Cancer Cells Cancer Research. 44: 2302-2308. PMID 6547074  0.64
1984 Miller MA, Lippman ME, Katzenellenbogen BS. Antiestrogen Binding in Antiestrogen Growth-resistant Estrogen-responsive Clonal Variants of MCF-7 Human Breast Cancer Cells Cancer Research. 44: 5038-5045. PMID 6488162  0.64
1984 Rorke EA, Katzenellenbogen BS. Dissociated regulation of growth and ornithine decarboxylase activity by estrogen in the rat uterus Biochemical and Biophysical Research Communications. 122: 1186-1193. PMID 6433909 DOI: 10.1016/0006-291X(84)91217-8  0.64
1984 Rorke EA, Kendra KL, Katzenellenbogen BS. Relationships among uterine growth, ornithine decarboxylase activity and polyamine levels: studies with estradiol and antiestrogens Molecular and Cellular Endocrinology. 38: 31-38. PMID 6394408 DOI: 10.1016/0303-7207(84)90142-4  0.64
1984 Katzenellenbogen JA, Katzenellenbogen BS. Affinity labeling of receptors for steroid and thyroid hormones Vitamins and Hormones. 213-274.  0.64
1983 Katzenellenbogen BS, Miller MA, Eckert RL, Sudo K. Antiestrogen pharmacology and mechanism of action Journal of Steroid Biochemistry. 19: 59-68. PMID 6887873  0.64
1983 Miller MA, Katzenellenbogen BS. Characterization and quantitation of antiestrogen binding sites in estrogen receptor-positive and -negative human breast cancer cell lines Cancer Research. 43: 3094-3100. PMID 6850618  0.64
1983 Sudo K, Monsma FJ, Katzenellenbogen BS. Antiestrogen-binding sites distinct from the estrogen receptor: subecellular localization, ligand specificity, and distribution in tissues of the rat. Endocrinology. 112: 425-34. PMID 6848356 DOI: 10.1210/endo-112-2-425  0.64
1983 Peltz SW, Katzenellenbogen BS, Kneifel MA, Mangel WF. Plasminogen activators in tissues of the immature and estrogen-stimulated rat uterus and in uterine luminal fluid: characterization and properties Endocrinology. 112: 890-897. PMID 6681601  0.64
1983 Eckert RL, Katzenellenbogen BS. Modulation of progestin binding activity in cultured human breast carcinoma cells: The effect of serum type and concentration Journal of Receptors and Signal Transduction. 3: 599-621. PMID 6672191 DOI: 10.3109/10799898309041950  0.64
1982 Eckert RL, Katzenellenbogen BS. Physical properties of estrogen receptor complexes in MCF-7 human breast cancer cells. Differences with anti-estrogen and estrogen Journal of Biological Chemistry. 257: 8840-8846. PMID 7096337  0.64
1982 Pavlik EJ, Katzenellenbogen BS. The intranuclear distribution of rat uterine estrogen receptors determined after nuclease treatment and chromatin fractionation Molecular and Cellular Endocrinology. 26: 201-216. PMID 7084560 DOI: 10.1016/0303-7207(82)90017-X  0.64
1982 Robertson DW, Katzenellenbogen JA, Long DJ, Rorke EA, Katzenellenbogen BS. Tamoxifen antiestrogens. A comparison of the activity, pharmacokinetics, and metabolic activation of the cis and trans isomers of tamoxifen. Journal of Steroid Biochemistry. 16: 1-13. PMID 7062732 DOI: 10.1016/0022-4731(82)90137-6  0.64
1982 Robertson DW, Katzenellenbogen JA, Hayes JR, Katzenellenbogen BS. Antiestrogen basicity-activity relationships: A comparison of the estrogen receptor binding and antiuterotrophic potencies of several analogues of (Z)-1,2-diphenyl-1-[4-[2-(dimethylamino)ethoxy]phenyl]-1-butene (tamoxifen, Nolvadex) having altered basicity Journal of Medicinal Chemistry. 25: 167-171. PMID 7057423  0.64
1982 Eckert RL, Katzenellenbogen BS. Effects of estrogens and antiestrogens on estrogen receptor dynamics and the induction of progesterone receptor in MCF-7 human breast cancer cells Cancer Research. 42: 139-144. PMID 7053842  0.64
1982 Hersey RM, Weisz J, Katzenellenbogen BS. Estrogenic potency, receptor interactions, and metabolism of catechol estrogens in the immature rat uterus in vitro Endocrinology. 111: 896-903. PMID 6286287  0.64
1982 Katzenellenbogen JA, Katzenellenbogen BS. Considerations in the design and evaluation of cytotoxic estrogens Breast Cancer Research and Treatment. 2: 347-353. DOI: 10.1007/BF01805876  0.64
1981 Katzenellenbogen BS, Rorke EA, Eckert RL. Mechanisms of estrogen and antiestrogen action in mammary cancer Journal of Steroid Biochemistry. 15: 219-229. PMID 7339248 DOI: 10.1016/0022-4731(81)90278-8  0.64
1981 Eckert RL, Katzenellenbogen BS. Human endometrial cells in primary tissue culture: Modulation of the progesterone receptor level by natural and synthetic estrogens in vitro Journal of Clinical Endocrinology and Metabolism. 52: 699-708. PMID 7204540  0.64
1981 Katzenellenbogen BS, Pavlik EJ, Robertson DW, Katzenellenbogen JA. Interaction of a high affinity anti-estrogen (α-[4-pyrrolidinoethoxy]phenyl-4-hydroxy-α'-nitrostilbene, CI628M) with uterine estrogen receptors Journal of Biological Chemistry. 256: 2908-2915. PMID 7204382  0.64
1981 de Boer W, Notides AC, Katzenellenbogen BS, Hayes JR, Katzenellenbogen JA. The capacity of the antiestrogen CI-628 to activate the estrogen receptor in vitro Endocrinology. 108: 206-212. PMID 7007019  0.64
1981 Hayes JR, Rorke EA, Robertson DW, Katzenellenbogen BS, Katzenellenbogen JA. Biological potency and uterine estrogen receptor interaction of the metabolites of the antiestrogens CI628 and U23,469 Endocrinology. 108: 164-172. PMID 7007017  0.64
1981 Kneifel MA, Katzenellenbogen BS. Comparative effects of estrogen and antiestrogen on plasma renin substrate levels and hepatic estrogen receptors in the rat Endocrinology. 108: 545-552. PMID 7004858  0.64
1981 Rorke EA, Katzenellenbogen BS. Antitumor Activities and Estrogen Receptor Interactions of the Metabolites of the Antiestrogens CI628 and U23,469 in the 7,12-Dimethylbenz(a)anthracene-Induced Rat Mammary Tumor System Cancer Research. 41: 1257-1262. PMID 6783294  0.64
1980 Pavlik EJ, Katzenellenbogen BS. The stability of the uterine estrogen receptor when complexed with estrogens or antiestrogens Molecular Pharmacology. 18: 406-412. PMID 7464805  0.64
1980 Katzenellenbogen BS, Lan NC, Rutledge SK. Estrogen receptors of human endometrium: characterization of nuclear and cytoplasmic forms and comparisons with rat uterine receptors Journal of Steroid Biochemistry. 13: 113-122. PMID 7382488 DOI: 10.1016/0022-4731(80)90181-8  0.64
1980 Katzenellenbogen BS. Dynamics of steroid hormone receptor action Annual Review of Physiology. 17-35. PMID 6996577  0.64
1980 Rorke EA, Katzenellenbogen BS. Comparative Effects of Estrogen and Antiestrogens on Enzyme Activities in R3230AC Rat Mammary Tumors and Uteri of Tumor-bearing Animals Cancer Research. 40: 3158-3162. PMID 6253055  0.64
1980 Eckert RL, Katzenellenbogen BS. The effects of estrogens and antiestrogens on estrogen receptor dynamics and induction of progesterone receptor in MCF-7 human breast cancer cells Journal of Cell Biology. 87.  0.64
1980 Eckert RL, Katzenellenbogen BS. Human endometrial cells in primary tissue culture: Modulation of progesterone receptor level by estrogens in vitro Biology of Reproduction. 22.  0.64
1979 Tatee T, Carlson KE, Katzenellenbogen JA, Robertson DW, Katzenellenbogen BS. Antiestrogens and antiestrogen metabolites: Preparation of tritium-labeled (±)-cis-3-[p-(1,2,3,4-tetrahydro-6-methoxy-2-phenyl-1-naphthyl)phenoxy]- 1,2-propanediol (U-23469) and characterization and synthesis of a biologically important metabolite Journal of Medicinal Chemistry. 22: 1509-1517. PMID 536996  0.64
1979 Schmidt WN, Katzenellenbogen BS. Androgen-uterine interactions: An assessment of androgen interaction with the testosterone- and estrogen-receptor systems and stimulation of uterine growth and progesterone-receptor synthesis Molecular and Cellular Endocrinology. 15: 91-108. PMID 499651 DOI: 10.1016/0303-7207(79)90010-8  0.64
1979 Pavlik EJ, Rutledge S, Eckert RL, Katzenellenbogen BS. Localization of estrogen receptors in uterine cells. An appraisal of translocation Experimental Cell Research. 123: 177-189. PMID 488181 DOI: 10.1016/0014-4827(79)90434-8  0.64
1979 Katzenellenbogen BS, Tsai TS, Tatee T, Katzenellenbogen JA. Estrogen and antiestrogen action: studies in reproductive target tissues and tumors Advances in Experimental Medicine and Biology. 117: 111-132. PMID 474274  0.64
1979 Katzenellenbogen BS, Katzenellenbogen JA, Mordecai D. Zearalenones: Characterization of the estrogenic potencies and receptor interactions of a series of fungal β-resorcylic acid lactones Endocrinology. 105: 33-40. PMID 446414  0.64
1979 Navickis RJ, Katzenellenbogen BS, Nalbandov AV. Effects of the sex steroid hormones and vitamin D3 on calcium-binding proteins in the chick shell gland. Biology of Reproduction. 21: 1153-62. PMID 229921  0.64
1979 Tsai TLS, Rutledge S, Katzenellenbogen BS. Antiestrogen Modulation of the Growth and Properties of Ovarian-Autonomous and Ovarian-Dependent Mammary Tumors in Rats Cancer Research. 39: 5043-5050. PMID 227594  0.64
1979 Navickis RJ, Dial OK, Katzenellenbogen BS, Nalbandov AV. Effects of gonadal hormones on calcium-binding protein in chick duodenum. The American Journal of Physiology. 237: E408-17. PMID 227275  0.64
1979 Hammond B, Katzenellenbogen BS, Krauthammer N, McConnell J. Estrogenic activity of the insecticide chlordecone (Kepone) and interaction with uterine estrogen receptors Proceedings of the National Academy of Sciences of the United States of America. 76: 6641-6645. PMID 93289  0.64
1978 Katzenellenbogen BS, Katzenellenbogen JA, Ferguson ER, Krauthammer N. Anti-estrogen interaction with uterine estrogen receptors. Studies with a radiolabeled anti-estrogen (CI-628) Journal of Biological Chemistry. 253: 697-707. PMID 621199  0.64
1978 Katzenellenbogen BS, Iwamoto HS, Heiman DF, Lan NC, Katzenellenbogen JA. Stilbestrols and stilbestrol derivatives: Estrogenic potency and temporal relationships between estrogen receptor binding and uterine growth Molecular and Cellular Endocrinology. 10: 103-113. PMID 564791 DOI: 10.1016/0303-7207(78)90063-1  0.64
1978 Pavlik EJ, Katzenellenbogen BS. Human endometrial cells in primary tissue culture: Estrogen interactions and modulation of cell proliferation Journal of Clinical Endocrinology and Metabolism. 47: 333-344. PMID 263301  0.64
1977 Bhakoo HS, Katzenellenbogen BS. Progesterone modulation of estrogen-stimulated uterine biosynthetic events and estrogen receptor levels Molecular and Cellular Endocrinology. 8: 121-134. PMID 924010 DOI: 10.1016/0303-7207(77)90024-7  0.64
1977 Katzenellenbogen BS, Ferguson ER, Lan NC. Fundamental differences in the action of estrogens and antiestrogens on the uterus: comparison between compounds with similar duration of action Endocrinology. 100: 1252-1259. PMID 849722  0.64
1977 Ferguson ER, Katzenellenbogen BS. A comparative study of antiestrogen action: temporal patterns of antagonism of estrogen stimulated uterine growth and effects on estrogen receptor levels Endocrinology. 100: 1242-1251. PMID 849721  0.64
1977 Tsai TLS, Katzenellenbogen BS. Antagonism of Development and Growth of 7, 12-Dimethylbenz(a)anthracene-induced Rat Mammary Tumors by the Antiestrogen U 23, 469 and Effects on Estrogen and Progesterone Receptors Cancer Research. 37: 1537-1543. PMID 404032  0.64
1977 Bhakoo HS, Katzenellenbogen BS. Progesterone antagonism of estradiol-stimulated uterine 'induced protein' synthesis Molecular and Cellular Endocrinology. 8: 105-120. PMID 72697 DOI: 10.1016/0303-7207(77)90023-5  0.64
1976 Schmidt WN, Sadler MA, Katzenellenbogen BS. Androgen uterine interaction: nuclear translocation of the estrogen receptor and induction of the synthesis of the uterine induced protein (IP) by high concentrations of androgens in vitro but not in vivo Endocrinology. 98: 702-716. PMID 177269  0.64
1976 Lan NC, Katzenellenbogen BS. Temporal relationships between hormone receptor binding and biological responses in the uterus: studies with short and long acting derivatives of estriol Endocrinology. 98: 220-227. PMID 174891  0.64
1975 Katzenellenbogen BS, Gorski J. [38] Methods for assessing estrogen effects on new uterine protein synthesis In Vitro Methods in Enzymology. 36: 444-455. PMID 1110635 DOI: 10.1016/S0076-6879(75)36041-2  0.64
1975 Katzenellenbogen BS, Ferguson ER. Antiestrogen action in the uterus: biological ineffectiveness of nuclear bound estradiol after antiestrogen Endocrinology. 97: 1-12. PMID 166821  0.64
1975 Katzenellenbogen BS. Synthesis and inducibility of the uterine estrogen induced protein, IP, during the rat estrous cycle: clues to uterine estrogen sensitivity Endocrinology. 96: 289-297. PMID 163181  0.64
1974 Katzenellenbogen BS, Greger NG. Ontogeny of uterine responsiveness to estrogen during early development in the rat Molecular and Cellular Endocrinology. 2: 31-42. PMID 4455530 DOI: 10.1016/0303-7207(74)90010-0  0.64
1974 Katzenellenbogen BS, Leake RE. Distribution of the oestrogen induced protein and of total protein between endometrial and myometrial fractions of the immature and mature rat uterus Journal of Endocrinology. 63: 439-449. PMID 4452816  0.64
1974 Katzenellenbogen BS, Williams LB. Uterine estrogen induced protein: physical and immunological comparison with ovalbumin Proceedings of the National Academy of Sciences of the United States of America. 71: 1281-1285. PMID 4133849  0.64
1973 Ruh TS, Katzenellenbogen BS, Katzenellenbogen JA, Gorski J. Estrone interaction with the rat uterus: in vitro response and nuclear uptake Endocrinology. 92: 125-134. PMID 4681918  0.64
1972 Katzenellenbogen BS, Gorski J. Estrogen action in vitro. Induction of the synthesis of a specific uterine protein Journal of Biological Chemistry. 247: 1299-1305. PMID 4335193  0.64
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